PYRIDINE COMPOUNDS AS FUNGICIDES

Description

The present invention relates to novel pyridine compounds and the N-oxides and the salts thereof, and to the use and methods for combating phytopathogenic fungi and to seeds coated with at least one such compound. The invention also relates to processes for preparing these compounds and to compositions comprising at least one compound I.

In many cases, in particular at low application rates, the fungicidal activity of the known fungicidal compounds is unsatisfactory. Based on this, it was an object of the present invention to provide compounds having improved activity and/or a broader activity spectrum against phyto- pathogenic harmful fungi.

Surprisingly, this objective is achieved by the use of the inventive pyridine compounds of formula I having favorable fungicidal activity against phytopathogenic fungi.

Accordingly, the present invention relates to the com ounds of the formula I

wherein

is selected from halogen, CN , N0 ₂ , SR ¹¹ , N H ₂ , N H(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-S0 ₂ -R ^{1 1} , Ci-C ₆ -alkyl, C ₂ -C ₆ -alkenyl, C ₂ -C ₆ -alkynyl, Ci-C ₆ -alkoxy, C(=0)-(R ¹² ), C3-C6-cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the het- eroaryl contains one, two or three heteroatoms selected from N, O and S; where- in

R ¹¹ is selected from Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, aryl or heteroaryl that is unsubsti- tuted or substituted by 1 , 2, 3, 4 or 5 substituents R ¹¹¹ independently selected from Ci-C ₄ -alkyl; and

R ¹² is independently selected from H , Ci-C6-alkyl, C ₂ -C6-alkenyl, C ₂ -C6-alkynyl, Cs- Cs-cycloalkyl, O-R ¹²¹ , N(R ²² )(R ¹²³ );

R ¹²¹ is independently selected from H , Ci-C6-alkyl, C ₂ -C6-alkenyl, C ₂ -C6- alkynyl, Cs-Cs-cycloalkyl;

R ¹²² , R ¹²³ are independently selected from H , Ci-C6-alkyl, Ci-C6-alkenyl, C1-C6- alkynyl and Cs-Cs-cycloalkyl;

wherein the aliphatic moieties of R ¹ are unsubstituted or substituted with identical or different groups R ^1a which independently of one another are selected from:

_R 1a halogen, OH , CN , Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, Ci-C ₄ - halogenalkoxy, Ci-C6-alkylthio, phenyl and phenoxy, wherein the phenyl and phe- noxy group is unsubstituted or carries 1 , 2, 3, 4 or 5 substituents R ^11a selected from the group consisting of halogen, OH , Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy and Ci-C4-halogenalkoxy; and

wherein the cycloalkyl, heteroaryl and aryl moieties of R ¹ are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups R ^1b which independently of one another are selected from:

R ^1b halogen, OH, CN , Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ - cycloalkyl, C3-C6-halogencycloalkyl, Ci-C4-halogenalkoxy and Ci-C6-alkylthio; R ² is selected from halogen, CN, N0 ₂ , SR ²¹ , NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-SO2- R ²¹ , Ci-C ₆ -alkyl, C ₂ -C ₆ -alkenyl, C ₂ -C ₆ -alkynyl, Ci-C ₆ -alkoxy, C(=0)-(R ²² ), C ₃ -C ₆ - cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein

R ²¹ is selected from Ci-C4-alkyl, Ci-C4-halogenalkyl, aryl or heteroaryl that is unsubsti- tuted or substituted by 1 , 2, 3, 4 or 5 substituents R ²¹¹ independently selected from

Ci-C4-alkyl; and

R ²² is independently selected from H , Ci-C6-alkyl, C ₂ -C6-alkenyl, C ₂ -C6-alkynyl, C ₃ -C ₃ - cycloalkyl, O-R ²²¹ , N(R ²²² )(R ²²³ );

R ²²¹ is independently selected from H, Ci-C6-alkyl, C ₂ -C6-alkenyl, C ₂ -C6- alkynyl, C ₃ -C8-cycloalkyl;

R ²²² , R ²²³ are independently selected from H, Ci-C6-alkyl, C ₂ -C6-alkenyl, C ₂ -C6- alkynyl, Cs-Cs-cycloalkyl;

wherein the aliphatic moieties of R ² are unsubstituted or substituted with identical or different groups R ^2a which independently of one another are selected from:

R ^2a halogen, OH, CN , Ci-C ₆ -alkoxy, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ -halogencycloalkyl, C1-C4- halogenalkoxy, Ci-C6-alkylthio, phenyl and phenoxy, wherein the phenyl and phenoxy group is unsubstituted or carries 1 , 2, 3, 4 or 5 substituents R ^21a selected from the group consisting of halogen, OH , Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy and Ci-C4-halogenalkoxy; and

wherein the cycloalkyl, heteroaryl and aryl moieties of R ² are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups R ^2b which independently of one another are selected from:

R ^2b halogen, OH, CN, Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ - halogencycloalkyl, Ci-C4-halogenalkoxy and Ci-C6-alkylthio;

R ³ is selected from H, halogen, OH, CN, N0 ₂ , SR ³¹ , NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-S0 ₂ -R ³¹ , Ci-C ₆ -alkyl, C ₂ -C ₆ -alkenyl, C ₂ -C ₆ -alkynyl, Ci-C ₆ -alkoxy, C ₃ -C ₆ -cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein R ³¹ is selected Ci-C4-alkyl, Ci-C4-halogenalkyl, aryl or heteroaryl that is unsubstituted or substituted by 1 , 2, 3, 4 or 5 substituents R ³¹¹ independently selected from Ci-C ₄ - alkyl;

and wherein the aliphatic moieties of R ³ are unsubstituted or substituted with identical or different groups R ^3a which independently of one another are selected from:

R ^3a halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, Ci-C ₄ - halogenalkoxy, Ci-C6-alkylthio, phenyl and phenoxy, wherein the phenyl and phe- noxy group is unsubstituted or carries 1 , 2, 3, 4 or 5 substituents R ^31a selected from the group consisting of halogen, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, Ci-C ₄ -alkoxy and Ci-C ₄ -halogenalkoxy;

and wherein the cycloalkyl, heteroaryl and aryl moieties of R ³ are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups R ^3b which independently of one another are selected from:

R ^3b halogen, OH, CN, Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ - cycloalkyl, C3-C6-halogencycloalkyl, Ci-C ₄ -halogenalkoxy and Ci-C6-alkylthio; ⁴ is selected from H, halogen, OH, CN, N0 ₂ , SR ⁴¹ , NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-S0 ₂ -R ⁴¹ , Ci-C ₆ -alkyl, C ₂ -C ₆ -alkenyl, C ₂ -C ₆ -alkynyl, Ci-C ₆ -alkoxy, C ₃ -C ₆ -cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein

R ⁴¹ is selected Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, aryl or heteroaryl that is unsubstituted or substituted by 1 , 2, 3, 4 or 5 substituents R ⁴¹¹ independently selected from Ci-C ₄ - alkyl;

and wherein the aliphatic moieties of R ⁴ are unsubstituted or substituted with identical or different groups R ^4a which independently of one another are selected from:

R ^4a halogen, OH, CN, Ci-C ₆ -alkoxy, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ -halogencycloalkyl, Ci-C ₄ - halogenalkoxy, Ci-C6-alkylthio, phenyland phenoxy, wherein the phenyl and phenoxy group is unsubstituted or carries 1 , 2, 3, 4 or 5 substituents R ^41a selected from the group consisting of halogen, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, Ci-C ₄ -alkoxy and Ci-C ₄ -halogenalkoxy;

and wherein the cycloalkyl, heteroaryl and aryl moieties of R ⁴ are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups R ^4b which independently of one another are selected from:

R ^4b halogen, OH, CN, Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ - cycloalkyl, C3-C6-halogencycloalkyl, Ci-C ₄ -halogenalkoxy and C1-C6- alkylthio;

Y is O or S(0) _n wherein

n is 0, 1 or 2; Q ¹ is selected from Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C6-cycloalkyl, five- or six- membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three het- eroatoms selected from N, O and S;

wherein the aliphatic moieties of Q ¹ are unsubstituted or substituted with identical or different groups Q ^1a which independently of one another are selected from:

Q ^1a halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, C1-C4- halogenalkoxy, Ci-C6-alkylthio, phenyl and phenoxy, wherein the phenyl and phe- noxy group is unsubstituted or carries 1 , 2, 3, 4 or 5 substituents Q ^11a selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy and Ci-C4-halogenalkoxy;

wherein the cycloalkyi, heteroaryl and aryl moieties of Q ¹ are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups Q ^1b which independently of one another are selected from:

Q ^1b halogen, OH, CN, Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ - cycloalkyl, C3-C6-halogencycloalkyl, Ci-C4-halogenalkoxy and Ci-C6-alkylthio;

Q ² is selected from H, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C6-cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N, O and S;

wherein the aliphatic moieties of Q ² are unsubstituted or substituted with identical or different groups Q ^2a which independently of one another are selected from:

Q ^2a halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, C1-C4- halogenalkoxy, Ci-C6-alkylthio, phenyl and phenoxy, wherein the phenyl and phenoxy group is unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ¹² selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy and Ci-C4-halogenalkoxy;

wherein the cycloalkyi, heteroaryl and aryl moieties of Q ² are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups Q ^2b which independently of one another are selected from:

Q ^2b halogen, OH, CN, Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ - cycloalkyl, C3-C6-halogencycloalkyl, Ci-C4-halogenalkoxy and Ci-C6-alkylthio;

Q ¹ and Q ² together with the carbon atom to which they are bound form a three- to seven- membered saturated or partially unsaturated carbo- or heterocycle

wherein the ring may further contain 1 , 2, 3 or 4 heteroatoms selected from N-R ^N , O and S, wherein R ^N is selected from H, Ci-C4-alkyl and S02R ^Q ; wherein

R ^Q is selected from Ci-C4-alkyl, Ci-C4-halogenalkyl, unsubstituted aryl or heteroaryl that is substituted by 1 , 2, 3, 4 or 5 substituents R ^Q1 independently selected from C1-C4- alkyl;

and wherein S may be in the form of its oxide SO or SO2; and wherein in each case one or two CH2 groups of the carbo- or heterocycle may be replaced by a group inde- pendently selected from C(=0) and C(=S);

and wherein the ring is unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups R ^QR which independently of one another are selected from:

Q ^QR halogen, OH, CN, Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ - cycloalkyl, C3-C6-halogencycloalkyl, Ci-C ₄ -halogenalkoxy and C1-C6- alkylthio;

is selected from H, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C6-cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N, O and S;

wherein the aliphatic moieties of Q ³ are unsubstituted or substituted with identical or different groups Q ^3a which independently of one another are selected from:

Q ^3a halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-cycloalkyloxy, C3-C6-halogencycloalkyl, Ci-C ₄ -halogenalkoxy, Ci-C6-alkylthio, phenyl, phe- noxy and five- to ten-membered heterocycle, heteroaryl, heterocycloxy, heteryloxy; wherein the heterocycle or heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein the cycloalkyl, cycloalkyloxy phenyl, phenoxy, heterocycleand heteroaryl groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^13a selected from the group consisting of halogen, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, Ci-C ₄ -alkoxy, Ci-C ₄ - halogenalkoxy, CR -NOR"; C3-C6-cycloalkyl, C3-C6-cycloalkyloxy, phenyl, phenoxy and five- to ten-membered heterocycle, heterocycloxy, heteroaryl and heteroaryloxy; wherein the heterocycle, heterocycloxy or heteroaryl, het- eroaryloxy contain one, two or three heteroatoms selected from N, O and S; and wherein the phenyl, phenoxy, heterocycle, cycloalkyl and heteroaryl groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^113a selected from the group consisting of halogen, OH, Ci-C ₄ -alkyl, Ci-C ₄ - halogenalkyl, Ci-C ₄ -alkoxy, CN, CR -NOR" and Ci-C ₄ -halogenalkoxy; wherein the cycloalkyl, heteroaryl and aryl moieties of Q ³ are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups Q ^3b which independently of one another are selected from:

Q ^3b halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-cycloalkyloxy, C3-C6-halogencycloalkyl, Ci-C ₄ -halogenalkoxy, Ci-C6-alkylthio, phenyl, phenoxy and five- to ten-membered heterocycle, heteroaryl, heterocycloxy, heteryloxy; wherein the heterocycle or heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein the phenyl, phenoxy, heterocycle, cycloalkyl and heteroaryl groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^13b selected from the group consisting of halogen, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkoxy, CR -NOR"; C3-C6-cycloalkyl, C3-C6-cycloalkyloxy, phenyl, phenoxy and five- to ten-membered heterocycle, heterocycloxy, heteroaryl and heteroaryloxy; wherein the heterocycle, heterocycloxy or heteroaryl, heteroaryloxy contain one, two or three heteroatoms selected from N, O and S; and wherein the phenyl, phenoxy, heterocycle, cycloalkyl and heteroaryl groups are unsubsti- tuted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^113b selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, C1-C4- alkoxy, CN, CR -NOR" and Ci-C4-halogenalkoxy; and wherein R' and R" are independently unsubstituted or substituted by R'" which is independently selected from halogen, OH, CN, N0 ₂ , SH, NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , Ci-C6-alkyl, Ci-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-halogenalkenyl, C2-C6- alkynyl, C2-C6-halogenalkynyl, Ci-C6-alkoxy, Ci-C6-halogenalkoxy, C3-C6- cycloalkyl, C3-C6-halogencycloalkyl and phenyl;

is O or S;

is selected from H, halogen, OH, CN, Ci-C4-alkyl, Ci-C4-alkoxy, Ci-C4-halogenalkyl, C3- C6-cycloalkyl, C3-C6-halogencycloalkyl, Ci-C4-halogenalkoxy and Ci-C6-alkylthio; wherein

n is 0, 1 , 2, 3 or 4;

with the proviso that if

R ¹ is CH ₃ ,

R ² is not CH ₃ ; and if

R ² is CHs,

R ¹ is not CHs. and the N-oxides and the agriculturally acceptable salts thereof.

Compounds of type I can be prepared by reacting compounds of type II with a suitable elec- trophile Q ³ -LG in an organic solvent, preferably NMP or a halocarbon and in the presence of a base at temperatures between -20 and 100 °C, most preferably between 0 and 40 °C. LG represents a suitable leavin group, preferably a halogen or a sulfonate.

II

Alternatively compounds I may be obtained by reacting compounds II ^* with compounds Q3-W- H under conditions described for the reaction between compounds II and Q3-LG yielding compounds I.

Compounds of type II may be accessed as described for example in J P2010/202530 or An- gewandte Chemie, International Edition, 45(35), 5803-5807; 2006 and as outlined below. Com- pounds of type III (where Hal is a halogen, most preferably Br or I) can be metallated by treatment with an appropriate organometallic reagent [M] in an ethereal solvent at low temperatures. Preferably, an organolithium or organomagnesium compound is used and the reaction is best performed in THF and between -78 °C and 0 °C. The intermediary organometallic species can be trapped with (thio)carbonyl compounds of type IV to furnish compounds of type II after aque- ous workup. Compounds of type IV are readily available either from commercial suppliers or through methods obvious to a person skilled in the art.

To access compounds of type III, it may be preferred to react compounds V in a nucleophilic aromatic substitution with compounds of type VI which are either commercially available or can be prepared following procedures that are obvious to a skilled person. LG represents a suitable leaving group, with special preference given to fluoride (for precedents see e.g.

WO2007/1 17381 , WO2012/037782, or Bioorganic & Medicinal Chemistry, 21 (4), 979-992;

2013). The reaction is best carried out at temperatures between 0 and 100 °C, preferably be- tween room temperature and 80 °C. Furthermore, it may be appropriate to perform the reaction in an organic solvent, preferably, but not limited to DMF or NMP and in the presence of a base, preferably, but not limited to potassium carbonate or sodium hydride.

V

Alternatively compounds III can be synthesized reacting compounds V ^* and VI ^* applying ditions already described for the reaction of compounds V with compounds VI

III

Alternatively compounds IN ^* can be accessed by reacting compounds V ^** with compounds VI ^** applying conditions already described for the reaction of V ^* with VI ^* yielding compounds III ^* . Compounds III ^* can subsequently be converted to compounds II using methods already described for the reaction of compounds III with compounds IV yielding compounds II.

Compounds of type V can be prepared from nitro compounds of type VII in a two-step sequence that has been previously described (for examples see Journal of Medicinal Chemistry, 35(20), 3667-71 ; 1992, WO2005/123668, or US20060293364). The first step seeks to achieve a chemoselective reduction of the nitro group to its amino congener by employing a suitable reducing agent, such as iron, zinc, or hydrogen in the presence of a transition metal catalyst such as palladium. Preferably, the reduction is performed in an organic solvent, more preferably in an alcoholic solvent, if appropriate at elevated temperatures and/or increased pressure. The respective amino compounds can be transformed into compounds of type V through a Sandmeyer reaction by reacting them first with a suitable nitrite source at low temperatures, preferably but not limited to sodium nitrite or t-BuONO. For the preparation of compounds in which Y is oxy- gen, the intermediary diazonium salt may be treated with a suitable acid, for example, but not limited to HCI or HBF4. It may be appropriate to increase the temperature upon addition of the acid. Compounds in which Y is S can be accessed by reacting said diazonium salt with a suitable sulfur source, preferably a alkali xanthate such as potassium xanthate, followed by base- mediated cleavage of the thioester. A precedent can be found for example in Journal of Medici- nal Chemistr 36(8), 953-66; 1993.

VII V

A person skilled in the art will realize that compounds of type VI I are either commercially available or be able to prepare said compounds following standard procedures. The N-oxides may be prepared from the inventive compounds according to conventional oxidation methods, e. g. by treating compounds I with an organic peracid such as metachloroper- benzoic acid (cf. WO 03/64572 or J. Med. Chem. 38(1 1 ), 1892-903, 1995); or with inorganic oxidizing agents such as hydrogen peroxide (cf. J. Heterocyc. Chem. 18(7), 1305-8, 1981 ) or oxone (cf. J. Am. Chem. Soc. 123(25), 5962-5973, 2001 ). The oxidation may lead to pure mono-N-oxides or to a mixture of different N-oxides, which can be separated by conventional methods such as chromatography.

If the synthesis yields mixtures of isomers, a separation is generally not necessarily required since in some cases the individual isomers can be interconverted during work-up for use or during application (e. g. under the action of light, acids or bases). Such conversions may also take place after use, e. g. in the treatment of plants in the treated plant, or in the harmful fungus to be controlled.

In the following, the intermediate compounds are further described. A skilled person will readily understand that the preferences for the substituents, also in particular the ones given in the tables below for the respective substituents, given herein in connection with compounds I apply for the intermediates accordingly. Thereby, the substituents in each case have independently of each other or more preferably in combination the meanings as defined herein.

In the definitions of the variables given above, collective terms are used which are generally representative for the substituents in question. The term "C _n -C _m " indicates the number of carbon atoms possible in each case in the substituent or substituent moiety in question.

The term "halogen" refers to fluorine, chlorine, bromine and iodine.

The term "Ci-C6-alkyl" refers to a straight-chained or branched saturated hydrocarbon group having 1 to 6 carbon atoms, e.g. methyl, ethyl, propyl, 1 -methylethyl, butyl, 1 -methyl propyl, 2- methylpropyl, 1 ,1 -dimethylethyl, pentyl, 1 -methylbutyl, 2-methylbutyl, 3-methylbutyl,

2,2-dimethylpropyl, 1 -ethylpropyl, 1 ,1 -dimethylpropyl, 1 ,2-dimethylpropyl, hexyl, 1 -methylpentyl, 2-methylpentyl, 3-methylpentyl, 4-methylpentyl, 1 ,1 -dimethylbutyl, 1 ,2-dimethylbutyl,

1 ,3-dimethylbutyl, 2,2-dimethylbutyl, 2,3-dimethylbutyl, 3,3-dimethylbutyl, 1 -ethylbutyl,

2- ethylbutyl, 1 ,1 ,2-trimethylpropyl, 1 ,2,2-trimethylpropyl, 1 -ethyl-1 -methylpropyl and 1 -ethyl-2- methylpropyl. Likewise, the term "C2-C4-alkyl" refers to a straight-chained or branched alkyl group having 2 to 4 carbon atoms, such as ethyl, propyl (n-propyl), 1 -methylethyl (iso-propoyl), butyl, 1 -methylpropyl (sec. -butyl), 2-methylpropyl (iso-butyl), 1 ,1 -dimethylethyl (tert. -butyl). The term "Ci-C6-halogenalkyl" refers to an alkyl group having 1 or 6 carbon atoms as defined above, wherein some or all of the hydrogen atoms in these groups may be replaced by halogen atoms as mentioned above. Examples are "Ci-C2-halogenalkyl" groups such as chloromethyl, bromomethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoromethyl, trifluoromethyl, chlorofluoromethyl, dichlorofluoromethyl, chlorodifluoromethyl, 1 -chloroethyl, 1 -bromoethyl, 1 - fluoroethyl, 2-fluoroethyl, 2,2-difluoroethyl, 2,2,2-trifluoroethyl, 2-chloro-2-fluoroethyl, 2-chloro- 2,2-difluoroethyl, 2,2-dichloro-2-fluoroethyl, 2,2,2-trichloroethyl or pentafluoroethyl.

The term "Ci-C6-hydroxyalkyl" refers to an alkyl group having 1 or 6 carbon atoms as defined above, wherein some or all of the hydrogen atoms in these groups may be replaced by OH groups.

The term "Ci-C4-alkoxy-Ci-C4-alkyl" refers to alkyl having 1 to 4 carbon atoms (as defined above), wherein one hydrogen atom of the alkyl radical is replaced by a Ci-C4-alkoxy group (as defined above). Likewise, the term "Ci-C6-alkoxy-Ci-C4-alkyl" refers to alkyl having 1 to 4 carbon atoms (as defined above), wherein one hydrogen atom of the alkyl radical is replaced by a Ci-C6-alkoxy group (as defined above).

The term "C2-C6-alkenyl" refers to a straight-chain or branched unsaturated hydrocarbon radical having 2 to 6 carbon atoms and a double bond in any position. Examples are "C2-C4-alkenyl" groups, such as ethenyl, 1 -propenyl, 2-propenyl (allyl), 1 -methylethenyl, 1 -butenyl, 2-butenyl,

3- butenyl, 1 -methyl-1 -propenyl, 2-methyl-1 -propenyl, 1 -methyl-2-propenyl, 2-methyl-2-propenyl.

The term "C2-C6-alkynyl" refers to a straight-chain or branched unsaturated hydrocarbon radical having 2 to 6 carbon atoms and containing at least one triple bond. Examples are "C2-C4- alkynyl" groups, such as ethynyl, prop-1 -ynyl, prop-2-ynyl (propargyl), but-1 -ynyl, but-2-ynyl, but-3-ynyl , 1 -methyl-prop-2-ynyl .

The term "Ci-C6-alkoxy" refers to a straight-chain or branched alkyl group having 1 to 6 carbon atoms which is bonded via an oxygen, at any position in the alkyl group. Examples are "C1-C4- alkoxy" groups, such as methoxy, ethoxy, n-propoxy, 1 -methylethoxy, butoxy, 1 - methyhpropoxy, 2-methylpropoxy or 1 ,1 -dimethylethoxy.

The term "Ci-C6-halogenalkoxy" refers to a Ci-C6-alkoxy radical as defined above, wherein some or all of the hydrogen atoms in these groups may be replaced by halogen atoms as mentioned above. Examples are "Ci-C4-halogenalkoxy" groups, such as OCH2F, OCHF2, OCF3, OCH2CI, OCHCI2, OCCI3, chlorofluoromethoxy, dichlorofluoromethoxy, chlorodifluoromethoxy, 2-fluoroethoxy, 2-chloroethoxy, 2-bromoethoxy, 2-iodoethoxy, 2,2-difluoroethoxy, 2,2,2-tri- fluoroethoxy, 2-chloro-2-fluoroethoxy, 2-chloro-2,2-difluoroethoxy, 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloro ^-, ethoxy, OC2F5, 2-fluoropropoxy, 3-fluoropropoxy, 2,2-difluoropropoxy,

2,3-difluoro ^-, propoxy, 2 chloropropoxy, 3-chloropropoxy, 2,3-dichloropropoxy, 2-bro- mo-'propoxy, 3 bromopropoxy, 3,3,3-trifluoropropoxy, 3,3,3-trichloropropoxy, OCH2-C2F5, OCF2-C2F5, 1 -fluoromethyl-2-fluoroethoxy, 1 -chloromethyl-2-chloroethoxy, 1 -bromomethyl-2- bromo-Othoxy, 4-fluorobutoxy, 4-chlorobutoxy, 4-bromobutoxy or nonafluorobutoxy.

The term "C2-C6-alkenyloxy" refers to a straight-chain or branched alkenyl group having 2 to 6 carbon atoms which is bonded via an oxygen, at any position in the alkenyl group. Examples are "C2-C4-alkenyloxy" groups.

The term "C2-C6-alkynyloxy" refers to a straight-chain or branched alkynyl group having 2 to 6 carbon atoms which is bonded via an oxygen, at any position in the alkynyl group. Examples are "C2-C4-alkynyloxy" groups.

The term "C3-C6-cycloalkyl" refers to monocyclic saturated hydrocarbon radicals having 3 to 6 carbon ring members, such as cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl. Accordingly, a saturated three-, four-, five-, six-, seven-, eight-, nine or ten-membered carbocyclyl or carbocycle is a "C3-Cio-cycloalkyl".

The term "C3-C6-cycloalkenyl" refers to a monocyclic partially unsaturated 3-, 4- 5- or 6- membered carbocycle having 3 to 6 carbon ring members and at least one double bond, such as cyclopentenyl, cyclopentadienyl, cyclohexadienyl. Accordingly, a partially unsaturated three-, four-, five-, six-, seven-, eight-, nine or ten-membered carbocyclyl or carbocycle is a "C3-C10- cycloalkenyl".

The term "C3-C6-cycloalkynyl" refers to a monocyclic partially unsaturated 3-, 4- 5- or 6- membered carbocycle having 3 to 6 carbon ring members and at least one triple bond.

The term "Ci-C6-alkylthio" as used herein refers to straight-chain or branched alkyl groups having 1 to 6 carbon atoms (as defined above) bonded via a sulfur atom. Accordingly, the term "Ci- C6-halogenalkylthio" as used herein refers to straight-chain or branched halogenalkyi group having 1 to 6 carbon atoms (as defined above) bonded through a sulfur atom, at any position in the halogenalkyi group.

The term "C(=0)-Ci-C6-alkyl" refers to a radical which is attached through the carbon atom of the group C(=0) as indicated by the number valence of the carbon atom. The number of va- lence of carbon is 4, that of nitrogen is 3. Likewise the following terms are to be construed: NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH(C ₃ -C ₆ -cycloalkyl), N(C ₃ -C ₆ -cycloalkyl) ₂ , C(=0)-NH(Ci-C ₆ - alkyl), C(=0)-N(Ci-C ₆ -alkyl) ₂ .

The term "saturated or partially unsaturated three-, four-, five-, six-, seven-, eight-, nine or ten- membered heterocyclyl or heterocycle, wherein the heterocyclyl or heterocycle contains 1 , 2, 3 or 4 heteroatoms selected from N, O and S" is to be understood as meaning both saturated and partially unsaturated heterocycles, wherein the ring member atoms of the heterocycle include besides carbon atoms 1 , 2, 3 or 4 heteroatoms independently selected from the group of O, N and S. For example:

a 3- or 4-membered saturated heterocycle which contains 1 or 2 heteroatoms from the group consisting of O, N and S as ring members such as oxirane, aziridine, thiirane, oxetane, azet- idine, thiethane, [1 ,2]dioxetane, [1 ,2]dithietane, [1 ,2]diazetidine; and a 5- or 6-membered saturated or partially unsaturated heterocycle which contains 1 , 2 or 3 het- eroatoms from the group consisting of O, N and S as ring members such as 2-tetrahydrofuranyl, 3-tetrahydrofuranyl, 2-tetrahydrothienyl, 3-tetrahydrothienyl, 2-pyrrolidinyl, 3-pyrrolidinyl, 3-isoxazolidinyl, 4-isoxazolidinyl, 5-isoxazolidinyl, 3-isothiazolidinyl, 4-isothiazolidinyl,

5-isothiazolidinyl, 3-pyrazolidinyl, 4-pyrazolidinyl, 5-pyrazolidinyl, 2-oxazolidinyl, 4-oxazolidinyl, 5-oxazolidinyl, 2-thiazolidinyl, 4-thiazolidinyl, 5-thiazolidinyl, 2-imidazolidinyl, 4-imidazolidinyl, 1 ,2,4-oxadiazolidin-3-yl, 1 ,2,4-oxadiazolidin-5-yl, 1 ,2,4-thiadiazolidin-3-yl, 1 ,2,4-thiadiazolidin-5- yl, 1 ,2,4-triazolidin-3-yl, 1 ,3,4-oxadiazolidin-2-yl, 1 ,3,4-thiadiazolidin-2-yl, 1 ,3,4-triazolidin-2-yl, 2,3-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,4-dihydrofur-2-yl, 2,4-dihydrofur-3-yl, 2,3-dihydrothien- 2-yl, 2,3-dihydrothien-3-yl, 2,4-dihydrothien-2-yl, 2,4-dihydrothien-3-yl, 2-pyrrolin-2-yl, 2-pyrrolin-

3- yl, 3-pyrrolin-2-yl, 3-pyrrolin-3-yl, 2-isoxazolin-3-yl, 3-isoxazolin-3-yl, 4-isoxazolin-3-yl, 2- isoxazolin-4-yl, 3-isoxazolin-4-yl, 4-isoxazolin-4-yl, 2-isoxazolin-5-yl, 3-isoxazolin-5-yl,

4- isoxazolin-5-yl, 2-isothiazolin-3-yl, 3-isothiazolin-3-yl, 4-isothiazolin-3-yl, 2-isothiazolin-4-yl, 3- isothiazolin-4-yl, 4-isothiazolin-4-yl, 2-isothiazolin-5-yl, 3-isothiazolin-5-yl, 4-isothiazolin-5-yl, 2,3- dihydropyrazol-1 -yl, 2,3-dihydropyrazol-2-yl, 2,3-dihydropyrazol-3-yl, 2,3-dihydropyrazol-4-yl, 2,3-dihydropyrazol-5-yl, 3,4-dihydropyrazol-1 -yl, 3,4-dihydropyrazol-3-yl, 3,4-dihydropyrazol-4- yl, 3,4-dihydropyrazol-5-yl, 4,5-dihydropyrazol-1 -yl, 4,5-dihydropyrazol-3-yl, 4,5-dihydropyrazol- 4-yl, 4,5-dihydropyrazol-5-yl, 2,3-dihydrooxazol-2-yl, 2,3-dihydrooxazol-3-yl, 2,3-dihydrooxazol- 4-yl, 2,3-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4- yl, 3,4-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4- yl, 2-piperidinyl, 3-piperidinyl, 4-piperidinyl, 1 ,3-dioxan-5-yl, 2-tetrahydropyranyl, 4- tetrahydropyranyl, 2-tetrahydrothienyl, 3-hexahydropyridazinyl, 4-hexahydropyridazinyl, 2-hexahydropyrimidinyl, 4-hexahydropyrimidinyl, 5-hexahydropyrimidinyl, 2-piperazinyl, 1 ,3,5- hexahydrotriazin-2-yl and 1 ,2,4-hexahydrotriazin-3-yl and also the corresponding -ylidene radi- cals; and

a 7-membered saturated or partially unsaturated heterocycle such as tetra- and hexahydroaze- pinyl, such as 2,3,4,5-tetrahydro[1 H]azepin-1 -,-2-,-3-,-4-,-5-,-6- or-7-yl, 3,4,5,6-tetra- hydro[2H]azepin-2-,-3-,-4-,-5-,-6- or-7-yl, 2,3,4,7-tetrahydro[1 H]azepin-1 -,-2-,-3-,-4-,-5-,-6- or-7- yl, 2,3,6,7-tetrahydro[1 H]azepin-1 -,-2-,-3-,-4-,-5-,-6- or-7-yl, hexahydroazepin-1 -,-2-,-3- or-4-yl, tetra- and hexahydrooxepinyl such as 2,3,4,5-tetrahydro[1 H]oxepin-2-,-3-,-4-,-5-,-6- or-7-yl,

2,3,4,7-tetrahydro[1 H]oxepin-2-,-3-,-4-,-5-,-6- or-7-yl, 2,3,6,7-tetrahydro[1 H]oxepin-2-, -3-,-4-,-5- ,-6- or-7-yl, hexahydroazepin-1 -,-2-,-3- or-4-yl, tetra- and hexahydro-1 ,3-diazepinyl, tetra- and hexahydro-1 ,4-diazepinyl, tetra- and hexahydro-1 ,3-oxazepinyl, tetra- and hexahydro-1 ,4- oxazepinyl, tetra- and hexahydro-1 ,3-dioxepinyl, tetra- and hexahydro-1 ,4-dioxepinyl and the corresponding -ylidene radicals.

The term "5-or 6-membered heteroaryl" refers to aromatic ring systems incuding besides carbon atoms, 1 , 2, 3 or 4 heteroatoms independently selected from the group consisting of N, O and S, for example,

a 5-membered heteroaryl such as pyrrol-1 -yl, pyrrol-2-yl, pyrrol-3-yl, thien-2-yl, thien-3-yl, furan- 2-yl, furan-3-yl, pyrazol-1 -yl, pyrazol-3-yl, pyrazol-4-yl, pyrazol-5-yl, imidazol-1 -yl, imidazol-2-yl, imidazol-4-yl, imidazol-5-yl, oxazol-2-yl, oxazol-4-yl, oxazol-5-yl, isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl, thiazol-2-yl, thiazol-4-yl, thiazol-5-yl, isothiazol-3-yl, isothiazol-4-yl, isothiazol-5-yl, 1 ,2,4-triazolyl-1 -yl, 1 ,2,4-triazol-3-yl 1 ,2,4-triazol-5-yl, 1 ,2,4-oxadiazol-3-yl, 1 ,2,4-oxadiazol-5-yl and 1 ,2,4-thiadiazol-3-yl, 1 ,2,4-thiadiazol-5-yl; or

a 6-membered heteroaryl, such as pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, pyridazin-3-yl, pyri- dazin-4-yl, pyrimidin-2-yl, pyrimidin-4-yl, pyrimidin-5-yl, pyrazin-2-yl and 1 ,3,5-triazin-2-yl and 1 ,2,4-triazin-3-yl.

Agriculturally acceptable salts of the inventive compounds encompass especially the salts of those cations or the acid addition salts of those acids whose cations and anions, respectively, have no adverse effect on the fungicidal action of said compounds. Suitable cations are thus in particular the ions of the alkali metals, preferably sodium and potassium, of the alkaline earth metals, preferably calcium, magnesium and barium, of the transition metals, preferably manganese, copper, zinc and iron, and also the ammonium ion which, if desired, may carry one to four Ci-C4-alkyl substituents and/or one phenyl or benzyl substituent, preferably diisopropylammoni- um, tetramethylammonium, tetrabutylammonium, trimethylbenzylammonium, furthermore phos- phonium ions, sulfonium ions, preferably tri(Ci-C4-alkyl)sulfonium, and sulfoxonium ions, prefer- ably tri(Ci-C4-alkyl)sulfoxonium. Anions of useful acid addition salts are primarily chloride, bromide, fluoride, hydrogensulfate, sulfate, dihydrogenphosphate, hydrogenphosphate, phosphate, nitrate, bicarbonate, carbonate, hexafluorosilicate, hexafluorophosphate, benzoate, and the anions of Ci-C4-alkanoic acids, preferably formate, acetate, propionate and butyrate. They can be formed by reacting such inventive compound with an acid of the corresponding anion, prefera- bly of hydrochloric acid, hydrobromic acid, sulfuric acid, phosphoric acid or nitric acid.

