Title:
NAPHTHALIMIDOBENZAMIDE DERIVATIVES
Document Type and Number:
WIPO Patent Application WO/2000/001672
Kind Code:
A1
Abstract:
Naphthalimidobenzamide derivatives represented by general formula (1) or salts thereof; and drugs containing both as the active ingredient: (wherein R?1¿ is hydrogen or the like; Y is hydrogen or -CON(R?4¿)-A?2¿-X?2¿; R?2¿ and R?4¿ are each independently hydrogen or the like; A?1¿ and A?2¿ are each independently alkylene which may be interrupted by -N(R?3¿)- (wherein R?3¿ is hydrogen or the like) at one or more positions; and X?1¿ and X?2¿ are each independently optionally substituted (hetero)aryl or the like). These compounds are useful as antitumor agents and so on.
Inventors:
NOGUCHI KAZUHARU (JP)
WAKIDA MOTOJI (JP)
SUZUKI KENJI (JP)
YAMADA YUJI (JP)
ASAO TETSUJI (JP)
WAKIDA MOTOJI (JP)
SUZUKI KENJI (JP)
YAMADA YUJI (JP)
ASAO TETSUJI (JP)
Application Number:
PCT/JP1999/003574
Publication Date:
January 13, 2000
Filing Date:
July 02, 1999
Export Citation:
Assignee:
TAIHO PHARMACEUTICAL CO LTD (JP)
NOGUCHI KAZUHARU (JP)
WAKIDA MOTOJI (JP)
SUZUKI KENJI (JP)
YAMADA YUJI (JP)
ASAO TETSUJI (JP)
NOGUCHI KAZUHARU (JP)
WAKIDA MOTOJI (JP)
SUZUKI KENJI (JP)
YAMADA YUJI (JP)
ASAO TETSUJI (JP)
International Classes:
C07D221/14; C07D401/14; C07D471/04; C07D519/00; (IPC1-7): C07D221/14; C07D401/12; C07D401/14; A61K31/47; A61K31/495; A61K31/535
Domestic Patent References:
| WO1993012092A1 | 1993-06-24 | |||
| WO1992017453A1 | 1992-10-15 | |||
| WO1991009850A1 | 1991-07-11 |
Foreign References:
| EP0125439A2 | 1984-11-21 |
Other References:
See also references of EP 1020446A4
Attorney, Agent or Firm:
Aruga, Mitsuyuki (Nihonbashiningyocho 1-chome Chuo-ku Tokyo, JP)
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