NOVEL PENAM DERIVATIVES OR SALTS THEREOF, PHARMACEUTICAL COMPOSITIONS AND USE THEREOF

WIPO Patent Application WO/2019/194306

A1

The problem addressed by the present invention is to provide compounds and pharmaceutical compositions that demonstrate strong antibacterial activity against gram-negative bacteria and drug-resistant gram-negative bacteria. Compounds represented by general formula [1] (in the formula, each symbol is as described in the specification.) or salts thereof have strong antibacterial activity against gram-negative bacteria, including Pseudomonas aeruginosa, and drug-resistant gram-negative bacteria, including multidrug-resistant Pseudomonas aeruginosa, and pharmaceutical compositions containing these compounds or salts are useful as antimicrobials.

SHOJI MUNEO (JP)
FURUYA KENTARO (JP)
MATSUURA KEI (JP)
NAKAE TOMOFUMI (JP)

PCT/JP2019/015176

October 10, 2019

April 05, 2019

Click for automatic bibliography generation  

FUJIFILM CORP (JP)

C07D499/00; A61K31/431; A61K31/4439; A61K31/497; A61P31/04

JPH0474182A	1992-03-09
JPH10130272A	1998-05-19
JPH072870A	1995-01-06
JPS63183588A	1988-07-28
JPH0474182A	1992-03-09
JPH10182654A	1998-07-07
US5185330A	1993-02-09

ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, vol. 52, 2008, pages 813 - 821
SCIENTIFIC REPORTS, no. 24, 2017
INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS, vol. 43, 2014, pages 533 - 539
W. GREENE ET AL.: "Protective Groups in Organic Synthesis", 2007, JOHN WILEY & SONS, INC., pages: 533 - 643
See also references of EP 3778609A4

SIKS & CO. (JP)

View/Download PDF      PDF Help

Previous Patent: SCANNING ELECTRON MICROSCOPE SYSTEM AND DEPTH MEASUREMENT METHOD FOR PATTERN

Next Patent: IMAGING DEVICE AND IMAGE TRANSMISSION/RECORDING SYSTEM