The inventive compounds can be present in atropisomers arising from restricted rotation about a single bond of asymmetric groups. They also form part of the subject matter of the present invention.

Depending on the substitution pattern, the compounds of formula I and their N-oxides may have one or more centers of chirality, in which case they are present as pure enantiomers or pure diastereomers or as enantiomer or diastereomer mixtures. Both, the pure enantiomers or dia- stereomers and their mixtures are subject matter of the present invention.

In the following, particular embodiments of the inventive compounds are described. Therein, specific meanings of the respective substituents are further detained, wherein the meanings are in each case on their own but also in any combination with one another, particular embodiments of the present invention.

Furthermore, in respect of the variables, generally, the embodiments of the compounds I also apply to the intermediates. R ¹ according to the invention is is in each case independently selected from halogen, CN,

N0 ₂ , SR ¹¹ ' NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-SO2-R ¹¹ , Ci-C ₆ -alkyl, C ₂ -C ₆ -alkenyl, C ₂ -C ₆ - alkynyl, Ci-C6-alkoxy, C(=0)-(R ¹² ), C3-C6-cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N , O and S;

wherein R ¹¹ is selected from Ci-C4-alkyl, Ci-C4-halogenalkyl, aryl or heteroaryl that is unsubsti- tuted or substituted by 1 , 2, 3, 4 or 5 substituents R ¹¹¹ independently selected from Ci-C ₄ -alkyl; and R ¹² is independently selected from H, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C ₃ -C ₃ - cycloalkyl, O-R ¹²¹ , N(R ²² )(R ¹²³ );

R ¹²¹ is independently selected from H, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C ₃ -C ₃ - cycloalkyl;

R ¹²² , R ¹²³ are independently selected from H, Ci-C6-alkyl, Ci-C6-alkenyl, Ci-C6-alkynyl and C ₃ - Cs-cycloalkyl;

wherein the aliphatic moieties of R ¹ are unsubstituted or substituted with identical or different groups R ^1a which independently of one another are selected from:

R ^1a halogen, OH, CN, Ci-C ₆ -alkoxy, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ -halogencycloalkyl, C1-C4- halogenalkoxy, Ci-C6-alkylthio, phenyl and phenoxy, wherein the phenyl and phenoxy group is unsubstituted or carries 1 , 2, 3, 4 or 5 substituents R ^11a selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy and Ci-C4-halogenalkoxy; and wherein the cycloalkyl, heteroaryl and aryl moieties of R ¹ are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups R ^1b which independently of one another are selected from:

R ^1b halogen, OH, CN, Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ - halogencycloalkyl, Ci-C4-halogenalkoxy and Ci-C6-alkylthio.

According to one specific embodiment, R ¹ is halogen, in particular Br, F or CI, more specifically F or CI.

According to a further specific embodiment, R ¹ is CN.

According to a further specific embodiment R ¹ is NH2, NH(Ci-C4-alkyl), N(Ci-C4-alkyl)2 or NH- SO2-R ¹¹ , wherein R ¹¹ is Ci-C4-alkyl, Ci-C4-halogenalkyl, unsubstituted aryl or aryl that is substituted by one, two, three, four or five substituents R ¹¹¹ independently selected from Ci-C4-alkyl. According to a further specific embodiment, R ¹ is Ci-C6-alkyl, in particular Ci-C4-alkyl, such as CH ₃ .

According to a further specific embodiment, R ¹ is Ci-C6-halogenalkyl, in particular C1-C4- halogenalkyl, such as CF ₃ , CHF ₂ , CH ₂ F, CCI ₃ , CHCI2 or CH ₂ CI.

According to still a further embodiment, R ¹ is C2-C6-alkenyl or C2-C6-halogenalkenyl, in particu- lar C2-C4-alkenyl or C2-C4-halogenalkenyl, such as CH=CH2.

According to still a further embodiment, R ¹ is C2-C6-alkynyl or C2-C6-halogenalkynyl, in particular C2-C4-alkynyl or C2-C4-halogenalkynyl, such as C CH.

According to a further specific embodiment, R ¹ is Ci-C6-alkoxy, in particular Ci-C4-alkoxy, more specifically Ci-C2-alkoxy such as OCH ₃ or OCH2CH ₃ .

According to a further specific embodiment, R ¹ is Ci-C6-halogenalkoxy, in particular C1-C4- halogenalkoxy, more specifically Ci-C2-halogenalkoxy such as OCF ₃ , OCHF2, OCH2F, OCCI ₃ , OCHC or OCH2CI, in particular OCF ₃ , OCHF ₂ , OCCI ₃ or OCHCI ₂ .

According to a further specific embodiment, R ¹ is C(=0)-(R ¹² ),

R ¹² is independently selected from H, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C ₃ -C ₃ - cycloalkyl, O-R ¹²¹ , N(R ²² )(R ¹²³ ); R ¹²¹ is independently selected from H, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8- cycloalkyl;

R ¹²² , R ¹²³ are independently selected from H, Ci-C6-alkyl, Ci-C6-alkenyl, Ci-C6-alkynyl and C3- Ce-cycloalkyl. Especially R ¹ is C(=0)NH ₂ , C(=0)NHCH ₃ , C(=0)N(CH ₃ ) ₂ .

According to a further specific embodiment R ¹ is C3-C6-cycloalkyl, in particular cyclopropyl.

In a further specific embodiment, R ¹ is C3-C6-cycloalkyl, for example cyclopropyl, substituted by one, two, three or up to the maximum possible number of identical or different groups R ^1b as defined and preferably herein.

According to a specific embodiment R ¹ is C3-C6-halogencycloalkyl. In a special embodiment R ¹ is fully or partially halogenated cyclopropyl.

According to still a further specific embodiment, R ¹ is unsubstituted aryl or aryl that is substituted by one, two, three or four R ^1b , as defined herein. In particular, R ¹ is unsubstituted phenyl or phenyl that is substituted by one, two, three or four R ^1b , as defined herein.

According to still a further specific embodiment, R ¹ is unsubstituted 5- or 6-membered heteroaryl. According to still a further embodiment, R ¹ is 5- or 6-membered heteroaryl that is substituted by one, two or three R ^1b , as defined herein.

According to one further embodiment R ¹ is in each case independently selected from halogen, OH, CN, N0 ₂ , SR ¹¹ , NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-S0 ₂ -R ^x , Ci-C ₆ -alkyl, C ₂ -C ₆ - alkenyl, C ₂ -C6-alkynyl, Ci-C6-alkoxy and C3-C6-cycloalkyl; wherein the aliphatic moieties of R ¹ are not further substituted or carry one, two, three, four or five identical or different groups R ^1a as defined below and wherein the cycloalkyl moieties of R ¹ are not further substituted or carry one, two, three, four or five identical or different groups R ^1b as defined below.

According to a further embodiment, R ¹ is independently selected from halogen, OH, Ci-C6-alkyl, Ci-C6-halogenalkyl, Ci-C6-alkoxy and Ci-C6-halogenalkoxy, in particular independently selected from F, CI, Br, CN, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, Ci-C ₄ -alkoxy and Ci-C ₄ -halogenalkoxy.

R ^1a are the possible substituents for the aliphatic moieties of R ¹ .

R ^1a according to the invention is independently selected from halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, Ci-C ₄ -halogenalkoxy, Ci-C6-alkylthio and phenoxy, wherein the phenyl group is unsubstituted or carries one, two, three, four or five substituents R ^11a selected from the group consisting of halogen, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, C1-C4- alkoxy and Ci-C ₄ -halogenalkoxy, in particular selected from halogen, Ci-C ₂ -alkyl, Ci-C ₂ - halogenalkyl, Ci-C ₂ -alkoxy and Ci-C ₂ -halogenalkoxy, more specifically selected from halogen, such as F, CI and Br.

According to one embodiment R ^1a is independently selected from halogen, OH, CN, Ci-C ₂ - alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and Ci-C ₂ -halogenalkoxy. Specifically, R ^1a is independently selected from F, CI, OH, CN, Ci-C ₂ -alkoxy, cyclopropyl, 1 -F-cyclopropyl, 1 -CI- cyclopropyl and Ci-C ₂ -halogenalkoxy.

According to one particular embodiment R ^1a is independently selected from halogen, such as F, CI, Br and I, more specifically F, CI and Br. According to a further embodiment, R ^1a is independently selected from OH, C3-C6-cycloalkyl, C3- C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, R ^1a is independently selected from OH, cyclopropyl and Ci-C2-halogenalkoxy.

R ^1b are the possible substituents for the cycloalkyi, heteroaryl and aryl moieties of R ¹ .

R ^1b according to the invention is independently selected from halogen, OH, CN , Ci-C4-alkyl, Ci- C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C4- halogenalkoxy.

According to one embodiment thereof R ^1b is independently selected from halogen, CN, C1-C2- alkyl, Ci-C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, R ^1b is independently selected from F, CI, OH, CN, CH ₃ , OCH ₃ , cyclopropyl, 1 -F-cyclopropyl, 1 -CI-cyclopropyl and halogenmethoxy.

According to a further embodiment thereof R ^1b is independently selected from Ci-C2-alkyl, Ci- C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, R ^1b is independently selected from OH, CH3, OCH3, cyclopropyl, 1 - F-cyclopropyl, 1 -CI-cyclopropyl and halogenmethoxy, more specifically independently selected from OH, CH3, OCH3, cyclopropyl, 1 -F-cyclopropyl, 1 -CI-cyclopropyl and OCHF2.

According to a further embodiment thereof R ^1b is independently selected from F, CI and Br.

R ² according to the invention is in each case independently selected from halogen, CN , NO2, SR ²¹ , NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-SO2-R ²¹ , Ci-C ₆ -alkyl, C ₂ -C ₆ -alkenyl, C ₂ -C ₆ - alkynyl, Ci-C6-alkoxy, C(=0)-(R ²² ), C3-C6-cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N , O and S;

wherein R ²¹ is selected from Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, aryl or heteroaryl that is unsubstituted or substituted by 1 , 2, 3, 4 or 5 substituents R ²¹¹ independently selected from C1-C4- alkyl; and

R ²² is independently selected from H , Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8- cycloalkyl, O-R ¹²¹ , N(R ²²² )(R ²²³ );

R ²²¹ is independently selected from H, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8- cycloalkyl;

R ²²² , R ²²³ are independently selected from H, Ci-C6-alkyl, Ci-C6-alkenyl, Ci-C6-alkynyl and C3- Cs-cycloalkyl;

wherein the aliphatic moieties of R ² are unsubstituted or substituted with identical or different groups R ^2a which independently of one another are selected from:

R ^2a halogen, OH, CN , Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, C1-C4- halogenalkoxy, Ci-C6-alkylthio, phenyl and phenoxy, wherein the phenyl and phenoxy group is unsubstituted or carries 1 , 2, 3, 4 or 5 substituents R ^11a selected from the group consisting of halogen, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, Ci-C ₄ -alkoxy and Ci-C ₄ -halogenalkoxy; and wherein the cycloalkyi, heteroaryl and aryl moieties of R ² are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups R ^2b which independently of one another are selected from:

R ^2b halogen, OH, CN , Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ - halogencycloalkyl, Ci-C ₄ -halogenalkoxy and Ci-C6-alkylthio.

According to one specific embodiment, R ² is halogen, in particular Br, F or CI, more specifically F or CI.

According to a further specific embodiment, R ² is CN.

According to a further specific embodiment R ² is NH2, NH(Ci-C4-alkyl), N(Ci-C4-alkyl)2 or NH- SO2-R ²¹ , wherein R ²¹ is Ci-C4-alkyl, Ci-C4-halogenalkyl, unsubstituted aryl or aryl that is substi- tuted by one, two, three, four or five substituents R ²¹¹ independently selected from Ci-C4-alkyl.

According to a further specific embodiment, R ² is Ci-C6-alkyl, in particular Ci-C4-alkyl, such as CH ₃ .

According to a further specific embodiment, R ² is Ci-C6-halogenalkyl, in particular C1-C4- halogenalkyl, such as CF ₃ , CHF ₂ , CH ₂ F, CCI ₃ , CHC or CH ₂ CI.

According to still a further embodiment, R ² is C2-C6-alkenyl or C2-C6-halogenalkenyl, in particular C2-C4-alkenyl or C2-C4-halogenalkenyl, such as CH=CH2.

According to still a further embodiment, R ² is C2-C6-alkynyl or C2-C6-halogenalkynyl, in particular C2-C4-alkynyl or C2-C4-halogenalkynyl, such as C CH.

According to a further specific embodiment, R ² is Ci-C6-alkoxy, in particular Ci-C4-alkoxy, more specifically Ci-C2-alkoxy such as OCH3 or OCH2CH3.

According to a further specific embodiment, R ² is Ci-C6-halogenalkoxy, in particular C1-C4- halogenalkoxy, more specifically Ci-C2-halogenalkoxy such as OCF3, OCHF2, OCH2F, OCCI3, OCHC or OCH2CI, in particular OCF ₃ , OCHF ₂ , OCCI ₃ or OCHCI ₂ .

According to a further specific embodiment, R ² is C(=0)-(R ¹² ),

R ¹² is independently selected from H, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, Cs-Cs-cycloalkyl, O-R ¹²¹ , N(R ²²² )(R ²²³ );

R ¹²¹ is independently selected from H, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, Cs-Cs- cycloalkyl;

R ²²² , R ²²³ are independently selected from H, Ci-C6-alkyl, Ci-C6-alkenyl, Ci-C6-alkynyl and C3- Ce-cycloalkyl. Especially R ² is C(=0)NH ₂ , C(=0)NHCH ₃ , C(=0)N(CH ₃ ) ₂ .

According to a further specific embodiment R ² is C3-C6-cycloalkyl, in particular cyclopropyl.

In a further specific embodiment, R ² is C3-C6-cycloalkyl, for example cyclopropyl, substituted by one, two, three or up to the maximum possible number of identical or different groups R ^2b as defined and preferably herein.

According to a specific embodiment R ² is C3-C6-halogencycloalkyl. In a special embodiment R ² is fully or partially halogenated cyclopropyl.

According to still a further specific embodiment, R ² is unsubstituted aryl or aryl that is substituted by one, two, three or four R ^2b , as defined herein. In particular, R ² is unsubstituted phenyl or phenyl that is substituted by one, two, three or four R ^1b , as defined herein.

According to still a further specific embodiment, R ² is unsubstituted 5- or 6-membered heteroaryl. According to still a further embodiment, R ² is 5- or 6-membered heteroaryl that is substituted by one, two or three R ^2b , as defined herein.

According to one further embodiment R ² is in each case independently selected from halogen, OH, CN, N0 ₂ , SR ²¹ , NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-S0 ₂ -R ^x , Ci-C ₆ -alkyl, C ₂ -C ₆ - alkenyl, C2-C6-alkynyl, Ci-C6-alkoxy and C3-C6-cycloalkyl; wherein the aliphatic moieties of R ² are not further substituted or carry one, two, three, four or five identical or different groups R ^2a as defined below and wherein the cycloalkyl moieties of R ² are not further substituted or carry one, two, three, four or five identical or different groups R ^2b as defined below.

According to a further embodiment, R ² is independently selected from halogen, OH, Ci-C6-alkyl, Ci-C6-halogenalkyl, Ci-C6-alkoxy and Ci-C6-halogenalkoxy, in particular independently selected from F, CI, Br, CN, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy and Ci-C4-halogenalkoxy.

R ^2a are the possible substituents for the aliphatic moieties of R ² .

R ^2a according to the invention is independently selected from halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, Ci-C4-halogenalkoxy, Ci-C6-alkylthio and phenoxy, wherein the phenyl group is unsubstituted or carries one, two, three, four or five substituents R ^21a selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, C1-C4- alkoxy and Ci-C4-halogenalkoxy, in particular selected from halogen, Ci-C2-alkyl, C1-C2- halogenalkyl, Ci-C2-alkoxy and Ci-C2-halogenalkoxy, more specifically selected from halogen, such as F, CI and Br.

According to one embodiment R ^2a is independently selected from halogen, OH, CN, C1-C2- alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, R ^2a is independently selected from F, CI, OH, CN, Ci-C2-alkoxy, cyclopropyl, 1 -F-cyclopropyl, 1 -CI- cyclopropyl and Ci-C2-halogenalkoxy.

According to one particular embodiment R ^2a is independently selected from halogen, such as F, CI, Br and I, more specifically F, CI and Br.

According to a further embodiment, R ^2a is independently selected from OH, C3-C6-cycloalkyl, C3- C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, R ^2a is independently selected from OH, cyclopropyl and Ci-C2-halogenalkoxy.

R ^2b are the possible substituents for the cycloalkyl, heteroaryl and aryl moieties of R ¹ .

R ^2b according to the invention is independently selected from halogen, OH, CN, Ci-C4-alkyl, Ci- C4-alkoxy, Ci-C4-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C4- halogenalkoxy.

According to one embodiment thereof R ^2b is independently selected from halogen, CN, C1-C2- alkyl, Ci-C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, R ^2b is independently selected from F, CI, OH, CN, CH3, OCH3, cyclopropyl, 1 -F-cyclopropyl, 1 -CI-cyclopropyl and halogenmethoxy.

According to a further embodiment thereof R ^2b is independently selected from Ci-C2-alkyl, Ci- C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, R ^2b is independently selected from OH, CH3, OCH3, cyclopropyl, 1 - F-cyclopropyl, 1 -CI-cyclopropyl and halogenmethoxy, more specifically independently selected from OH, CH3, OCH3, cyclopropyl, 1 -F-cyclopropyl, 1 -CI-cyclopropyl and OCHF2.

According to a further embodiment thereof R ^2b is independently selected from F, CI and Br.

According to a further embodiment if R ¹ is CH ₃ ,

R ² is not Ci-Ce-alkyl.

According to a further embodiment if

R ² is CH ₃ ,

R ¹ is not Ci-Ce-alkyl.

R ² according to the invention is is in each case independently selected from halogen, CN, NO2, SR ²¹ , NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-SO2-R ²¹ , C ₂ -C ₆ -alkenyl, C ₂ -C ₆ -alkynyl, Ci-C ₆ - alkoxy, C(=0)-(R ²² ), C3-C6-cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein R ²¹ is selected from Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, aryl or heteroaryl that is unsubstituted or substituted by 1 , 2, 3, 4 or 5 substituents R ²¹¹ independently selected from Ci-C ₄ -alkyl; and

R ²² is independently selected from H, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8- cycloalkyl, O-R ¹²¹ , N(R ²²² )(R ²²³ );

R ²²¹ is independently selected from H, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C8- cycloalkyl;

R ²²² , R ²²³ are independently selected from H, Ci-C6-alkyl, Ci-C6-alkenyl, Ci-C6-alkynyl and C3- Cs-cycloalkyl;

wherein the aliphatic moieties of R ² are unsubstituted or substituted with identical or different groups R ^2a which independently of one another are selected from:

R ^2a halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, Ci-C ₄ - halogenalkoxy, Ci-C6-alkylthio, phenyl and phenoxy, wherein the phenyl and phenoxy group is unsubstituted or carries 1 , 2, 3, 4 or 5 substituents R ^11a selected from the group consisting of halogen, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, Ci-C ₄ -alkoxy and Ci-C ₄ -halogenalkoxy; and wherein the cycloalkyi, heteroaryl and aryl moieties of R ² are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups R ^2b which independently of one another are selected from:

R ^2b halogen, OH, CN, Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ - halogencycloalkyl, Ci-C ₄ -halogenalkoxy and Ci-C6-alkylthio.

According to one specific embodiment, R ² is halogen, in particular Br, F or CI, more specifically F or CI.

R ³ according to the invention is in each case independently selected from H, halogen, OH, CN, N0 ₂ , SR ³¹ , NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-SO2-R ³¹ , Ci-Ce-alkyl, C ₂ -C ₆ -alkenyl, C2-C6-alkynyl, Ci-C6-alkoxy, C3-C6-cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein R ³¹ is selected from Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, aryl or heteroaryl that is unsubstituted or substituted by 1 , 2, 3, 4 or 5 substituents R ³¹¹ independently selected from Ci-C ₄ -alkyl; and wherein the aliphatic moieties of R ³ are unsubstituted or substituted with identical or different groups R ^3a which independently of one another are selected from:

R ^3a halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, C1-C4- halogenalkoxy, Ci-C6-alkylthio, phenyl and phenoxy, wherein the phenyl and phenoxy group is unsubstituted or carries 1 , 2, 3, 4 or 5 substituents R ^31a selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy and Ci-C4-halogenalkoxy; and wherein the cycloalkyl, heteroaryl and aryl moieties of R ³ are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups R ^3b which independently of one another are selected from:

R ^3b halogen, OH, CN, Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ - halogencycloalkyl, Ci-C4-halogenalkoxy and Ci-C6-alkylthio.

According to one specific embodiment, R ³ is H.

According to one specific embodiment, R ³ is halogen, in particular Br, F or CI, more specifically F or CI.

According to a further specific embodiment, R ³ is CN.

According to a further specific embodiment R ³ is NH2, NH(Ci-C4-alkyl), N(Ci-C4-alkyl)2 or NH- SO2-R ³¹ , wherein R ³¹ is Ci-C4-alkyl, Ci-C4-halogenalkyl, unsubstituted aryl or aryl that is substituted by one, two, three, four or five substituents R ³¹¹ independently selected from Ci-C4-alkyl. According to a further specific embodiment, R ³ is Ci-C6-alkyl, in particular Ci-C4-alkyl, such as CH ₃ .

According to a further specific embodiment, R ³ is Ci-C6-halogenalkyl, in particular C1-C4- halogenalkyl, such as CF ₃ , CHF ₂ , CH ₂ F, CCI ₃ , CHCI2 or CH ₂ CI.

According to still a further embodiment, R ³ is C2-C6-alkenyl or C2-C6-halogenalkenyl, in particu- lar C2-C4-alkenyl or C2-C4-halogenalkenyl, such as CH=CH2.

According to still a further embodiment, R ³ is C2-C6-alkynyl or C2-C6-halogenalkynyl, in particular C2-C4-alkynyl or C2-C4-halogenalkynyl, such as C CH.

According to a further specific embodiment, R ³ is Ci-C6-alkoxy, in particular Ci-C4-alkoxy, more specifically Ci-C2-alkoxy such as OCH ₃ or OCH2CH ₃ .

According to a further specific embodiment, R ³ is Ci-C6-halogenalkoxy, in particular C1-C4- halogenalkoxy, more specifically Ci-C2-halogenalkoxy such as OCF ₃ , OCHF2, OCH2F, OCCI ₃ , OCHC or OCH2CI, in particular OCF ₃ , OCHF ₂ , OCCI ₃ or OCHCI ₂ .

According to a further specific embodiment R ³ is C ₃ -C6-cycloalkyl, in particular cyclopropyl.

In a further specific embodiment, R ³ is C ₃ -C6-cycloalkyl, for example cyclopropyl, substituted by one, two, three or up to the maximum possible number of identical or different groups R ^3b as defined and preferably herein.

According to a specific embodiment R ³ is C ₃ -C6-halogencycloalkyl. In a special embodiment R ³ is fully or partially halogenated cyclopropyl.

According to still a further specific embodiment, R ³ is unsubstituted aryl or aryl that is substituted by one, two, three or four R ^3b , as defined herein. In particular, R ³ is unsubstituted phenyl or phenyl that is substituted by one, two, three or four R ^3b , as defined herein.

According to still a further specific embodiment, R ³ is unsubstituted 5- or 6-membered heteroaryl. According to still a further embodiment, R ³ is 5- or 6-membered heteroaryl that is substituted by one, two or three R ^3b , as defined herein.

According to one further embodiment R ³ is in each case independently selected from H, halogen, OH, CN, N0 ₂ , SR ³¹ , NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-SO2-R ³¹ , Ci-C ₆ -alkyl, C ₂ -C ₆ - alkenyl, C2-C6-alkynyl, Ci-C6-alkoxy and C3-C6-cycloalkyl; wherein the aliphatic moieties of R ³ are not further substituted or carry one, two, three, four or five identical or different groups R ^3a as defined below and wherein the cycloalkyl moieties of R ³ are not further substituted or carry one, two, three, four or five identical or different groups R ^3b as defined below.

According to a further embodiment, R ³ is independently selected from H, halogen, OH, C1-C6- alkyl, Ci-C6-halogenalkyl, Ci-C6-alkoxy and Ci-C6-halogenalkoxy, in particular independently selected from F, CI, Br, CN, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, Ci-C ₄ -alkoxy and Ci-C ₄ - halogenalkoxy.

R ^3a are the possible substituents for the aliphatic moieties of R ³ .

R ^3a according to the invention is independently selected from halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, Ci-C ₄ -halogenalkoxy, Ci-C6-alkylthio and phenoxy, wherein the phenyl group is unsubstituted or carries one, two, three, four or five substituents R ^31a selected from the group consisting of halogen, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, Ci-C ₄ - alkoxy and Ci-C ₄ -halogenalkoxy, in particular selected from halogen, Ci-C2-alkyl, C1-C2- halogenalkyl, Ci-C2-alkoxy and Ci-C2-halogenalkoxy, more specifically selected from halogen, such as F, CI and Br.

According to one embodiment R ^3a is independently selected from halogen, OH, CN, C1-C2- alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, R ^3a is independently selected from F, CI, OH, CN, Ci-C2-alkoxy, cyclopropyl, 1 -F-cyclopropyl, 1 -CI- cyclopropyl and Ci-C2-halogenalkoxy.

According to one particular embodiment R ^3a is independently selected from halogen, such as F, CI, Br and I, more specifically F, CI and Br.

According to a further embodiment, R ^3a is independently selected from OH, C3-C6-cycloalkyl, C3- C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, R ^3a is independently selected from OH, cyclopropyl and Ci-C2-halogenalkoxy.

R ^3b are the possible substituents for the cycloalkyl, heteroaryl and aryl moieties of R ³ .

R ^3b according to the invention is independently selected from halogen, OH, CN, Ci-C ₄ -alkyl, Ci- C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and Ci-C ₄ - halogenalkoxy.

According to one embodiment thereof R ^3b is independently selected from halogen, CN, C1-C2- alkyl, Ci-C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, R ^3b is independently selected from F, CI, OH, CN, CH3, OCH3, cyclopropyl, 1 -F-cyclopropyl, 1 -CI-cyclopropyl and halogenmethoxy. According to a further embodiment thereof R ^3b is independently selected from Ci-C2-alkyl, Ci- C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, R ^3b is independently selected from OH, CH3, OCH3, cyclopropyl, 1 - F-cyclopropyl, 1 -CI-cyclopropyl and halogenmethoxy, more specifically independently selected from OH, CH3, OCH3, cyclopropyl, 1 -F-cyclopropyl, 1 -CI-cyclopropyl and OCHF2.

According to a further embodiment thereof R ^3b is independently selected from F, CI and Br.

R ⁴ according to the invention is in each case independently selected from H, halogen, OH, CN, N0 ₂ , SR ⁴¹ , NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-SO2-R ⁴¹ , Ci-C ₆ -alkyl, C ₂ -C ₆ -alkenyl, C ₂ -C ₆ - alkynyl, Ci-C6-alkoxy, C3-C6-cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein R ⁴¹ is selected from Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, aryl or heteroaryl that is unsubstituted or substituted by 1 , 2, 3, 4 or 5 substituents R ⁴¹¹ independently selected from Ci-C ₄ -alkyl; and

wherein the aliphatic moieties of R ⁴ are unsubstituted or substituted with identical or different groups R ^4a which independently of one another are selected from:

R ^4a halogen, OH, CN, Ci-C ₆ -alkoxy, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ -halogencycloalkyl, C1-C4- halogenalkoxy, Ci-C6-alkylthio, phenyl and phenoxy, wherein the phenyl and phenoxy group is unsubstituted or carries 1 , 2, 3, 4 or 5 substituents R ^41a selected from the group consisting of halogen, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, Ci-C ₄ -alkoxy and Ci-C ₄ -halogenalkoxy; and wherein the cycloalkyi, heteroaryl and aryl moieties of R ⁴ are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups R ^4b which independently of one another are selected from:

R ⁴ halogen, OH, CN, Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ - halogencycloalkyl, Ci-C ₄ -halogenalkoxy and Ci-C6-alkylthio. According to one specific embodiment, R ⁴ is H.

According to one specific embodiment, R ⁴ is halogen, in particular Br, F or CI, more specifically F or CI.

According to a further specific embodiment, R ⁴ is CN.

According to a further specific embodiment R ⁴ is NH2, NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl)2 or NH- SO2-R ⁴¹ , wherein R ⁴¹ is Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, unsubstituted aryl or aryl that is substituted by one, two, three, four or five substituents R ⁴¹¹ independently selected from Ci-C ₄ -alkyl.

According to a further specific embodiment, R ⁴ is Ci-C6-alkyl, in particular Ci-C ₄ -alkyl, such as CH ₃ .

According to a further specific embodiment, R ⁴ is Ci-C6-halogenalkyl, in particular C1-C4- halogenalkyl, such as CF ₃ , CHF ₂ , CH ₂ F, CCI ₃ , CHCI2 or CH ₂ CI.

According to still a further embodiment, R ⁴ is C2-C6-alkenyl or C2-C6-halogenalkenyl, in particular C2-C ₄ -alkenyl or C2-C ₄ -halogenalkenyl, such as CH=CH2.

According to still a further embodiment, R ⁴ is C2-C6-alkynyl or C2-C6-halogenalkynyl, in particular C2-C ₄ -alkynyl or C2-C ₄ -halogenalkynyl, such as C CH.

According to a further specific embodiment, R ⁴ is Ci-C6-alkoxy, in particular Ci-C ₄ -alkoxy, more specifically Ci-C2-alkoxy such as OCH3 or OCH2CH3.

According to a further specific embodiment, R ⁴ is Ci-C6-halogenalkoxy, in particular C1-C4- halogenalkoxy, more specifically Ci-C2-halogenalkoxy such as OCF3, OCHF2, OCH2F, OCCI3, OCHC or OCH2CI, in particular OCF ₃ , OCHF ₂ , OCCI ₃ or OCHCI ₂ .

According to a further specific embodiment R ⁴ is C3-C6-cycloalkyl, in particular cyclopropyl.

In a further specific embodiment, R ⁴ is C3-C6-cycloalkyl, for example cyclopropyl, substituted by one, two, three or up to the maximum possible number of identical or different groups R ^4b as defined and preferably herein.

According to a specific embodiment R ⁴ is C3-C6-halogencycloalkyl. In a special embodiment R ⁴ is fully or partially halogenated cyclopropyl.

According to still a further specific embodiment, R ⁴ is unsubstituted aryl or aryl that is substituted by one, two, three or four R ^4b , as defined herein. In particular, R ⁴ is unsubstituted phenyl or phenyl that is substituted by one, two, three or four R ^4b , as defined herein.

According to still a further specific embodiment, R ⁴ is unsubstituted 5- or 6-membered heteroaryl. According to still a further embodiment, R ⁴ is 5- or 6-membered heteroaryl that is substituted by one, two or three R ^4b , as defined herein.

According to one further embodiment R ⁴ is in each case independently selected from H, halogen, OH, CN, N0 ₂ , SR ⁴¹ NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , NH-SO2-R ⁴¹ , Ci-C ₆ -alkyl, C ₂ -C ₆ - alkenyl, C2-C6-alkynyl, Ci-C6-alkoxy and C3-C6-cycloalkyl; wherein the aliphatic moieties of R ⁴ are not further substituted or carry one, two, three, four or five identical or different groups R ^4a as defined below and wherein the cycloalkyl moieties of R ⁴ are not further substituted or carry one, two, three, four or five identical or different groups R ^4b as defined below.

According to a further embodiment, R ⁴ is independently selected from H, halogen, OH, C1-C6- alkyl, Ci-C6-halogenalkyl, Ci-C6-alkoxy and Ci-C6-halogenalkoxy, in particular independently selected from F, CI, Br, CN, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, Ci-C ₄ -alkoxy and C1-C4- halogenalkoxy.

R ^4a are the possible substituents for the aliphatic moieties of R ⁴ .

R ^4a according to the invention is independently selected from halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, Ci-C ₄ -halogenalkoxy, Ci-C6-alkylthio and phenoxy, wherein the phenyl group is unsubstituted or carries one, two, three, four or five substituents R ^41a selected from the group consisting of halogen, OH, Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, C1-C4- alkoxy and Ci-C ₄ -halogenalkoxy, in particular selected from halogen, Ci-C2-alkyl, C1-C2- halogenalkyl, Ci-C2-alkoxy and Ci-C2-halogenalkoxy, more specifically selected from halogen, such as F, CI and Br.

According to one embodiment R ^4a is independently selected from halogen, OH, CN, C1-C2- alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, R ^4a is independently selected from F, CI, OH, CN, Ci-C2-alkoxy, cyclopropyl, 1 -F-cyclopropyl, 1 -CI- cyclopropyl and Ci-C2-halogenalkoxy.

According to one particular embodiment R ^4a is independently selected from halogen, such as F, CI, Br and I, more specifically F, CI and Br. According to a further embodiment, R ^4a is independently selected from OH, C3-C6-cycloalkyl, C3- C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, R ^4a is independently selected from OH, cyclopropyl and Ci-C2-halogenalkoxy.

R ^4b are the possible substituents for the cycloalkyi, heteroaryl and aryl moieties of R ⁴ .

R ^4b according to the invention is independently selected from halogen, OH, CN , Ci-C4-alkyl, Ci- C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C4- halogenalkoxy.

According to one embodiment thereof R ^4b is independently selected from halogen, CN, C1-C2- alkyl, Ci-C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, R ^4b is independently selected from F, CI, OH, CN, CH ₃ , OCH ₃ , cyclopropyl, 1 -F-cyclopropyl, 1 -CI-cyclopropyl and halogenmethoxy.

According to a further embodiment thereof R ^4b is independently selected from Ci-C2-alkyl, Ci- C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, R ^4b is independently selected from OH, CH3, OCH3, cyclopropyl, 1 - F-cyclopropyl, 1 -CI-cyclopropyl and halogenmethoxy, more specifically independently selected from OH, CH3, OCH3, cyclopropyl, 1 -F-cyclopropyl, 1 -CI-cyclopropyl and OCHF2.

According to a further embodiment thereof R ^4b is independently selected from F, CI and Br.

Y according to the invention is O.

According to a further embodiment thereof Y is S.

According to a further embodiment thereof Y is S(O).

According to a further embodiment thereof Y is S(0)2.

Q ¹ according to the invention is in each case independently selected from Ci-C6-alkyl, C2-C6- alkenyl, C2-C6-alkynyl, C3-C6-cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N , O and S;

wherein the aliphatic moieties of Q ¹ are unsubstituted or substituted with identical or different groups Q ^1a which independently of one another are selected from:

Q ^1a halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, C1-C4- halogenalkoxy, Ci-C6-alkylthio, phenyl and phenoxy, wherein the phenyl and phenoxy group is unsubstituted or carries 1 , 2, 3, 4 or 5 substituents Q ^11a selected from the group consisting of halogen, OH , Ci-C ₄ -alkyl, Ci-C ₄ -halogenalkyl, Ci-C ₄ -alkoxy and C1-C4- halogenalkoxy; and

wherein the cycloalkyi, heteroaryl and aryl moieties of Q ¹ are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups Q ^1b which independently of one another are selected from:

Q ^{1 b} halogen, OH, CN , Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ - halogencycloalkyl, Ci-C ₄ -halogenalkoxy and Ci-C6-alkylthio.

