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Title:
N-(2-ARYLETHYL)BENZYLAMINES AS ANTAGONISTS OF THE 5-HT6 RECEPTOR
Document Type and Number:
WIPO Patent Application WO2002078693
Kind Code:
A3
Abstract:
The present invention provides compounds of formula (I), which are antagonists of the 5-HT6 receptor.

Inventors:
CHEN ZHAOGEN (US)
COHEN MICHAEL PHILIP (US)
FISHER MATTHEW JOSEPH (US)
GIETHLEN BRUNO (FR)
GILLIG JAMES RONALD (US)
MCCOWAN JEFFERSON RAY (US)
MILLER SHAWN CHRISTOPHER (US)
SCHAUS JOHN MEHNERT (US)
Application Number:
PCT/US2002/005115
Publication Date:
December 05, 2002
Filing Date:
March 15, 2002
Export Citation:
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Assignee:
LILLY CO ELI (US)
CHEN ZHAOGEN (US)
COHEN MICHAEL PHILIP (US)
FISHER MATTHEW JOSEPH (US)
GIETHLEN BRUNO (FR)
GILLIG JAMES RONALD (US)
MCCOWAN JEFFERSON RAY (US)
MILLER SHAWN CHRISTOPHER (US)
SCHAUS JOHN MEHNERT (US)
International Classes:
A61K31/137; A61K31/18; A61K31/343; A61K31/381; A61K31/4045; A61K31/417; A61K31/426; A61K31/427; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4439; A61K31/505; A61K31/506; A61P25/18; A61P25/22; A61P25/28; C07C211/52; C07C211/56; C07C215/32; C07D233/64; C07C215/50; C07C217/58; C07C217/60; C07C225/16; C07C309/73; C07C311/37; C07C317/32; C07C317/34; C07C323/32; C07D209/00; C07D209/08; C07D209/14; C07D209/16; C07D209/86; C07D213/30; C07D213/38; C07D213/63; C07D213/64; C07D213/65; C07D213/68; C07D213/74; C07D233/24; C07D239/34; C07D277/20; C07D277/34; C07D307/91; C07D333/20; C07D401/12; C07D403/06; C07D403/12; C07D405/12; C07D417/12; C07D471/04; C07F7/08; (IPC1-7): A61K31/4045; C07D209/16; A61P25/18; A61P25/28; C07D403/12; C07D401/12; A61K31/4406; A61K31/4409; A61K31/506; A61K31/4402; C07C217/54; C07C323/01; C07C317/14; C07D213/64; C07D277/34; C07D239/34; C07D233/24; C07D333/20; C07D307/91; C07D209/14
Domestic Patent References:
WO2000034242A12000-06-15
Foreign References:
US6187805B12001-02-13
Other References:
DATABASE CROSSFIRE BEILSTEIN [online] Beilstein Institut zur Förderung der Chemischen Wissenschaften, Frankfurt am Main, DE; IDE, BUCK, XP002209139, Database accession no. 3365864
DATABASE CROSSFIRE BEILSTEIN [online] Beilstein Institut zur Förderung der Chemischen Wissenschaften, Frankfurt am Main, DE; XP002209140, Database accession no. 3365863
DATABASE CROSSFIRE BEILSTEIN [online] Beilstein Institut zur Förderung der Chemischen Wissenschaften, Frankfurt am Main, DE; IDE, BUCK, XP002209141, Database accession no. 3380345
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