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Title:
NEW (HETERO)ARYL-SUBSTITUTED-PIPERIDINYL DERIVATIVES, A PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
Document Type and Number:
WIPO Patent Application WO/2017/212010
Kind Code:
A1
Abstract:
Compounds of formula (I) wherein R1, R2, J, K, L, n and W are as defined in the description. Medicaments.

Inventors:
KOTSCHY ANDRÁS (HU)
WÉBER CSABA (HU)
VASAS ATTILA (HU)
MOLNÁR BALÁZS (HU)
KISS ÁRPÁD (HU)
MACIAS ALBA (GB)
MURRAY JAMES BROOKE (GB)
LEWKOWICZ ELODIE (FR)
GENESTE OLIVIER (FR)
CHANRION MAÏA (FR)
DEMARLES DIDIER (FR)
IVANSCHITZ LISA (FR)
Application Number:
PCT/EP2017/064062
Publication Date:
December 14, 2017
Filing Date:
June 09, 2017
Export Citation:
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Assignee:
SERVIER LAB (FR)
VERNALIS R&D LTD (GB)
International Classes:
C07D471/04; A61K31/519; A61P35/00; C07D487/04; C07D495/04
Domestic Patent References:
WO2013030218A12013-03-07
WO2008108957A22008-09-12
Other References:
EDELMAN ET AL., EXPERT REV. MOL. MED., vol. 13, 2011, pages 1 - 17
PAL ET AL., CANCER RES., vol. 74, 2014, pages 4955 - 4966
LUISE ET AL., PLOS ONE, vol. 6, 2011, pages e15891
ROLEN ET AL., MOL. CARCINOG., vol. 45, 2006, pages 260 - 269
NICHOLSON ET AL., CELL BIOCHEM. BIOPHYS., vol. 60, 2011, pages 61 - 68
VAN LOOSDREGT ET AL., IMMUNITY, vol. 39, 2013, pages 259 - 27
COLLERAN ET AL., PROC. NATL. ACAD. SCI. USA, vol. 110, 2013, pages 618 - 623
HAO ET AL., MOL. CELL, vol. 59, 2015, pages 956 - 969
HOLOWATY ET AL., BIOCHEM. SOC. TRANS., vol. 32, 2004, pages 731 - 732
KEMP ET AL., PROGRESS IN MEDICINAL CHEMISTRY, vol. 55, 2016, pages 149 - 192
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