Title:
NOVEL HETEROARYL AND HETEROCYCLE COMPOUNDS, COMPOSITIONS AND METHODS
Document Type and Number:
WIPO Patent Application WO/2016/119707
Kind Code:
A1
Abstract:
The invention relates to novel heteroaryl and heterocycle compounds of formula I and pharmaceutical compositions comprising them, uses and methods thereof for inhibiting the activity of PI3K and for treating inflammatory and autoimmune diseases and cancer.
Inventors:
SU WEI-GUO (CN)
DAI GUANGXIU (CN)
JIA HONG (CN)
ZHANG ZHULIN (CN)
WENG JIANYANG (CN)
VENABLE JENNIFER DIANE (US)
BEMBENEK SCOTT DAMIAN (US)
CHAI WENYING (US)
MEDUNA STEVEN PAUL (US)
KEITH JOHN MATTHEW (US)
ECCLES WENDY (US)
LEBSACK ALEC DONALD (US)
JONES WILLIAM MOORE (US)
SMITH RUSSELL CHRISTOPHER (US)
DAI GUANGXIU (CN)
JIA HONG (CN)
ZHANG ZHULIN (CN)
WENG JIANYANG (CN)
VENABLE JENNIFER DIANE (US)
BEMBENEK SCOTT DAMIAN (US)
CHAI WENYING (US)
MEDUNA STEVEN PAUL (US)
KEITH JOHN MATTHEW (US)
ECCLES WENDY (US)
LEBSACK ALEC DONALD (US)
JONES WILLIAM MOORE (US)
SMITH RUSSELL CHRISTOPHER (US)
Application Number:
PCT/CN2016/072474
Publication Date:
August 04, 2016
Filing Date:
January 28, 2016
Export Citation:
Assignee:
HUTCHISON MEDIPHARMA LTD (CN)
International Classes:
C07D473/34; A61K31/437; A61P35/00; C07D487/04
Domestic Patent References:
WO2014015830A1 | 2014-01-30 |
Attorney, Agent or Firm:
ZHONGZI LAW OFFICE (26 Pinganli Xidajie Xicheng District, Beijing 4, CN)
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