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Title:
NUCLEOSIDE DERIVATIVE AND USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2017/047594
Kind Code:
A1
Abstract:
Provided is a nucleoside derivative represented by formula (1). (In formula (1), Y represents an unfused aromatic or heterocyclic hydrocarbon group or a fused polycyclic based hydrocarbon group, W1 represents a hydrogen atom, a hydroxyl group-protecting group, or a phosphate ester group, W2 represents a hydrogen atom, a hydroxyl group-protecting group, or a phosphate ester group, and R1, R2, and R3 each independently represent a hydrogen atom or a linear saturated hydrocarbon group having 1-4 carbon atoms.)

Inventors:
UENO YOSHIHITO (JP)
Application Number:
PCT/JP2016/077006
Publication Date:
March 23, 2017
Filing Date:
September 13, 2016
Export Citation:
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Assignee:
UNIV GIFU (JP)
International Classes:
C07D239/47; A61K31/7088; A61K48/00; A61P43/00; C07D239/54; C07D473/18; C07D473/34; C07H21/02; C07H21/04; C12N15/09
Domestic Patent References:
WO1997029077A11997-08-14
WO2007094135A12007-08-23
WO2011071078A12011-06-16
Foreign References:
JPH02161422A1990-06-21
EP0665223A11995-08-02
JP2010189276A2010-09-02
Other References:
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BREDIHHINA, J. ET AL.: "Hydrolytic and Aminolytic Kinetic Resolution of Terminal Bis- Epoxides", J. ORG. CHEM., vol. 78, no. 6, 2013, pages 2379 - 2385, XP055372559, ISSN: 0022-3263
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SHIN, S. H. ET AL.: "An Easy and Covenient Synthesis of Optically Active beta-Amino Alcohols and 1,2-Diamines. Applications in Enantioselective Deprotonation of Cyclohexene Oxide", BULL. KOREAN CHEM. SOC., vol. 24, no. 11, 2003, pages 1695 - 1698, XP055372565, ISSN: 0253-2964
DATABASE REGISTRY 16 November 1984 (1984-11-16), retrieved from STN Database accession no. 65446-03-9
DATABASE REGISTRY 18 December 1984 (1984-12-18), retrieved from STN Database accession no. 93727-38-9
DATABASE REGISTRY 3 June 2015 (2015-06-03), retrieved from STN Database accession no. 1772627-66-3
DATABASE REGISTRY 8 October 2010 (2010-10-08), retrieved from STN Database accession no. 1245831-23-5
Attorney, Agent or Firm:
KAI-U PATENT LAW FIRM (JP)
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