Title:
PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING GLAUCOMA
Document Type and Number:
WIPO Patent Application WO/2010/113957
Kind Code:
A1
Abstract:
Provided is a pharmaceutical composition for treating or preventing glaucoma, comprising a pyridylamino acetic acid compound represented by general formula (1) or a pharmacologically acceptable salt thereof as an active ingredient. In formula (1), R1, R2, and R3 each independently represent a hydrogen atom or the like; Y represents a group: -Q1-Q2 (wherein Q1 represents an arylene group or the like; and Q2 represents a group such as an aromatic ring group which may be substituted by a halogen atom or the like) or a dicyclic heteroaromatic ring which may be substituted by a halogen atom or the like; and Z represents a group such as an aromatic ring group which may be substituted by a halogen atom or the like.
Inventors:
HAGIHARA MASAHIKO
YONEDA KENJI
OKANARI EIJI
SHIGETOMI MANABU
YONEDA KENJI
OKANARI EIJI
SHIGETOMI MANABU
Application Number:
PCT/JP2010/055719
Publication Date:
October 07, 2010
Filing Date:
March 30, 2010
Export Citation:
Assignee:
UBE INDUSTRIES (JP)
HAGIHARA MASAHIKO
YONEDA KENJI
OKANARI EIJI
SHIGETOMI MANABU
HAGIHARA MASAHIKO
YONEDA KENJI
OKANARI EIJI
SHIGETOMI MANABU
International Classes:
C07D213/83; A61K31/44; A61K31/443; A61K31/4439; A61K31/444; A61K31/501; A61K31/506; A61P27/06; C07D401/12; C07D405/14; C07D409/14; C07D417/12; C07D417/14; C07D401/14
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Other References:
CHRISTOPHER P. HOLMES, ET AL.: "PTP1B inhibitors: Synthesis and evaluation of difluoro-methylenephosphonate bioisosteres on a sulfonamide scaffold", BIOORG.MED.CHEM.LETT., vol. 18, no. 8, 2008, pages 2719 - 2724, XP022606378
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 20, 1985, pages 16
THE JOURNAL OF ORGANIC CHEMISTRY, vol. 60, 1995, pages 7508
THE JOURNAL OF ORGANIC CHEMISTRY, vol. 65, 2000, pages 64
ABRAANOVITZ ET AL., BIOCHIMICA ET BIOPHYSICA ACTA, vol. 1483, 2000, pages 285
WILSON ET AL., EUROPEAN JOURNAL OFPHARMACOLOGY, vol. 501, 2004, pages 49
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, vol. 20, 1985, pages 16
THE JOURNAL OF ORGANIC CHEMISTRY, vol. 60, 1995, pages 7508
THE JOURNAL OF ORGANIC CHEMISTRY, vol. 65, 2000, pages 64
ABRAANOVITZ ET AL., BIOCHIMICA ET BIOPHYSICA ACTA, vol. 1483, 2000, pages 285
WILSON ET AL., EUROPEAN JOURNAL OFPHARMACOLOGY, vol. 501, 2004, pages 49
Attorney, Agent or Firm:
TSUKUNI, HAJIME (JP)
Hajime Tsukuni (JP)
Hajime Tsukuni (JP)
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