Title:
PROCESS FOR THE PREPARATION OF 6-O-PROPARGYL ERYTHROMYCIN DERIVATIVES
Document Type and Number:
WIPO Patent Application WO2001077134
Kind Code:
A3
Abstract:
Disclosed herein is a process for the preparation of erythromycin derivatives, or pharmaceutically acceptable salts thereof, which contain an optionally substituted propargyl group at the 6-O-position.
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Inventors:
KERDESKY FRANCIS A J
PREMCHANDRAN RAMIYA
WAYNE GREGORY S
CHANG SOU-JEN
PEASE JONATHAN P
BHAGAVATULA LAKSHMI
LALLAMAN JOHN E
MORTON HOWARD E
KING STEVEN A
PREMCHANDRAN RAMIYA
WAYNE GREGORY S
CHANG SOU-JEN
PEASE JONATHAN P
BHAGAVATULA LAKSHMI
LALLAMAN JOHN E
MORTON HOWARD E
KING STEVEN A
Application Number:
PCT/US2001/008842
Publication Date:
August 08, 2002
Filing Date:
March 20, 2001
Export Citation:
Assignee:
ABBOTT LAB (US)
International Classes:
C07H17/08; A61P31/04; C07B61/00; C07D407/14; C07D409/04; C07D498/04; (IPC1-7): C07H17/08; A61K31/7048; A61P31/04
Domestic Patent References:
WO1997042204A1 | 1997-11-13 | |||
WO1999021871A1 | 1999-05-06 |
Foreign References:
US5866549A | 1999-02-02 |
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