Title:
PROCESSES FOR PREPARATION OF ZIPRASIDONE
Document Type and Number:
WIPO Patent Application WO2005040160
Kind Code:
A3
Abstract:
Provided are processes for preparing ziprasidone from 1, 2-benzothiazole-3-piperazinyl (BITP) and 5-(2-chloroethyl)-6-chloro-1, 3-dihydro-indole-2(2H) one (CEI) using various solvents, bases and promoters.
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Inventors:
PILARSKY GIDEON (IL)
SHENKAR NATALIA (IL)
MENDELOVICI MARIOARA (IL)
NIDAM TAMAR (IL)
BALANOV ANNA (IL)
SHENKAR NATALIA (IL)
MENDELOVICI MARIOARA (IL)
NIDAM TAMAR (IL)
BALANOV ANNA (IL)
Application Number:
PCT/US2004/035604
Publication Date:
July 07, 2005
Filing Date:
October 25, 2004
Export Citation:
Assignee:
TEVA PHARMA (US)
TEVA PHARMA (US)
PILARSKY GIDEON (IL)
SHENKAR NATALIA (IL)
MENDELOVICI MARIOARA (IL)
NIDAM TAMAR (IL)
BALANOV ANNA (IL)
TEVA PHARMA (US)
PILARSKY GIDEON (IL)
SHENKAR NATALIA (IL)
MENDELOVICI MARIOARA (IL)
NIDAM TAMAR (IL)
BALANOV ANNA (IL)
International Classes:
A61K31/519; C07D417/12; C07D487/04; (IPC1-7): C07D417/12
Domestic Patent References:
WO2003070246A1 | 2003-08-28 |
Foreign References:
US4831031A | 1989-05-16 | |||
US5338846A | 1994-08-16 |
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