NOVEL DERIVATIVES OF ANDROSTANE AND ANDROSTENE WITH ASCORBIC A CID AND USE THEREOF IN TREATING OR PREVENTING VARIOUS CONDITIONS, DISEASES, AND DISORDERS

Title:

NOVEL DERIVATIVES OF ANDROSTANE AND ANDROSTENE WITH ASCORBIC A CID AND USE THEREOF IN TREATING OR PREVENTING VARIOUS CONDITIONS, DISEASES, AND DISORDERS

Document Type and Number:

WIPO Patent Application WO2003104254

Kind Code:

A3

Abstract:

The present invention provides novel derivatives comprising compounds in the androstane and androstene series, coupled with ascorbic acid, including salts thereof, and represented by one or more of the general formulae (I), (II), (III): wherein R1, R2, R3, R4, R5, R6 may individually be chosen from hydrogen, OH, carbonyl, and an ascorbyl moiety; and R7 may be hydrogen or any halogen.

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Inventors:

KUTNEY JAMES P
CHEN HONGMING
HOU DUANJIE
WANG CHANGQING

Application Number:

PCT/CA2003/000824

Publication Date:

May 06, 2004

Filing Date:

June 06, 2003

Export Citation:

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Assignee:

FORBES MEDI TECH INC (CA)

International Classes:

A61K31/58; A61K31/585; A61K31/663; A61K47/48; A61K31/6615; A61P3/04; A61P3/06; A61P3/10; A61P9/00; A61P29/00; A61P35/00; A61P37/04; C07J1/00; C07J17/00; C07J19/00; (IPC1-7): C07J1/00; C07J19/00; A61K31/58; A61P3/04

Domestic Patent References:

WO2003035023A1	2003-05-01
WO2003026672A1	2003-04-03
WO2001000653A1	2001-01-04

Foreign References:

EP0665238A1	1995-08-02
US5318987A	1994-06-07

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