According to a further specific embodiment, Q ¹ is Ci-C6-alkyl, in particular Ci-C ₄ -alkyl, such as CH ₃ .

According to a further specific embodiment, Q ¹ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which is unsubstitituted. According to a further specific embodiment, Q ¹ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries 1 , 2 or 3 halogen.

According to a further specific embodiment, Q ¹ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries 1 , 2 or 3 Ci-C4-alkoxy groups.

According to a further specific embodiment, Q ¹ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries 1 , 2 or 3 Ci-C4-alkyl groups.

According to a further specific embodiment, Q ¹ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries 1 , 2 or 3 Ci-C4-halogenalkyl groups.

According to a further specific embodiment, Q ¹ is Ci-C6-halogenalkyl, in particular C1-C4- halogenalkyl, such as CF ₃ , CHF ₂ , CH ₂ F, CCI ₃ , CHC or CH ₂ CI.

According to still a further embodiment, Q ¹ is C2-C6-alkenyl or C2-C6-halogenalkenyl, in particular C2-C4-alkenyl or C2-C4-halogenalkenyl, such as CH=CH2.

According to still a further embodiment, Q ¹ is C2-C6-alkynyl or C2-C6-halogenalkynyl, in particular C2-C4-alkynyl or C2-C4-halogenalkynyl, such as C CH.

According to a further specific embodiment Q ¹ is C3-C6-cycloalkyl, in particular cyclopropyl.

In a further specific embodiment, Q ¹ is C3-C6-cycloalkyl, for example cyclopropyl, substituted by one, two, three or up to the maximum possible number of identical or different groups Q ^1b as defined and preferably herein.

According to a specific embodiment Q ¹ is C3-C6-halogencycloalkyl. In a special embodiment Q ¹ is fully or partially halogenated cyclopropyl.

According to still a further specific embodiment, Q ¹ is unsubstituted aryl or aryl that is substituted by one, two, three or four Q ^1b , as defined herein. In particular, Q ¹ is unsubstituted phenyl or phenyl that is substituted by one, two, three or four Q ^1b , as defined herein.

According to still a further specific embodiment, Q ¹ is unsubstituted 5- or 6-membered heteroaryl. According to still a further embodiment, Q ¹ is 5- or 6-membered heteroaryl that is substituted by one, two or three Q ^1b , as defined herein.

According to one further embodiment Q ¹ according to the invention is in each case independently selected from Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C6-cycloalkyl, five- or six- membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein Q ^1a is selected from halogen, Ci-C6-alkoxy, Cs-Ce- halogencycloalkyl, phenyl that is unsubstituted or substituted by 1 , 2, 3, 4 or 5 substituents Q ^11a independently selected from Ci-C4-alkyl; and

wherein the aliphatic moieties of Q ¹ are unsubstituted or substituted with identical or different groups Q ^1a as defined below and wherein the cycloalkyl moieties of Q ¹ are not further substitut- ed or carry one, two, three, four or five identical or different groups Q ^1b as defined below.

According to a further embodiment

Q ^1a are the possible substituents for the aliphatic moieties of Q ¹ .

Q ^1a according to the invention is independently selected from halogen, Ci-C6-alkoxy, Cs-Ce- halogencycloalkyl, and phenyl, wherein the phenyl group is unsubstituted or carries one, two, three, four or five substituents R ^11a selected from the group consisting of halogen, OH, C1-C4- alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy and Ci-C4-halogenalkoxy, in particular selected from halogen, Ci-C2-alkyl, Ci-C2-halogenalkyl, Ci-C2-alkoxy and Ci-C2-halogenalkoxy, more specifically selected from halogen, such as F, CI and Br.

According to one embodiment Q ^1a is independently selected from halogen, OH, CN, C1-C2- alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, Q ^1a is independently selected from F, CI, OH, CN, Ci-C2-alkoxy, cyclopropyl, 1 -F-cyclopropyl, 1-CI- cyclopropyl and Ci-C2-halogenalkoxy.

According to one particular embodiment Q ^1a is independently selected from halogen, such as F, CI, Br and I, more specifically F, CI and Br.

According to a further embodiment, Q ^1a is independently selected from OH, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, Q ^1a is independently selected from OH, cyclopropyl and Ci-C2-halogenalkoxy.

Q ^{1 b} are the possible substituents for the cycloalkyl, heteroaryl and aryl moieties of Q ¹ .

Q ^1b according to the invention is independently selected from halogen, OH, CN, Ci-C4-alkyl, Ci- C4-alkoxy, Ci-C4-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C4- halogenalkoxy.

According to one embodiment thereof Q ^1b is independently selected from halogen, CN, C1-C2- alkyl, Ci-C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, Q ^1b is independently selected from F, CI, OH, CN, CH ₃ , OCH ₃ , cyclopropyl, 1 -F-cyclopropyl, 1-CI-cyclopropyl and halogenmethoxy.

According to a further embodiment thereof Q ^1b is independently selected from Ci-C2-alkyl, Ci- C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, Q ^1b is independently selected from OH, CH3, OCH3, cyclopropyl, 1- F-cyclopropyl, 1-CI-cyclopropyl and halogenmethoxy, more specifically independently selected from OH, CH3, OCH3, cyclopropyl, 1 -F-cyclopropyl, 1-CI-cyclopropyl and OCHF2.

According to a further embodiment thereof R ^{1 b} is independently selected from F, CI and Br.

Q ² according to the invention is in each case independently selected from H, Ci-C6-alkyl, C2- C6-alkenyl, C2-C6-alkynyl, C3-C6-cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N, O and S

wherein the aliphatic moieties of Q ² are unsubstituted or substituted with identical or different groups Q ^2a which independently of one another are selected from:

Q ^2a halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, C1-C4- halogenalkoxy, Ci-C6-alkylthio, phenyl and phenoxy, wherein the phenyl and phenoxy group is unsubstituted or carries 1 , 2, 3, 4 or 5 substituents Q ^11a selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy and Ci-C4-halogenalkoxy; and wherein the cycloalkyl, heteroaryl and aryl moieties of Q ² are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups Q ^2b which inde- pendently of one another are selected from: Q ^2b halogen, OH, CN, Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ -cycloalkyl, Cs-Ce- halogencycloalkyl, Ci-C ₄ -halogenalkoxy and Ci-C6-alkylthio.

According to a further specific embodiment, Q ² is H.

According to a further specific embodiment, Q ² is Ci-C6-alkyl, in particular Ci-C ₄ -alkyl, such as CHs.

According to a further specific embodiment, Q ² is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which is unsubstitituted.

According to a further specific embodiment, Q ² is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries 1 , 2 or 3 halogen.

According to a further specific embodiment, Q ² is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries 1 , 2 or 3 Ci-C ₄ -alkoxy groups.

According to a further specific embodiment, Q ² is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries 1 , 2 or 3 Ci-C ₄ -alkyl groups.

According to a further specific embodiment, Q ² is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries 1 , 2 or 3 Ci-C ₄ -halogenalkyl groups.

According to a further specific embodiment, Q ² is Ci-C6-halogenalkyl, in particular Ci-C ₄ - halogenalkyl, such as CF ₃ , CHF ₂ , CH ₂ F, CCI ₃ , CHC or CH ₂ CI.

According to still a further embodiment, Q ² is C2-C6-alkenyl or C2-C6-halogenalkenyl, in particular C2-C ₄ -alkenyl or C2-C ₄ -halogenalkenyl, such as CH=CH2.

According to still a further embodiment, Q ² is C2-C6-alkynyl or C2-C6-halogenalkynyl, in particular C2-C ₄ -alkynyl or C2-C ₄ -halogenalkynyl, such as C CH.

According to a further specific embodiment Q ² is C3-C6-cycloalkyl, in particular cyclopropyl.

In a further specific embodiment, Q ² is C3-C6-cycloalkyl, for example cyclopropyl, substituted by one, two, three or up to the maximum possible number of identical or different groups Q ^2b as defined and preferably herein.

According to a specific embodiment Q ² is C3-C6-halogencycloalkyl. In a special embodiment Q ¹ is fully or partially halogenated cyclopropyl.

According to still a further specific embodiment, Q ² is unsubstituted aryl or aryl that is substituted by one, two, three or four Q ^2b , as defined herein. In particular, Q ² is unsubstituted phenyl or phenyl that is substituted by one, two, three or four Q ^2b , as defined herein.

According to still a further specific embodiment, Q ² is unsubstituted 5- or 6-membered heteroaryl. According to still a further embodiment, Q ² is 5- or 6-membered heteroaryl that is substituted by one, two or three Q ^2b , as defined herein.

According to one further embodiment Q ² according to the invention is in each case inde- pendently selected from Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C6-cycloalkyl, five- or six- membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein the aliphatic moieties of Q ² are unsubstituted or substituted with identical or different groups Q ^2a as defined below and wherein the cycloalkyl moieties of Q ² are not further substituted or carry one, two, three, four or five identical or different groups Q ^2b as defined below.

According to a further embodiment, Q ² is independently selected from halogen, OH, Ci-C6-alkyl, Ci-C6-halogenalkyl, Ci-C6-alkoxy and Ci-C6-halogenalkoxy, in particular independently selected from F, CI, Br, CN, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy and Ci-C4-halogenalkoxy.

Q ^2a are the possible substituents for the aliphatic moieties of Q ² .

Q ^2a according to the invention is independently selected from halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, Ci-C4-halogenalkoxy, Ci-C6-alkylthio and phenoxy, wherein the phenyl group is unsubstituted or carries one, two, three, four or five substituents ^Q2a selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, C1-C4- alkoxy and Ci-C4-halogenalkoxy, in particular selected from halogen, Ci-C2-alkyl, C1-C2- halogenalkyl, Ci-C2-alkoxy and Ci-C2-halogenalkoxy, more specifically selected from halogen, such as F, CI and Br.

According to one embodiment Q ^2a is independently selected from halogen, OH, CN, C1-C2- alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, Q ^2a is independently selected from F, CI, OH, CN, Ci-C2-alkoxy, cyclopropyl, 1-F-cyclopropyl, 1-CI- cyclopropyl and Ci-C2-halogenalkoxy.

According to one particular embodiment Q ^2a is independently selected from halogen, such as F, CI, Br and I, more specifically F, CI and Br.

According to a further embodiment, Q ^2a is independently selected from OH, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, Q ^2a is independently selected from OH, cyclopropyl and Ci-C2-halogenalkoxy.

Q ^2b are the possible substituents for the cycloalkyl, heteroaryl and aryl moieties of Q ² .

Q ^2b according to the invention is independently selected from halogen, OH, CN, Ci-C4-alkyl, Ci- C4-alkoxy, Ci-C4-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C4- halogenalkoxy.

According to one embodiment thereof Q ^2b is independently selected from halogen, CN, C1-C2- alkyl, Ci-C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, Q ^2b is independently selected from F, CI, OH, CN, CH3, OCH3, cyclopropyl, 1-F-cyclopropyl, 1-CI-cyclopropyl and halogenmethoxy.

According to a further embodiment thereof Q ^2b is independently selected from Ci-C2-alkyl, Ci- C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, Q ^2b is independently selected from OH, CH3, OCH3, cyclopropyl, 1- F-cyclopropyl, 1-CI-cyclopropyl and halogenmethoxy, more specifically independently selected from OH, CH3, OCH3, cyclopropyl, 1-F-cyclopropyl, 1-CI-cyclopropyl and OCHF2.

According to a further embodiment thereof R ^2b is independently selected from F, CI and Br. Q ¹ and Q ² according to the present invention form, together with the carbon atom to which they are bound form a three- to seven- membered saturated or partially unsaturated carbo- or heter- ocycle, wherein the ring may further contain 1 , 2, 3 or 4 heteroatoms selected from N-R ^N , O and S, wherein R ^N is selected from H, Ci-C4-alkyl and S02R ^Q ; wherein

R ^Q is selected from Ci-C4-alkyl, Ci-C4-halogenalkyl, unsubstituted aryl or heteroaryl that is substituted by 1 , 2, 3, 4 or 5 substituents R ^Q1 independently selected from Ci-C4-alkyl; and wherein S may be in the form of its oxide SO or SO2; and wherein in each case one or two CH2 groups of the carbo- or heterocycle may be replaced by a group independently selected from C(=0) and C(=S);

and wherein the ring is unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups R ^QR which independently of one another are selected from:

Q ^QR halogen, OH, CN, Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, Ci-C ₄ -halogenalkyl, C ₃ -C ₆ -cycloalkyl, C ₃ -C ₆ - halogencycloalkyl, Ci-C4-halogenalkoxy and Ci-C6-alkylthio.

According to one embodiment, the carbocycle formed by Q ¹ and Q ² is saturated.

According to a further embodiment, the carbocycle formed by Q ¹ and Q ² is a saturated unsubstituted or substituted carbocycle. According to one embodiment, this saturated carbocycle is unsubstituted. According to a further embodiment, the saturated carbocycle carries one, two, three or four substituents Q ^QR . In one further particular embodiment, said carbocycle is cyclopropane. In one further particular embodiment, said carbocycle is cyclobutane. In one further particular embodiment, said carbocycle is cyclohexane. In one further particular embodiment, said carbocycle is cyclopentane. In one further particular embodiment, said carbocycle is cyclopropane substituted by halogene or Ci-C4-alkyl. In one further particular embodiment, said carbocycle is cyclobutane substituted by halogene or Ci-C4-alkyl. In one further particular embodiment, said carbocycle is cyclohexane substituted by halogene or Ci-C4-alkyl. In one further particular embodiment, said carbocycle is cyclopentane substituted by halogene or Ci-C4-alkyl.

According to a further embodiment, the unsubstituted or substituted and saturated or partially unsaturated heterocycle is three-, four-, five- or six-membered and contains one, two or three, more particularly one or two, heteroatoms selected from NH, NR ^N , O, S, S(=0) and S(=0)2, wherein R ^N is as defined above or preferably selected from Ci-C2-alkyl, Ci-C2-halogenalkyl and S02Ph, wherein Ph is unsubstituted phenyl or phenyl that is substituted by one Ci-C2-alkyl. In one further particular embodiment, said heterocycle is four- or six-membered.

According to a further embodiment, the heterocycle formed by Q ¹ and Q ² contains one, two or three, more specifically one or two, heteroatoms selected from NH and NR ^N , wherein R ^N is as defined and preferably defined below, more particularly selected from Ci-C2-alkyl, C1-C2- halogenalkyl and S02Ph, wherein Ph is unsubstituted phenyl or phenyl that is substituted by one methyl. In one embodiment thereof, it contains one or two heteroatoms NH, in particular one NH. In another embodiment, it contains one or two heteroatoms NR ^N , in particular one NR ^N , wherein R ^N in each case is as defined and preferably defined above.

According to a further embodiment, the heterocycle formed by Q ¹ and Q ² contains one, two or three, more specifically one or two, in particular one, heteroatom(s) selected from S, S(=0) and S(=0)2. In one embodiment thereof, it contains one or two heteroatoms S, in particular one S. In another embodiment, it contains one or two heteroatoms S(=0), in particular one S(=0). In still another embodiment, it contains one or two heteroatoms S(=0)2, in particular one S(=0)2.

According to a further embodiment, the heterocycle formed by Q ¹ and Q ² contains one or two heteroatoms O. In one embodiment thereof, it contains one heteroatom O. In another embodi- ment, it contains two heteroatoms O.

According to a further embodiment, the heterocycle formed by Q ¹ and Q ² is unsubstituted, i.e. it does not carry any substituent Q ^QR . According to a further embodiment, it carries one, two, three or four Q ^QR .

According to one particular embodiment, Q ¹ and Q ² together form a 4-membered saturated het- erocycle which contains 1 or 2 heteroatoms, in particular 1 heteroatom, from the group consisting of NH, NR ^N , O, S, S(=0) and S(=0)2, as ring members, wherein R ^N is defined and preferably defined above. In one embodiment, the heterocycle contains one O as heteroatom. For example, the formed heterocycle is oxetane. According to one embodiment thereof, the heterocycle is unsubstituted, i.e. it does not carry any substituent Q ^QR . According to a further embodiment, it carries one, two, three or four Q ^QR .

According to a further particular embodiment, Q ¹ and Q ² together form a 5-membered saturated heterocycle which contains 1 , 2 or 3, in particular 1 or 2, heteroatoms from the group consisting of NH, NR ^N , O, S, S(=0) and S(=0)2, as ring members, wherein R ^N is as defined and preferably defined above. According to one embodiment thereof, the heterocycle is unsubstituted, i.e. it does not carry any substituent Q ^QR . According to a further embodiment, it carries one, two, three or four Q ^QR .

According to a further particular embodiment, Q ¹ and Q ² together form a 6-membered saturated heterocycle which contains 1 , 2 or 3, in particular 1 or 2, heteroatoms from the group consisting of NH, NR ^N , O, S, S(=0) and S(=0)2, as ring members, wherein R ^N is as defined and preferably defined below. According to one embodiment thereof, the heterocycle is unsubstituted, i.e. it does not carry any substituent Q ^QR . According to a further embodiment, it carries one, two, three or four Q ^QR . According to one specific embodiment thereof, said 6-membered saturated heterocycle contains 1 or 2 heteroatoms selected from NH and NR ^N . According to a further specific embodiment thereof, said 6-membered saturated heterocycle contains 1 or 2 heteroatoms O. According to a further specific embodiment thereof, said 6-membered saturated heterocycle contains 1 or 2 heteroatoms selected from S, S(=0) and S(=0)2. According to one embodiment thereof, the respective 6-membered heterocycle is unsubstituted, i.e. it does not carry any substituent Q ^QR . According to a further embodiment, it carries one, two, three or four Q ^QR .

Q ^QR are the possible substituents for the heterocycle formed by Q ¹ and Q ² and are independent- ly selected from halogen, OH, CN, N0 ₂ , SH, NH ₂ , Ci-C ₆ -alkyl, d-C ₆ -halogenalkyl, Ci-C ₆ -alkoxy, Ci-C6-halogenalkoxy, Ci-C6-alkylthio, Ci-C6-halogenalkylthio, Ci-C4-alkoxy-Ci-C4-alkyl, phenyl and phenoxy, wherein the phenyl groups are unsubstituted or carry one, two, three, four or five substituents Q ^QR selected from the group consisting of halogen, OH, Ci-C4-alkyl, C1-C4- halogenalkyl, Ci-C4-alkoxy and Ci-C4-halogenalkoxy; and wherein in each case one or two CH2 groups of the carbo- or heterocycle may be replaced by a group independently selected from C(=0) and C(=S).

In one preferred embodiment, Q ^QR is in each case independently selected from halogen, OH, CN, SH, Ci-C6-alkyl, Ci-C6-halogenalkyl, Ci-C6-alkoxy, Ci-C6-halogenalkoxy and C1-C6- alkylthio. In one further preferred embodiment, Q ^QR is in each case independently selected from halogen, Ci-C6-alkyl and Ci-C6-halogenalkyl. In one further particular embodiment, Q ^QR is in each case independently selected from Ci-C6-alkyl, such as methyl and ethyl.

R ^N is the substituent of the heteroatom NR ^N that is contained in the heterocycle formed by Q ² and Q ³ in some of the inventive compounds. R ^N is selected from Ci-C4-alkyl, Ci-C4-halogenalk and S02Ph, wherein Ph is unsubstituted phenyl or phenyl that is substituted by one, two or three substituents selected from Ci-C4-alkyl. In one preferred embodiment, R ^N is in each case independently selected from Ci-C2-alkyl, Ci-C2-halogenalkyl and S02Ph, wherein Ph is unsubstituted phenyl or phenyl that is substituted by one methyl substituents. In one particular embodiment, R ^N is in each case independently selected from Ci-C2-alkyl, more particularly methyl. In one particular embodiment, R ^N is in each case independently selected from S02Ph, wherein Ph is unsubstituted phenyl or phenyl that is substituted by one methyl.

Particularly preferred embodiments of the heterocycles formed by Q ¹ and Q ² and according to the invention are in Table P1 below, wherein each line of lines P1 -1 to P1 -15 corresponds to one particular embodiment of the invention, wherein P1 -1 to P1 -15 are also in any combination with one another a preferred embodiment of the present invention. The carbon atom, to which Q ² and Q ³ are bound is marked with # in the drawings.

Table P1 :

Q ³ according to the invention is in each case independently selected from Q ³ is selected from H, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, C3-C6-cycloalkyl, five- or six-membered heteroaryl and aryl; wherein the heteroaryl contains one, two or three heteroatoms selected from N, O and S;

wherein the aliphatic moieties of Q ³ are unsubstituted or substituted with identical or different groups Q ^3a which independently of one another are selected from:

Q ^3a halogen, OH, CN , Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-cycloalkyloxy, C3-C6-halogencycloalkyl, Ci-C4-halogenalkoxy, Ci-C6-alkylthio, phenyl, phe- noxy and five- to ten-membered heterocycle, heteroaryl, heterocycloxy, heteryloxy; wherein the heterocycle or heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein the cycloalkyl, cycloalkyloxy phenyl, phenoxy, heterocycleand heteroaryl groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^13a selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy, C1-C4- halogenalkoxy, CR -NOR"; C3-C6-cycloalkyl, C3-C6-cycloalkyloxy, phenyl, phenoxy and five- to ten-membered heterocycle, heterocycloxy, heteroaryl and heteroaryloxy; wherein the heterocycle, heterocycloxy or heteroaryl, het- eroaryloxy contain one, two or three heteroatoms selected from N , O and S; and wherein the phenyl, phenoxy, heterocycle, cycloalkyl and heteroaryl groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^113a selected from the group consisting of halogen, OH , Ci-C4-alkyl, C1-C4- halogenalkyl, Ci-C ₄ -alkoxy, CN, CR -NOR" and Ci-C ₄ -halogenalkoxy;

wherein the cycloalkyl, heteroaryl and aryl moieties of Q ³ are unsubstituted or substituted with 1 , 2, 3, 4, 5 or up to the maximum number of identical or different groups Q ^3b which independently of one another are selected from:

Q ^3b halogen, OH, CN , Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-cycloalkyloxy, C3-C6-halogencycloalkyl, Ci-C4-halogenalkoxy, Ci-C6-alkylthio, phenyl, phenoxy and five- to ten-membered heterocycle, heteroaryl, heterocycloxy, heteryloxy; wherein the heterocycle or heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein the phenyl, phenoxy, heterocycle, cycloalkyl and heteroaryl groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^13b selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy, Ci-C4-halogenalkoxy, CR -NOR"; C3-C6-cycloalkyl, C3-C6-cycloalkyloxy, phenyl, phenoxy and five- to ten-membered heterocycle, heterocycloxy, heteroaryl and heteroaryloxy; wherein the heterocycle, heterocycloxy or heteroaryl, heteroaryloxy contain one, two or three heteroatoms selected from N, O and S; and wherein the phenyl, phenoxy, heterocycle, cycloalkyl and heteroaryl groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^113b selected from the group consisting of halogen, OH , Ci-C4-alkyl, Ci-C4-halogenalkyl, C1-C4- alkoxy, CN, CR -NOR" and Ci-C4-halogenalkoxy; and wherein R' and R" are independently unsubstituted or substituted by R'" which is independently selected from halogen, OH, CN, N0 ₂ , SH, NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C ₄ -alkyl) ₂ , Ci-C6-alkyl, Ci-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-halogenalkenyl, C2-C6- alkynyl, C2-C6-halogenalkynyl, Ci-C6-alkoxy, Ci-C6-halogenalkoxy, C3-C6- cycloalkyl, C3-C6-halogencycloalkyl and phenyl.

According to a further specific embodiment, Q ³ is H.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular Ci-C ₄ -alkyl, such as According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which is unsubstitituted.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries 1 , 2 or 3 halogen.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries 1 , 2 or 3 Ci-C ₄ -alkoxy groups.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries 1 , 2 or 3 Ci-C ₄ -alkyl groups.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries 1 , 2 or 3 Ci-C ₄ -halogenalkyl groups.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries a further phenyl group which can be unsubstituted or substituted by halogen or Ci-C ₄ -alkyl. In one embodiment the phenyl is attached to phenyl directly. In one further embodiment the phenyl is attached to the phenyl via O.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenoxy which carries a phenyl group which can be unsubstituted or substituted by halogen or Ci-C ₄ -alkyl. In one embodiment the phenyl is attached to phenoxy directly. In one further embodiment the phenyl is attached to the phenyl via O.

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially CH2 subsitited by a 5-membered saturated heteroaryl which contains 1 , 2 or 3, in particular 1 or 2, heteroatoms from the group consisting of N, O and S as ring members.

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially CH2 subsitited by a 5-membered saturated heteroaryl which contains one N as ring member.

According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by Q ^13a . According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially CH2 subsitited by a 5-membered saturated heteroaryl which contains two N as ring members.

According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by Q ^13a .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially CH2 subsitited by a 5-membered saturated heteroaryl which contains three N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by Q ^13a . According to one specific embodiment thereof, said 5-membered saturated heterocycle contains 1 or 2, in particular 1 , heteroatom(s) O.

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains one S as ring member.

According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by Q ^13a .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains one S and one N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by Q ^13a .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains one S and two N as ring mem- bers. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by Q ^13a .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains one oxygen and one N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains one oxygen and two N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 6-membered saturated heteroaryl which contains 1 , 2 or 3, in particular 1 or 2, heteroatoms from the group consisting of N, O and S as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by Q ^13a .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 6-membered saturated heteroaryl which one N as ring member. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by Q ^13a .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 6-membered saturated heteroaryl which two N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by Q ^13a .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 10-membered saturated heteroaryl which contains 1 , 2 or 3, in particular 1 or 2, heteroatoms from the group consisting of N, O and S as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by Q ^13a . According to one specific embodiment thereof, said 10-membered saturated heterocycle contains 1 or 2, in par- ticular 1 , heteroatom(s) N.

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 10-membered saturated heteroaryl which one N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13a . According to still another embodiment of formula I, it is substituted by Q ^13a .

According to still another embodiment of formula I, Q ³ is Chb substituted by a 5-membered heteroaryl such as pyrrol-1-yl, pyrrol-2-yl, pyrrol-3-yl, thien-2-yl, thien-3-yl, furan-2-yl, furan-3-yl, pyrazol-1-yl, pyrazol-3-yl, pyrazol-4-yl, pyrazol-5-yl, imidazol-1-yl, imidazol-2-yl, imidazol-4-yl, imidazol-5-yl, oxazol-2-yl, oxazol-4-yl, oxazol-5-yl, isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl, thiazol-2-yl, thiazol-4-yl, thiazol-5-yl, isothiazol-3-yl, isothiazol-4-yl, isothiazol-5-yl, 1 ,2,4-triazolyl- 1-yl, 1 ,2,4-triazol-3-yl 1 ,2,4-triazol-5-yl, 1 ,2,4-oxadiazol-3-yl, 1 ,2,4-oxadiazol-5-yl and 1 ,2,4- thiadiazol-3-yl, 1 ,2,4-thiadiazol-5-yl.

According to still another embodiment of formula I, Q ³ is Chb substituted by a 6-membered heteroaryl, such as pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, pyridazin-3-yl, pyridazin-4-yl, pyrimidin-2- yl, pyrimidin-4-yl, pyrimidin-5-yl, pyrazin-2-yl and 1 ,3,5-triazin-2-yl and 1 ,2,4-triazin-3-yl.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular CH(CH3), substituted by phenyl which unsubstitituted.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular CH(CH3), substituted by phenyl which carries 1 , 2 or 3 halogen.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular CH(CH3), substituted by phenyl which carries 1 , 2 or 3 Ci-C4-alkoxy groups.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular CH(CH3), substituted by phenyl which carries 1 , 2 or 3 Ci-C4-alkyl groups.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular CH(CH3), substituted by phenyl which carries 1 , 2 or 3 Ci-C4-halogenalkyl groups.

According to a further specific embodiment, Q ³ is Ci-C6-halogenalkyl, in particular C1-C4- halogenalkyl, such as CF ₃ , CHF ₂ , CH ₂ F, CCI ₃ , CHC or CH ₂ CI.

According to still a further embodiment, Q ³ is C2-C6-alkenyl or C2-C6-halogenalkenyl, in particu- lar C2-C4-alkenyl or C2-C4-halogenalkenyl, such as CH=CH2.

According to still a further embodiment, Q ³ is C2-C6-alkynyl or C2-C6-halogenalkynyl, in particular C2-C4-alkynyl or C2-C4-halogenalkynyl, such as C CH.

According to a further specific embodiment Q ³ is C3-C6-cycloalkyl, in particular cyclopropyl. In a further specific embodiment, Q ³ is C3-C6-cycloalkyl, for example cyclopropyl, substituted by one, two, three or up to the maximum possible number of identical or different groups Q ^13b as defined and preferably herein.

According to a further specific embodiment Q ³ is C3-C6-cycloalkoxy, in particular cyclopropyloxy. In a further specific embodiment, Q ³ is C3-C6-cycloalkoxy, for example cyclopropyloxy, substituted by one, two, three or up to the maximum possible number of identical or different groups Q ^3b as defined and preferably herein.

According to a specific embodiment Q ³ is C3-C6-halogencycloalkyl. In a special embodiment Q ¹ is fully or partially halogenated cyclopropyl.

According to still a further specific embodiment, Q ³ is unsubstituted aryl or aryl that is substituted by one, two, three or four Q ^3b , as defined herein. In particular, Q ³ is unsubstituted phenyl or phenyl that is substituted by one, two, three or four Q ^3b , as defined herein.

According to still a further specific embodiment, Q ³ is unsubstituted 5- or 6-membered heteroaryl. According to still a further embodiment, Q ³ is 5- or 6-membered heteroaryl that is substituted by one, two or three Q ^3b , as defined herein.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenyl which carries a further phenyl group which can be unsubstituted or substituted by halogen or Ci-C4-alkyl. In one embodiment the phenyl is attached to phenyl directly. In one further embodiment the phenyl is attached to the phenyl via O.

According to a further specific embodiment, Q ³ is Ci-C6-alkyl, in particular Ci-alkyl, substituted by phenoxy which carries a phenyl group which can be unsubstituted or substituted by halogen or Ci-C4-alkyl. In one embodiment the phenyl is attached to phenoxy directly. In one further embodiment the phenyl is attached to the phenyl via O.

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains 1 , 2 or 3, in particular 1 or 2, heteroatoms from the group consisting of N, O and S as ring members.

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains one N as ring member.

According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by Q ^13b .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains two N as ring members.

According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by Q ^13b . According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains three N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by Q ^13b . According to one specific embodiment thereof, said 5-membered saturated heterocycle contains 1 or 2, in particular 1 , heteroatom(s) O. According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains one S as ring member.

According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by Q ^13b . According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains one S and one N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by Q ^13b .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains one S and two N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by Q ^13b .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains one oxygen and one N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 5-membered saturated heteroaryl which contains one oxygen and two N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 6-membered saturated heteroaryl which contains 1 , 2 or 3, in particular 1 or 2, heteroatoms from the group consisting of N, O and S as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by Q ^13b .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 6-membered saturated heteroaryl which one N as ring member. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by Q ^13b .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 6-membered saturated heteroaryl which two N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by Q ^13b .

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 10-membered saturated heteroaryl which contains 1 , 2 or 3, in particular 1 or 2, heteroatoms from the group consisting of N, O and S as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by Q ^13b . According to one specific embodiment thereof, said 10-membered saturated heterocycle contains 1 or 2, in par- ticular 1 , heteroatom(s) N.

According to a further specific embodiment of formula I, Q ³ is Ci-C6-alkyl, especially Chb subsitited by a 10-membered saturated heteroaryl which one N as ring members. According to one embodiment thereof, the heteroaryl is unsubstituted, i.e. it does not carry any substituent Q ^13b . According to still another embodiment of formula I, it is substituted by Q ^13b .

According to still another embodiment of formula I, Q ³ is Chb substituted by a 5-membered heteroaryl such as pyrrol-1 -yl, pyrrol-2-yl, pyrrol-3-yl, thien-2-yl, thien-3-yl, furan-2-yl, furan-3-yl, pyrazol-1 -yl, pyrazol-3-yl, pyrazol-4-yl, pyrazol-5-yl, imidazol-1 -yl, imidazol-2-yl, imidazol-4-yl, imidazol-5-yl, oxazol-2-yl, oxazol-4-yl, oxazol-5-yl, isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl, thiazol-2-yl, thiazol-4-yl, thiazol-5-yl, isothiazol-3-yl, isothiazol-4-yl, isothiazol-5-yl, 1 ,2,4-triazolyl- 1 -yl, 1 ,2,4-triazol-3-yl 1 ,2,4-triazol-5-yl, 1 ,2,4-oxadiazol-3-yl, 1 ,2,4-oxadiazol-5-yl and 1 ,2,4- thiadiazol-3-yl, 1 ,2,4-thiadiazol-5-yl.

According to still another embodiment of formula I, Q ³ is Chb substituted by a 6-membered heteroaryl, such as pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, pyridazin-3-yl, pyridazin-4-yl, pyrimidin-2- yl, pyrimidin-4-yl, pyrimidin-5-yl, pyrazin-2-yl and 1 ,3,5-triazin-2-yl and 1 ,2,4-triazin-3-yl.

Q ^3a are the possible substituents for the aliphatic moieties of OA

Q ^3a according to the invention is independently selected from halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-cycloalkyloxy, C3-C6-halogencycloalkyl, Ci-C4-halogenalkoxy, C1-C6- alkylthio, phenyl, phenoxy and five- to ten-membered heterocycle, heteroaryl, heterocycloxy, heteryloxy; wherein the heterocycle or heteroaryl contains one, two or three heteroatoms selected from N, O and S; wherein the cycloalkyl, cycloalkyloxy phenyl, phenoxy, heterocycleand heteroaryl groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^13a selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy, C1-C4- halogenalkoxy, CR'=NOR"; C3-C6-cycloalkyl, C3-C6-cycloalkyloxy, phenyl, phenoxy and five- to ten-membered heterocycle, heterocycloxy, heteroaryl and heteroaryloxy; wherein the heterocycle, heterocycloxy or heteroaryl, heteroaryloxy contain one, two or three heteroatoms selected from N, O and S; and wherein the phenyl, phenoxy, heterocycle, cycloalkyl and heteroaryl groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^113a selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy, CN, CR -NOR" and Ci-C4-halogenalkoxy;

, in particular selected from halogen, Ci-C2-alkyl, Ci-C2-halogenalkyl, Ci-C2-alkoxy and C1-C2- halogenalkoxy, more specifically selected from halogen, such as F, CI and Br.

According to one embodiment Q ^3a is independently selected from halogen, OH, CN, C1-C2- alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, Q ^3a is independently selected from F, CI, OH, CN, Ci-C2-alkoxy, cyclopropyl, 1 -F-cyclopropyl, 1 -CI- cyclopropyl and Ci-C2-halogenalkoxy, phenyl and five- to ten-membered heterocycle and heteroaryl.

According to one particular embodiment Q ^3a is independently selected from halogen, such as F, CI, Br and I, more specifically F, CI and Br.

According to one embodiment Q ^3a is independently selected from halogen, OH, CN, C1-C2- alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, Q ^3a is independently selected from F, CI, OH, CN, Ci-C2-alkoxy, cyclopropyl, 1 -F-cyclopropyl, 1 -CI- cyclopropyl, Ci-C2-halogenalkoxy, phenyl, five- and sex-membered heteroaryl.

According to one embodiment Q ^3a is independently selected from halogen, OH, CN, C1-C2- alkoxy, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, Ci-C2-halogenalkoxy, phenyl and five- to ten- membered heterocycle and heteroaryl. Specifically, Q ^3a is independently selected from F, CI, OH, CN, Ci-C2-alkoxy, cyclopropyl, 1 -F-cyclopropyl, 1 -CI-cyclopropyl, Ci-C2-halogenalkoxy, phenyl, five- and sex-membered heteroaryl.

In the embodiments in which Q ^3a phenyl, phenoxy, heterocycle and heteroaryl groups, these groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^13a selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy, C1-C4- halogenalkoxy; phenyl, phenoxy and five- to ten-membered heterocycle and heteroaryl; wherein the heterocycle or heteroaryl contains one, two or three heteroatoms selected from N, O and S; and wherein the phenyl, phenoxy, heterocycle and heteroaryl groups can be attached directly to Q ^3a or via O; and wherein the phenyl, phenoxy, heterocycle and heteroaryl groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^113a selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy and Ci-C4-halogenalkoxy.

According to one particular embodiment Q ^3a is phenyl.

According to one particular embodiment Q ^3a is heteroaryl.

According to one particular embodiment Q ^3a is cycloalkyl.

According to one particular embodiment Q ^3a is heterocyclyl.

According to one particular embodiment Q ^3a is phenoxy.

According to one particular embodiment Q ^3a is heteroaryloxy.

According to one particular embodiment Q ^3a is cycloalkoxy.

According to one particular embodiment Q ^3a is heterocyclyloxy.

According to a further embodiment, Q ^3a is independently selected from OH, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and Ci-C2-halogenalkoxy. Specifically, Q ^3a is independently selected from OH, cyclopropyl and Ci-C2-halogenalkoxy.

Q ^3b are the possible substituents for the cycloalkyl, heteroaryl and aryl moieties of Q ³ .

Q ^3b according to the invention is independently selected from halogen, OH, CN, Ci-C6-alkoxy, C3-C6-cycloalkyl, C3-C6-cycloalkyloxy, C3-C6-halogencycloalkyl, Ci-C4-halogenalkoxy, C1-C6- alkylthio, phenyl, phenoxy and five- to ten-membered heterocycle, heteroaryl, heterocycloxy, heteryloxy; wherein the heterocycle or heteroaryl contains one, two or three heteroatoms se- lected from N, O and S; wherein the phenyl, phenoxy, heterocycle, cycloalkyl and heteroaryl groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^13b selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy, C1-C4- halogenalkoxy, CR -NOR"; C3-C6-cycloalkyl, C3-C6-cycloalkyloxy, phenyl, phenoxy and five- to ten-membered heterocycle, heterocycloxy, heteroaryl and heteroaryloxy; wherein the heterocy- cle, heterocycloxy or heteroaryl, heteroaryloxy contain one, two or three heteroatoms selected from N, O and S; and wherein the phenyl, phenoxy, heterocycle, cycloalkyl and heteroaryl groups are unsubstituted or substituted with 1 , 2, 3, 4 or 5 substituents Q ^113b selected from the group consisting of halogen, OH, Ci-C4-alkyl, Ci-C4-halogenalkyl, Ci-C4-alkoxy, CN, CR'=NOR" and Ci-C4-halogenalkoxy; and wherein R' and R" are independently unsubstituted or substituted by R'" which is independently selected from halogen, OH, CN, N0 ₂ , SH, NH ₂ , NH(Ci-C ₄ -alkyl), N(Ci-C4-alkyl)2, Ci-C6-alkyl, Ci-C6-halogenalkyl, C2-C6-alkenyl, C2-C6-halogenalkenyl, C2-C6- alkynyl, C2-C6-halogenalkynyl, Ci-C6-alkoxy, Ci-C6-halogenalkoxy, C3-C6-cycloalkyl, C3-C6- halogencycloalkyl and phenyl.

According to one embodiment thereof Q ^3b is independently selected from halogen, OH, CN, Ci- C4-alkyl, Ci-C4-alkoxy, Ci-C4-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C4- halogenalkoxy.

According to one embodiment thereof Q ^3b is independently selected from halogen, CN, C1-C2- alkyl, Ci-C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, Q ^3b is independently selected from F, CI, OH, CN, CH3, OCH3, cyclopropyl, 1 -F-cyclopropyl, 1 -CI-cyclopropyl and halogenmethoxy.

According to a further embodiment thereof Q ^3b is independently selected from Ci-C2-alkyl, Ci- C2-alkoxy, Ci-C2-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl and C1-C2- halogenalkoxy. Specifically, Q ^3b is independently selected from OH, CH3, OCH3, cyclopropyl, 1 - F-cyclopropyl, 1 -CI-cyclopropyl and halogenmethoxy, more specifically independently selected from OH, CH3, OCH3, cyclopropyl, 1 -F-cyclopropyl, 1 -CI-cyclopropyl and OCHF2.

According to a further embodiment thereof R ^3b is independently selected from F, CI and Br

Particularly preferred embodiments of Q ³ according to the invention are in Table P4 below, wherein each line of lines Q3-1 to Q3-180 corresponds to one particular embodiment of the in- vention, wherein Q3-1 to Q3-180 are also in any combination with one another a preferred embodiment of the present invention. The connection point to the W group, to which Q ³ is bound is marked with "#" in the drawings.

Table Q3:

According to one embodiment of the invention W is O.

According to one further embodiment of the invention W is S.

X according to the invention is is in each case independently selected from H, halogen, OH, CN, Ci-C4-alkyl, Ci-C4-alkoxy, Ci-C4-halogenalkyl, C3-C6-cycloalkyl, C3-C6-halogencycloalkyl, Ci-C4-halogenalkoxy and Ci-C6-alkylthio.

X according to the invention is in each case independently selected from H, halogen, CN, C1-C4- alkyl, Ci-C4-halogenalkyl.

According to one specific embodiment, X ist H.

According to a further specific embodiment X is halogen, in particular Br, F or CI, more specifically F or CI.

According to a further specific embodiment, X is CN.

According to a further specific embodiment, X is Ci-C6-alkyl, in particular Ci-C4-alkyl, such as According to a further specific embodiment, X is Ci-C6-alkoxy, in particular Ci-C4-alkoxy, more specifically Ci-C2-alkoxy such as OCH3 or OCH2CH3.

According to a further specific embodiment, X is Ci-C6-halogenalkyl, in particular C1-C4- halogenalkyl, such as CF ₃ , CHF ₂ , CH ₂ F, CCI ₃ , CHC or CH ₂ CI.

According to a further specific embodiment X is C3-C6-cycloalkyl, in particular cyclopropyl.

In a further specific embodiment, X is C3-C6-cycloalkyl, for example cyclopropyl, substituted by one, two, three or up to the maximum possible number of identical or different groups R ^1b as defined and preferably herein.

According to a specific embodiment X is C3-C6-halogencycloalkyl. In a special embodiment R ¹ is fully or partially halogenated cyclopropyl.

According to a further specific embodiment, X is Ci-C6-halogenalkoxy, in particular C1-C4- halogenalkoxy, more specifically Ci-C2-halogenalkoxy such as OCF3, OCHF2, OCH2F, OCCI3, OCHC or OCH2CI, in particular OCF ₃ , OCHF ₂ , OCCI ₃ or OCHCI ₂ .

According to a further specific embodiment, X is selected from H, F, CI, CN, CH3, CF3'.

According to the invention, there can be zero, one, two, three or four X present, namely for n is 0, 1 , 2, 3 or 4.

According to one embodiment, n is 0 or 1.

According to a further embodiment, n is 0.

According to still a further embodiment, n is 1. According to still a further embodiment, n is 2.

According to still a further embodiment, n is 3.

According to still a further embodiment, n is 4.

According to one embodiment of the invention, one X is attached to the 3-position as numbered in formula I above.

According to a further embodiment of the invention, one X is attached to the 4-position as numbered in formula I above.

According to a further embodiment of the invention, one X is attached to the 5-position as numbered in formula I above.

According to a further embodiment of the invention, one X is attached to the 6-position as numbered in formula I above.

According to a further embodiment of the invention, two X are attached in 3,4- -position as numbered in formula I above.

According to a further embodiment of the invention, two X are attached in 3,5- -position as numbered in formula I above.

According to a further embodiment of the invention, two X are attached in 4,5- -position as numbered in formula I above.

According to a further embodiment of the invention, two X are attached in 3,6- -position as numbered in formula I above.

According to a further embodiment of the invention, two X are attached in 4,6- -position as numbered in formula I above.

According to a further embodiment of the invention, two X are attached in 5,6- -position as numbered in formula I above.

For every X that is present in the inventive compounds, the following embodiments and preferences apply independently of the meaning of the other X that may be present in the ring. Furthermore, the particular embodiments and preferences given herein for X apply inde- pendently for each of n=1 and n=2.

According to one specific embodiment, X is halogen, in particular Br, F or CI, more specifically F or CI.

According to a further specific embodiment, X is CN.

According to a further specific embodiment, X is Ci-C6-alkyl, in particular Ci-C4-alkyl, such as CHs.

According to a further specific embodiment, X is Ci-C6-halogenalkyl, in particular C1-C4- halogenalkyl, such as CF ₃ , CHF ₂ , CH ₂ F, CCI ₃ , CHC or CH ₂ CI.

According to a further specific embodiment, X is Ci-C6-alkoxy, in particular Ci-C4-alkoxy, more specifically Ci-C2-alkoxy such as OCH ₃ or OCH2CH3.

According to a further specific embodiment X is C3-C6-cycloalkyl, in particular cyclopropyl.

In a further specific embodiment, X is C3-C6-cycloalkyl, for example cyclopropyl, substituted by one, two, three or up to the maximum possible number of identical or different groups R ^2b as defined and preferably herein.

According to a specific embodiment X is C3-C6-halogencycloalkyl. In a special embodiment X is fully or partially halogenated cyclopropyl.

According to still a further specific embodiment, X is Ci-C6-halogenalkoxy, in particular C1-C4- halogenalkoxy, more specifically Ci-C2-halogenalkoxy such as OCF3, OCHF2, OCH2F, OCCI3, OCHC or OCH2CI, in particular OCF ₃ , OCHF ₂ , OCCI ₃ or OCHCI ₂ .

Preferred embodiments of the present invention are the following compounds I .A, I.B, I.C, I.D, I.E, I.F and I.G. In these formulae, the substituents R ¹ R ² , R ³ , R ⁴ , Q ³ X and n are independently as defined or preferably defined herein:

I.G

Preferred embodiments of the present invention are the following compounds I.A-2 to I.A-12, I.B-2 to I.B-12, I.C-2 to I.C-12, I.D-2 to I.D-12, I.E-2 to I.E-12, I.F-2 to I.F-12, I.G-2 to I.G-12. In these formulae, the substituents R ¹ ,R ² , R ³ , R ⁴ , Q ³ , X and n are independently as defined or preferably defined herein:

I.G-2

I.G-3

I.G-4

I.G-5

PCT/EP2016/078958

PCT/EP2016/078958

I.G-9

.G-12

In particular with a view to their use, according to one embodiment, preference is given to the compounds of the formula I.A-1 to I.A-12, I.B-1 to I.B-12, I.C-1 to I.C-12, I.D-1 to I.D-12, I.E-1 to I.E-12, I.F-1 to I.F-12, I.G-1 to I.G-12 that are compiled in the Tables 1 a to 6a, Tables 1 b to 6b, Tables 1 c to 6c, Tables 1 d to 6d, Tables 1 e to 6e, Tables 1f to 6f, Tables 1 g to 6g, Tables 1 h to 6h, Tables 1 i to 6i and Tables 1j to 6j. Each of the groups mentioned for a substituent in the tables is furthermore per se, independently of the combination in which it is mentioned, a particularly preferred aspect of the substituent in question.

Table 1 a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-1 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(

compounds .A-2.X-1 .A-1 to

compounds .C-2.X-1.A-1 to

compounds .E-2.X-1 .A-1 to

compounds .G-2.X-1.A-- to

compounds .A-3.X-1 .A-1 to

compounds .C-3.X-1.A-1 to

compounds .E-3.X-1.A-1 to

compounds .G-3.X-1.A-1 to

compounds .A-4.X-1 .A-1 to

compounds .C-4.X-1.A-1 to

compounds .E-4.X-1 .A-1 to

compounds .G-4.X-1.A-1 to

compounds .A-5.X-1.A-1 to

compounds .C-5.X-1.A-1 to

compounds .E-5.X-1 .A-1 to

compounds .G-5.X-1.A-1 to

compounds .A-6.X-1 .A-1 to

compounds .C-6.X-1.A-1 to

compounds .E-6.X-1 .A-1 to

compounds .G-6.X-1.A-1 to

compounds .A-7.X-1 .A-1 to

compounds .C-7.X-1.A-1 to

compounds .E-7.X-1 .A-1 to

compounds .G-7.X-1.A-1 to compounds I.A-8.X-1 .A-1 to I.A-8.X-1.A-3600; compounds I.B-8.X-1.A-1 to I.B-8.X-1.A-3600; compounds I.C-8.X-1.A-1 to I.C-8.X-1.A-3600; compounds I.D-8.X-1.A-1 to I.D-8.X-1.A-3600; compounds I.E-8.X-1.A-1 to I.E-8.X-1.A-3600; compounds I.F-8.X-1 .A-1 to I.F-8.X-1 .A-3600; compounds I.G-8.X-1.A-1 to I.G-8.X-1.A-3600;

compounds I.A-9.X-1 .A-1 to I.A-9.X-1.A-3600; compounds I.B-9.X-1.A-1 to I.B-9.X-1.A-3600; compounds I.C-9.X-1.A-1 to I. C-9.X-1.A-3600; compounds I.D-9.X-1.A-1 to I. D-9.X-1.A-3600; compounds I.E-9.X-1 .A-1 to I. E-9.X-1.A-3600; compounds I.F-9.X-1 .A-1 to I. F-9.X-1 .A-3600; compounds I.G-9.X-1.A-1 to I.G-9.X-1.A-3600;

compounds I.A-10.X-1.A-1 to I.A-10.X-1.A-3600; compounds I.B-10.X-1.A-1 to I.B-10.X-1.A- 3600; compounds I.C-10.X-1.A-1 to I.C-10.X-1.A-3600; compounds I.D-10.X-1.A-1 to I.D-10.X- 1 . A-3600; compounds I.E-10.X-1 .A-1 to I.E-10.X-1.A-3600; compounds I.F-10.X-1 .A-1 to I.F- 10.X-1.A-3600; compounds I.G-10.X-1.A-1 to I.G-10.X-1.A-3600;

compounds I.A-1 1 .X-1.A-1 to I. A-1 1.X-1. A-3600; compounds I.B-1 1 .X-1.A-1 to I.B-1 1 .X-1.A- 3600; compounds I.C-1 1.X-1.A-1 to I.C-1 1.X-1 .A-3600; compounds I.D-1 1.X-1.A-1 to I.D-1 1.X- 1 . A-3600; compounds I.E-1 1.X-1 .A-1 to I. E-1 1.X-1. A-3600; compounds I.F-1 1.X-1 .A-1 to I.F- 1 1.X-1 .A-3600; compounds I.G-1 1.X-1.A-1 to I.G-1 1.X-1.A-3600;

compounds I.A-12.X-1.A-1 to I.A-12.X-1.A-3600; compounds I.B-12.X-1.A-1 to I.B-12.X-1.A- 3600; compounds I.C-12.X-1.A-1 to I.C-12.X-1 .A-3600; compounds I.D-12.X-1.A-1 to I.D-12.X- 1 .A-3600; compounds I.E-12.X-1 .A-1 to I.E-12.X-1.A-3600; compounds I.F-12.X-1 .A-1 to I.F- 12.X-1.A-3600; compounds I.G-12.X-1.A-1 to I.G-12.X-1.A-3600).

Table 2a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-2 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (

compounds I.A-2.X-2.A-1 to I.A-2.X-2.A-3600; compounds I.B-2.X-2.A-1 to I.B-2.X-2.A-3600; compounds I.C-2.X-2.A-1 to I.C-2.X-2.A-3600; compounds I.D-2.X-2.A-1 to I.D-2.X-2.A-3600; compounds I.E-2.X-2.A-1 to I.E-2.X-2.A-3600; compounds I.F-2.X-2.A-1 to I.F-2.X-2.A-3600; compounds I.G-2.X-2.A-1 to I.G-2.X-2.A-3600;

compounds I.A-3.X-2.A-1 to I.A-3.X-2.A-3600; compounds I.B-3.X-2.A-1 to I.B-3.X-2.A-3600; compounds I.C-3.X-2.A-1 to I.C-3.X-2.A-3600; compounds I.D-3.X-2.A-1 to I.D-3.X-2.A-3600; compounds I.E-3.X-2.A-1 to I.E-3.X-2.A-3600; compounds I.F-3.X-2.A-1 to I.F-3.X-2.A-3600; compounds I.G-3.X-2.A-1 to I.G-3.X-2.A-3600;

compounds I.A-4.X-2.A-1 to I.A-4.X-2.A-3600; compounds I.B-4.X-2.A-1 to I. B-4.X-2. A-3600; compounds I.C-4.X-2.A-1 to I.C-4.X-2.A-3600; compounds I.D-4.X-2.A-1 to I.D-4.X-2.A-3600; compounds I.E-4.X-2.A-1 to I.E-4.X-2.A-3600; compounds I.F-4.X-2.A-1 to I.F-4.X-2.A-3600; compounds I.G-4.X-2.A-1 to I.G-4.X-2.A-3600;

compounds I.A-5.X-2.A-1 to I.A-5.X-2.A-3600; compounds I.B-5.X-2.A-1 to I.B-5.X-2.A-3600; compounds I.C-5.X-2.A-1 to I.C-5.X-2.A-3600; compounds I.D-5.X-2.A-1 to I.D-5.X-2.A-3600; compounds I.E-5.X-2.A-1 to I.E-5.X-2.A-3600; compounds I.F-5.X-2.A-1 to I.F-5.X-2.A-3600; compounds I.G-5.X-2.A-1 to I.G-5.X-2.A-3600;

compounds I.A-6.X-2.A-1 to I.A-6.X-2.A-3600; compounds I.B-6.X-2.A-1 to I.B-6.X-2.A-3600; compounds I.C-6.X-2.A-1 to I.C-6.X-2.A-3600; compounds I.D-6.X-2.A-1 to I.D-6.X-2.A-3600; compounds I.E-6.X-2.A-1 to I.E-6.X-2.A-3600; compounds I.F-6.X-2.A-1 to I.F-6.X-2.A-3600; compounds I.G-6.X-2.A-1 to I.G-6.X-2.A-3600;

compounds I.A-7.X-2.A-1 to I.A-7.X-2.A-3600; compounds I.B-7.X-2.A-1 to I.B-7.X-2.A-3600; compounds I.C-7.X-2.A-1 to I.C-7.X-2.A-3600; compounds I.D-7.X-2.A-1 to I.D-7.X-2.A-3600; compounds I.E-7.X-2.A-1 to I.E-7.X-2.A-3600; compounds I.F-7.X-2.A-1 to I.F-7.X-2.A-3600; compounds I.G-7.X-2.A-1 to I.G-7.X-2.A-3600;

compounds I.A-8.X-2.A-1 to I.A-8.X-2.A-3600; compounds I.B-8.X-2.A-1 to I.B-8.X-2.A-3600; compounds I.C-8.X-2.A-1 to I.C-8.X-2.A-3600; compounds I.D-8.X-2.A-1 to I.D-8.X-2.A-3600; compounds I.E-8.X-2.A-1 to I.E-8.X-2.A-3600; compounds I.F-8.X-2.A-1 to I.F-8.X-2.A-3600; compounds I.G-8.X-2.A-1 to I.G-8.X-2.A-3600;

compounds I.A-9.X-2.A-1 to I.A-9.X-2.A-3600; compounds I.B-9.X-2.A-1 to I.B-9.X-2.A-3600; compounds I.C-9.X-2.A-1 to I.C-9.X-2.A-3600; compounds I.D-9.X-2.A-1 to I.D-9.X-2.A-3600; compounds I.E-9.X-2.A-1 to I.E-9.X-2.A-3600; compounds I.F-9.X-2.A-1 to I.F-9.X-2.A-3600; compounds I.G-9.X-2.A-1 to I.G-9.X-2.A-3600;

compounds I.A-10.X-2.A-1 to I.A-10.X-2.A-3600; compounds I.B-10.X-2.A-1 to I.B-10.X-2.A- 3600; compounds I.C-10.X-2.A-1 to I.C-10.X-2.A-3600; compounds I.D-10.X-2.A-1 to I.D-10.X- 2.A-3600; compounds I.E-10.X-2.A-1 to I.E-10.X-2.A-3600; compounds I.F-10.X-2.A-1 to I.F- 10.X-2.A-3600; compounds I.G-10.X-2.A-1 to I.G-10.X-2.A-3600;

compounds I.A-1 1.X-2.A-1 to I.A-1 1.X-2.A-3600; compounds I.B-1 1 .X-2.A-1 to I.B-1 1 .X-2.A- 3600; compounds I.C-1 1.X-2.A-1 to I.C-1 1.X-2.A-3600; compounds I.D-1 1.X-2.A-1 to I.D-1 1.X- 2.A-3600; compounds I.E-1 1.X-2.A-1 to I.E-1 1.X-2.A-3600; compounds I.F-1 1.X-2.A-1 to I.F- 1 1.X-2.A-3600; compounds I.G-1 1.X-2.A-1 to I.G-1 1.X-2.A-3600;

compounds I.A-12.X-2.A-1 to I.A-12.X-2.A-3600; compounds I.B-12.X-2.A-1 to I.B-12.X-2.A- 3600; compounds I.C-12.X-2.A-1 to I.C-12.X-2.A-3600; compounds I.D-12.X-2.A-1 to I.D-12.X- 2.A-3600; compounds I.E-12.X-2.A-1 to I.E-12.X-2.A-3600; compounds I.F-12.X-2.A-1 to I.F- 12.X-2.A-3600; compounds I.G-12.X-2.A-1 to I.G-12.X-2.A-3600).

Table 3a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12; in which X _n is as defined in line X-3 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-3.A-1 to I.A-2.X-3.A-3600; compounds I.B-2.X-3.A-1 to I.B-2.X-3.A-3600; compounds I.C-2.X-3.A-1 to I.C-2.X-3.A-3600; compounds I.D-2.X-3.A-1 to I.D-2.X-3.A-3600; compounds I.E-2.X-3.A-1 to I.E-2.X-3.A-3600; compounds I.F-2.X-3.A-1 to I.F-2.X-3.A-3600; compounds I.G-2.X-3.A-1 to I.G-2.X-3.A-3600;

compounds I.A-3.X-3.A-1 to I.A-3.X-3.A-3600; compounds I.B-3.X-3.A-1 to I.B-3.X-3.A-3600; compounds I.C-3.X-3.A-1 to I.C-3.X-3.A-3600; compounds I.D-3.X-3.A-1 to I.D-3.X-3.A-3600; compounds I.E-3.X-3.A-1 to I.E-3.X-3.A-3600; compounds I.F-3.X-3.A-1 to I.F-3.X-3.A-3600; compounds I.G-3.X-3.A-1 to I.G-3.X-3.A-3600;

compounds I.A-4.X-3.A-1 to I.A-4.X-3.A-3600; compounds I.B-4.X-3.A-1 to I.B-4.X-3.A-3600; compounds I.C-4.X-3.A-1 to I.C-4.X-3.A-3600; compounds I.D-4.X-3.A-1 to I.D-4.X-3.A-3600; compounds I.E-4.X-3.A-1 to I.E-4.X-3.A-3600; compounds I.F-4.X-3.A-1 to I.F-4.X-3.A-3600; compounds I.G-4.X-3.A-1 to I.G-4.X-3.A-3600;

compounds I.A-5.X-3.A-1 to I.A-5.X-3.A-3600; compounds I.B-5.X-3.A-1 to I.B-5.X-3.A-3600; compounds I.C-5.X-3.A-1 to I.C-5.X-3.A-3600; compounds I.D-5.X-3.A-1 to I.D-5.X-3.A-3600; compounds I.E-5.X-3.A-1 to I.E-5.X-3.A-3600; compounds I.F-5.X-3.A-1 to I.F-5.X-3.A-3600; compounds I.G-5.X-3.A-1 to I.G-5.X-3.A-3600;

compounds I.A-6.X-3.A-1 to I.A-6.X-3.A-3600; compounds I.B-6.X-3.A-1 to I.B-6.X-3.A-3600; compounds I.C-6.X-3.A-1 to I.C-6.X-3.A-3600; compounds I.D-6.X-3.A-1 to I.D-6.X-3.A-3600; compounds I.E-6.X-3.A-1 to I.E-6.X-3.A-3600; compounds I.F-6.X-3.A-1 to I.F-6.X-3.A-3600; compounds I.G-6.X-3.A-1 to I.G-6.X-3.A-3600;

compounds I.A-7.X-3.A-1 to I.A-7.X-3.A-3600; compounds I.B-7.X-3.A-1 to I.B-7.X-3.A-3600; compounds I.C-7.X-3.A-1 to I.C-7.X-3.A-3600; compounds I.D-7.X-3.A-1 to I.D-7.X-3.A-3600; compounds I.E-7.X-3.A-1 to I.E-7.X-3.A-3600; compounds I.F-7.X-3.A-1 to I.F-7.X-3.A-3600; compounds I.G-7.X-3.A-1 to I.G-7.X-3.A-3600;

compounds I.A-8.X-3.A-1 to I.A-8.X-3.A-3600; compounds I.B-8.X-3.A-1 to I.B-8.X-3.A-3600; compounds I.C-8.X-3.A-1 to I.C-8.X-3.A-3600; compounds I.D-8.X-3.A-1 to I.D-8.X-3.A-3600; compounds I.E-8.X-3.A-1 to I.E-8.X-3.A-3600; compounds I.F-8.X-3.A-1 to I.F-8.X-3.A-3600; compounds I.G-8.X-3.A-1 to I.G-8.X-3.A-3600;

compounds I.A-9.X-3.A-1 to I.A-9.X-3.A-3600; compounds I.B-9.X-3.A-1 to I.B-9.X-3.A-3600; compounds I.C-9.X-3.A-1 to I.C-9.X-3.A-3600; compounds I.D-9.X-3.A-1 to I.D-9.X-3.A-3600; compounds I.E-9.X-3.A-1 to I.E-9.X-3.A-3600; compounds I.F-9.X-3.A-1 to I.F-9.X-3.A-3600; compounds I.G-9.X-3.A-1 to I.G-9.X-3.A-3600;

compounds I.A-10.X-3.A-1 to I.A-10.X-3.A-3600; compounds I.B-10.X-3.A-1 to I.B-10.X-3.A- 3600; compounds I.C-10.X-3.A-1 to I.C-10.X-3.A-3600; compounds I.D-10.X-3.A-1 to I.D-10.X- 3.A-3600; compounds I.E-10.X-3.A-1 to I.E-10.X-3.A-3600; compounds I.F-10.X-3.A-1 to I.F- 10.X-3.A-3600; compounds I.G-10.X-3.A-1 to I.G-10.X-3.A-3600;

compounds I.A-1 1.X-3.A-1 to I.A-1 1.X-3.A-3600; compounds I.B-1 1 .X-3.A-1 to I.B-1 1 .X-3.A- 3600; compounds I.C-1 1.X-3.A-1 to I.C-1 1.X-3.A-3600; compounds I.D-1 1.X-3.A-1 to I.D-1 1.X- 3.A-3600; compounds I.E-1 1.X-3.A-1 to I.E-1 1.X-3.A-3600; compounds I.F-1 1.X-3.A-1 to I.F- 1 1.X-3.A-3600; compounds I.G-1 1.X-3.A-1 to I.G-1 1.X-3.A-3600;

compounds I.A-12.X-3.A-1 to I.A-12.X-3.A-3600; compounds I.B-12.X-3.A-1 to I.B-12.X-3.A- 3600; compounds I.C-12.X-3.A-1 to I.C-12.X-3.A-3600; compounds I.D-12.X-3.A-1 to I.D-12.X- 3.A-3600; compounds I.E-12.X-3.A-1 to I.E-12.X-3.A-3600; compounds I.F-12.X-3.A-1 to I.F- 12.X-3.A-3600; compounds I.G-12.X-3.A-1 to I.G-12.X-3.A-3600).

Table 4a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-4 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (compounds I.A-2.X-4.A-1 to I.A-2.X-4.A-3600; compounds I.B-2.X-4.A-1 to I.B-2.X-4.A-3600; compounds I.C-2.X-4.A-1 to I.C-2.X-4.A-3600; compounds I.D-2.X-4.A-1 to I.D-2.X-4.A-3600; compounds I.E-2.X-4.A-1 to I.E-2.X-4.A-3600; compounds I.F-2.X-4.A-1 to I.F-2.X-4.A-3600; compounds I.G-2.X-4.A-1 to I.G-2.X-4.A-3600;

compounds I.A-3.X-4.A-1 to I.A-3.X-4.A-3600; compounds I.B-3.X-4.A-1 to I.B-3.X-4.A-3600; compounds I.C-3.X-4.A-1 to I.C-3.X-4.A-3600; compounds I.D-3.X-4.A-1 to I.D-3.X-4.A-3600; compounds I.E-3.X-4.A-1 to I.E-3.X-4.A-3600; compounds I.F-3.X-4.A-1 to I.F-3.X-4.A-3600; compounds I.G-3.X-4.A-1 to I.G-3.X-4.A-3600;

compounds I.A-4.X-4.A-1 to I.A-4.X-4.A-3600; compounds I.B-4.X-4.A-1 to I.B-4.X-4.A-3600; compounds I.C-4.X-4.A-1 to I.C-4.X-4.A-3600; compounds I.D-4.X-4.A-1 to I.D-4.X-4.A-3600; compounds I.E-4.X-4.A-1 to I.E-4.X-4.A-3600; compounds I.F-4.X-4.A-1 to I.F-4.X-4.A-3600; compounds I.G-4.X-4.A-1 to I.G-4.X-4.A-3600;

compounds I.A-5.X-4.A-1 to I.A-5.X-4.A-3600; compounds I.B-5.X-4.A-1 to I.B-5.X-4.A-3600; compounds I.C-5.X-4.A-1 to I.C-5.X-4.A-3600; compounds I.D-5.X-4.A-1 to I.D-5.X-4.A-3600; compounds I.E-5.X-4.A-1 to I.E-5.X-4.A-3600; compounds I.F-5.X-4.A-1 to I.F-5.X-4.A-3600; compounds I.G-5.X-4.A-1 to I.G-5.X-4.A-3600;

compounds I.A-6.X-4.A-1 to I.A-6.X-4.A-3600; compounds I.B-6.X-4.A-1 to I.B-6.X-4.A-3600; compounds I.C-6.X-4.A-1 to I.C-6.X-4.A-3600; compounds I.D-6.X-4.A-1 to I.D-6.X-4.A-3600; compounds I.E-6.X-4.A-1 to I.E-6.X-4.A-3600; compounds I.F-6.X-4.A-1 to I.F-6.X-4.A-3600; compounds I.G-6.X-4.A-1 to I.G-6.X-4.A-3600;

compounds I.A-7.X-4.A-1 to I.A-7.X-4.A-3600; compounds I.B-7.X-4.A-1 to I.B-7.X-4.A-3600; compounds I.C-7.X-4.A-1 to I.C-7.X-4.A-3600; compounds I.D-7.X-4.A-1 to I.D-7.X-4.A-3600; compounds I.E-7.X-4.A-1 to I.E-7.X-4.A-3600; compounds I.F-7.X-4.A-1 to I.F-7.X-4.A-3600; compounds I.G-7.X-4.A-1 to I.G-7.X-4.A-3600;

compounds I.A-8.X-4.A-1 to I.A-8.X-4.A-3600; compounds I.B-8.X-4.A-1 to I.B-8.X-4.A-3600; compounds I.C-8.X-4.A-1 to I.C-8.X-4.A-3600; compounds I.D-8.X-4.A-1 to I.D-8.X-4.A-3600; compounds I.E-8.X-4.A-1 to I.E-8.X-4.A-3600; compounds I.F-8.X-4.A-1 to I.F-8.X-4.A-3600; compounds I.G-8.X-4.A-1 to I.G-8.X-4.A-3600;

compounds I.A-9.X-4.A-1 to I.A-9.X-4.A-3600; compounds I.B-9.X-4.A-1 to I.B-9.X-4.A-3600; compounds I.C-9.X-4.A-1 to I.C-9.X-4.A-3600; compounds I.D-9.X-4.A-1 to I.D-9.X-4.A-3600; compounds I.E-9.X-4.A-1 to I.E-9.X-4.A-3600; compounds I.F-9.X-4.A-1 to I.F-9.X-4.A-3600; compounds I.G-9.X-4.A-1 to I.G-9.X-4.A-3600;

compounds I.A-10.X-4.A-1 to I.A-10.X-4.A-3600; compounds I.B-10.X-4.A-1 to I.B-10.X-4.A- 3600; compounds I.C-10.X-4.A-1 to I.C-10.X-4.A-3600; compounds I.D-10.X-4.A-1 to I.D-10.X- 4.A-3600; compounds I.E-10.X-4.A-1 to I.E-10.X-4.A-3600; compounds I.F-10.X-4.A-1 to I.F- 10.X-4.A-3600; compounds I.G-10.X-4.A-1 to I.G-10.X-4.A-3600;

compounds I.A-1 1.X-4.A-1 to I.A-1 1.X-4.A-3600; compounds I.B-1 1 .X-4.A-1 to I.B-1 1 .X-4.A- 3600; compounds I.C-1 1.X-4.A-1 to I.C-1 1.X-4.A-3600; compounds I.D-1 1.X-4.A-1 to I.D-1 1.X- 4.A-3600; compounds I.E-1 1.X-4.A-1 to I.E-1 1.X-4.A-3600; compounds I.F-1 1.X-4.A-1 to I.F- 1 1.X-4.A-3600; compounds I.G-1 1.X-4.A-1 to I.G-1 1.X-4.A-3600;

compounds I.A-12.X-4.A-1 to I.A-12.X-4.A-3600; compounds I.B-12.X-4.A-1 to I.B-12.X-4.A- 3600; compounds I.C-12.X-4.A-1 to I.C-12.X-4.A-3600; compounds I.D-12.X-4.A-1 to I.D-12.X- 4.A-3600; compounds I.E-12.X-4.A-1 to I.E-12.X-4.A-3600; compounds I.F-12.X-4.A-1 to I.F- 12.X-4.A-3600; compounds I.G-12.X-4.A-1 to I.G-12.X-4.A-3600).

