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Title:
PROCESSES FOR PREPARING TETRAHYDROISOQUINOLINES
Document Type and Number:
WIPO Patent Application WO/2014/159501
Kind Code:
A3
Abstract:
Disclosed are processes for preparing tetrahydroisoquinolines, intermediates useful in the preparation of tetrahydroisoquinolines, processes for preparing such intermediates, and compositions comprising the tetrahydroisoquinolines and other compounds, e.g, intermediates and by-products of the processes described herein. Pharmaceutical compositions comprising tetrahydroisoquinolines, methods of using tetrahydroisoquinolines in the treatment of depression are also disclosed.

Inventors:
GONZALEZ-BOBES FRANCISCO (US)
CONLON DAVID ALAN (US)
LOBBEN PAUL C (US)
BURT JUSTIN LOCKHEART (US)
ENGSTROM JOSHUA (US)
WEI CAROLYN S (US)
ZHU JASON J (US)
FAN YU (US)
Application Number:
PCT/US2014/023938
Publication Date:
November 20, 2014
Filing Date:
March 12, 2014
Export Citation:
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Assignee:
BRISTOL MYERS SQUIBB CO (US)
International Classes:
A61K31/501; C07D217/04; C07D401/04; A61P25/00
Domestic Patent References:
WO2009149258A22009-12-10
WO2006020049A22006-02-23
Foreign References:
US20110281842A12011-11-17
Attorney, Agent or Firm:
VOLLES, Warren et al. (Route 206 and Province Line RoadPrinceton, New Jersey, US)
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