Title:
PHARMACEUTICAL COMPOSITION OF FUSED AMINODIHYDROTHIAZINE DERIVATIVE
Document Type and Number:
WIPO Patent Application WO/2016/056638
Kind Code:
A1
Abstract:
The present invention provides a pharmaceutical composition which includes: a compound represented by formula (1), or N-[3-((4aS, 5R, 7aS)-2-amino-5-methyl-4a, 5, 7, 7a-tetrahydro-4H-furo[3, 4-d][1, 3]thiazine-7a-yl)-4-fluorophenyl]-5-difluoromethylpyrazine-2-carboxamide, or pharmaceutically acceptable salts of these; and a salt of a compound provided with a C12-22 saturated aliphatic hydrocarbon group.
Inventors:
ZAIMA YASUHIRO (JP)
KAZAMA KAZUO (JP)
ARASE SHUNTARO (JP)
NAGANE KENTARO (JP)
HORIE KANTA (JP)
UEKI YOSUKE (JP)
KAZAMA KAZUO (JP)
ARASE SHUNTARO (JP)
NAGANE KENTARO (JP)
HORIE KANTA (JP)
UEKI YOSUKE (JP)
Application Number:
PCT/JP2015/078688
Publication Date:
April 14, 2016
Filing Date:
October 08, 2015
Export Citation:
Assignee:
EISAI R&D MAN CO LTD (JP)
International Classes:
A61K31/542; A61K9/20; A61K47/14; A61K47/20; A61P25/28
Domestic Patent References:
| WO2009091016A1 | 2009-07-23 |
Other References:
JAPAN PHARMACEUTICAL EXCIPIENTS COUNCIL, HANDBOOK OF PHARMACEUTICAL EXCIPIENTS, 2007, pages 465, 468, 471, 762, 1007, XP009501743, ISBN: 978-4-8408-0968-9
KANA TAKAHASHI ET AL.: "Kattakuzai no Butsuri Kagakuteki Tokusei ga Jozai kara no Yakubutsu Hoshutsu ni Oyobosu Eikyo", ABSTRACTS OF 132TH ANNUAL MEETING OF PHARMACEUTICAL SOCIETY OF JAPAN (SAPPORO) PROGRUM-SHU, 2012, pages 169, XP009501736
KANA TAKAHASHI ET AL.: "Kattakuzai no Butsuri Kagakuteki Tokusei ga Jozai kara no Yakubutsu Hoshutsu ni Oyobosu Eikyo", ABSTRACTS OF 132TH ANNUAL MEETING OF PHARMACEUTICAL SOCIETY OF JAPAN (SAPPORO) PROGRUM-SHU, 2012, pages 169, XP009501736
Attorney, Agent or Firm:
INABA, Yoshiyuki et al. (JP)
Yoshiyuki Inaba (JP)
Yoshiyuki Inaba (JP)
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