Title:
NOVEL M-AMINO-PHENYLIMINO-IMIDAZOLIDINE DERIVATIVES FOR TREATING URINARY INCONTINENCE
Document Type and Number:
WIPO Patent Application WO2002032876
Kind Code:
A3
Abstract:
The invention relates to m-amino-phenylimino-imidazolidine derivatives with a novel substituent pattern on the phenyl ring, of general formula (I) or of general formula (II), wherein R1 is F, Cl, Br, CH2F, CF2H or CF3, R2 is NR6R7, R6 being Me, Et, Pr or iPr and R7 being Me, Et or Pr; and R3, R4 and R5 are each, independently of each other, H, Me, F, Cl, Br, CH2F, CF2H and/or CF3 and if R4 is Me, F, Cl, Br, CH2F, CF2H or CF3, then R1 is additionally also H or Me; and or their pharmacologically compatible salts, to the use thereof for producing medicaments, especially for treating urinary incontinence, and to a method for producing the same.
Inventors:
ESSER FRANZ
POUZET PASCALE ARIELLE JANE-JO
KITAGAWA HISATO
SAKAI KENJI
MURAMATSU IKUNOBU
POUZET PASCALE ARIELLE JANE-JO
KITAGAWA HISATO
SAKAI KENJI
MURAMATSU IKUNOBU
Application Number:
PCT/EP2001/011764
Publication Date:
July 18, 2002
Filing Date:
October 11, 2001
Export Citation:
Assignee:
BOEHRINGER INGELHEIM PHARMA (DE)
International Classes:
A61K31/4168; A61P13/00; A61P13/10; C07D233/50; (IPC1-7): C07D233/50; A61K31/415; A61P13/00
Domestic Patent References:
| WO1996032939A1 | 1996-10-24 |
Foreign References:
| EP0081924A1 | 1983-06-22 | |||
| DE2806811A1 | 1979-08-23 |
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