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Title:
N-SUBSTITUTED BENZENE SULFONAMIDES
Document Type and Number:
WIPO Patent Application WO2005090296
Kind Code:
A3
Abstract:
The invention provides N-substituted benzenesulfonamides for use in treating or preventing cognitive disorders, such as Alzheimer's Disease. Compounds of particular interest are defined by Formula (I), wherein R1, R2, R3, R4, and R3, are as described in the specification. The invention also encompasses pharmaceutical compositions comprising compounds of Formula (I) as well as methods of treating cognitive disorders, including Alzheimer's disease using compounds of Formula (I).

Inventors:
NEITZEL MARTIN (US)
MARUGG JENNIFER (US)
Application Number:
PCT/US2005/007811
Publication Date:
November 24, 2005
Filing Date:
March 11, 2005
Export Citation:
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Assignee:
ELAN PHARM INC (US)
NEITZEL MARTIN (US)
MARUGG JENNIFER (US)
International Classes:
A61K31/185; A61K31/4172; A61K31/426; A61K31/445; C07C311/15; C07C311/16; C07C311/17; C07C311/18; C07C311/19; C07C311/20; C07C311/21; C07C311/31; C07C311/51; C07C317/32; C07D209/14; C07D211/58; C07D231/06; C07D277/24; C07D307/52; C07D307/81; (IPC1-7): C07C311/15; A61K31/18; A61P25/28
Domestic Patent References:
WO2003103660A12003-12-18
WO2003053912A12003-07-03
Foreign References:
CH246983A1947-02-15
Other References:
DATABASE BEILSTEIN Beilstein Institut zur Förderung der Chemischen Wissenschaften, Frankfurt am Main, DE; XP002343799, Database accession no. BRN 2149884
DATABASE BEILSTEIN Beilstein Institut zur Förderung der Chemischen Wissenschaften, Frankfurt am Main, DE; XP002343800, Database accession no. 6432097
DATABASE BEILSTEIN Beilstein Institut zur Förderung der Chemischen Wissenschaften, Frankfurt am Main, DE; XP002343801, Database accession no. BRN 2128431
DATABASE BEILSTEIN Beilstein Institut zur Förderung der Chemischen Wissenschaften; XP002343802, Database accession no. BRN 2136785
DATABASE BEILSTEIN Beilstein Institut zur Förderung der Chemischen Wissenschaften, Frankfurt am Main, DE; XP002343803, Database accession no. BRN 2852299
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