Title:
PYRAZOLE COMPOUNDS
Document Type and Number:
WIPO Patent Application WO/2004/029043
Kind Code:
A1
Abstract:
Pyrazole compounds represented by the general formula (I) or pharmacologically acceptable salts thereof, and pharmaceutical compositions containing the same as the active ingredient: (I) wherein R1 is optionally substituted phenyl; R2 is H, halogeno, alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, or substituted amino; Q is CH or N; R3 is H, alkyl, or amino; and R4 is a group represented by the general formula (II), (III), (IV), or (V): (II) (III) (III) (V) (wherein R7 is H or alkyl; R8 is H, alkyl, or substituted amino; R9 is H or alkyl; and R12 is H, alkyl, halogenoalkyl, or substituted amino).
Inventors:
HAGIHARA MASAHIKO (JP)
SHIBAKAWA NOBUHIKO (JP)
NISHIHARA MASAMICHI (JP)
SHIRAI TOSHIYUKI (JP)
SHIMIZU MOTOHISA (JP)
HASEGAWA TOHRU (JP)
TOKUNAGA YASUNORI (JP)
SUZUKI NAOTO (JP)
WADA YUKINORI (JP)
SHIBAKAWA NOBUHIKO (JP)
NISHIHARA MASAMICHI (JP)
SHIRAI TOSHIYUKI (JP)
SHIMIZU MOTOHISA (JP)
HASEGAWA TOHRU (JP)
TOKUNAGA YASUNORI (JP)
SUZUKI NAOTO (JP)
WADA YUKINORI (JP)
Application Number:
PCT/JP2003/012254
Publication Date:
April 08, 2004
Filing Date:
September 25, 2003
Export Citation:
Assignee:
UBE INDUSTRIES (JP)
HAGIHARA MASAHIKO (JP)
SHIBAKAWA NOBUHIKO (JP)
NISHIHARA MASAMICHI (JP)
SHIRAI TOSHIYUKI (JP)
SHIMIZU MOTOHISA (JP)
HASEGAWA TOHRU (JP)
TOKUNAGA YASUNORI (JP)
SUZUKI NAOTO (JP)
WADA YUKINORI (JP)
HAGIHARA MASAHIKO (JP)
SHIBAKAWA NOBUHIKO (JP)
NISHIHARA MASAMICHI (JP)
SHIRAI TOSHIYUKI (JP)
SHIMIZU MOTOHISA (JP)
HASEGAWA TOHRU (JP)
TOKUNAGA YASUNORI (JP)
SUZUKI NAOTO (JP)
WADA YUKINORI (JP)
International Classes:
A61K31/501; A61K31/5025; A61K31/506; A61P1/04; A61P3/10; A61P9/10; A61P17/06; A61P19/02; A61P19/10; A61P25/00; A61P29/00; A61P37/08; A61P43/00; C07D401/14; C07D403/14; C07D487/04; (IPC1-7): C07D401/14; A61K31/501; A61K31/5025; A61K31/506; A61P1/04; A61P3/10; A61P9/10; A61P17/06; A61P19/02; A61P19/10; A61P25/00; A61P29/00; A61P37/08; A61P43/00; C07D403/14; C07D487/04
Domestic Patent References:
| WO2000039116A1 | 2000-07-06 | |||
| WO2000031063A1 | 2000-06-02 | |||
| WO1995031451A1 | 1995-11-23 | |||
| WO2002057265A1 | 2002-07-25 | |||
| WO2001021591A1 | 2001-03-29 | |||
| WO1999057101A1 | 1999-11-11 | |||
| WO1998056377A1 | 1998-12-17 | |||
| WO1998052941A1 | 1998-11-26 | |||
| WO1998052937A2 | 1998-11-26 | |||
| WO1995031451A1 | 1995-11-23 | |||
| WO2000031451A1 | 2000-06-02 | |||
| WO2000031451A1 | 2000-06-02 | |||
| WO2000039116A1 | 2000-07-06 |
Foreign References:
| EP1142890A1 | 2001-10-10 |
Other References:
See also references of EP 1553096A4
Attorney, Agent or Firm:
Tsukuni, Hajime (22-12 Toranomon 1-chom, Minato-ku Tokyo, JP)
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