Table 5a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-5 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-5.A-1 to I.A-2.X-5.A-3600; compounds I.B-2.X-5.A-1 to I.B-2.X-5.A-3600; compounds I.C-2.X-5.A-1 to I.C-2.X-5.A-3600; compounds I.D-2.X-5.A-1 to I.D-2.X-5.A-3600; compounds I.E-2.X-5.A-1 to I.E-2.X-5.A-3600; compounds I.F-2.X-5.A-1 to I.F-2.X-5.A-3600; compounds I.G-2.X-5.A-1 to I.G-2.X-5.A-3600;

compounds I.A-3.X-5.A-1 to I.A-3.X-5.A-3600; compounds I.B-3.X-5.A-1 to I.B-3.X-5.A-3600; compounds I.C-3.X-5.A-1 to I.C-3.X-5.A-3600; compounds I.D-3.X-5.A-1 to I.D-3.X-5.A-3600; compounds I.E-3.X-5.A-1 to I.E-3.X-5.A-3600; compounds I.F-3.X-5.A-1 to I.F-3.X-5.A-3600; compounds I.G-3.X-5.A-1 to I.G-3.X-5.A-3600;

compounds I.A-4.X-5.A-1 to I.A-4.X-5.A-3600; compounds I.B-4.X-5.A-1 to I.B-4.X-5.A-3600; compounds I.C-4.X-5.A-1 to I.C-4.X-5.A-3600; compounds I.D-4.X-5.A-1 to I.D-4.X-5.A-3600; compounds I.E-4.X-5.A-1 to I.E-4.X-5.A-3600; compounds I.F-4.X-5.A-1 to I.F-4.X-5.A-3600; compounds I.G-4.X-5.A-1 to I.G-4.X-5.A-3600;

compounds I.A-5.X-5.A-1 to I.A-5.X-5.A-3600; compounds I.B-5.X-5.A-1 to I.B-5.X-5.A-3600; compounds I.C-5.X-5.A-1 to I.C-5.X-5.A-3600; compounds I.D-5.X-5.A-1 to I.D-5.X-5.A-3600; compounds I.E-5.X-5.A-1 to I.E-5.X-5.A-3600; compounds I.F-5.X-5.A-1 to I.F-5.X-5.A-3600; compounds I.G-5.X-5.A-1 to I.G-5.X-5.A-3600;

compounds I.A-6.X-5.A-1 to I.A-6.X-5.A-3600; compounds I.B-6.X-5.A-1 to I.B-6.X-5.A-3600; compounds I.C-6.X-5.A-1 to I.C-6.X-5.A-3600; compounds I.D-6.X-5.A-1 to I.D-6.X-5.A-3600; compounds I.E-6.X-5.A-1 to I.E-6.X-5.A-3600; compounds I.F-6.X-5.A-1 to I.F-6.X-5.A-3600; compounds I.G-6.X-5.A-1 to I.G-6.X-5.A-3600;

compounds I.A-7.X-5.A-1 to I.A-7.X-5.A-3600; compounds I.B-7.X-5.A-1 to I.B-7.X-5.A-3600; compounds I.C-7.X-5.A-1 to I.C-7.X-5.A-3600; compounds I.D-7.X-5.A-1 to I.D-7.X-5.A-3600; compounds I.E-7.X-5.A-1 to I.E-7.X-5.A-3600; compounds I.F-7.X-5.A-1 to I.F-7.X-5.A-3600; compounds I.G-7.X-5.A-1 to I.G-7.X-5.A-3600;

compounds I.A-8.X-5.A-1 to I.A-8.X-5.A-3600; compounds I.B-8.X-5.A-1 to I.B-8.X-5.A-3600; compounds I.C-8.X-5.A-1 to I.C-8.X-5.A-3600; compounds I.D-8.X-5.A-1 to I.D-8.X-5.A-3600; compounds I.E-8.X-5.A-1 to I.E-8.X-5.A-3600; compounds I.F-8.X-5.A-1 to I.F-8.X-5.A-3600; compounds I.G-8.X-5.A-1 to I.G-8.X-5.A-3600;

compounds I.A-9.X-5.A-1 to I.A-9.X-5.A-3600; compounds I.B-9.X-5.A-1 to I.B-9.X-5.A-3600; compounds I.C-9.X-5.A-1 to I.C-9.X-5.A-3600; compounds I.D-9.X-5.A-1 to I.D-9.X-5.A-3600; compounds I.E-9.X-5.A-1 to I.E-9.X-5.A-3600; compounds I.F-9.X-5.A-1 to I.F-9.X-5.A-3600; compounds I.G-9.X-5.A-1 to I.G-9.X-5.A-3600;

compounds I.A-10.X-5.A-1 to I.A-10.X-5.A-3600; compounds I.B-10.X-5.A-1 to I.B-10.X-5.A- 3600; compounds I.C-10.X-5.A-1 to I.C-10.X-5.A-3600; compounds I.D-10.X-5.A-1 to I.D-10.X- 5.A-3600; compounds I.E-10.X-5.A-1 to I.E-10.X-5.A-3600; compounds I.F-10.X-5.A-1 to I.F- 10.X-5.A-3600; compounds I.G-10.X-5.A-1 to I.G-10.X-5.A-3600;

compounds I.A-1 1.X-5.A-1 to I.A-1 1.X-5.A-3600; compounds I.B-1 1 .X-5.A-1 to I.B-1 1 .X-5.A- 3600; compounds I.C-1 1.X-5.A-1 to I.C-1 1.X-5.A-3600; compounds I.D-1 1.X-5.A-1 to I.D-1 1.X- 5.A-3600; compounds I.E-1 1.X-5.A-1 to I.E-1 1.X-5.A-3600; compounds I.F-1 1.X-5.A-1 to I.F- 1 1.X-5.A-3600; compounds I.G-1 1.X-5.A-1 to I.G-1 1.X-5.A-3600;

compounds I.A-12.X-5.A-1 to I.A-12.X-5.A-3600; compounds I.B-12.X-5.A-1 to I.B-12.X-5.A- 3600; compounds I.C-12.X-5.A-1 to I.C-12.X-5.A-3600; compounds I.D-12.X-5.A-1 to I.D-12.X- 5.A-3600; compounds I.E-12.X-5.A-1 to I.E-12.X-5.A-3600; compounds I.F-12.X-5.A-1 to I.F- 12.X-5.A-3600; compounds I.G-12.X-5.A-1 to I.G-12.X-5.A-3600).

Table 6a

Compounds of the formula; I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-6 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (compounds I.A-2.X-6.A-1 to I.A-2.X-6.A-3600; compounds I.B-2.X-6.A-1 to I.B-2.X-6.A-3600; compounds I.C-2.X-6.A-1 to I.C-2.X-6.A-3600; compounds I.D-2.X-6.A-1 to I.D-2.X-6.A-3600; compounds I.E-2.X-6.A-1 to I.E-2.X-6.A-3600; compounds I.F-2.X-6.A-1 to I.F-2.X-6.A-3600; compounds I.G-2.X-6.A-1 to I.G-2.X-6.A-3600;

compounds I.A-3.X-6.A-1 to I.A-3.X-6.A-3600; compounds I.B-3.X-6.A-1 to I.B-3.X-6.A-3600; compounds I.C-3.X-6.A-1 to I.C-3.X-6.A-3600; compounds I.D-3.X-6.A-1 to I.D-3.X-6.A-3600; compounds I.E-3.X-6.A-1 to I.E-3.X-6.A-3600; compounds I.F-3.X-6.A-1 to I.F-3.X-6.A-3600; compounds I.G-3.X-6.A-1 to I.G-3.X-6.A-3600;

compounds I.A-4.X-6.A-1 to I.A-4.X-6.A-3600; compounds I.B-4.X-6.A-1 to I.B-4.X-6.A-3600; compounds I.C-4.X-6.A-1 to I.C-4.X-6.A-3600; compounds I.D-4.X-6.A-1 to I.D-4.X-6.A-3600; compounds I.E-4.X-6.A-1 to I.E-4.X-6.A-3600; compounds I.F-4.X-6.A-1 to I.F-4.X-6.A-3600; compounds I.G-4.X-6.A-1 to I.G-4.X-6.A-3600;

compounds I.A-5.X-6.A-1 to I.A-5.X-6.A-3600; compounds I.B-5.X-6.A-1 to I.B-5.X-6.A-3600; compounds I.C-5.X-6.A-1 to I.C-5.X-6.A-3600; compounds I.D-5.X-6.A-1 to I.D-5.X-6.A-3600; compounds I.E-5.X-6.A-1 to I.E-5.X-6.A-3600; compounds I.F-5.X-6.A-1 to I.F-5.X-6.A-3600; compounds I.G-5.X-6.A-1 to I.G-5.X-6.A-3600;

compounds I.A-6.X-6.A-1 to I.A-6.X-6.A-3600; compounds I.B-6.X-6.A-1 to I.B-6.X-6.A-3600; compounds I.C-6.X-6.A-1 to I.C-6.X-6.A-3600; compounds I.D-6.X-6.A-1 to I.D-6.X-6.A-3600; compounds I.E-6.X-6.A-1 to I.E-6.X-6.A-3600; compounds I.F-6.X-6.A-1 to I.F-6.X-6.A-3600; compounds I.G-6.X-6.A-1 to I.G-6.X-6.A-3600;

compounds I.A-7.X-6.A-1 to I.A-7.X-6.A-3600; compounds I.B-7.X-6.A-1 to I.B-7.X-6.A-3600; compounds I.C-7.X-6.A-1 to I.C-7.X-6.A-3600; compounds I.D-7.X-6.A-1 to I.D-7.X-6.A-3600; compounds I.E-7.X-6.A-1 to I.E-7.X-6.A-3600; compounds I.F-7.X-6.A-1 to I.F-7.X-6.A-3600; compounds I.G-7.X-6.A-1 to I.G-7.X-6.A-3600;

compounds I.A-8.X-6.A-1 to I.A-8.X-6.A-3600; compounds I.B-8.X-6.A-1 to I.B-8.X-6.A-3600; compounds I.C-8.X-6.A-1 to I.C-8.X-6.A-3600; compounds I.D-8.X-6.A-1 to I.D-8.X-6.A-3600; compounds I.E-8.X-6.A-1 to I.E-8.X-6.A-3600; compounds I.F-8.X-6.A-1 to I.F-8.X-6.A-3600; compounds I.G-8.X-6.A-1 to I.G-8.X-6.A-3600;

compounds I.A-9.X-6.A-1 to I.A-9.X-6.A-3600; compounds I.B-9.X-6.A-1 to I.B-9.X-6.A-3600; compounds I.C-9.X-6.A-1 to I.C-9.X-6.A-3600; compounds I.D-9.X-6.A-1 to I.D-9.X-6.A-3600; compounds I.E-9.X-6.A-1 to I.E-9.X-6.A-3600; compounds I.F-9.X-6.A-1 to I.F-9.X-6.A-3600; compounds I.G-9.X-6.A-1 to I.G-9.X-6.A-3600;

compounds I.A-10.X-6.A-1 to I.A-10.X-6.A-3600; compounds I.B-10.X-6.A-1 to I.B-10.X-6.A- 3600; compounds I.C-10.X-6.A-1 to I.C-10.X-6.A-3600; compounds I.D-10.X-6.A-1 to I.D-10.X- 6.A-3600; compounds I.E-10.X-6.A-1 to I.E-10.X-6.A-3600; compounds I.F-10.X-6.A-1 to I.F- 10.X-6.A-3600; compounds I.G-10.X-6.A-1 to I.G-10.X-6.A-3600;

compounds I.A-1 1.X-6.A-1 to I.A-1 1.X-6.A-3600; compounds I.B-1 1 .X-6.A-1 to I.B-1 1 .X-6.A- 3600; compounds I.C-1 1.X-6.A-1 to I.C-1 1 .X-6.A-3600; compounds I.D-1 1.X-6.A-1 to I.D-1 1.X- 6.A-3600; compounds I.E-1 1.X-6.A-1 to I.E-1 1.X-6.A-3600; compounds I.F-1 1.X-6.A-1 to I.F- 1 1.X-6.A-3600; compounds I.G-1 1.X-6.A-1 to I.G-1 1.X-6.A-3600;

compounds I.A-12.X-6.A-1 to I.A-12.X-6.A-3600; compounds I.B-12.X-6.A-1 to I.B-12.X-6.A- 3600; compounds I.C-12.X-6.A-1 to I.C-12.X-6.A-3600; compounds I.D-12.X-6.A-1 to I.D-12.X- 6.A-3600; compounds I.E-12.X-6.A-1 to I.E-12.X-6.A-3600; compounds I.F-12.X-6.A-1 to I.F- 12.X-6.A-3600; compounds I.G-12.X-6.A-1 to I.G-12.X-6.A-3600).

Table 7a

Compounds of the formula; I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-7 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(

compounds I.A-2.X-7.A-1 to I.A-2.X-7.A-3600; compounds I.B-2.X-7.A-1 to I.B-2.X-7.A-3600; compounds I.C-2.X-7.A-1 to I.C-2.X-7.A-3600; compounds I.D-2.X-7.A-1 to I.D-2.X-7.A-3600; compounds I.E-2.X-7.A-1 to I.E-2.X-7.A-3600; compounds I.F-2.X-7.A-1 to I.F-2.X-7.A-3600; compounds I.G-2.X-7.A-1 to I.G-2.X-7.A-3600;

compounds I.A-3.X-7.A-1 to I.A-3.X-7.A-3600; compounds I.B-3.X-7.A-1 to I.B-3.X-7.A-3600; compounds I.C-3.X-7.A-1 to I.C-3.X-7.A-3600; compounds I.D-3.X-7.A-1 to I.D-3.X-7.A-3600; compounds I.E-3.X-7.A-1 to I.E-3.X-7.A-3600; compounds I.F-3.X-7.A-1 to I.F-3.X-7.A-3600; compounds I.G-3.X-7.A-1 to I.G-3.X-7.A-3600;

compounds I.A-4.X-7.A-1 to I.A-4.X-7.A-3600; compounds I.B-4.X-7.A-1 to I.B-4.X-7.A-3600; compounds I.C-4.X-7.A-1 to I.C-4.X-7.A-3600; compounds I.D-4.X-7.A-1 to I.D-4.X-7.A-3600; compounds I.E-4.X-7.A-1 to I.E-4.X-7.A-3600; compounds I.F-4.X-7.A-1 to I.F-4.X-7.A-3600; compounds I.G-4.X-7.A-1 to I.G-4.X-7.A-3600;

compounds I.A-5.X-7.A-1 to I.A-5.X-7.A-3600; compounds I.B-5.X-7.A-1 to I.B-5.X-7.A-3600; compounds I.C-5.X-7.A-1 to I.C-5.X-7.A-3600; compounds I.D-5.X-7.A-1 to I.D-5.X-7.A-3600; compounds I.E-5.X-7.A-1 to I.E-5.X-7.A-3600; compounds I.F-5.X-7.A-1 to I.F-5.X-7.A-3600; compounds I.G-5.X-7.A-1 to I.G-5.X-7.A-3600;

compounds I.A-6.X-7.A-1 to I.A-6.X-7.A-3600; compounds I.B-6.X-7.A-1 to I.B-6.X-7.A-3600; compounds I.C-6.X-7.A-1 to I.C-6.X-7.A-3600; compounds I.D-6.X-7.A-1 to I.D-6.X-7.A-3600; compounds I.E-6.X-7.A-1 to I.E-6.X-7.A-3600; compounds I.F-6.X-7.A-1 to I.F-6.X-7.A-3600; compounds I.G-6.X-7.A-1 to I.G-6.X-7.A-3600;

compounds I.A-7.X-7.A-1 to I.A-7.X-7.A-3600; compounds I.B-7.X-7.A-1 to I.B-7.X-7.A-3600; compounds I.C-7.X-7.A-1 to I.C-7.X-7.A-3600; compounds I.D-7.X-7.A-1 to I.D-7.X-7.A-3600; compounds I.E-7.X-7.A-1 to I.E-7.X-7.A-3600; compounds I.F-7.X-7.A-1 to I.F-7.X-7.A-3600; compounds I.G-7.X-7.A-1 to I.G-7.X-7.A-3600;

compounds I.A-8.X-7.A-1 to I.A-8.X-7.A-3600; compounds I.B-8.X-7.A-1 to I.B-8.X-7.A-3600; compounds I.C-8.X-7.A-1 to I.C-8.X-7.A-3600; compounds I.D-8.X-7.A-1 to I.D-8.X-7.A-3600; compounds I.E-8.X-7.A-1 to I.E-8.X-7.A-3600; compounds I.F-8.X-7.A-1 to I.F-8.X-7.A-3600; compounds I.G-8.X-7.A-1 to I.G-8.X-7.A-3600;

compounds I.A-9.X-7.A-1 to I.A-9.X-7.A-3600; compounds I.B-9.X-7.A-1 to I.B-9.X-7.A-3600; compounds I.C-9.X-7.A-1 to I.C-9.X-7.A-3600; compounds I.D-9.X-7.A-1 to I.D-9.X-7.A-3600; compounds I.E-9.X-7.A-1 to I.E-9.X-7.A-3600; compounds I.F-9.X-7.A-1 to I.F-9.X-7.A-3600; compounds I.G-9.X-7.A-1 to I.G-9.X-7.A-3600;

compounds I.A-10.X-7.A-1 to I.A-10.X-7.A-3600; compounds I.B-10.X-7.A-1 to I.B-10.X-7.A- 3600; compounds I.C-10.X-7.A-1 to I.C-10.X-7.A-3600; compounds I.D-10.X-7.A-1 to I.D-10.X- 7.A-3600; compounds I.E-10.X-7.A-1 to I.E-10.X-7.A-3600; compounds I.F-10.X-7.A-1 to I.F- 10.X-7.A-3600; compounds I.G-10.X-7.A-1 to I.G-10.X-7.A-3600;

compounds I.A-1 1.X-7.A-1 to I.A-1 1.X-7.A-3600; compounds I.B-1 1 .X-7.A-1 to I.B-1 1 .X-7.A- 3600; compounds I.C-1 1.X-7.A-1 to I.C-1 1.X-7.A-3600; compounds I.D-1 1.X-7.A-1 to I.D-1 1.X- 7.A-3600; compounds I.E-1 1.X-7.A-1 to I.E-1 1.X-7.A-3600; compounds I.F-1 1.X-7.A-1 to I.F- 1 1.X-7.A-3600; compounds I.G-1 1.X-7.A-1 to I.G-1 1.X-7.A-3600;

compounds I.A-12.X-7.A-1 to I.A-12.X-7.A-3600; compounds I.B-12.X-7.A-1 to I.B-12.X-7.A- 3600; compounds I.C-12.X-7.A-1 to I.C-12.X-7.A-3600; compounds I.D-12.X-7.A-1 to I.D-12.X-

7. A-3600; compounds I.E-12.X-7.A-1 to I.E-12.X-7.A-3600; compounds I.F-12.X-7.A-1 to I.F- 12.X-7.A-3600; compounds I.G-12.X-7.A-1 to I.G-12.X-7.A-3600).

Table 8a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A-

8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-8 of Table X and the meaning for the combination of ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(

compounds I.A-2.X-8.A-1 to I.A-2.X-8.A-3600; compounds I.B-2.X-8.A-1 to I.B-2.X-8.A-3600; compounds I.C-2.X-8.A-1 to I.C-2.X-8.A-3600; compounds I.D-2.X-8.A-1 to I.D-2.X-8.A-3600; compounds I.E-2.X-8.A-1 to I.E-2.X-8.A-3600; compounds I.F-2.X-8.A-1 to I.F-2.X-8.A-3600; compounds I.G-2.X-8.A-1 to I.G-2.X-8.A-3600;

compounds I.A-3.X-8.A-1 to I.A-3.X-8.A-3600; compounds I.B-3.X-8.A-1 to I.B-3.X-8.A-3600; compounds I.C-3.X-8.A-1 to I.C-3.X-8.A-3600; compounds I.D-3.X-8.A-1 to I.D-3.X-8.A-3600; compounds I.E-3.X-8.A-1 to I.E-3.X-8.A-3600; compounds I.F-3.X-8.A-1 to I.F-3.X-8.A-3600; compounds I.G-3.X-8.A-1 to I.G-3.X-8.A-3600;

compounds I.A-4.X-8.A-1 to I.A-4.X-8.A-3600; compounds I.B-4.X-8.A-1 to I.B-4.X-8.A-3600; compounds I.C-4.X-8.A-1 to I.C-4.X-8.A-3600; compounds I.D-4.X-8.A-1 to I.D-4.X-8.A-3600; compounds I.E-4.X-8.A-1 to I.E-4.X-8.A-3600; compounds I.F-4.X-8.A-1 to I.F-4.X-8.A-3600; compounds I.G-4.X-8.A-1 to I.G-4.X-8.A-3600;

compounds I.A-5.X-8.A-1 to I.A-5.X-8.A-3600; compounds I.B-5.X-8.A-1 to I.B-5.X-8.A-3600; compounds I.C-5.X-8.A-1 to I.C-5.X-8.A-3600; compounds I.D-5.X-8.A-1 to I.D-5.X-8.A-3600; compounds I.E-5.X-8.A-1 to I.E-5.X-8.A-3600; compounds I.F-5.X-8.A-1 to I.F-5.X-8.A-3600; compounds I.G-5.X-8.A-1 to I.G-5.X-8.A-3600;

compounds I.A-6.X-8.A-1 to I.A-6.X-8.A-3600; compounds I.B-6.X-8.A-1 to I.B-6.X-8.A-3600; compounds I.C-6.X-8.A-1 to I.C-6.X-8.A-3600; compounds I.D-6.X-8.A-1 to I.D-6.X-8.A-3600; compounds I.E-6.X-8.A-1 to I.E-6.X-8.A-3600; compounds I.F-6.X-8.A-1 to I.F-6.X-8.A-3600; compounds I.G-6.X-8.A-1 to I.G-6.X-8.A-3600;

compounds I.A-7.X-8.A-1 to I.A-7.X-8.A-3600; compounds I.B-7.X-8.A-1 to I.B-7.X-8.A-3600; compounds I.C-7.X-8.A-1 to I.C-7.X-8.A-3600; compounds I.D-7.X-8.A-1 to I.D-7.X-8.A-3600; compounds I.E-7.X-8.A-1 to I.E-7.X-8.A-3600; compounds I.F-7.X-8.A-1 to I.F-7.X-8.A-3600; compounds I.G-7.X-8.A-1 to I.G-7.X-8.A-3600;

compounds I.A-8.X-8.A-1 to I.A-8.X-8.A-3600; compounds I.B-8.X-8.A-1 to I.B-8.X-8.A-3600; compounds I.C-8.X-8.A-1 to I.C-8.X-8.A-3600; compounds I.D-8.X-8.A-1 to I.D-8.X-8.A-3600; compounds I.E-8.X-8.A-1 to I.E-8.X-8.A-3600; compounds I.F-8.X-8.A-1 to I.F-8.X-8.A-3600; compounds I.G-8.X-8.A-1 to I.G-8.X-8.A-3600;

compounds I.A-9.X-8.A-1 to I.A-9.X-8.A-3600; compounds I.B-9.X-8.A-1 to I.B-9.X-8.A-3600; compounds I.C-9.X-8.A-1 to I.C-9.X-8.A-3600; compounds I.D-9.X-8.A-1 to I.D-9.X-8.A-3600; compounds I.E-9.X-8.A-1 to I.E-9.X-8.A-3600; compounds I.F-9.X-8.A-1 to I.F-9.X-8.A-3600; compounds I.G-9.X-8.A-1 to I.G-9.X-8.A-3600;

compounds I.A-10.X-8.A-1 to I.A-10.X-8.A-3600; compounds I.B-10.X-8.A-1 to I.B-10.X-8.A- 3600; compounds I.C-10.X-8.A-1 to I.C-10.X-8.A-3600; compounds I.D-10.X-8.A-1 to I.D-10.X- 8.A-3600; compounds I.E-10.X-8.A-1 to I.E-10.X-8.A-3600; compounds I.F-10.X-8.A-1 to I.F- 10.X-8.A-3600; compounds I.G-10.X-8.A-1 to I.G-10.X-8.A-3600;

compounds I.A-1 1.X-8.A-1 to I.A-1 1.X-8.A-3600; compounds I.B-1 1 .X-8.A-1 to I.B-1 1 .X-8.A- 3600; compounds I.C-1 1.X-8.A-1 to I.C-1 1.X-8.A-3600; compounds I.D-1 1.X-8.A-1 to I.D-1 1.X- 8.A-3600; compounds I.E-1 1.X-8.A-1 to I.E-1 1.X-8.A-3600; compounds I.F-1 1.X-8.A-1 to I.F- 1 1.X-8.A-3600; compounds I.G-1 1.X-8.A-1 to I.G-1 1.X-8.A-3600;

compounds I.A-12.X-8.A-1 to I.A-12.X-8.A-3600; compounds I.B-12.X-8.A-1 to I.B-12.X-8.A- 3600; compounds I.C-12.X-8.A-1 to I.C-12.X-8.A-3600; compounds I.D-12.X-8.A-1 to I.D-12.X- 8.A-3600; compounds I.E-12.X-8.A-1 to I.E-12.X-8.A-3600; compounds I.F-12.X-8.A-1 to I.F- 12.X-8.A-3600; compounds I.G-12.X-8.A-1 to I.G-12.X-8.A-3600).

Table 9a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-9 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (compounds I.A-2.X-9.A-1 to I.A-2.X-9.A-3600; compounds I.B-2.X-9.A-1 to I.B-2.X-9.A-3600; compounds I.C-2.X-9.A-1 to I.C-2.X-9.A-3600; compounds I.D-2.X-9.A-1 to I.D-2.X-9.A-3600; compounds I.E-2.X-9.A-1 to I.E-2.X-9.A-3600; compounds I.F-2.X-9.A-1 to I.F-2.X-9.A-3600; compounds I.G-2.X-9.A-1 to I.G-2.X-9.A-3600;

compounds I.A-3.X-9.A-1 to I.A-3.X-9.A-3600; compounds I.B-3.X-9.A-1 to I.B-3.X-9.A-3600; compounds I.C-3.X-9.A-1 to I.C-3.X-9.A-3600; compounds I.D-3.X-9.A-1 to I.D-3.X-9.A-3600; compounds I.E-3.X-9.A-1 to I.E-3.X-9.A-3600; compounds I.F-3.X-9.A-1 to I.F-3.X-9.A-3600; compounds I.G-3.X-9.A-1 to I.G-3.X-9.A-3600;

compounds I.A-4.X-9.A-1 to I.A-4.X-9.A-3600; compounds I.B-4.X-9.A-1 to I.B-4.X-9.A-3600; compounds I.C-4.X-9.A-1 to I.C-4.X-9.A-3600; compounds I.D-4.X-9.A-1 to I.D-4.X-9.A-3600; compounds I.E-4.X-9.A-1 to I.E-4.X-9.A-3600; compounds I.F-4.X-9.A-1 to I.F-4.X-9.A-3600; compounds I.G-4.X-9.A-1 to I.G-4.X-9.A-3600;

compounds I.A-5.X-9.A-1 to I.A-5.X-9.A-3600; compounds I.B-5.X-9.A-1 to I.B-5.X-9.A-3600; compounds I.C-5.X-9.A-1 to I.C-5.X-9.A-3600; compounds I.D-5.X-9.A-1 to I.D-5.X-9.A-3600; compounds I.E-5.X-9.A-1 to I.E-5.X-9.A-3600; compounds I.F-5.X-9.A-1 to I.F-5.X-9.A-3600; compounds I.G-5.X-9.A-1 to I.G-5.X-9.A-3600;

compounds I.A-6.X-9.A-1 to I.A-6.X-9.A-3600; compounds I.B-6.X-9.A-1 to I.B-6.X-9.A-3600; compounds I.C-6.X-9.A-1 to I.C-6.X-9.A-3600; compounds I.D-6.X-9.A-1 to I.D-6.X-9.A-3600; compounds I.E-6.X-9.A-1 to I.E-6.X-9.A-3600; compounds I.F-6.X-9.A-1 to I.F-6.X-9.A-3600; compounds I.G-6.X-9.A-1 to I.G-6.X-9.A-3600;

compounds I.A-7.X-9.A-1 to I.A-7.X-9.A-3600; compounds I.B-7.X-9.A-1 to I.B-7.X-9.A-3600; compounds I.C-7.X-9.A-1 to I.C-7.X-9.A-3600; compounds I.D-7.X-9.A-1 to I.D-7.X-9.A-3600; compounds I.E-7.X-9.A-1 to I.E-7.X-9.A-3600; compounds I.F-7.X-9.A-1 to I.F-7.X-9.A-3600; compounds I.G-7.X-9.A-1 to I.G-7.X-9.A-3600;

compounds I.A-8.X-9.A-1 to I.A-8.X-9.A-3600; compounds I.B-8.X-9.A-1 to I.B-8.X-9.A-3600; compounds I.C-8.X-9.A-1 to I.C-8.X-9.A-3600; compounds I.D-8.X-9.A-1 to I.D-8.X-9.A-3600; compounds I.E-8.X-9.A-1 to I.E-8.X-9.A-3600; compounds I.F-8.X-9.A-1 to I.F-8.X-9.A-3600; compounds I.G-8.X-9.A-1 to I.G-8.X-9.A-3600;

compounds I.A-9.X-9.A-1 to I.A-9.X-9.A-3600; compounds I.B-9.X-9.A-1 to I.B-9.X-9.A-3600; compounds I.C-9.X-9.A-1 to I.C-9.X-9.A-3600; compounds I.D-9.X-9.A-1 to I.D-9.X-9.A-3600; compounds I.E-9.X-9.A-1 to I.E-9.X-9.A-3600; compounds I.F-9.X-9.A-1 to I.F-9.X-9.A-3600; compounds I.G-9.X-9.A-1 to I.G-9.X-9.A-3600;

compounds I.A-10.X-9.A-1 to I.A-10.X-9.A-3600; compounds I.B-10.X-9.A-1 to I.B-10.X-9.A- 3600; compounds I.C-10.X-9.A-1 to I.C-10.X-9.A-3600; compounds I.D-10.X-9.A-1 to I.D-10.X- 9.A-3600; compounds I.E-10.X-9.A-1 to I.E-10.X-9.A-3600; compounds I.F-10.X-9.A-1 to I.F- 10.X-9.A-3600; compounds I.G-10.X-9.A-1 to I.G-10.X-9.A-3600;

compounds I.A-1 1.X-9.A-1 to I.A-1 1.X-9.A-3600; compounds I.B-1 1 .X-9.A-1 to I.B-1 1 .X-9.A- 3600; compounds I.C-1 1.X-9.A-1 to I.C-1 1.X-9.A-3600; compounds I.D-1 1.X-9.A-1 to I.D-1 1.X- 9.A-3600; compounds I.E-1 1.X-9.A-1 to I.E-1 1.X-9.A-3600; compounds I.F-1 1.X-9.A-1 to I.F- 1 1.X-9.A-3600; compounds I.G-1 1.X-9.A-1 to I.G-1 1.X-9.A-3600;

compounds I.A-12.X-9.A-1 to I.A-12.X-9.A-3600; compounds I.B-12.X-9.A-1 to I.B-12.X-9.A- 3600; compounds I.C-12.X-9.A-1 to I.C-12.X-9.A-3600; compounds I.D-12.X-9.A-1 to I.D-12.X-

9. A-3600; compounds I.E-12.X-9.A-1 to I.E-12.X-9.A-3600; compounds I.F-12.X-9.A-1 to I.F- 12.X-9.A-3600; compounds I.G-12.X-9.A-1 to I.G-12.X-9.A-3600).

