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Patent Searching and Data


Title:
PYRAZOLE DERIVATIVES, PREPARATION METHOD THEREOF, AND COMPOSITION FOR PREVENTING AND TREATING OSTEOPOROSIS CONTAINING SAME
Document Type and Number:
WIPO Patent Application WO/2012/118309
Kind Code:
A2
Abstract:
The present invention provides a pyrazole derivative compound and pharmaceutically acceptable salts thereof. The compound of the invention is remarkably effective for preventing and treating osteoporosis.

Inventors:
BAE YUN SOO (KR)
LEE KEE IN (KR)
LEE JEE HYUN (KR)
LEE SOO YOUNG (KR)
CHOI SUN (KR)
Application Number:
PCT/KR2012/001457
Publication Date:
September 07, 2012
Filing Date:
February 27, 2012
Export Citation:
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Assignee:
UNIV EWHA IND COLLABORATION (KR)
BAE YUN SOO (KR)
LEE KEE IN (KR)
LEE JEE HYUN (KR)
LEE SOO YOUNG (KR)
CHOI SUN (KR)
International Classes:
C07D401/04; A61K31/454; A61P19/10
Foreign References:
KR100942382B12010-02-12
Other References:
DARDEN, A. G. ET AL., J. BONE MINER, RES., vol. 11, 1996, pages 671 - 675
YANG, S. ET AL., J. BIOL. CHEM., vol. 276, 2001, pages 5452 - 5458
FRASER, J. H. ET AL., BONE, vol. 19, 1996, pages 223 - 226
YANG, S. ET AL., CALCIF. TISSUE INT., vol. 63, 1998, pages 346 - 350
BOYLE, N. J. ET AL., NATURE, vol. 423, 2003, pages 337 - 342
J. ORG. CHEM., vol. 43, no. 10, 1978, pages 2087 - 2088
J. CHEM. SOC., PERKIN TRANS., vol. 1, 1986, pages 1139 - 1143
See also references of EP 2682392A4
Attorney, Agent or Firm:
AHN, So-Young (KR)
안소영 (KR)
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Claims: