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Title:
PEPTIDE COMPOUND AND PHARMACEUTICAL COMPOSITIONS AND MEDICINES CONTAINING THE SAME AS THE ACTIVE INGREDIENT
Document Type and Number:
WIPO Patent Application WO/2002/000688
Kind Code:
A1
Abstract:
Peptide compound (I) or pharmacologically acceptable salts thereof exhibit selective antagonism against oxytocin receptor more than against vasopressin receptor and are effective in the prevention or treatment of threatened premature delivery.

Inventors:
Inoue, Takashi (102 20-1, Hirado 3-chome Totsuka-ku Yokohama-shi Kanagawa, Hirado 3-chome Totsuka-ku Yokohama-shi Kanagawa, 244-0802, JP)
Nakanishi, Akihiro (1-14, Suwacho 2-chome Arai-shi, Niigata, 944-0018, JP)
Kamiya, Seiji (Mitsubishi-Tokyo Pharmaceuticals, Inc. Kazusa Research Center 100-5 Yana, Kisarazu-shi Chiba, 292-0812, JP)
Ohno, Norio (Mitsubishi-Tokyo Pharmaceuticals, Inc. 2-6 Nihonbashi-Honcho 2-chome Chuo-ku, Tokyo, 103-8405, JP)
Application Number:
PCT/JP2001/005461
Publication Date:
January 03, 2002
Filing Date:
June 26, 2001
Export Citation:
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Assignee:
DAICEL CHEMICAL INDUSTRIES, LTD. (1 Teppocho Sakai-shi Osaka, 590-0905, JP)
MITSUBISHI-TOKYO PHARMACEUTICALS, INC. (2-6 Nihonbashi-Honcho 2-chome Chuo-ku Tokyo, 103-8405, JP)
Inoue, Takashi (102 20-1, Hirado 3-chome Totsuka-ku Yokohama-shi Kanagawa, Hirado 3-chome Totsuka-ku Yokohama-shi Kanagawa, 244-0802, JP)
Nakanishi, Akihiro (1-14, Suwacho 2-chome Arai-shi, Niigata, 944-0018, JP)
Kamiya, Seiji (Mitsubishi-Tokyo Pharmaceuticals, Inc. Kazusa Research Center 100-5 Yana, Kisarazu-shi Chiba, 292-0812, JP)
Ohno, Norio (Mitsubishi-Tokyo Pharmaceuticals, Inc. 2-6 Nihonbashi-Honcho 2-chome Chuo-ku, Tokyo, 103-8405, JP)
International Classes:
A61K38/11; A61P5/12; A61P15/06; C07K7/06; C07K7/16; A61K38/00; A61K38/10; A61P5/00; A61P15/00; C07K7/00; A61K38/00; (IPC1-7): C07K7/16; A61K38/08; A61P15/06
Attorney, Agent or Firm:
Miura, Yoshikazu (Kurosusaido Kojimachi 4, Kojimachi 5-chome Chiyoda-ku Tokyo, 102-0083, JP)
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