Table 10a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10,

1. C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-10 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-10.A-1 to I.A-2.X-10.A-3600; compounds I.B-2.X-10.A-1 to I.B-2.X-10.A- 3600; compounds I.C-2.X-10.A-1 to I.C-2.X-10.A-3600; compounds I.D-2.X-10.A-1 to I.D-2.X- 10.A-3600; compounds I.E-2.X-10.A-1 to I.E-2.X-10.A-3600; compounds I.F-2.X-10.A-1 to I.F-

2. X-10.A-3600; compounds I.G-2.X-10.A-1 to I.G-2.X-10.A-3600;

compounds I.A-3.X-10.A-1 to I.A-3.X-10.A-3600; compounds I.B-3.X-10.A-1 to I.B-3.X-10.A- 3600; compounds I.C-3.X-10.A-1 to I.C-3.X-10.A-3600; compounds I.D-3.X-10.A-1 to I.D-3.X-

10. A-3600; compounds I.E-3.X-10.A-1 to I.E-3.X-10.A-3600; compounds I.F-3.X-10.A-1 to I.F- 3.X-10.A-3600; compounds I.G-3.X-10.A-1 to I.G-3.X-10.A-3600;

compounds I.A-4.X-10.A-1 to I.A-4.X-10.A-3600; compounds I.B-4.X-10.A-1 to I.B-4.X-10.A- 3600; compounds I.C-4.X-10.A-1 to I.C-4.X-10.A-3600; compounds I.D-4.X-10.A-1 to I.D-4.X- 10.A-3600; compounds I.E-4.X-10.A-1 to I.E-4.X-10.A-3600; compounds I.F-4.X-10.A-1 to I.F-

4. X-10.A-3600; compounds I.G-4.X-10.A-1 to I.G-4.X-10.A-3600;

compounds I.A-5.X-10.A-1 to I.A-5.X-10.A-3600; compounds I.B-5.X-10.A-1 to I.B-5.X-10.A- 3600; compounds I.C-5.X-10.A-1 to I.C-5.X-10.A-3600; compounds I.D-5.X-10.A-1 to I.D-5.X- 10.A-3600; compounds I.E-5.X-10.A-1 to I.E-5.X-10.A-3600; compounds I.F-5.X-10.A-1 to I.F-

5. X-10.A-3600; compounds I.G-5.X-10.A-1 to I.G-5.X-10.A-3600;

compounds I.A-6.X-10.A-1 to I.A-6.X-10.A-3600; compounds I.B-6.X-10.A-1 to I.B-6.X-10.A- 3600; compounds I.C-6.X-10.A-1 to I.C-6.X-10.A-3600; compounds I.D-6.X-10.A-1 to I.D-6.X- 10.A-3600; compounds I.E-6.X-10.A-1 to I.E-6.X-10.A-3600; compounds I.F-6.X-10.A-1 to I.F-

6. X-10.A-3600; compounds I.G-6.X-10.A-1 to I.G-6.X-10.A-3600;

compounds I.A-7.X-10.A-1 to I.A-7.X-10.A-3600; compounds I.B-7.X-10.A-1 to I.B-7.X-10.A- 3600; compounds I.C-7.X-10.A-1 to I.C-7.X-10.A-3600; compounds I.D-7.X-10.A-1 to I.D-7.X- 10.A-3600; compounds I.E-7.X-10.A-1 to I.E-7.X-10.A-3600; compounds I.F-7.X-10.A-1 to I.F-

7. X-10.A-3600; compounds I.G-7.X-10.A-1 to I.G-7.X-10.A-3600;

compounds I.A-8.X-10.A-1 to I.A-8.X-10.A-3600; compounds I.B-8.X-10.A-1 to I.B-8.X-10.A- 3600; compounds I.C-8.X-10.A-1 to I.C-8.X-10.A-3600; compounds I.D-8.X-10.A-1 to I.D-8.X- 10.A-3600; compounds I.E-8.X-10.A-1 to I.E-8.X-10.A-3600; compounds I.F-8.X-10.A-1 to I.F- 8.X-10.A-3600; compounds I.G-8.X-10.A-1 to I.G-8.X-10.A-3600; compounds I.A-9.X-10.A-1 to I.A-9.X-10.A-3600; compounds I.B-9.X-10.A-1 to I.B-9.X-10.A- 3600; compounds I.C-9.X-10.A-1 to I.C-9.X-10.A-3600; compounds I.D-9.X-10.A-1 to I.D-9.X- 10.A-3600; compounds I.E-9.X-10.A-1 to I.E-9.X-10.A-3600; compounds I.F-9.X-10.A-1 to I.F-

9. X-10.A-3600; compounds I.G-9.X-10.A-1 to I.G-9.X-10.A-3600;

compounds I.A-10.X-10.A-1 to I.A-10.X-10.A-3600; compounds I.B-10.X-10.A-1 to I.B-10.X-

10. A-3600; compounds I.C-10.X-10.A-1 to I.C-10.X-10.A-3600; compounds I.D-10.X-10.A-1 to I.D-10.X-10.A-3600; compounds I.E-10.X-10.A-1 to I.E-10.X-10.A-3600; compounds I.F-10.X- 10.A-1 to I.F-10.X-10.A-3600; compounds I.G-10.X-10.A-1 to I.G-10.X-10.A-3600;

compounds I.A-1 1.X-10.A-1 to I.A-1 1.X-10.A-3600; compounds I.B-1 1.X-10.A-1 to I.B-1 1.X- 10.A-3600; compounds I.C-1 1.X-10.A-1 to I.C-1 1 .X-10.A-3600; compounds I.D-1 1.X-10.A-1 to I.D-1 1.X-10.A-3600; compounds I.E-1 1 .X-10.A-1 to I.E-1 1.X-10.A-3600; compounds I.F-1 1.X- 10.A-1 to I.F-1 1.X-10.A-3600; compounds I.G-1 1.X-10.A-1 to I.G-1 1.X-10.A-3600;

compounds I.A-12.X-10.A-1 to I.A-12.X-10.A-3600; compounds I.B-12.X-10.A-1 to I.B-12.X- 10.A-3600; compounds I.C-12.X-10.A-1 to I.C-12.X-10.A-3600; compounds I.D-12.X-10.A-1 to I.D-12.X-10.A-3600; compounds I.E-12.X-10.A-1 to I.E-12.X-10.A-3600; compounds I.F-12.X-

10. A-1 to I.F-12.X-10.A-3600; compounds I.G-12.X-10.A-1 to I.G-12.X-10.A-3600).

Table 1 1 a

Compounds of the formula I.A-1 , I.B-1 , I.C-1 , I.D-1 , I.E-1 , I.F-1 , I.G-1 ; I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A- 7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A-8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 ,

1. C-1 1 , I.D-1 1 , I.E-1 1. I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-1 1 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-1.X-1 1.A-1 to I.A-1.X-1 1.A-3600; compounds I.B-1 . X-1 1 .A-1 to I.B-1 .X-1 1 .A- 3600; compounds I.C-1 .X-1 1.A-1 to I.C-1. X-1 1.A-3600; compounds I.D-1 .X-1 1.A-1 to I.D-1.X-

1 1. A-3600; compounds I.E-1 .X-1 1.A-1 to I.E-1 .X-1 1.A-3600; compounds I.F-1 .X-1 1.A-1 to I.F- 1 .X-1 1 .A-3600; compounds I.G-1 .X-1 1 .A-1 to I.G-1 .X-1 1 .A-3600;

compounds I.A-2.X-1 1.A-1 to I. A-2.X-1 1 .A-3600; compounds I.B-2.X-1 1 .A-1 to I.B-2. X-1 1 .A- 3600; compounds I.C-2.X-1 1.A-1 to I. C-2.X-1 1. A-3600; compounds I.D-2.X-1 1.A-1 to I.D-2.X- 1 1. A-3600; compounds I.E-2.X-1 1.A-1 to I. E-2.X-1 1. A-3600; compounds I.F-2.X-1 1.A-1 to I.F-

2. X-1 1 . A-3600; compounds I.G-2.X-1 1 .A-1 to I. G-2.X-1 1 .A-3600;

compounds I.A-3.X-1 1.A-1 to I. A-3.X-1 1 .A-3600; compounds I.B-3.X-1 1 .A-1 to I.B-3. X-1 1 .A- 3600; compounds I.C-3.X-1 1.A-1 to I. C-3.X-1 1. A-3600; compounds I.D-3.X-1 1.A-1 to I.D-3.X- 1 1. A-3600; compounds I.E-3.X-1 1.A-1 to I. E-3.X-1 1. A-3600; compounds I.F-3.X-1 1.A-1 to I.F-

3. X-1 1 . A-3600; compounds I.G-3.X-1 1 .A-1 to I. G-3.X-1 1 .A-3600;

compounds I.A-4.X-1 1.A-1 to I. A-4.X-1 1 .A-3600; compounds I.B-4.X-1 1 .A-1 to I.B-4. X-1 1 .A- 3600; compounds I.C-4.X-1 1.A-1 to I. C-4.X-1 1. A-3600; compounds I.D-4.X-1 1.A-1 to I.D-4.X- 1 1. A-3600; compounds I.E-4.X-1 1.A-1 to I. E-4.X-1 1. A-3600; compounds I.F-4.X-1 1.A-1 to I.F-

4. X-1 1 . A-3600; compounds I.G-4.X-1 1 .A-1 to I. G-4.X-1 1 .A-3600; compounds I.A-5.X-1 1.A-1 to I.A-5.X-1 1 .A-3600; compounds I.B-5.X-1 1 .A-1 to I.B-5.X-1 1 .A- 3600; compounds I.C-5.X-1 1.A-1 to I. C-5.X-1 1. A-3600; compounds I.D-5.X-1 1.A-1 to I.D-5.X- 1 1. A-3600; compounds I.E-5.X-1 1.A-1 to I. E-5.X-1 1. A-3600; compounds I.F-5.X-1 1.A-1 to I.F-

5. X-1 1 . A-3600; compounds I.G-5.X-1 1 .A-1 to I. G-5.X-1 1 .A-3600;

compounds I.A-6.X-1 1.A-1 to I. A-6.X-1 1 .A-3600; compounds I.B-6.X-1 1 .A-1 to I.B-6.X-1 1 .A- 3600; compounds I.C-6.X-1 1.A-1 to I. C-6.X-1 1. A-3600; compounds I.D-6.X-1 1.A-1 to I.D-6.X- 1 1. A-3600; compounds I.E-6.X-1 1.A-1 to I. E-6.X-1 1. A-3600; compounds I.F-6.X-1 1.A-1 to I.F-

6. X-1 1 .A-3600; compounds I.G-6.X-1 1 .A-1 to I. G-6.X-1 1 .A-3600;

compounds I.A-7.X-1 1.A-1 to I. A-7.X-1 1 .A-3600; compounds I.B-7.X-1 1 .A-1 to I. B-7.X-1 I .A- 3600; compounds I.C-7.X-1 1.A-1 to I. C-7.X-1 1. A-3600; compounds I.D-7.X-1 1.A-1 to I.D-7.X- 1 1. A-3600; compounds I.E-7.X-1 1.A-1 to I. E-7.X-1 1. A-3600; compounds I.F-7.X-1 1.A-1 to I.F-

7. X-1 1 .A-3600; compounds I.G-7.X-1 1 .A-1 to I. G-7.X-1 1 .A-3600;

compounds I.A-8.X-1 1.A-1 to I. A-8.X-1 1 .A-3600; compounds I.B-8.X-1 1 .A-1 to I.B-8.X-1 1 .A- 3600; compounds I.C-8.X-1 1.A-1 to I. C-8.X-1 1. A-3600; compounds I.D-8.X-1 1.A-1 to I.D-8.X- 1 1. A-3600; compounds I.E-8.X-1 1.A-1 to I. E-8.X-1 1. A-3600; compounds I.F-8.X-1 1.A-1 to I.F-

8. X-1 1 .A-3600; compounds I.G-8.X-1 1 .A-1 to I. G-8.X-1 1 .A-3600;

compounds I.A-9.X-1 1.A-1 to I. A-9.X-1 1 .A-3600; compounds I.B-9.X-1 1 .A-1 to I.B-9.X-1 1 .A- 3600; compounds I.C-9.X-1 1.A-1 to I. C-9.X-1 1. A-3600; compounds I.D-9.X-1 1.A-1 to I.D-9.X- 1 1. A-3600; compounds I.E-9.X-1 1.A-1 to I. E-9.X-1 1. A-3600; compounds I.F-9.X-1 1.A-1 to I.F- 9.X-1 1 .A-3600; compounds I.G-9.X-1 1 .A-1 to I.G-9.X-1 1 .A-3600;

compounds I.A-10.X-1 1.A-1 to I. A-10.X-1 1. A-3600; compounds I.B-10.X-1 1.A-1 to I.B-10.X- 1 1. A-3600; compounds I.C-10.X-1 1.A-1 to I. C-10.X-1 1. A-3600; compounds I.D-10.X-1 1.A-1 to

I. D-10.X-1 1. A-3600; compounds I.E-10.X-1 1.A-1 to I.E-10.X-1 1 . A-3600; compounds I.F-10.X-

I I . A-1 to I. F-10.X-1 1. A-3600; compounds I.G-10.X-1 1.A-1 to I. G-10.X-1 1. A-3600;

compounds I.A-1 1.X-1 1.A-1 to I .A-1 1.X-1 1.A-3600; compounds I.B-1 1.X-1 1.A-1 to I.B-1 1.X- 1 1.A-3600; compounds I.C-1 1.X-1 1.A-1 to I.C-1 1 .X-1 1.A-3600; compounds I.D-1 1.X-1 1.A-1 to I.D-1 1.X-1 1.A-3600; compounds I.E-1 1 .X-1 1.A-1 to I.E-1 1.X-1 1 .A-3600; compounds I.F-1 1.X- 1 1.A-1 to I.F-1 1.X-1 1.A-3600; compounds I.G-1 1.X-1 1.A-1 to I.G-1 1.X-1 1.A-3600;

compounds I.A-12.X-1 1.A-1 to I. A-12.X-1 1. A-3600; compounds I.B-12.X-1 1.A-1 to I.B-12.X- 1 1. A-3600; compounds I.C-12.X-1 1. A-1 to I. C-12.X-1 1. A-3600; compounds I.D-12.X-1 1.A-1 to

I. D-12.X-1 1. A-3600; compounds I.E-12.X-1 1.A-1 to I.E-12.X-1 1 .A-3600; compounds I.F-12.X-

I I . A-1 to I. F-12.X-1 1. A-3600; compounds I.G-12.X-1 1. A-1 to I. G-12.X-1 1. A-3600).

Table 12a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-12 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (compounds I.A-2.X-12.A-1 to I.A-2.X-12.A-3600; compounds I.B-2.X-12.A-1 to I.B-2.X-12.A- 3600; compounds I.C-2.X-12.A-1 to I.C-2.X-12.A-3600; compounds I.D-2.X-12.A-1 to I.D-2.X- 12.A-3600; compounds I.E-2.X-12.A-1 to I.E-2.X-12.A-3600; compounds I.F-2.X-12.A-1 to I.F-

2. X-12.A-3600; compounds I.G-2.X-12.A-1 to I.G-2.X-12.A-3600;

compounds I.A-3.X-12.A-1 to I.A-3.X-12.A-3600; compounds I.B-3.X-12.A-1 to I.B-3.X-12.A- 3600; compounds I.C-3.X-12.A-1 to I.C-3.X-12.A-3600; compounds I.D-3.X-12.A-1 to I.D-3.X- 12.A-3600; compounds I.E-3.X-12.A-1 to I.E-3.X-12.A-3600; compounds I.F-3.X-12.A-1 to I.F-

3. X-12.A-3600; compounds I.G-3.X-12.A-1 to I.G-3.X-12.A-3600;

compounds I.A-4.X-12.A-1 to I.A-4.X-12.A-3600; compounds I.B-4.X-12.A-1 to I.B-4.X-12.A- 3600; compounds I.C-4.X-12.A-1 to I.C-4.X-12.A-3600; compounds I.D-4.X-12.A-1 to I.D-4.X- 12.A-3600; compounds I.E-4.X-12.A-1 to I.E-4.X-12.A-3600; compounds I.F-4.X-12.A-1 to I.F-

4. X-12.A-3600; compounds I.G-4.X-12.A-1 to I.G-4.X-12.A-3600;

compounds I.A-5.X-12.A-1 to I.A-5.X-12.A-3600; compounds I.B-5.X-12.A-1 to I.B-5.X-12.A- 3600; compounds I.C-5.X-12.A-1 to I.C-5.X-12.A-3600; compounds I.D-5.X-12.A-1 to I.D-5.X- 12.A-3600; compounds I.E-5.X-12.A-1 to I.E-5.X-12.A-3600; compounds I.F-5.X-12.A-1 to I.F-

5. X-12.A-3600; compounds I.G-5.X-12.A-1 to I.G-5.X-12.A-3600;

compounds I.A-6.X-12.A-1 to I.A-6.X-12.A-3600; compounds I.B-6.X-12.A-1 to I.B-6.X-12.A- 3600; compounds I.C-6.X-12.A-1 to I.C-6.X-12.A-3600; compounds I.D-6.X-12.A-1 to I.D-6.X- 12.A-3600; compounds I.E-6.X-12.A-1 to I.E-6.X-12.A-3600; compounds I.F-6.X-12.A-1 to I.F- 6.X-12.A-3600; compounds I.G-6.X-12.A-1 to I.G-6.X-12.A-3600;

compounds I.A-7.X-12.A-1 to I.A-7.X-12.A-3600; compounds I.B-7.X-12.A-1 to I.B-7.X-12.A- 3600; compounds I.C-7.X-12.A-1 to I.C-7.X-12.A-3600; compounds I.D-7.X-12.A-1 to I.D-7.X- 12.A-3600; compounds I.E-7.X-12.A-1 to I.E-7.X-12.A-3600; compounds I.F-7.X-12.A-1 to I.F-

7. X-12.A-3600; compounds I.G-7.X-12.A-1 to I.G-7.X-12.A-3600;

compounds I.A-8.X-12.A-1 to I.A-8.X-12.A-3600; compounds I.B-8.X-12.A-1 to I.B-8.X-12.A- 3600; compounds I.C-8.X-12.A-1 to I.C-8.X-12.A-3600; compounds I.D-8.X-12.A-1 to I.D-8.X- 12.A-3600; compounds I.E-8.X-12.A-1 to I.E-8.X-12.A-3600; compounds I.F-8.X-12.A-1 to I.F-

8. X-12.A-3600; compounds I.G-8.X-12.A-1 to I.G-8.X-12.A-3600;

compounds I.A-9.X-12.A-1 to I.A-9.X-12.A-3600; compounds I.B-9.X-12.A-1 to I.B-9.X-12.A- 3600; compounds I.C-9.X-12.A-1 to I.C-9.X-12.A-3600; compounds I.D-9.X-12.A-1 to I.D-9.X- 12.A-3600; compounds I.E-9.X-12.A-1 to I.E-9.X-12.A-3600; compounds I.F-9.X-12.A-1 to I.F-

9. X-12.A-3600; compounds I.G-9.X-12.A-1 to I.G-9.X-12.A-3600;

compounds I.A-10.X-12.A-1 to I.A-10.X-12.A-3600; compounds I.B-10.X-12.A-1 to I.B-10.X- 12.A-3600; compounds I.C-10.X-12.A-1 to I.C-10.X-12.A-3600; compounds I.D-10.X-12.A-1 to I.D-10.X-12.A-3600; compounds I.E-10.X-12.A-1 to I.E-10.X-12.A-3600; compounds I.F-10.X- 12.A-1 to I.F-10.X-12.A-3600; compounds I.G-10.X-12.A-1 to I.G-10.X-12.A-3600;

compounds I.A-1 1.X-12.A-1 to I.A-1 1.X-12.A-3600; compounds I.B-1 1.X-12.A-1 to I.B-1 1.X- 12.A-3600; compounds I.C-1 1.X-12.A-1 to I.C-1 1 .X-12.A-3600; compounds I.D-1 1.X-12.A-1 to I.D-1 1.X-12.A-3600; compounds I.E-1 1 .X-12.A-1 to I.E-1 1.X-12.A-3600; compounds I.F-1 1.X- 12.A-1 to I.F-1 1.X-12.A-3600; compounds I.G-1 1.X-12.A-1 to I.G-1 1.X-12.A-3600;

compounds I.A-12.X-12.A-1 to I.A-12.X-12.A-3600; compounds I.B-12.X-12.A-1 to I.B-12.X- 12.A-3600; compounds I.C-12.X-12.A-1 to I.C-12.X-12.A-3600; compounds I.D-12.X-12.A-1 to I.D-12.X-12.A-3600; compounds I.E-12.X-12.A-1 to I.E-12.X-12.A-3600; compounds I.F-12.X-

12. A-1 to I.F-12.X-12.A-3600; compounds I.G-12.X-12.A-1 to I.G-12.X-12.A-3600).

Table 13a

Compounds of the formula I.A-1 , I.B-1 , I.C-1 , I.D-1 , I.E-1 , I.F-1 , I.G-1 ; I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A- 7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A-8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1. I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-13 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-1.X-13.A-1 to I.A-1.X-13.A-3600; compounds I.B-1 .X-13.A-1 to I.B-1 .X-13.A- 3600; compounds I.C-1 .X-13.A-1 to I.C-1.X-13.A-3600; compounds I.D-1 .X-13.A-1 to I.D-1.X- 13.A-3600; compounds I.E-1 .X-13.A-1 to I.E-1 .X-13.A-3600; compounds I.F-1 .X-13.A-1 to I.F- 1 .X-13.A-3600; compounds I.G-1 .X-13.A-1 to I.G-1 .X-13.A-3600;

compounds I.A-2.X-13.A-1 to I.A-2.X-13.A-3600; compounds I.B-2.X-13.A-1 to I.B-2.X-13.A- 3600; compounds I.C-2.X-13.A-1 to I.C-2.X-13.A-3600; compounds I.D-2.X-13.A-1 to I.D-2.X-

13. A-3600; compounds I.E-2.X-13.A-1 to I.E-2.X-13.A-3600; compounds I.F-2.X-13.A-1 to I.F- 2.X-13.A-3600; compounds I.G-2.X-13.A-1 to I.G-2.X-13.A-3600;

compounds I.A-3.X-13.A-1 to I.A-3.X-13.A-3600; compounds I.B-3.X-13.A-1 to I.B-3.X-13.A- 3600; compounds I.C-3.X-13.A-1 to I.C-3.X-13.A-3600; compounds I.D-3.X-13.A-1 to I.D-3.X- 13.A-3600; compounds I.E-3.X-13.A-1 to I.E-3.X-13.A-3600; compounds I.F-3.X-13.A-1 to I.F-

3. X-13.A-3600; compounds I.G-3.X-13.A-1 to I.G-3.X-13.A-3600;

compounds I.A-4.X-13.A-1 to I.A-4.X-13.A-3600; compounds I.B-4.X-13.A-1 to I.B-4.X-13.A- 3600; compounds I.C-4.X-13.A-1 to I.C-4.X-13.A-3600; compounds I.D-4.X-13.A-1 to I.D-4.X- 13.A-3600; compounds I.E-4.X-13.A-1 to I.E-4.X-13.A-3600; compounds I.F-4.X-13.A-1 to I.F-

4. X-13.A-3600; compounds I.G-4.X-13.A-1 to I.G-4.X-13.A-3600;

compounds I.A-5.X-13.A-1 to I.A-5.X-13.A-3600; compounds I.B-5.X-13.A-1 to I.B-5.X-13.A- 3600; compounds I.C-5.X-13.A-1 to I.C-5.X-13.A-3600; compounds I.D-5.X-13.A-1 to I.D-5.X- 13.A-3600; compounds I.E-5.X-13.A-1 to I.E-5.X-13.A-3600; compounds I.F-5.X-13.A-1 to I.F-

5. X-13.A-3600; compounds I.G-5.X-13.A-1 to I.G-5.X-13.A-3600;

compounds I.A-6.X-13.A-1 to I.A-6.X-13.A-3600; compounds I.B-6.X-13.A-1 to I.B-6.X-13.A- 3600; compounds I.C-6.X-13.A-1 to I.C-6.X-13.A-3600; compounds I.D-6.X-13.A-1 to I.D-6.X- 13.A-3600; compounds I.E-6.X-13.A-1 to I.E-6.X-13.A-3600; compounds I.F-6.X-13.A-1 to I.F-

6. X-13.A-3600; compounds I.G-6.X-13.A-1 to I.G-6.X-13.A-3600;

compounds I.A-7.X-13.A-1 to I.A-7.X-13.A-3600; compounds I.B-7.X-13.A-1 to I.B-7.X-13.A- 3600; compounds I.C-7.X-13.A-1 to I.C-7.X-13.A-3600; compounds I.D-7.X-13.A-1 to I.D-7.X- 13.A-3600; compounds I.E-7.X-13.A-1 to I.E-7.X-13.A-3600; compounds I.F-7.X-13.A-1 to I.F- 7.X-13.A-3600; compounds I.G-7.X-13.A-1 to I.G-7.X-13.A-3600; compounds I.A-8.X-13.A-1 to I.A-8.X-13.A-3600; compounds I.B-8.X-13.A-1 to I.B-8.X-13.A- 3600; compounds I.C-8.X-13.A-1 to I.C-8.X-13.A-3600; compounds I.D-8.X-13.A-1 to I.D-8.X- 13.A-3600; compounds I.E-8.X-13.A-1 to I.E-8.X-13.A-3600; compounds I.F-8.X-13.A-1 to I.F-

8. X-13.A-3600; compounds I.G-8.X-13.A-1 to I.G-8.X-13.A-3600;

compounds I.A-9.X-13.A-1 to I.A-9.X-13.A-3600; compounds I.B-9.X-13.A-1 to I.B-9.X-13.A- 3600; compounds I.C-9.X-13.A-1 to I.C-9.X-13.A-3600; compounds I.D-9.X-13.A-1 to I.D-9.X- 13.A-3600; compounds I.E-9.X-13.A-1 to I.E-9.X-13.A-3600; compounds I.F-9.X-13.A-1 to I.F-

9. X-13.A-3600; compounds I.G-9.X-13.A-1 to I.G-9.X-13.A-3600;

compounds I.A-10.X-13.A-1 to I.A-10.X-13.A-3600; compounds I.B-10.X-13.A-1 to I.B-10.X- 13.A-3600; compounds I.C-10.X-13.A-1 to I.C-10.X-13.A-3600; compounds I.D-10.X-13.A-1 to I.D-10.X-13.A-3600; compounds I.E-10.X-13.A-1 to I.E-10.X-13.A-3600; compounds I.F-10.X- 13.A-1 to I.F-10.X-13.A-3600; compounds I.G-10.X-13.A-1 to I.G-10.X-13.A-3600;

compounds I.A-1 1.X-13.A-1 to I.A-1 1.X-13.A-3600; compounds I.B-1 1 .X-13.A-1 to I.B-1 1.X- 13.A-3600; compounds I.C-1 1.X-13.A-1 to I.C-1 1 .X-13.A-3600; compounds I.D-1 1.X-13.A-1 to I.D-1 1.X-13.A-3600; compounds I.E-1 1 .X-13.A-1 to I.E-1 1.X-13.A-3600; compounds I.F-1 1.X- 13.A-1 to I.F-1 1.X-13.A-3600; compounds I.G-1 1.X-13.A-1 to I.G-1 1.X-13.A-3600;

compounds I.A-12.X-13.A-1 to I.A-12.X-13.A-3600; compounds I.B-12.X-13.A-1 to I.B-12.X-

13. A-3600; compounds I.C-12.X-13.A-1 to I.C-12.X-13.A-3600; compounds I.D-12.X-13.A-1 to I.D-12.X-13.A-3600; compounds I.E-12.X-13.A-1 to I.E-12.X-13.A-3600; compounds I.F-12.X- 13.A-1 to I.F-12.X-13.A-3600; compounds I.G-12.X-13.A-1 to I.G-12.X-13.A-3600).

Table 14a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-14 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (compounds I.A-2.X-14.A-1 to I.A-2.X-14.A-3600; compounds I.B-2.X-14.A-1 to I.B-2.X-14.A- 3600; compounds I.C-2.X-14.A-1 to I.C-2.X-14.A-3600; compounds I.D-2.X-14.A-1 to I.D-2.X-

14. A-3600; compounds I.E-2.X-14.A-1 to I.E-2.X-14.A-3600; compounds I.F-2.X-14.A-1 to I.F-

2. X-14.A-3600; compounds I.G-2.X-14.A-1 to I.G-2.X-14.A-3600;

compounds I.A-3.X-14.A-1 to I.A-3.X-14.A-3600; compounds I.B-3.X-14.A-1 to I.B-3.X-14.A- 3600; compounds I.C-3.X-14.A-1 to I.C-3.X-14.A-3600; compounds I.D-3.X-14.A-1 to I.D-3.X- 14.A-3600; compounds I.E-3.X-14.A-1 to I.E-3.X-14.A-3600; compounds I.F-3.X-14.A-1 to I.F-

3. X-14.A-3600; compounds I.G-3.X-14.A-1 to I.G-3.X-14.A-3600;

compounds I.A-4.X-14.A-1 to I.A-4.X-14.A-3600; compounds I.B-4.X-14.A-1 to I.B-4.X-14.A- 3600; compounds I.C-4.X-14.A-1 to I.C-4.X-14.A-3600; compounds I.D-4.X-14.A-1 to I.D-4.X- 14.A-3600; compounds I.E-4.X-14.A-1 to I.E-4.X-14.A-3600; compounds I.F-4.X-14.A-1 to I.F-

4. X-14.A-3600; compounds I.G-4.X-14.A-1 to I.G-4.X-14.A-3600; compounds I.A-5.X-14.A-1 to I.A-5.X-14.A-3600; compounds I.B-5.X-14.A-1 to I.B-5.X-14.A- 3600; compounds I.C-5.X-14.A-1 to I.C-5.X-14.A-3600; compounds I.D-5.X-14.A-1 to I.D-5.X- 14.A-3600; compounds I.E-5.X-14.A-1 to I.E-5.X-14.A-3600; compounds I.F-5.X-14.A-1 to I.F-

5. X-14.A-3600; compounds I.G-5.X-14.A-1 to I.G-5.X-14.A-3600;

compounds I.A-6.X-14.A-1 to I.A-6.X-14.A-3600; compounds I.B-6.X-14.A-1 to I.B-6.X-14.A- 3600; compounds I.C-6.X-14.A-1 to I.C-6.X-14.A-3600; compounds I.D-6.X-14.A-1 to I.D-6.X- 14.A-3600; compounds I.E-6.X-14.A-1 to I.E-6.X-14.A-3600; compounds I.F-6.X-14.A-1 to I.F-

6. X-14.A-3600; compounds I.G-6.X-14.A-1 to I.G-6.X-14.A-3600;

compounds I.A-7.X-14.A-1 to I.A-7.X-14.A-3600; compounds I.B-7.X-14.A-1 to I.B-7.X-14.A- 3600; compounds I.C-7.X-14.A-1 to I.C-7.X-14.A-3600; compounds I.D-7.X-14.A-1 to I.D-7.X- 14.A-3600; compounds I.E-7.X-14.A-1 to I.E-7.X-14.A-3600; compounds I.F-7.X-14.A-1 to I.F-

7. X-14.A-3600; compounds I.G-7.X-14.A-1 to I.G-7.X-14.A-3600;

compounds I.A-8.X-14.A-1 to I.A-8.X-14.A-3600; compounds I.B-8.X-14.A-1 to I.B-8.X-14.A- 3600; compounds I.C-8.X-14.A-1 to I.C-8.X-14.A-3600; compounds I.D-8.X-14.A-1 to I.D-8.X- 14.A-3600; compounds I.E-8.X-14.A-1 to I.E-8.X-14.A-3600; compounds I.F-8.X-14.A-1 to I.F-

8. X-14.A-3600; compounds I.G-8.X-14.A-1 to I.G-8.X-14.A-3600;

compounds I.A-9.X-14.A-1 to I.A-9.X-14.A-3600; compounds I.B-9.X-14.A-1 to I.B-9.X-14.A- 3600; compounds I.C-9.X-14.A-1 to I.C-9.X-14.A-3600; compounds I.D-9.X-14.A-1 to I.D-9.X- 14.A-3600; compounds I.E-9.X-14.A-1 to I.E-9.X-14.A-3600; compounds I.F-9.X-14.A-1 to I.F- 9.X-14.A-3600; compounds I.G-9.X-14.A-1 to I.G-9.X-14.A-3600;

compounds I.A-10.X-14.A-1 to I.A-10.X-14.A-3600; compounds I.B-10.X-14.A-1 to I.B-10.X- 14.A-3600; compounds I.C-10.X-14.A-1 to I.C-10.X-14.A-3600; compounds I.D-10.X-14.A-1 to I.D-10.X-14.A-3600; compounds I.E-10.X-14.A-1 to I.E-10.X-14.A-3600; compounds I.F-10.X- 14.A-1 to I.F-10.X-14.A-3600; compounds I.G-10.X-14.A-1 to I.G-10.X-14.A-3600;

compounds I.A-1 1.X-14.A-1 to I.A-1 1.X-14.A-3600; compounds I.B-1 1.X-14.A-1 to I.B-1 1.X- 14.A-3600; compounds I.C-1 1.X-14.A-1 to I.C-1 1 .X-14.A-3600; compounds I.D-1 1.X-14.A-1 to I.D-1 1.X-14.A-3600; compounds I.E-1 1 .X-14.A-1 to I.E-1 1.X-14.A-3600; compounds I.F-1 1.X- 14.A-1 to I.F-1 1.X-14.A-3600; compounds I.G-1 1.X-14.A-1 to I.G-1 1.X-14.A-3600;

compounds I.A-12.X-14.A-1 to I.A-12.X-14.A-3600; compounds I.B-12.X-14.A-1 to I.B-12.X- 14.A-3600; compounds I.C-12.X-14.A-1 to I.C-12.X-14.A-3600; compounds I.D-12.X-14.A-1 to I.D-12.X-14.A-3600; compounds I.E-12.X-14.A-1 to I.E-12.X-14.A-3600; compounds I.F-12.X- 14.A-1 to I.F-12.X-14.A-3600; compounds I.G-12.X-14.A-1 to I.G-12.X-14.A-3600).

Table 15a

Compounds of the formula I.A-1 , I.B-1 , I.C-1 , I.D-1 , I.E-1 , I.F-1 , I.G-1 ; I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A- 7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A-8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-15 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (compounds I.A-1.X-15.A-1 to I.A-1.X-15.A-3600; compounds I.B-1 .X-15.A-1 to I.B-1 .X-15.A- 3600; compounds I.C-1 .X-15.A-1 to I.C-1.X-15.A-3600; compounds I.D-1 .X-15.A-1 to I.D-1.X- 15.A-3600; compounds I.E-1 .X-15.A-1 to I.E-1 .X-15.A-3600; compounds I.F-1 .X-15.A-1 to I.F-

1 . X-15.A-3600; compounds I.G-1 .X-15.A-1 to I.G-1 .X-15.A-3600;

compounds I.A-2.X-15.A-1 to I.A-2.X-15.A-3600; compounds I.B-2.X-15.A-1 to I.B-2.X-15.A- 3600; compounds I.C-2.X-15.A-1 to I.C-2.X-15.A-3600; compounds I.D-2.X-15.A-1 to I.D-2.X- 15.A-3600; compounds I.E-2.X-15.A-1 to I.E-2.X-15.A-3600; compounds I.F-2.X-15.A-1 to I.F-

2. X-15.A-3600; compounds I.G-2.X-15.A-1 to I.G-2.X-15.A-3600;

compounds I.A-3.X-15.A-1 to I.A-3.X-15.A-3600; compounds I.B-3.X-15.A-1 to I.B-3.X-15.A- 3600; compounds I.C-3.X-15.A-1 to I.C-3.X-15.A-3600; compounds I.D-3.X-15.A-1 to I.D-3.X- 15.A-3600; compounds I.E-3.X-15.A-1 to I.E-3.X-15.A-3600; compounds I.F-3.X-15.A-1 to I.F-

3. X-15.A-3600; compounds I.G-3.X-15.A-1 to I.G-3.X-15.A-3600;

compounds I.A-4.X-15.A-1 to I.A-4.X-15.A-3600; compounds I.B-4.X-15.A-1 to I.B-4.X-15.A- 3600; compounds I.C-4.X-15.A-1 to I.C-4.X-15.A-3600; compounds I.D-4.X-15.A-1 to I.D-4.X- 15.A-3600; compounds I.E-4.X-15.A-1 to I.E-4.X-15.A-3600; compounds I.F-4.X-15.A-1 to I.F-

4. X-15.A-3600; compounds I.G-4.X-15.A-1 to I.G-4.X-15.A-3600;

compounds I.A-5.X-15.A-1 to I.A-5.X-15.A-3600; compounds I.B-5.X-15.A-1 to I.B-5.X-15.A- 3600; compounds I.C-5.X-15.A-1 to I.C-5.X-15.A-3600; compounds I.D-5.X-15.A-1 to I.D-5.X- 15.A-3600; compounds I.E-5.X-15.A-1 to I.E-5.X-15.A-3600; compounds I.F-5.X-15.A-1 to I.F- 5.X-15.A-3600; compounds I.G-5.X-15.A-1 to I.G-5.X-15.A-3600;

compounds I.A-6.X-15.A-1 to I.A-6.X-15.A-3600; compounds I.B-6.X-15.A-1 to I.B-6.X-15.A- 3600; compounds I.C-6.X-15.A-1 to I.C-6.X-15.A-3600; compounds I.D-6.X-15.A-1 to I.D-6.X- 15.A-3600; compounds I.E-6.X-15.A-1 to I.E-6.X-15.A-3600; compounds I.F-6.X-15.A-1 to I.F-

6. X-15.A-3600; compounds I.G-6.X-15.A-1 to I.G-6.X-15.A-3600;

compounds I.A-7.X-15.A-1 to I.A-7.X-15.A-3600; compounds I.B-7.X-15.A-1 to I.B-7.X-15.A- 3600; compounds I.C-7.X-15.A-1 to I.C-7.X-15.A-3600; compounds I.D-7.X-15.A-1 to I.D-7.X- 15.A-3600; compounds I.E-7.X-15.A-1 to I.E-7.X-15.A-3600; compounds I.F-7.X-15.A-1 to I.F-

7. X-15.A-3600; compounds I.G-7.X-15.A-1 to I.G-7.X-15.A-3600;

compounds I.A-8.X-15.A-1 to I.A-8.X-15.A-3600; compounds I.B-8.X-15.A-1 to I.B-8.X-15.A- 3600; compounds I.C-8.X-15.A-1 to I.C-8.X-15.A-3600; compounds I.D-8.X-15.A-1 to I.D-8.X- 15.A-3600; compounds I.E-8.X-15.A-1 to I.E-8.X-15.A-3600; compounds I.F-8.X-15.A-1 to I.F-

8. X-15.A-3600; compounds I.G-8.X-15.A-1 to I.G-8.X-15.A-3600;

compounds I.A-9.X-15.A-1 to I.A-9.X-15.A-3600; compounds I.B-9.X-15.A-1 to I.B-9.X-15.A- 3600; compounds I.C-9.X-15.A-1 to I.C-9.X-15.A-3600; compounds I.D-9.X-15.A-1 to I.D-9.X- 15.A-3600; compounds I.E-9.X-15.A-1 to I.E-9.X-15.A-3600; compounds I.F-9.X-15.A-1 to I.F-

9. X-15.A-3600; compounds I.G-9.X-15.A-1 to I.G-9.X-15.A-3600;

compounds I.A-10.X-15.A-1 to I.A-10.X-15.A-3600; compounds I.B-10.X-15.A-1 to I.B-10.X- 15.A-3600; compounds I.C-10.X-15.A-1 to I.C-10.X-15.A-3600; compounds I.D-10.X-15.A-1 to I.D-10.X-15.A-3600; compounds I.E-10.X-15.A-1 to I.E-10.X-15.A-3600; compounds I.F-10.X- 15.A-1 to I.F-10.X-15.A-3600; compounds I.G-10.X-15.A-1 to I.G-10.X-15.A-3600;

compounds I.A-1 1.X-15.A-1 to I.A-1 1 .X-15.A-3600; compounds I.B-1 1.X-15.A-1 to I.B-1 1.X- 15.A-3600; compounds I.C-1 1.X-15.A-1 to I.C-1 1 .X-15.A-3600; compounds I.D-1 1.X-15.A-1 to I.D-1 1.X-15.A-3600; compounds I.E-1 1 .X-15.A-1 to I.E-1 1.X-15.A-3600; compounds I.F-1 1.X- 15.A-1 to I.F-1 1.X-15.A-3600; compounds I.G-1 1.X-15.A-1 to I.G-1 1.X-15.A-3600;

compounds I.A-12.X-15.A-1 to I.A-12.X-15.A-3600; compounds I.B-12.X-15.A-1 to I.B-12.X- 15.A-3600; compounds I.C-12.X-15.A-1 to I.C-12.X-15.A-3600; compounds I.D-12.X-15.A-1 to I.D-12.X-15.A-3600; compounds I.E-12.X-15.A-1 to I.E-12.X-15.A-3600; compounds I.F-12.X-

15. A-1 to I.F-12.X-15.A-3600; compounds I.G-12.X-15.A-1 to I.G-12.X-15.A-3600).

Table 16a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-16 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(

compounds I.A-2.X-16.A-1 to I.A-2.X-16.A-3600; compounds I.B-2.X-16.A-1 to I.B-2.X-16.A- 3600; compounds I.C-2.X-16.A-1 to I.C-2.X-16.A-3600; compounds I.D-2.X-16.A-1 to I.D-2.X- 16.A-3600; compounds I.E-2.X-16.A-1 to I.E-2.X-16.A-3600; compounds I.F-2.X-16.A-1 to I.F-

2. X-16.A-3600; compounds I.G-2.X-16.A-1 to I.G-2.X-16.A-3600;

compounds I.A-3.X-16.A-1 to I.A-3.X-16.A-3600; compounds I.B-3.X-16.A-1 to I.B-3.X-16.A- 3600; compounds I.C-3.X-16.A-1 to I.C-3.X-16.A-3600; compounds I.D-3.X-16.A-1 to I.D-3.X-

16. A-3600; compounds I.E-3.X-16.A-1 to I.E-3.X-16.A-3600; compounds I.F-3.X-16.A-1 to I.F- 3.X-16.A-3600; compounds I.G-3.X-16.A-1 to I.G-3.X-16.A-3600;

compounds I.A-4.X-16.A-1 to I.A-4.X-16.A-3600; compounds I.B-4.X-16.A-1 to I.B-4.X-16.A- 3600; compounds I.C-4.X-16.A-1 to I.C-4.X-16.A-3600; compounds I.D-4.X-16.A-1 to I.D-4.X- 16.A-3600; compounds I.E-4.X-16.A-1 to I.E-4.X-16.A-3600; compounds I.F-4.X-16.A-1 to I.F-

4. X-16.A-3600; compounds I.G-4.X-16.A-1 to I.G-4.X-16.A-3600;

compounds I.A-5.X-16.A-1 to I.A-5.X-16.A-3600; compounds I.B-5.X-16.A-1 to I.B-5.X-16.A- 3600; compounds I.C-5.X-16.A-1 to I.C-5.X-16.A-3600; compounds I.D-5.X-16.A-1 to I.D-5.X- 16.A-3600; compounds I.E-5.X-16.A-1 to I.E-5.X-16.A-3600; compounds I.F-5.X-16.A-1 to I.F-

5. X-16.A-3600; compounds I.G-5.X-16.A-1 to I.G-5.X-16.A-3600;

compounds I.A-6.X-16.A-1 to I.A-6.X-16.A-3600; compounds I.B-6.X-16.A-1 to I.B-6.X-16.A- 3600; compounds I.C-6.X-16.A-1 to I.C-6.X-16.A-3600; compounds I.D-6.X-16.A-1 to I.D-6.X- 16.A-3600; compounds I.E-6.X-16.A-1 to I.E-6.X-16.A-3600; compounds I.F-6.X-16.A-1 to I.F-

6. X-16.A-3600; compounds I.G-6.X-16.A-1 to I.G-6.X-16.A-3600;

compounds I.A-7.X-16.A-1 to I.A-7.X-16.A-3600; compounds I.B-7.X-16.A-1 to I.B-7.X-16.A- 3600; compounds I.C-7.X-16.A-1 to I.C-7.X-16.A-3600; compounds I.D-7.X-16.A-1 to I.D-7.X- 16.A-3600; compounds I.E-7.X-16.A-1 to I.E-7.X-16.A-3600; compounds I.F-7.X-16.A-1 to I.F- 7. X-16.A-3600; compounds I.G-7.X-16.A-1 to I.G-7.X-16.A-3600;

compounds I.A-8.X-16.A-1 to I.A-8.X-16.A-3600; compounds I.B-8.X-16.A-1 to I.B-8.X-16.A- 3600; compounds I.C-8.X-16.A-1 to I.C-8.X-16.A-3600; compounds I.D-8.X-16.A-1 to I.D-8.X- 16.A-3600; compounds I.E-8.X-16.A-1 to I.E-8.X-16.A-3600; compounds I.F-8.X-16.A-1 to I.F- 8.X-16.A-3600; compounds I.G-8.X-16.A-1 to I.G-8.X-16.A-3600;

compounds I.A-9.X-16.A-1 to I.A-9.X-16.A-3600; compounds I.B-9.X-16.A-1 to I.B-9.X-16.A- 3600; compounds I.C-9.X-16.A-1 to I.C-9.X-16.A-3600; compounds I.D-9.X-16.A-1 to I.D-9.X- 16.A-3600; compounds I.E-9.X-16.A-1 to I.E-9.X-16.A-3600; compounds I.F-9.X-16.A-1 to I.F- 9.X-16.A-3600; compounds I.G-9.X-16.A-1 to I.G-9.X-16.A-3600;

compounds I.A-10.X-16.A-1 to I.A-10.X-16.A-3600; compounds I.B-10.X-16.A-1 to I.B-10.X- 16.A-3600; compounds I.C-10.X-16.A-1 to I.C-10.X-16.A-3600; compounds I.D-10.X-16.A-1 to I.D-10.X-16.A-3600; compounds I.E-10.X-16.A-1 to I.E-10.X-16.A-3600; compounds I.F-10.X- 16.A-1 to I.F-10.X-16.A-3600; compounds I.G-10.X-16.A-1 to I.G-10.X-16.A-3600;

compounds I.A-1 1.X-16.A-1 to I.A-1 1.X-16.A-3600; compounds I.B-1 1.X-16.A-1 to I.B-1 1.X- 16.A-3600; compounds I.C-1 1.X-16.A-1 to I.C-1 1 .X-16.A-3600; compounds I.D-1 1.X-16.A-1 to I.D-1 1.X-16.A-3600; compounds I.E-1 1 .X-16.A-1 to I.E-1 1.X-16.A-3600; compounds I.F-1 1.X- 16.A-1 to I.F-1 1.X-16.A-3600; compounds I.G-1 1.X-16.A-1 to I.G-1 1.X-16.A-3600;

compounds I.A-12.X-16.A-1 to I.A-12.X-16.A-3600; compounds I.B-12.X-16.A-1 to I.B-12.X- 16.A-3600; compounds I.C-12.X-16.A-1 to I.C-12.X-16.A-3600; compounds I.D-12.X-16.A-1 to I.D-12.X-16.A-3600; compounds I.E-12.X-16.A-1 to I.E-12.X-16.A-3600; compounds I.F-12.X-

16. A-1 to I.F-12.X-16.A-3600; compounds I.G-12.X-16.A-1 to I.G-12.X-16.A-3600).

Table 17a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A-

8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-17 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-17.A-1 to I.A-2.X-17.A-3600; compounds I.B-2.X-17.A-1 to I.B-2.X-17.A- 3600; compounds I.C-2.X-17.A-1 to I.C-2.X-17.A-3600; compounds I.D-2.X-17.A-1 to I.D-2.X-

17. A-3600; compounds I.E-2.X-17.A-1 to I.E-2.X-17.A-3600; compounds I.F-2.X-17.A-1 to I.F-

2. X-17.A-3600; compounds I.G-2.X-17.A-1 to I.G-2.X-17.A-3600;

compounds I.A-3.X-17.A-1 to I.A-3.X-17.A-3600; compounds I.B-3.X-17.A-1 to I.B-3.X-17.A- 3600; compounds I.C-3.X-17.A-1 to I.C-3.X-17.A-3600; compounds I.D-3.X-17.A-1 to I.D-3.X- 17.A-3600; compounds I.E-3.X-17.A-1 to I.E-3.X-17.A-3600; compounds I.F-3.X-17.A-1 to I.F-

3. X-17.A-3600; compounds I.G-3.X-17.A-1 to I.G-3.X-17.A-3600;

compounds I.A-4.X-17.A-1 to I.A-4.X-17.A-3600; compounds I.B-4.X-17.A-1 to I.B-4.X-17.A- 3600; compounds I.C-4.X-17.A-1 to I.C-4.X-17.A-3600; compounds I.D-4.X-17.A-1 to I.D-4.X- 17.A-3600; compounds I.E-4.X-17.A-1 to I.E-4.X-17.A-3600; compounds I.F-4.X-17.A-1 to I.F-

4. X-17.A-3600; compounds I.G-4.X-17.A-1 to I.G-4.X-17.A-3600;

compounds I.A-5.X-17.A-1 to I.A-5.X-17.A-3600; compounds I.B-5.X-17.A-1 to I.B-5.X-17.A- 3600; compounds I.C-5.X-17.A-1 to I.C-5.X-17.A-3600; compounds I.D-5.X-17.A-1 to I.D-5.X- 17.A-3600; compounds I.E-5.X-17.A-1 to I.E-5.X-17.A-3600; compounds I.F-5.X-17.A-1 to I.F-

5. X-17.A-3600; compounds I.G-5.X-17.A-1 to I.G-5.X-17.A-3600;

compounds I.A-6.X-17.A-1 to I.A-6.X-17.A-3600; compounds I.B-6.X-17.A-1 to I.B-6.X-17.A- 3600; compounds I.C-6.X-17.A-1 to I.C-6.X-17.A-3600; compounds I.D-6.X-17.A-1 to I.D-6.X- 17.A-3600; compounds I.E-6.X-17.A-1 to I.E-6.X-17.A-3600; compounds I.F-6.X-17.A-1 to I.F- 6.X-17.A-3600; compounds I.G-6.X-17.A-1 to I.G-6.X-17.A-3600;

compounds I.A-7.X-17.A-1 to I.A-7.X-17.A-3600; compounds I.B-7.X-17.A-1 to I.B-7.X-17.A- 3600; compounds I.C-7.X-17.A-1 to I.C-7.X-17.A-3600; compounds I.D-7.X-17.A-1 to I.D-7.X- 17.A-3600; compounds I.E-7.X-17.A-1 to I.E-7.X-17.A-3600; compounds I.F-7.X-17.A-1 to I.F-

7. X-17.A-3600; compounds I.G-7.X-17.A-1 to I.G-7.X-17.A-3600;

compounds I.A-8.X-17.A-1 to I.A-8.X-17.A-3600; compounds I.B-8.X-17.A-1 to I.B-8.X-17.A- 3600; compounds I.C-8.X-17.A-1 to I.C-8.X-17.A-3600; compounds I.D-8.X-17.A-1 to I.D-8.X- 17.A-3600; compounds I.E-8.X-17.A-1 to I.E-8.X-17.A-3600; compounds I.F-8.X-17.A-1 to I.F-

8. X-17.A-3600; compounds I.G-8.X-17.A-1 to I.G-8.X-17.A-3600;

compounds I.A-9.X-17.A-1 to I.A-9.X-17.A-3600; compounds I.B-9.X-17.A-1 to I.B-9.X-17.A- 3600; compounds I.C-9.X-17.A-1 to I.C-9.X-17.A-3600; compounds I.D-9.X-17.A-1 to I.D-9.X- 17.A-3600; compounds I.E-9.X-17.A-1 to I.E-9.X-17.A-3600; compounds I.F-9.X-17.A-1 to I.F-

9. X-17.A-3600; compounds I.G-9.X-17.A-1 to I.G-9.X-17.A-3600;

compounds I.A-10.X-17.A-1 to I.A-10.X-17.A-3600; compounds I.B-10.X-17.A-1 to I.B-10.X- 17.A-3600; compounds I.C-10.X-17.A-1 to I.C-10.X-17.A-3600; compounds I.D-10.X-17.A-1 to I.D-10.X-17.A-3600; compounds I.E-10.X-17.A-1 to I.E-10.X-17.A-3600; compounds I.F-10.X- 17.A-1 to I.F-10.X-17.A-3600; compounds I.G-10.X-17.A-1 to I.G-10.X-17.A-3600;

compounds I.A-1 1.X-17.A-1 to I.A-1 1.X-17.A-3600; compounds I.B-1 1.X-17.A-1 to I.B-1 1.X- 17.A-3600; compounds I.C-1 1.X-17.A-1 to I.C-1 1 .X-17.A-3600; compounds I.D-1 1.X-17.A-1 to I.D-1 1.X-17.A-3600; compounds I.E-1 1 .X-17.A-1 to I.E-1 1.X-17.A-3600; compounds I.F-1 1.X- 17.A-1 to I.F-1 1.X-17.A-3600; compounds I.G-1 1.X-17.A-1 to I.G-1 1.X-17.A-3600;

compounds I.A-12.X-17.A-1 to I.A-12.X-17.A-3600; compounds I.B-12.X-17.A-1 to I.B-12.X- 17.A-3600; compounds I.C-12.X-17.A-1 to I.C-12.X-17.A-3600; compounds I.D-12.X-17.A-1 to I.D-12.X-17.A-3600; compounds I.E-12.X-17.A-1 to I.E-12.X-17.A-3600; compounds I.F-12.X- 17.A-1 to I.F-12.X-17.A-3600; compounds I.G-12.X-17.A-1 to I.G-12.X-17.A-3600).

Table 18a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12; in which X _n is as defined in line X-18 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-18.A-1 to I.A-2.X-18.A-3600; compounds I.B-2.X-18.A-1 to I.B-2.X-18.A- 3600; compounds I.C-2.X-18.A-1 to I.C-2.X-18.A-3600; compounds I.D-2.X-18.A-1 to I.D-2.X- 18.A-3600; compounds I.E-2.X-18.A-1 to I.E-2.X-18.A-3600; compounds I.F-2.X-18.A-1 to I.F- 2.X-18.A-3600; compounds I.G-2.X-18.A-1 to I.G-2.X-18.A-3600;

compounds I.A-3.X-18.A-1 to I.A-3.X-18.A-3600; compounds I.B-3.X-18.A-1 to I.B-3.X-18.A- 3600; compounds I.C-3.X-18.A-1 to I.C-3.X-18.A-3600; compounds I.D-3.X-18.A-1 to I.D-3.X- 18.A-3600; compounds I.E-3.X-18.A-1 to I.E-3.X-18.A-3600; compounds I.F-3.X-18.A-1 to I.F- 3.X-18.A-3600; compounds I.G-3.X-18.A-1 to I.G-3.X-18.A-3600;

compounds I.A-4.X-18.A-1 to I.A-4.X-18.A-3600; compounds I.B-4.X-18.A-1 to I.B-4.X-18.A- 3600; compounds I.C-4.X-18.A-1 to I.C-4.X-18.A-3600; compounds I.D-4.X-18.A-1 to I.D-4.X- 18.A-3600; compounds I.E-4.X-18.A-1 to I.E-4.X-18.A-3600; compounds I.F-4.X-18.A-1 to I.F-

4. X-18.A-3600; compounds I.G-4.X-18.A-1 to I.G-4.X-18.A-3600;

compounds I.A-5.X-18.A-1 to I.A-5.X-18.A-3600; compounds I.B-5.X-18.A-1 to I.B-5.X-18.A- 3600; compounds I.C-5.X-18.A-1 to I.C-5.X-18.A-3600; compounds I.D-5.X-18.A-1 to I.D-5.X- 18.A-3600; compounds I.E-5.X-18.A-1 to I.E-5.X-18.A-3600; compounds I.F-5.X-18.A-1 to I.F-

5. X-18.A-3600; compounds I.G-5.X-18.A-1 to I.G-5.X-18.A-3600;

compounds I.A-6.X-18.A-1 to I.A-6.X-18.A-3600; compounds I.B-6.X-18.A-1 to I.B-6.X-18.A- 3600; compounds I.C-6.X-18.A-1 to I.C-6.X-18.A-3600; compounds I.D-6.X-18.A-1 to I.D-6.X- 18.A-3600; compounds I.E-6.X-18.A-1 to I.E-6.X-18.A-3600; compounds I.F-6.X-18.A-1 to I.F-

6. X-18.A-3600; compounds I.G-6.X-18.A-1 to I.G-6.X-18.A-3600;

compounds I.A-7.X-18.A-1 to I.A-7.X-18.A-3600; compounds I.B-7.X-18.A-1 to I.B-7.X-18.A- 3600; compounds I.C-7.X-18.A-1 to I.C-7.X-18.A-3600; compounds I.D-7.X-18.A-1 to I.D-7.X- 18.A-3600; compounds I.E-7.X-18.A-1 to I.E-7.X-18.A-3600; compounds I.F-7.X-18.A-1 to I.F-

7. X-18.A-3600; compounds I.G-7.X-18.A-1 to I.G-7.X-18.A-3600;

compounds I.A-8.X-18.A-1 to I.A-8.X-18.A-3600; compounds I.B-8.X-18.A-1 to I.B-8.X-18.A- 3600; compounds I.C-8.X-18.A-1 to I.C-8.X-18.A-3600; compounds I.D-8.X-18.A-1 to I.D-8.X- 18.A-3600; compounds I.E-8.X-18.A-1 to I.E-8.X-18.A-3600; compounds I.F-8.X-18.A-1 to I.F- 8.X-18.A-3600; compounds I.G-8.X-18.A-1 to I.G-8.X-18.A-3600;

compounds I.A-9.X-18.A-1 to I.A-9.X-18.A-3600; compounds I.B-9.X-18.A-1 to I.B-9.X-18.A- 3600; compounds I.C-9.X-18.A-1 to I.C-9.X-18.A-3600; compounds I.D-9.X-18.A-1 to I.D-9.X- 18.A-3600; compounds I.E-9.X-18.A-1 to I.E-9.X-18.A-3600; compounds I.F-9.X-18.A-1 to I.F- 9.X-18.A-3600; compounds I.G-9.X-18.A-1 to I.G-9.X-18.A-3600;

compounds I.A-10.X-18.A-1 to I.A-10.X-18.A-3600; compounds I.B-10.X-18.A-1 to I.B-10.X- 18.A-3600; compounds I.C-10.X-18.A-1 to I.C-10.X-18.A-3600; compounds I.D-10.X-18.A-1 to I.D-10.X-18.A-3600; compounds I.E-10.X-18.A-1 to I.E-10.X-18.A-3600; compounds I.F-10.X- 18.A-1 to I.F-10.X-18.A-3600; compounds I.G-10.X-18.A-1 to I.G-10.X-18.A-3600;

compounds I.A-1 1.X-18.A-1 to I.A-1 1.X-18.A-3600; compounds I.B-1 1.X-18.A-1 to I.B-1 1.X- 18.A-3600; compounds I.C-1 1.X-18.A-1 to I.C-1 1 .X-18.A-3600; compounds I.D-1 1.X-18.A-1 to I.D-1 1.X-18.A-3600; compounds I.E-1 1 .X-18.A-1 to I.E-1 1.X-18.A-3600; compounds I.F-1 1.X- 18.A-1 to I.F-1 1.X-18.A-3600; compounds I.G-1 1.X-18.A-1 to I.G-1 1.X-18.A-3600; compounds I.A-12.X-18.A-1 to I.A-12.X-18.A-3600; compounds I.B-12.X-18.A-1 to I.B-12.X-

18. A-3600; compounds I.C-12.X-18.A-1 to I.C-12.X-18.A-3600; compounds I.D-12.X-18.A-1 to I.D-12.X-18.A-3600; compounds I.E-12.X-18.A-1 to I.E-12.X-18.A-3600; compounds I.F-12.X- 18.A-1 to I.F-12.X-18.A-3600; compounds I.G-12.X-18.A-1 to I.G-12.X-18.A-3600).

Table 19a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-19 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (compounds I.A-2.X-19.A-1 to I.A-2.X-19.A-3600; compounds I.B-2.X-19.A-1 to I.B-2.X-19.A- 3600; compounds I.C-2.X-19.A-1 to I.C-2.X-19.A-3600; compounds I.D-2.X-19.A-1 to I.D-2.X-

19. A-3600; compounds I.E-2.X-19.A-1 to I.E-2.X-19.A-3600; compounds I.F-2.X-19.A-1 to I.F-

2. X-19.A-3600; compounds I.G-2.X-19.A-1 to I.G-2.X-19.A-3600;

compounds I.A-3.X-19.A-1 to I.A-3.X-19.A-3600; compounds I.B-3.X-19.A-1 to I.B-3.X-19.A- 3600; compounds I.C-3.X-19.A-1 to I.C-3.X-19.A-3600; compounds I.D-3.X-19.A-1 to I.D-3.X- 19.A-3600; compounds I.E-3.X-19.A-1 to I.E-3.X-19.A-3600; compounds I.F-3.X-19.A-1 to I.F-

3. X-19.A-3600; compounds I.G-3.X-19.A-1 to I.G-3.X-19.A-3600;

compounds I.A-4.X-19.A-1 to I.A-4.X-19.A-3600; compounds I.B-4.X-19.A-1 to I.B-4.X-19.A- 3600; compounds I.C-4.X-19.A-1 to I.C-4.X-19.A-3600; compounds I.D-4.X-19.A-1 to I.D-4.X- 19.A-3600; compounds I.E-4.X-19.A-1 to I.E-4.X-19.A-3600; compounds I.F-4.X-19.A-1 to I.F-

4. X-19.A-3600; compounds I.G-4.X-19.A-1 to I.G-4.X-19.A-3600;

compounds I.A-5.X-19.A-1 to I.A-5.X-19.A-3600; compounds I.B-5.X-19.A-1 to I.B-5.X-19.A- 3600; compounds I.C-5.X-19.A-1 to I.C-5.X-19.A-3600; compounds I.D-5.X-19.A-1 to I.D-5.X- 19.A-3600; compounds I.E-5.X-19.A-1 to I.E-5.X-19.A-3600; compounds I.F-5.X-19.A-1 to I.F- 5.X-19.A-3600; compounds I.G-5.X-19.A-1 to I.G-5.X-19.A-3600;

compounds I.A-6.X-19.A-1 to I.A-6.X-19.A-3600; compounds I.B-6.X-19.A-1 to I.B-6.X-19.A- 3600; compounds I.C-6.X-19.A-1 to I.C-6.X-19.A-3600; compounds I.D-6.X-19.A-1 to I.D-6.X- 19.A-3600; compounds I.E-6.X-19.A-1 to I.E-6.X-19.A-3600; compounds I.F-6.X-19.A-1 to I.F-

6. X-19.A-3600; compounds I.G-6.X-19.A-1 to I.G-6.X-19.A-3600;

compounds I.A-7.X-19.A-1 to I.A-7.X-19.A-3600; compounds I.B-7.X-19.A-1 to I.B-7.X-19.A- 3600; compounds I.C-7.X-19.A-1 to I.C-7.X-19.A-3600; compounds I.D-7.X-19.A-1 to I.D-7.X- 19.A-3600; compounds I.E-7.X-19.A-1 to I.E-7.X-19.A-3600; compounds I.F-7.X-19.A-1 to I.F-

7. X-19.A-3600; compounds I.G-7.X-19.A-1 to I.G-7.X-19.A-3600;

compounds I.A-8.X-19.A-1 to I.A-8.X-19.A-3600; compounds I.B-8.X-19.A-1 to I.B-8.X-19.A- 3600; compounds I.C-8.X-19.A-1 to I.C-8.X-19.A-3600; compounds I.D-8.X-19.A-1 to I.D-8.X- 19.A-3600; compounds I.E-8.X-19.A-1 to I.E-8.X-19.A-3600; compounds I.F-8.X-19.A-1 to I.F-

8. X-19.A-3600; compounds I.G-8.X-19.A-1 to I.G-8.X-19.A-3600;

compounds I.A-9.X-19.A-1 to I.A-9.X-19.A-3600; compounds I.B-9.X-19.A-1 to I.B-9.X-19.A- 3600; compounds I.C-9.X-19.A-1 to I.C-9.X-19.A-3600; compounds I.D-9.X-19.A-1 to I.D-9.X- 19.A-3600; compounds I.E-9.X-19.A-1 to I.E-9.X-19.A-3600; compounds I.F-9.X-19.A-1 to I.F-

9. X-19.A-3600; compounds I.G-9.X-19.A-1 to I.G-9.X-19.A-3600;

compounds I.A-10.X-19.A-1 to I.A-10.X-19.A-3600; compounds I.B-10.X-19.A-1 to I.B-10.X- 19.A-3600; compounds I.C-10.X-19.A-1 to I.C-10.X-19.A-3600; compounds I.D-10.X-19.A-1 to I.D-10.X-19.A-3600; compounds I.E-10.X-19.A-1 to I.E-10.X-19.A-3600; compounds I.F-10.X- 19.A-1 to I.F-10.X-19.A-3600; compounds I.G-10.X-19.A-1 to I.G-10.X-19.A-3600;

compounds I.A-1 1.X-19.A-1 to I.A-1 1.X-19.A-3600; compounds I.B-1 1.X-19.A-1 to I.B-1 1.X- 19.A-3600; compounds I.C-1 1.X-19.A-1 to I.C-1 1 .X-19.A-3600; compounds I.D-1 1.X-19.A-1 to I.D-1 1.X-19.A-3600; compounds I.E-1 1 .X-19.A-1 to I.E-1 1.X-19.A-3600; compounds I.F-1 1.X- 19.A-1 to I.F-1 1.X-19.A-3600; compounds I.G-1 1.X-19.A-1 to I.G-1 1.X-19.A-3600;

compounds I.A-12.X-19.A-1 to I.A-12.X-19.A-3600; compounds I.B-12.X-19.A-1 to I.B-12.X- 19.A-3600; compounds I.C-12.X-19.A-1 to I.C-12.X-19.A-3600; compounds I.D-12.X-19.A-1 to I.D-12.X-19.A-3600; compounds I.E-12.X-19.A-1 to I.E-12.X-19.A-3600; compounds I.F-12.X-

19. A-1 to I.F-12.X-19.A-3600; compounds I.G-12.X-19.A-1 to I.G-12.X-19.A-3600).

Table 20a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10,

1. C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-20 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-20.A-1 to I.A-2.X-20.A-3600; compounds I.B-2.X-20.A-1 to I.B-2.X-20.A- 3600; compounds I.C-2.X-20.A-1 to I.C-2.X-20.A-3600; compounds I.D-2.X-20.A-1 to I.D-2.X- 20.A-3600; compounds I.E-2.X-20.A-1 to I.E-2.X-20.A-3600; compounds I.F-2.X-20.A-1 to I.F-

2. X-20.A-3600; compounds I.G-2.X-20.A-1 to I.G-2.X-20.A-3600;

compounds I.A-3.X-20.A-1 to I.A-3.X-20.A-3600; compounds I.B-3.X-20.A-1 to I.B-3.X-20.A- 3600; compounds I.C-3.X-20.A-1 to I.C-3.X-20.A-3600; compounds I.D-3.X-20.A-1 to I.D-3.X-

20. A-3600; compounds I.E-3.X-20.A-1 to I.E-3.X-20.A-3600; compounds I.F-3.X-20.A-1 to I.F- 3.X-20.A-3600; compounds I.G-3.X-20.A-1 to I.G-3.X-20.A-3600;

compounds I.A-4.X-20.A-1 to I.A-4.X-20.A-3600; compounds I.B-4.X-20.A-1 to I.B-4.X-20.A- 3600; compounds I.C-4.X-20.A-1 to I.C-4.X-20.A-3600; compounds I.D-4.X-20.A-1 to I.D-4.X- 20.A-3600; compounds I.E-4.X-20.A-1 to I.E-4.X-20.A-3600; compounds I.F-4.X-20.A-1 to I.F- 4.X-20.A-3600; compounds I.G-4.X-20.A-1 to I.G-4.X-20.A-3600;

compounds I.A-5.X-20.A-1 to I.A-5.X-20.A-3600; compounds I.B-5.X-20.A-1 to I.B-5.X-20.A- 3600; compounds I.C-5.X-20.A-1 to I.C-5.X-20.A-3600; compounds I.D-5.X-20.A-1 to I.D-5.X- 20.A-3600; compounds I.E-5.X-20.A-1 to I.E-5.X-20.A-3600; compounds I.F-5.X-20.A-1 to I.F-

5. X-20.A-3600; compounds I.G-5.X-20.A-1 to I.G-5.X-20.A-3600;

compounds I.A-6.X-20.A-1 to I.A-6.X-20.A-3600; compounds I.B-6.X-20.A-1 to I.B-6.X-20.A- 3600; compounds I.C-6.X-20.A-1 to I.C-6.X-20.A-3600; compounds I.D-6.X-20.A-1 to I.D-6.X- 20.A-3600; compounds I.E-6.X-20.A-1 to I.E-6.X-20.A-3600; compounds I.F-6.X-20.A-1 to I.F-

6. X-20.A-3600; compounds I.G-6.X-20.A-1 to I.G-6.X-20.A-3600;

compounds I.A-7.X-20.A-1 to I.A-7.X-20.A-3600; compounds I.B-7.X-20.A-1 to I.B-7.X-20.A- 3600; compounds I.C-7.X-20.A-1 to I.C-7.X-20.A-3600; compounds I.D-7.X-20.A-1 to I.D-7.X- 20.A-3600; compounds I.E-7.X-20.A-1 to I.E-7.X-20.A-3600; compounds I.F-7.X-20.A-1 to I.F-

7. X-20.A-3600; compounds I.G-7.X-20.A-1 to I.G-7.X-20.A-3600;

compounds I.A-8.X-20.A-1 to I.A-8.X-20.A-3600; compounds I.B-8.X-20.A-1 to I.B-8.X-20.A- 3600; compounds I.C-8.X-20.A-1 to I.C-8.X-20.A-3600; compounds I.D-8.X-20.A-1 to I.D-8.X- 20.A-3600; compounds I.E-8.X-20.A-1 to I.E-8.X-20.A-3600; compounds I.F-8.X-20.A-1 to I.F- 8.X-20.A-3600; compounds I.G-8.X-20.A-1 to I.G-8.X-20.A-3600;

compounds I.A-9.X-20.A-1 to I.A-9.X-20.A-3600; compounds I.B-9.X-20.A-1 to I.B-9.X-20.A- 3600; compounds I.C-9.X-20.A-1 to I.C-9.X-20.A-3600; compounds I.D-9.X-20.A-1 to I.D-9.X- 20.A-3600; compounds I.E-9.X-20.A-1 to I.E-9.X-20.A-3600; compounds I.F-9.X-20.A-1 to I.F- 9.X-20.A-3600; compounds I.G-9.X-20.A-1 to I.G-9.X-20.A-3600;

compounds I.A-10.X-20.A-1 to I.A-10.X-20.A-3600; compounds I.B-10.X-20.A-1 to I.B-10.X- 20.A-3600; compounds I.C-10.X-20.A-1 to I.C-10.X-20.A-3600; compounds I.D-10.X-20.A-1 to I.D-10.X-20.A-3600; compounds I.E-10.X-20.A-1 to I.E-10.X-20.A-3600; compounds I.F-10.X- 20.A-1 to I.F-10.X-20.A-3600; compounds I.G-10.X-20.A-1 to I.G-10.X-20.A-3600;

compounds I.A-1 1.X-20.A-1 to I.A-1 1.X-20.A-3600; compounds I.B-1 1.X-20.A-1 to I.B-1 1.X- 20.A-3600; compounds I.C-1 1.X-20.A-1 to I.C-1 1 .X-20.A-3600; compounds I.D-1 1.X-20.A-1 to I.D-1 1.X-20.A-3600; compounds I.E-1 1 .X-20.A-1 to I.E-1 1.X-20.A-3600; compounds I.F-1 1.X- 20.A-1 to I.F-1 1.X-20.A-3600; compounds I.G-1 1.X-20.A-1 to I.G-1 1.X-20.A-3600;

compounds I.A-12.X-20.A-1 to I.A-12.X-20.A-3600; compounds I.B-12.X-20.A-1 to I.B-12.X- 20.A-3600; compounds I.C-12.X-20.A-1 to I.C-12.X-20.A-3600; compounds I.D-12.X-20.A-1 to I.D-12.X-20.A-3600; compounds I.E-12.X-20.A-1 to I.E-12.X-20.A-3600; compounds I.F-12.X- 20.A-1 to I.F-12.X-20.A-3600; compounds I.G-12.X-20.A-1 to I.G-12.X-20.A-3600).

