Title:
PROCESS FOR THE PREPARATION OF [4-(2-CHLORO-4-METHOXY-5-METHYLPHENYL)-5-METHYL-THIAZOLO-2-YL]-[2-CYCLOPROPYL-1-(3-FLUORO-4-METHYLPHENYL)-ETHYL]-AMINE
Document Type and Number:
WIPO Patent Application WO/2010/125414
Kind Code:
A8
Abstract:
The subject of the present invention is a novel process for the preparation of the [4-(2-chloro-4-methoxy-5-methylphenyl)-5-methyl-thiazolo-2-yl]-[2-cyclopropyl-1-(3-fluoro-4-methylphenyl)-ethyl]-amine of formula (I) and the new intermediates of the preparation process.
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Inventors:
PARKANYI ZSOLT (HU)
FAZEKAS JANOS (HU)
MISKOLCZI PETER (HU)
MOLNAR ANNAMARIA (HU)
AGAI BEIA (HU)
FAZEKAS JANOS (HU)
MISKOLCZI PETER (HU)
MOLNAR ANNAMARIA (HU)
AGAI BEIA (HU)
Application Number:
PCT/HU2010/000047
Publication Date:
April 07, 2011
Filing Date:
April 26, 2010
Export Citation:
Assignee:
SANOFI AVENTIS (FR)
PARKANYI ZSOLT (HU)
FAZEKAS JANOS (HU)
MISKOLCZI PETER (HU)
MOLNAR ANNAMARIA (HU)
AGAI BEIA (HU)
PARKANYI ZSOLT (HU)
FAZEKAS JANOS (HU)
MISKOLCZI PETER (HU)
MOLNAR ANNAMARIA (HU)
AGAI BEIA (HU)
International Classes:
C07D277/42; C07C331/04; C07D327/04
Attorney, Agent or Firm:
SANOFI-AVENTIS (Tó u. 1-5, Budapest, HU)
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