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Title:
PLANT EXTRACTS ENRICHED WITH IPOLAMIIDE DERIVATIVES AS IMMUNOSUPPRESSANTS FOR TREATING IMMUNOLOGICAL DISORDERS
Document Type and Number:
WIPO Patent Application WO/2018/148816
Kind Code:
A3
Abstract:
The invention describes extracts from plants of the genus Stachytarpheta enriched with ipolamiide derivatives as immunosuppressants for treating immunological disorders. The isolated active compounds and a process of producing these are also disclosed.

Inventors:
GUIMARÃES CRISTIANO RUCH WERNECK (BR)
VITOR CARLOS EDUARDO (BR)
PESSA LISANDRA RAVANELLI (BR)
REIS ROMULO DRAGANI (BR)
MASCARELLO ALESSANDRA (BR)
GAMA FERNANDO HENRIQUE DE SOUZA (BR)
Application Number:
PCT/BR2018/050037
Publication Date:
October 18, 2018
Filing Date:
February 19, 2018
Export Citation:
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Assignee:
ACHE LABORATORIOS FARMACEUTICOS SA (BR)
International Classes:
C07D311/94; A61K31/201; A61K31/215; A61K31/352; A61P37/06; C07C59/42; C07C69/608
Domestic Patent References:
WO2016128471A12016-08-18
WO2008098325A12008-08-21
WO2003094946A12003-11-20
Foreign References:
CN103690551A2014-04-02
CN103120699A2013-05-29
EP1145709A12001-10-17
EP0045837A11982-02-17
US3703543A1972-11-21
DE19644422A11998-04-30
EP1371372A12003-12-17
Other References:
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Attorney, Agent or Firm:
DANIEL ADVOGADOS (BR)
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