Title:
OXONE-ACETONE MEDIATED METAL FREE PREPARATION OF SYN-DIOLS
Document Type and Number:
WIPO Patent Application WO/2014/207766
Kind Code:
A9
Abstract:
The present invention disclose a simple and high yielding process of Oxone-acetone mediated metal free syn-dihydroxylation of benzo fused olefins of formula (II) to obtain library of dioxolo compounds of formula (I). The invention further disclsoe a simple and high yielding process of Oxone-acetone mediated metal free syn-dihydroxylation of stilbene and its derivatives of formula (III) thereof. Also disclosed herein is Wacker-type oxidation of benzo-fused olefins of formula (X). The invention further disclose compounds of formula (I) which can be useful for the treatment of HIV, cancer or malaria.
Inventors:
RAMANA CHEPURI VENKATA (IN)
PHATAKE RAVINDRA SURESH (IN)
PHATAKE RAVINDRA SURESH (IN)
Application Number:
PCT/IN2014/000425
Publication Date:
March 19, 2015
Filing Date:
June 25, 2014
Export Citation:
Assignee:
COUNCIL SCIENT IND RES (IN)
International Classes:
C07D317/12; A61K31/352; A61K31/357; A61P31/18; A61P33/06; A61P35/00; C07C13/38; C07D317/70; C07D493/04
Attorney, Agent or Firm:
KOUL, Sunaina et al. (Plot No. B-28 Sector-32,Institutional Area, Gurgaon 1, IN)
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