Title:
PYRAZOLE DERIVATIVES, PREPARATION METHOD THEREOF, AND COMPOSITION FOR PREVENTING AND TREATING OSTEOPOROSIS CONTAINING SAME
Document Type and Number:
WIPO Patent Application WO/2012/118309
Kind Code:
A2
Abstract:
The present invention provides a pyrazole derivative compound and pharmaceutically acceptable salts thereof. The compound of the invention is remarkably effective for preventing and treating osteoporosis.
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Inventors:
BAE YUN SOO (KR)
LEE KEE IN (KR)
LEE JEE HYUN (KR)
LEE SOO YOUNG (KR)
CHOI SUN (KR)
LEE KEE IN (KR)
LEE JEE HYUN (KR)
LEE SOO YOUNG (KR)
CHOI SUN (KR)
Application Number:
PCT/KR2012/001457
Publication Date:
September 07, 2012
Filing Date:
February 27, 2012
Export Citation:
Assignee:
UNIV EWHA IND COLLABORATION (KR)
BAE YUN SOO (KR)
LEE KEE IN (KR)
LEE JEE HYUN (KR)
LEE SOO YOUNG (KR)
CHOI SUN (KR)
BAE YUN SOO (KR)
LEE KEE IN (KR)
LEE JEE HYUN (KR)
LEE SOO YOUNG (KR)
CHOI SUN (KR)
International Classes:
C07D401/04; A61K31/454; A61P19/10
Foreign References:
KR100942382B1 | 2010-02-12 |
Other References:
DARDEN, A. G. ET AL., J. BONE MINER, RES., vol. 11, 1996, pages 671 - 675
YANG, S. ET AL., J. BIOL. CHEM., vol. 276, 2001, pages 5452 - 5458
FRASER, J. H. ET AL., BONE, vol. 19, 1996, pages 223 - 226
YANG, S. ET AL., CALCIF. TISSUE INT., vol. 63, 1998, pages 346 - 350
BOYLE, N. J. ET AL., NATURE, vol. 423, 2003, pages 337 - 342
J. ORG. CHEM., vol. 43, no. 10, 1978, pages 2087 - 2088
J. CHEM. SOC., PERKIN TRANS., vol. 1, 1986, pages 1139 - 1143
See also references of EP 2682392A4
YANG, S. ET AL., J. BIOL. CHEM., vol. 276, 2001, pages 5452 - 5458
FRASER, J. H. ET AL., BONE, vol. 19, 1996, pages 223 - 226
YANG, S. ET AL., CALCIF. TISSUE INT., vol. 63, 1998, pages 346 - 350
BOYLE, N. J. ET AL., NATURE, vol. 423, 2003, pages 337 - 342
J. ORG. CHEM., vol. 43, no. 10, 1978, pages 2087 - 2088
J. CHEM. SOC., PERKIN TRANS., vol. 1, 1986, pages 1139 - 1143
See also references of EP 2682392A4
Attorney, Agent or Firm:
AHN, So-Young (KR)
안소영 (KR)
안소영 (KR)
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Claims: