Title:
PLATINUM COMPLEX AND MEDICAL COMPOUND CONTAINING SAME
Document Type and Number:
WIPO Patent Application WO/2010/026711
Kind Code:
A1
Abstract:
Disclosed is a new platinum complex, and medical compound containing same, which has strong antineoplastic activity and is efficacious at smaller doses. The platinum complex has a spiro [4,4]nonane-1,6-diamine represented by general formula (A) as the platinum complex’s ligand. (In the formula, X and Y are the same or different, and each represents a halogen atom, or X and Y jointly represent a bivalent residue represented by formula (Z).) Said platinum complex has strong antineoplastic activity and is efficacious as a therapeutic agent for malignant tumors.
Inventors:
ARAI, Hisae (LTD. 367-2 Kashiwa, Kashiwa-sh, Chiba 05, 〒2770005, JP)
新井久枝 (〒05 千葉県柏市柏367-2 ユニーテック株式会社内 Chiba, 〒2770005, JP)
OHNO, Masaji (LTD. 367-2 Kashiwa, Kashiwa-sh, Chiba 05, 〒2770005, JP)
大野雅二 (〒05 千葉県柏市柏367-2 ユニーテック株式会社内 Chiba, 〒2770005, JP)
新井久枝 (〒05 千葉県柏市柏367-2 ユニーテック株式会社内 Chiba, 〒2770005, JP)
OHNO, Masaji (LTD. 367-2 Kashiwa, Kashiwa-sh, Chiba 05, 〒2770005, JP)
大野雅二 (〒05 千葉県柏市柏367-2 ユニーテック株式会社内 Chiba, 〒2770005, JP)
Application Number:
JP2009/004077
Publication Date:
March 11, 2010
Filing Date:
August 25, 2009
Export Citation:
Assignee:
UNITECH CO., LTD. (367-2, Kashiwa Kashiwa-sh, Chiba 05, 〒2770005, JP)
ユニーテック株式会社 (〒05 千葉県柏市柏367-2 Chiba, 〒2770005, JP)
ARAI, Hisae (LTD. 367-2 Kashiwa, Kashiwa-sh, Chiba 05, 〒2770005, JP)
新井久枝 (〒05 千葉県柏市柏367-2 ユニーテック株式会社内 Chiba, 〒2770005, JP)
OHNO, Masaji (LTD. 367-2 Kashiwa, Kashiwa-sh, Chiba 05, 〒2770005, JP)
ユニーテック株式会社 (〒05 千葉県柏市柏367-2 Chiba, 〒2770005, JP)
ARAI, Hisae (LTD. 367-2 Kashiwa, Kashiwa-sh, Chiba 05, 〒2770005, JP)
新井久枝 (〒05 千葉県柏市柏367-2 ユニーテック株式会社内 Chiba, 〒2770005, JP)
OHNO, Masaji (LTD. 367-2 Kashiwa, Kashiwa-sh, Chiba 05, 〒2770005, JP)
International Classes:
C07C211/38; A61K31/555; A61P35/00; C07C55/06; C07C61/04; C07F15/00
Attorney, Agent or Firm:
MORIYA, Kazuo (Daiichi Teikei Bldg, 1-13-4 Nihonbashi-Kakigaracho, Chuo-k, Tokyo 14, 〒1030014, JP)
