Title:
NOVEL MCH RECEPTOR ANTAGONISTS
Document Type and Number:
WIPO Patent Application WO2006066173
Kind Code:
A3
Abstract:
The present invention relates to a melanin concentrating hormone antagonist compound of formula (I); wherein Ar1, L1, R1, q, X, R2, R3, R4, and R5 are as defined, or a pharmaceutically acceptable salt, solvate, or enantiomer thereof useful in the treatment, prevention or amelioration of symptoms associated with obesity and related diseases.
Inventors:
BECK JAMES PETER (US)
WAKEFIELD BRIAN DAVID (US)
CORDIER FREDERIC LAURENT (ES)
DOMINGUEZ-MANZANARES ESTEBAN (ES)
GARDINIER KEVIN MATTHEW (US)
GREENEN PETER MICHAEL (US)
SAVIN KENNETH ALLEN (US)
WAKEFIELD BRIAN DAVID (US)
CORDIER FREDERIC LAURENT (ES)
DOMINGUEZ-MANZANARES ESTEBAN (ES)
GARDINIER KEVIN MATTHEW (US)
GREENEN PETER MICHAEL (US)
SAVIN KENNETH ALLEN (US)
Application Number:
PCT/US2005/045864
Publication Date:
July 27, 2006
Filing Date:
December 16, 2005
Export Citation:
Assignee:
LILLY CO ELI (US)
BECK JAMES PETER (US)
WAKEFIELD BRIAN DAVID (US)
CORDIER FREDERIC LAURENT (ES)
DOMINGUEZ-MANZANARES ESTEBAN (ES)
GARDINIER KEVIN MATTHEW (US)
GREENEN PETER MICHAEL (US)
SAVIN KENNETH ALLEN (US)
BECK JAMES PETER (US)
WAKEFIELD BRIAN DAVID (US)
CORDIER FREDERIC LAURENT (ES)
DOMINGUEZ-MANZANARES ESTEBAN (ES)
GARDINIER KEVIN MATTHEW (US)
GREENEN PETER MICHAEL (US)
SAVIN KENNETH ALLEN (US)
International Classes:
C07D417/04; A61K31/41; A61K31/435; A61K31/495; A61P3/04; A61P3/06; A61P3/10; C07D263/58; C07D277/68; C07D277/82; C07D413/04; C07D413/12; C07D417/14
Domestic Patent References:
WO2004011440A1 | 2004-02-05 | |||
WO2001057008A1 | 2001-08-09 | |||
WO2002042273A2 | 2002-05-30 | |||
WO2004063155A1 | 2004-07-29 | |||
WO2003049702A2 | 2003-06-19 |
Foreign References:
EP1553089A1 | 2005-07-13 |
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