N-ALKYLATED GABA COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS

Title:

N-ALKYLATED GABA COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS MEDICAMENTS

Document Type and Number:

WIPO Patent Application WO2002042256

Kind Code:

A3

Abstract:

The present invention relates to N-alkylated GABA (Gamma-aminobutyric acid) compounds of Formula I, to processes for their preparation, to their use in therapy and to pharmaceutical compositions containing them. More particularly these compounds are useful for treatment of disorders of the central and/or peripheral nervous system. Of particular interest is their potent anticonvulsant activity.

Inventors:

KENDA BENOIT (BE)
MICHEL PHILIPPE (BE)
QUERE LUC (BE)

Application Number:

PCT/EP2001/013162

Publication Date:

May 01, 2003

Filing Date:

November 14, 2001

Export Citation:

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Assignee:

UCB SA (BE)
KENDA BENOIT (BE)
MICHEL PHILIPPE (BE)
QUERE LUC (BE)

International Classes:

A61K31/16; A61K31/197; A61P25/00; C07C237/06; C07C327/22; (IPC1-7): C07C237/06; A61K31/195; A61K31/22; A61P25/00

Foreign References:

US4639468A	1987-01-27
EP0165919A1	1985-12-27
EP0162036A1	1985-11-21
GB2126224A	1984-03-21

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