Table 21 a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A-

8. I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-21 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (compounds I.A-2.X-21.A-1 to I.A-2.X-21.A-3600; compounds I.B-2.X-21.A-1 to I.B-2.X-21 .A- 3600; compounds I.C-2.X-21.A-1 to I.C-2.X-21.A-3600; compounds I.D-2.X-21.A-1 to I.D-2.X- 21.A-3600; compounds I.E-2.X-21.A-1 to I.E-2.X-21.A-3600; compounds I.F-2.X-21.A-1 to I.F-

2. X-21 .A-3600; compounds I.G-2.X-21 .A-1 to I.G-2.X-21 .A-3600;

compounds I.A-3.X-21.A-1 to I. A-3.X-21 .A-3600; compounds I.B-3.X-21 .A-1 to I.B-3.X-21 .A- 3600; compounds I.C-3.X-21.A-1 to I.C-3.X-21. A-3600; compounds I.D-3.X-21.A-1 to I.D-3.X- 21. A-3600; compounds I.E-3.X-21.A-1 to I. E-3.X-21. A-3600; compounds I.F-3.X-21.A-1 to I.F-

3. X-21 . A-3600; compounds I.G-3.X-21 .A-1 to I. G-3.X-21 .A-3600;

compounds I.A-4.X-21.A-1 to I. A-4.X-21 .A-3600; compounds I.B-4.X-21 .A-1 to I.B-4.X-21 .A- 3600; compounds I.C-4.X-21.A-1 to I. C-4.X-21. A-3600; compounds I.D-4.X-21.A-1 to I.D-4.X- 21. A-3600; compounds I.E-4.X-21.A-1 to I. E-4.X-21. A-3600; compounds I.F-4.X-21.A-1 to I.F-

4. X-21 . A-3600; compounds I.G-4.X-21 .A-1 to I. G-4.X-21 .A-3600;

compounds I.A-5.X-21.A-1 to I. A-5.X-21 .A-3600; compounds I.B-5.X-21 .A-1 to I.B-5.X-21 .A- 3600; compounds I.C-5.X-21.A-1 to I. C-5.X-21. A-3600; compounds I.D-5.X-21.A-1 to I.D-5.X- 21. A-3600; compounds I.E-5.X-21.A-1 to I. E-5.X-21. A-3600; compounds I.F-5.X-21.A-1 to I.F-

5. X-21 . A-3600; compounds I.G-5.X-21 .A-1 to I. G-5.X-21 .A-3600;

compounds I.A-6.X-21.A-1 to I. A-6.X-21 .A-3600; compounds I.B-6.X-21 .A-1 to I.B-6.X-21 .A- 3600; compounds I.C-6.X-21.A-1 to I. C-6.X-21. A-3600; compounds I.D-6.X-21.A-1 to I.D-6.X- 21. A-3600; compounds I.E-6.X-21.A-1 to I. E-6.X-21. A-3600; compounds I.F-6.X-21.A-1 to I.F- 6.X-21 .A-3600; compounds I.G-6.X-21 .A-1 to I.G-6.X-21 .A-3600;

compounds I.A-7.X-21.A-1 to I. A-7.X-21 .A-3600; compounds I.B-7.X-21 .A-1 to I.B-7.X-21 .A- 3600; compounds I.C-7.X-21.A-1 to I. C-7.X-21. A-3600; compounds I.D-7.X-21.A-1 to I.D-7.X- 21. A-3600; compounds I.E-7.X-21.A-1 to I. E-7.X-21. A-3600; compounds I.F-7.X-21.A-1 to I.F-

7. X-21 . A-3600; compounds I.G-7.X-21 .A-1 to I. G-7.X-21 .A-3600;

compounds I.A-8.X-21.A-1 to I. A-8.X-21 .A-3600; compounds I.B-8.X-21 .A-1 to I.B-8.X-21 .A- 3600; compounds I.C-8.X-21.A-1 to I. C-8.X-21. A-3600; compounds I.D-8.X-21.A-1 to I.D-8.X- 21. A-3600; compounds I.E-8.X-21.A-1 to I. E-8.X-21. A-3600; compounds I.F-8.X-21.A-1 to I.F-

8. X-21 . A-3600; compounds I.G-8.X-21 .A-1 to I. G-8.X-21 .A-3600;

compounds I.A-9.X-21.A-1 to I. A-9.X-21 .A-3600; compounds I.B-9.X-21 .A-1 to I.B-9.X-21 .A- 3600; compounds I.C-9.X-21.A-1 to I. C-9.X-21. A-3600; compounds I.D-9.X-21.A-1 to I.D-9.X- 21. A-3600; compounds I.E-9.X-21.A-1 to I. E-9.X-21. A-3600; compounds I.F-9.X-21.A-1 to I.F-

9. X-21 . A-3600; compounds I.G-9.X-21 .A-1 to I. G-9.X-21 .A-3600;

compounds I.A-10.X-21.A-1 to I.A-10.X-21. A-3600; compounds I.B-10.X-21.A-1 to I.B-10.X- 21.A-3600; compounds I.C-10.X-21. A-1 to I.C-10.X-21. A-3600; compounds I.D-10.X-21. A-1 to I.D-10.X-21. A-3600; compounds I.E-10.X-21.A-1 to I.E-10.X-21 .A-3600; compounds I.F-10.X- 21. A-1 to I. F-10.X-21. A-3600; compounds I.G-10.X-21.A-1 to I.G-10.X-21. A-3600;

compounds I.A-1 1.X-21.A-1 to I. A-1 1.X-21. A-3600; compounds I.B-1 1.X-21.A-1 to I.B-1 1.X- 21. A-3600; compounds I.C-1 1.X-21. A-1 to I. C-1 1 .X-21. A-3600; compounds I.D-1 1.X-21. A-1 to I.D-1 1.X-21. A-3600; compounds I.E-1 1 .X-21.A-1 to I. E-1 1.X-21 . A-3600; compounds I.F-1 1.X- 21. A-1 to I. F-1 1.X-21. A-3600; compounds I.G-1 1.X-21.A-1 to I.G-1 1.X-21. A-3600;

compounds I.A-12.X-21. A-1 to I.A-12.X-21. A-3600; compounds I.B-12.X-21. A-1 to I.B-12.X- 21.A-3600; compounds I.C-12.X-21.A-1 to I.C-12.X-21.A-3600; compounds I.D-12.X-21.A-1 to I.D-12.X-21.A-3600; compounds I.E-12.X-21.A-1 to I.E-12.X-21 .A-3600; compounds I.F-12.X-

21. A-1 to I. F-12.X-21. A-3600; compounds I.G-12.X-21.A-1 to I.G-12.X-21. A-3600).

Table 22a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10,

1. C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-22 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-22.A-1 to I.A-2.X-22.A-3600; compounds I.B-2.X-22.A-1 to I.B-2.X-22.A- 3600; compounds I.C-2.X-22.A-1 to I.C-2.X-22.A-3600; compounds I.D-2.X-22.A-1 to I.D-2.X- 22.A-3600; compounds I.E-2.X-22.A-1 to I.E-2.X-22.A-3600; compounds I.F-2.X-22.A-1 to I.F-

2. X-22.A-3600; compounds I.G-2.X-22.A-1 to I.G-2.X-22.A-3600;

compounds I.A-3.X-22.A-1 to I.A-3.X-22.A-3600; compounds I.B-3.X-22.A-1 to I.B-3.X-22.A- 3600; compounds I.C-3.X-22.A-1 to I.C-3.X-22.A-3600; compounds I.D-3.X-22.A-1 to I.D-3.X-

22. A-3600; compounds I.E-3.X-22.A-1 to I.E-3.X-22.A-3600; compounds I.F-3.X-22.A-1 to I.F- 3.X-22.A-3600; compounds I.G-3.X-22.A-1 to I.G-3.X-22.A-3600;

compounds I.A-4.X-22.A-1 to I.A-4.X-22.A-3600; compounds I.B-4.X-22.A-1 to I.B-4.X-22.A- 3600; compounds I.C-4.X-22.A-1 to I.C-4.X-22.A-3600; compounds I.D-4.X-22.A-1 to I.D-4.X- 22.A-3600; compounds I.E-4.X-22.A-1 to I.E-4.X-22.A-3600; compounds I.F-4.X-22.A-1 to I.F-

4. X-22.A-3600; compounds I.G-4.X-22.A-1 to I.G-4.X-22.A-3600;

compounds I.A-5.X-22.A-1 to I.A-5.X-22.A-3600; compounds I.B-5.X-22.A-1 to I.B-5.X-22.A- 3600; compounds I.C-5.X-22.A-1 to I.C-5.X-22.A-3600; compounds I.D-5.X-22.A-1 to I.D-5.X- 22.A-3600; compounds I.E-5.X-22.A-1 to I.E-5.X-22.A-3600; compounds I.F-5.X-22.A-1 to I.F-

5. X-22.A-3600; compounds I.G-5.X-22.A-1 to I.G-5.X-22.A-3600;

compounds I.A-6.X-22.A-1 to I.A-6.X-22.A-3600; compounds I.B-6.X-22.A-1 to I.B-6.X-22.A- 3600; compounds I.C-6.X-22.A-1 to I.C-6.X-22.A-3600; compounds I.D-6.X-22.A-1 to I.D-6.X- 22.A-3600; compounds I.E-6.X-22.A-1 to I.E-6.X-22.A-3600; compounds I.F-6.X-22.A-1 to I.F-

6. X-22.A-3600; compounds I.G-6.X-22.A-1 to I.G-6.X-22.A-3600;

compounds I.A-7.X-22.A-1 to I.A-7.X-22.A-3600; compounds I.B-7.X-22.A-1 to I.B-7.X-22.A- 3600; compounds I.C-7.X-22.A-1 to I.C-7.X-22.A-3600; compounds I.D-7.X-22.A-1 to I.D-7.X- 22.A-3600; compounds I.E-7.X-22.A-1 to I.E-7.X-22.A-3600; compounds I.F-7.X-22.A-1 to I.F-

7. X-22.A-3600; compounds I.G-7.X-22.A-1 to I.G-7.X-22.A-3600;

compounds I.A-8.X-22.A-1 to I.A-8.X-22.A-3600; compounds I.B-8.X-22.A-1 to I.B-8.X-22.A- 3600; compounds I.C-8.X-22.A-1 to I.C-8.X-22.A-3600; compounds I.D-8.X-22.A-1 to I.D-8.X- 22.A-3600; compounds I.E-8.X-22.A-1 to I.E-8.X-22.A-3600; compounds I.F-8.X-22.A-1 to I.F- 8.X-22.A-3600; compounds I.G-8.X-22.A-1 to I.G-8.X-22.A-3600; compounds I.A-9.X-22.A-1 to I.A-9.X-22.A-3600; compounds I.B-9.X-22.A-1 to I.B-9.X-22.A- 3600; compounds I.C-9.X-22.A-1 to I.C-9.X-22.A-3600; compounds I.D-9.X-22.A-1 to I.D-9.X- 22.A-3600; compounds I.E-9.X-22.A-1 to I.E-9.X-22.A-3600; compounds I.F-9.X-22.A-1 to I.F- 9.X-22.A-3600; compounds I.G-9.X-22.A-1 to I.G-9.X-22.A-3600;

compounds I.A-10.X-22.A-1 to I.A-10.X-22.A-3600; compounds I.B-10.X-22.A-1 to I.B-10.X- 22.A-3600; compounds I.C-10.X-22.A-1 to I.C-10.X-22.A-3600; compounds I.D-10.X-22.A-1 to I.D-10.X-22.A-3600; compounds I.E-10.X-22.A-1 to I.E-10.X-22.A-3600; compounds I.F-10.X- 22.A-1 to I.F-10.X-22.A-3600; compounds I.G-10.X-22.A-1 to I.G-10.X-22.A-3600;

compounds I.A-1 1.X-22.A-1 to I.A-1 1.X-22.A-3600; compounds I.B-1 1.X-22.A-1 to I.B-1 1.X- 22.A-3600; compounds I.C-1 1.X-22.A-1 to I.C-1 1 .X-22.A-3600; compounds I.D-1 1.X-22.A-1 to I.D-1 1.X-22.A-3600; compounds I.E-1 1 .X-22.A-1 to I.E-1 1.X-22.A-3600; compounds I.F-1 1.X- 22.A-1 to I.F-1 1.X-22.A-3600; compounds I.G-1 1.X-22.A-1 to I.G-1 1.X-22.A-3600;

compounds I.A-12.X-22.A-1 to I.A-12.X-22.A-3600; compounds I.B-12.X-22.A-1 to I.B-12.X- 22.A-3600; compounds I.C-12.X-22.A-1 to I.C-12.X-22.A-3600; compounds I.D-12.X-22.A-1 to I.D-12.X-22.A-3600; compounds I.E-12.X-22.A-1 to I.E-12.X-22.A-3600; compounds I.F-12.X-

22. A-1 to I.F-12.X-22.A-3600; compounds I.G-12.X-22.A-1 to I.G-12.X-22.A-3600).

Table 23a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-23 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-23.A-1 to I.A-2.X-23.A-3600; compounds I.B-2.X-23.A-1 to I.B-2.X-23.A- 3600; compounds I.C-2.X-23.A-1 to I.C-2.X-23.A-3600; compounds I.D-2.X-23.A-1 to I.D-2.X-

23. A-3600; compounds I.E-2.X-23.A-1 to I.E-2.X-23.A-3600; compounds I.F-2.X-23.A-1 to I.F-

2. X-23.A-3600; compounds I.G-2.X-23.A-1 to I.G-2.X-23.A-3600;

compounds I.A-3.X-23.A-1 to I.A-3.X-23.A-3600; compounds I.B-3.X-23.A-1 to I.B-3.X-23.A- 3600; compounds I.C-3.X-23.A-1 to I.C-3.X-23.A-3600; compounds I.D-3.X-23.A-1 to I.D-3.X- 23.A-3600; compounds I.E-3.X-23.A-1 to I.E-3.X-23.A-3600; compounds I.F-3.X-23.A-1 to I.F-

3. X-23.A-3600; compounds I.G-3.X-23.A-1 to I.G-3.X-23.A-3600;

compounds I.A-4.X-23.A-1 to I.A-4.X-23.A-3600; compounds I.B-4.X-23.A-1 to I.B-4.X-23.A- 3600; compounds I.C-4.X-23.A-1 to I.C-4.X-23.A-3600; compounds I.D-4.X-23.A-1 to I.D-4.X- 23.A-3600; compounds I.E-4.X-23.A-1 to I.E-4.X-23.A-3600; compounds I.F-4.X-23.A-1 to I.F-

4. X-23.A-3600; compounds I.G-4.X-23.A-1 to I.G-4.X-23.A-3600;

compounds I.A-5.X-23.A-1 to I.A-5.X-23.A-3600; compounds I.B-5.X-23.A-1 to I.B-5.X-23.A- 3600; compounds I.C-5.X-23.A-1 to I.C-5.X-23.A-3600; compounds I.D-5.X-23.A-1 to I.D-5.X- 23.A-3600; compounds I.E-5.X-23.A-1 to I.E-5.X-23.A-3600; compounds I.F-5.X-23.A-1 to I.F-

5. X-23.A-3600; compounds I.G-5.X-23.A-1 to I.G-5.X-23.A-3600; compounds I.A-6.X-23.A-1 to I.A-6.X-23.A-3600; compounds I.B-6.X-23.A-1 to I.B-6.X-23.A- 3600; compounds I.C-6.X-23.A-1 to I.C-6.X-23.A-3600; compounds I.D-6.X-23.A-1 to I.D-6.X- 23.A-3600; compounds I.E-6.X-23.A-1 to I.E-6.X-23.A-3600; compounds I.F-6.X-23.A-1 to I.F-

6. X-23.A-3600; compounds I.G-6.X-23.A-1 to I.G-6.X-23.A-3600;

compounds I.A-7.X-23.A-1 to I.A-7.X-23.A-3600; compounds I.B-7.X-23.A-1 to I.B-7.X-23.A- 3600; compounds I.C-7.X-23.A-1 to I.C-7.X-23.A-3600; compounds I.D-7.X-23.A-1 to I.D-7.X- 23.A-3600; compounds I.E-7.X-23.A-1 to I.E-7.X-23.A-3600; compounds I.F-7.X-23.A-1 to I.F-

7. X-23.A-3600; compounds I.G-7.X-23.A-1 to I.G-7.X-23.A-3600;

compounds I.A-8.X-23.A-1 to I.A-8.X-23.A-3600; compounds I.B-8.X-23.A-1 to I.B-8.X-23.A- 3600; compounds I.C-8.X-23.A-1 to I.C-8.X-23.A-3600; compounds I.D-8.X-23.A-1 to I.D-8.X- 23.A-3600; compounds I.E-8.X-23.A-1 to I.E-8.X-23.A-3600; compounds I.F-8.X-23.A-1 to I.F-

8. X-23.A-3600; compounds I.G-8.X-23.A-1 to I.G-8.X-23.A-3600;

compounds I.A-9.X-23.A-1 to I.A-9.X-23.A-3600; compounds I.B-9.X-23.A-1 to I.B-9.X-23.A- 3600; compounds I.C-9.X-23.A-1 to I.C-9.X-23.A-3600; compounds I.D-9.X-23.A-1 to I.D-9.X- 23.A-3600; compounds I.E-9.X-23.A-1 to I.E-9.X-23.A-3600; compounds I.F-9.X-23.A-1 to I.F-

9. X-23.A-3600; compounds I.G-9.X-23.A-1 to I.G-9.X-23.A-3600;

compounds I.A-10.X-23.A-1 to I.A-10.X-23.A-3600; compounds I.B-10.X-23.A-1 to I.B-10.X- 23.A-3600; compounds I.C-10.X-23.A-1 to I.C-10.X-23.A-3600; compounds I.D-10.X-23.A-1 to I.D-10.X-23.A-3600; compounds I.E-10.X-23.A-1 to I.E-10.X-23.A-3600; compounds I.F-10.X- 23.A-1 to I.F-10.X-23.A-3600; compounds I.G-10.X-23.A-1 to I.G-10.X-23.A-3600;

compounds I.A-1 1.X-23.A-1 to I.A-1 1.X-23.A-3600; compounds I.B-1 1.X-23.A-1 to I.B-1 1.X- 23.A-3600; compounds I.C-1 1.X-23.A-1 to I.C-1 1 .X-23.A-3600; compounds I.D-1 1.X-23.A-1 to I.D-1 1.X-23.A-3600; compounds I.E-1 1 .X-23.A-1 to I.E-1 1.X-23.A-3600; compounds I.F-1 1.X- 23.A-1 to I.F-1 1.X-23.A-3600; compounds I.G-1 1.X-23.A-1 to I.G-1 1.X-23.A-3600;

compounds I.A-12.X-23.A-1 to I.A-12.X-23.A-3600; compounds I.B-12.X-23.A-1 to I.B-12.X- 23.A-3600; compounds I.C-12.X-23.A-1 to I.C-12.X-23.A-3600; compounds I.D-12.X-23.A-1 to I.D-12.X-23.A-3600; compounds I.E-12.X-23.A-1 to I.E-12.X-23.A-3600; compounds I.F-12.X- 23.A-1 to I.F-12.X-23.A-3600; compounds I.G-12.X-23.A-1 to I.G-12.X-23.A-3600).

Table 24a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10,

1. C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-24 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-24.A-1 to I.A-2.X-24.A-3600; compounds I.B-2.X-24.A-1 to I.B-2.X-24.A- 3600; compounds I.C-2.X-24.A-1 to I.C-2.X-24.A-3600; compounds I.D-2.X-24.A-1 to I.D-2.X- 24.A-3600; compounds I.E-2.X-24.A-1 to I.E-2.X-24.A-3600; compounds I.F-2.X-24.A-1 to I.F-

2. X-24.A-3600; compounds I.G-2.X-24.A-1 to I.G-2.X-24.A-3600; compounds I.A-3.X-24.A-1 to I.A-3.X-24.A-3600; compounds I.B-3.X-24.A-1 to I.B-3.X-24.A- 3600; compounds I.C-3.X-24.A-1 to I.C-3.X-24.A-3600; compounds I.D-3.X-24.A-1 to I.D-3.X- 24.A-3600; compounds I.E-3.X-24.A-1 to I.E-3.X-24.A-3600; compounds I.F-3.X-24.A-1 to I.F-

3. X-24.A-3600; compounds I.G-3.X-24.A-1 to I.G-3.X-24.A-3600;

compounds I.A-4.X-24.A-1 to I.A-4.X-24.A-3600; compounds I.B-4.X-24.A-1 to I.B-4.X-24.A- 3600; compounds I.C-4.X-24.A-1 to I.C-4.X-24.A-3600; compounds I.D-4.X-24.A-1 to I.D-4.X- 24.A-3600; compounds I.E-4.X-24.A-1 to I.E-4.X-24.A-3600; compounds I.F-4.X-24.A-1 to I.F-

4. X-24.A-3600; compounds I.G-4.X-24.A-1 to I.G-4.X-24.A-3600;

compounds I.A-5.X-24.A-1 to I.A-5.X-24.A-3600; compounds I.B-5.X-24.A-1 to I.B-5.X-24.A- 3600; compounds I.C-5.X-24.A-1 to I.C-5.X-24.A-3600; compounds I.D-5.X-24.A-1 to I.D-5.X- 24.A-3600; compounds I.E-5.X-24.A-1 to I.E-5.X-24.A-3600; compounds I.F-5.X-24.A-1 to I.F-

5. X-24.A-3600; compounds I.G-5.X-24.A-1 to I.G-5.X-24.A-3600;

compounds I.A-6.X-24.A-1 to I.A-6.X-24.A-3600; compounds I.B-6.X-24.A-1 to I.B-6.X-24.A- 3600; compounds I.C-6.X-24.A-1 to I.C-6.X-24.A-3600; compounds I.D-6.X-24.A-1 to I.D-6.X- 24.A-3600; compounds I.E-6.X-24.A-1 to I.E-6.X-24.A-3600; compounds I.F-6.X-24.A-1 to I.F-

6. X-24.A-3600; compounds I.G-6.X-24.A-1 to I.G-6.X-24.A-3600;

compounds I.A-7.X-24.A-1 to I.A-7.X-24.A-3600; compounds I.B-7.X-24.A-1 to I.B-7.X-24.A- 3600; compounds I.C-7.X-24.A-1 to I.C-7.X-24.A-3600; compounds I.D-7.X-24.A-1 to I.D-7.X- 24.A-3600; compounds I.E-7.X-24.A-1 to I.E-7.X-24.A-3600; compounds I.F-7.X-24.A-1 to I.F- 7.X-24.A-3600; compounds I.G-7.X-24.A-1 to I.G-7.X-24.A-3600;

compounds I.A-8.X-24.A-1 to I.A-8.X-24.A-3600; compounds I.B-8.X-24.A-1 to I.B-8.X-24.A- 3600; compounds I.C-8.X-24.A-1 to I.C-8.X-24.A-3600; compounds I.D-8.X-24.A-1 to I.D-8.X- 24.A-3600; compounds I.E-8.X-24.A-1 to I.E-8.X-24.A-3600; compounds I.F-8.X-24.A-1 to I.F-

8. X-24.A-3600; compounds I.G-8.X-24.A-1 to I.G-8.X-24.A-3600;

compounds I.A-9.X-24.A-1 to I.A-9.X-24.A-3600; compounds I.B-9.X-24.A-1 to I.B-9.X-24.A- 3600; compounds I.C-9.X-24.A-1 to I.C-9.X-24.A-3600; compounds I.D-9.X-24.A-1 to I.D-9.X- 24.A-3600; compounds I.E-9.X-24.A-1 to I.E-9.X-24.A-3600; compounds I.F-9.X-24.A-1 to I.F-

9. X-24.A-3600; compounds I.G-9.X-24.A-1 to I.G-9.X-24.A-3600;

compounds I.A-10.X-24.A-1 to I.A-10.X-24.A-3600; compounds I.B-10.X-24.A-1 to I.B-10.X- 24.A-3600; compounds I.C-10.X-24.A-1 to I.C-10.X-24.A-3600; compounds I.D-10.X-24.A-1 to I.D-10.X-24.A-3600; compounds I.E-10.X-24.A-1 to I.E-10.X-24.A-3600; compounds I.F-10.X- 24.A-1 to I.F-10.X-24.A-3600; compounds I.G-10.X-24.A-1 to I.G-10.X-24.A-3600;

compounds I.A-1 1.X-24.A-1 to I.A-1 1.X-24.A-3600; compounds I.B-1 1.X-24.A-1 to I.B-1 1.X- 24.A-3600; compounds I.C-1 1.X-24.A-1 to I.C-1 1 .X-24.A-3600; compounds I.D-1 1.X-24.A-1 to I.D-1 1.X-24.A-3600; compounds I.E-1 1 .X-24.A-1 to I.E-1 1.X-24.A-3600; compounds I.F-1 1.X- 24.A-1 to I.F-1 1.X-24.A-3600; compounds I.G-1 1.X-24.A-1 to I.G-1 1 .X-24.A-3600;

compounds I.A-12.X-24.A-1 to I.A-12.X-24.A-3600; compounds I.B-12.X-24.A-1 to I.B-12.X- 24.A-3600; compounds I.C-12.X-24.A-1 to I.C-12.X-24.A-3600; compounds I.D-12.X-24.A-1 to I.D-12.X-24.A-3600; compounds I.E-12.X-24.A-1 to I.E-12.X-24.A-3600; compounds I.F-12.X- 24.A-1 to I.F-12.X-24.A-3600; compounds I.G-12.X-24.A-1 to I.G-12.X-24.A-3600).

Table 25a Compounds of the formula I.G-1 ; I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G- 7; I.A-8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ;

1. A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-25 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-25.A-1 to I.A-2.X-25.A-3600; compounds I.B-2.X-25.A-1 to I.B-2.X-25.A- 3600; compounds I.C-2.X-25.A-1 to I.C-2.X-25.A-3600; compounds I.D-2.X-25.A-1 to I.D-2.X- 25.A-3600; compounds I.E-2.X-25.A-1 to I.E-2.X-25.A-3600; compounds I.F-2.X-25.A-1 to I.F-

2. X-25.A-3600; compounds I.G-2.X-25.A-1 to I.G-2.X-25.A-3600;

compounds I.A-3.X-25.A-1 to I.A-3.X-25.A-3600; compounds I.B-3.X-25.A-1 to I.B-3.X-25.A- 3600; compounds I.C-3.X-25.A-1 to I.C-3.X-25.A-3600; compounds I.D-3.X-25.A-1 to I.D-3.X- 25.A-3600; compounds I.E-3.X-25.A-1 to I.E-3.X-25.A-3600; compounds I.F-3.X-25.A-1 to I.F-

3. X-25.A-3600; compounds I.G-3.X-25.A-1 to I.G-3.X-25.A-3600;

compounds I.A-4.X-25.A-1 to I.A-4.X-25.A-3600; compounds I.B-4.X-25.A-1 to I.B-4.X-25.A- 3600; compounds I.C-4.X-25.A-1 to I.C-4.X-25.A-3600; compounds I.D-4.X-25.A-1 to I.D-4.X- 25.A-3600; compounds I.E-4.X-25.A-1 to I.E-4.X-25.A-3600; compounds I.F-4.X-25.A-1 to I.F- 4.X-25.A-3600; compounds I.G-4.X-25.A-1 to I.G-4.X-25.A-3600;

compounds I.A-5.X-25.A-1 to I.A-5.X-25.A-3600; compounds I.B-5.X-25.A-1 to I.B-5.X-25.A- 3600; compounds I.C-5.X-25.A-1 to I.C-5.X-25.A-3600; compounds I.D-5.X-25.A-1 to I.D-5.X- 25.A-3600; compounds I.E-5.X-25.A-1 to I.E-5.X-25.A-3600; compounds I.F-5.X-25.A-1 to I.F-

5. X-25.A-3600; compounds I.G-5.X-25.A-1 to I.G-5.X-25.A-3600;

compounds I.A-6.X-25.A-1 to I.A-6.X-25.A-3600; compounds I.B-6.X-25.A-1 to I.B-6.X-25.A- 3600; compounds I.C-6.X-25.A-1 to I.C-6.X-25.A-3600; compounds I.D-6.X-25.A-1 to I.D-6.X- 25.A-3600; compounds I.E-6.X-25.A-1 to I.E-6.X-25.A-3600; compounds I.F-6.X-25.A-1 to I.F-

6. X-25.A-3600; compounds I.G-6.X-25.A-1 to I.G-6.X-25.A-3600;

compounds I.A-7.X-25.A-1 to I.A-7.X-25.A-3600; compounds I.B-7.X-25.A-1 to I.B-7.X-25.A- 3600; compounds I.C-7.X-25.A-1 to I.C-7.X-25.A-3600; compounds I.D-7.X-25.A-1 to I.D-7.X- 25.A-3600; compounds I.E-7.X-25.A-1 to I.E-7.X-25.A-3600; compounds I.F-7.X-25.A-1 to I.F-

7. X-25.A-3600; compounds I.G-7.X-25.A-1 to I.G-7.X-25.A-3600;

compounds I.A-8.X-25.A-1 to I.A-8.X-25.A-3600; compounds I.B-8.X-25.A-1 to I.B-8.X-25.A- 3600; compounds I.C-8.X-25.A-1 to I.C-8.X-25.A-3600; compounds I.D-8.X-25.A-1 to I.D-8.X- 25.A-3600; compounds I.E-8.X-25.A-1 to I.E-8.X-25.A-3600; compounds I.F-8.X-25.A-1 to I.F-

8. X-25.A-3600; compounds I.G-8.X-25.A-1 to I.G-8.X-25.A-3600;

compounds I.A-9.X-25.A-1 to I.A-9.X-25.A-3600; compounds I.B-9.X-25.A-1 to I.B-9.X-25.A- 3600; compounds I.C-9.X-25.A-1 to I.C-9.X-25.A-3600; compounds I.D-9.X-25.A-1 to I.D-9.X- 25.A-3600; compounds I.E-9.X-25.A-1 to I.E-9.X-25.A-3600; compounds I.F-9.X-25.A-1 to I.F- 9.X-25.A-3600; compounds I.G-9.X-25.A-1 to I.G-9.X-25.A-3600;

compounds I.A-10.X-25.A-1 to I.A-10.X-25.A-3600; compounds I.B-10.X-25.A-1 to I.B-10.X- 25.A-3600; compounds I.C-10.X-25.A-1 to I.C-10.X-25.A-3600; compounds I.D-10.X-25.A-1 to I.D-10.X-25.A-3600; compounds I.E-10.X-25.A-1 to I.E-10.X-25.A-3600; compounds I.F-10.X- 25.A-1 to I.F-10.X-25.A-3600; compounds I.G-10.X-25.A-1 to I.G-10.X-25.A-3600;

compounds I.A-1 1.X-25.A-1 to I.A-1 1.X-25.A-3600; compounds I.B-1 1.X-25.A-1 to I.B-1 1.X- 25.A-3600; compounds I.C-1 1.X-25.A-1 to I.C-1 1 .X-25.A-3600; compounds I.D-1 1.X-25.A-1 to I.D-1 1.X-25.A-3600; compounds I.E-1 1 .X-25.A-1 to I.E-1 1.X-25.A-3600; compounds I.F-1 1.X- 25.A-1 to I.F-1 1.X-25.A-3600; compounds I.G-1 1.X-25.A-1 to I.G-1 1.X-25.A-3600;

compounds I.A-12.X-25.A-1 to I.A-12.X-25.A-3600; compounds I.B-12.X-25.A-1 to I.B-12.X- 25.A-3600; compounds I.C-12.X-25.A-1 to I.C-12.X-25.A-3600; compounds I.D-12.X-25.A-1 to I.D-12.X-25.A-3600; compounds I.E-12.X-25.A-1 to I.E-12.X-25.A-3600; compounds I.F-12.X-

25. A-1 to I.F-12.X-25.A-3600; compounds I.G-12.X-25.A-1 to I.G-12.X-25.A-3600).

Table 26a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-26 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-26.A-1 to I.A-2.X-26.A-3600; compounds I.B-2.X-26.A-1 to I.B-2.X-26.A- 3600; compounds I.C-2.X-26.A-1 to I.C-2.X-26.A-3600; compounds I.D-2.X-26.A-1 to I.D-2.X-

26. A-3600; compounds I.E-2.X-26.A-1 to I.E-2.X-26.A-3600; compounds I.F-2.X-26.A-1 to I.F-

2. X-26.A-3600; compounds I.G-2.X-26.A-1 to I.G-2.X-26.A-3600;

compounds I.A-3.X-26.A-1 to I.A-3.X-26.A-3600; compounds I.B-3.X-26.A-1 to I.B-3.X-26.A- 3600; compounds I.C-3.X-26.A-1 to I.C-3.X-26.A-3600; compounds I.D-3.X-26.A-1 to I.D-3.X- 26.A-3600; compounds I.E-3.X-26.A-1 to I.E-3.X-26.A-3600; compounds I.F-3.X-26.A-1 to I.F-

3. X-26.A-3600; compounds I.G-3.X-26.A-1 to I.G-3.X-26.A-3600;

compounds I.A-4.X-26.A-1 to I.A-4.X-26.A-3600; compounds I.B-4.X-26.A-1 to I.B-4.X-26.A- 3600; compounds I.C-4.X-26.A-1 to I.C-4.X-26.A-3600; compounds I.D-4.X-26.A-1 to I.D-4.X- 26.A-3600; compounds I.E-4.X-26.A-1 to I.E-4.X-26.A-3600; compounds I.F-4.X-26.A-1 to I.F-

4. X-26.A-3600; compounds I.G-4.X-26.A-1 to I.G-4.X-26.A-3600;

compounds I.A-5.X-26.A-1 to I.A-5.X-26.A-3600; compounds I.B-5.X-26.A-1 to I.B-5.X-26.A- 3600; compounds I.C-5.X-26.A-1 to I.C-5.X-26.A-3600; compounds I.D-5.X-26.A-1 to I.D-5.X- 26.A-3600; compounds I.E-5.X-26.A-1 to I.E-5.X-26.A-3600; compounds I.F-5.X-26.A-1 to I.F-

5. X-26.A-3600; compounds I.G-5.X-26.A-1 to I.G-5.X-26.A-3600;

compounds I.A-6.X-26.A-1 to I.A-6.X-26.A-3600; compounds I.B-6.X-26.A-1 to I.B-6.X-26.A- 3600; compounds I.C-6.X-26.A-1 to I.C-6.X-26.A-3600; compounds I.D-6.X-26.A-1 to I.D-6.X- 26.A-3600; compounds I.E-6.X-26.A-1 to I.E-6.X-26.A-3600; compounds I.F-6.X-26.A-1 to I.F- 6.X-26.A-3600; compounds I.G-6.X-26.A-1 to I.G-6.X-26.A-3600; compounds I.A-7.X-26.A-1 to I.A-7.X-26.A-3600; compounds I.B-7.X-26.A-1 to I.B-7.X-26.A- 3600; compounds I.C-7.X-26.A-1 to I.C-7.X-26.A-3600; compounds I.D-7.X-26.A-1 to I.D-7.X- 26.A-3600; compounds I.E-7.X-26.A-1 to I.E-7.X-26.A-3600; compounds I.F-7.X-26.A-1 to I.F-

7. X-26.A-3600; compounds I.G-7.X-26.A-1 to I.G-7.X-26.A-3600;

compounds I.A-8.X-26.A-1 to I.A-8.X-26.A-3600; compounds I.B-8.X-26.A-1 to I.B-8.X-26.A- 3600; compounds I.C-8.X-26.A-1 to I.C-8.X-26.A-3600; compounds I.D-8.X-26.A-1 to I.D-8.X- 26.A-3600; compounds I.E-8.X-26.A-1 to I.E-8.X-26.A-3600; compounds I.F-8.X-26.A-1 to I.F-

8. X-26.A-3600; compounds I.G-8.X-26.A-1 to I.G-8.X-26.A-3600;

compounds I.A-9.X-26.A-1 to I.A-9.X-26.A-3600; compounds I.B-9.X-26.A-1 to I.B-9.X-26.A- 3600; compounds I.C-9.X-26.A-1 to I.C-9.X-26.A-3600; compounds I.D-9.X-26.A-1 to I.D-9.X- 26.A-3600; compounds I.E-9.X-26.A-1 to I.E-9.X-26.A-3600; compounds I.F-9.X-26.A-1 to I.F-

9. X-26.A-3600; compounds I.G-9.X-26.A-1 to I.G-9.X-26.A-3600;

compounds I.A-10.X-26.A-1 to I.A-10.X-26.A-3600; compounds I.B-10.X-26.A-1 to I.B-10.X- 26.A-3600; compounds I.C-10.X-26.A-1 to I.C-10.X-26.A-3600; compounds I.D-10.X-26.A-1 to I.D-10.X-26.A-3600; compounds I.E-10.X-26.A-1 to I.E-10.X-26.A-3600; compounds I.F-10.X- 26.A-1 to I.F-10.X-26.A-3600; compounds I.G-10.X-26.A-1 to I.G-10.X-26.A-3600;

compounds I.A-1 1.X-26.A-1 to I.A-1 1.X-26.A-3600; compounds I.B-1 1.X-26.A-1 to I.B-1 1.X- 26.A-3600; compounds I.C-1 1.X-26.A-1 to I.C-1 1 .X-26.A-3600; compounds I.D-1 1.X-26.A-1 to I.D-1 1.X-26.A-3600; compounds I.E-1 1 .X-26.A-1 to I.E-1 1.X-26.A-3600; compounds I.F-1 1.X- 26.A-1 to I.F-1 1.X-26.A-3600; compounds I.G-1 1.X-26.A-1 to I.G-1 1.X-26.A-3600;

compounds I.A-12.X-26.A-1 to I.A-12.X-26.A-3600; compounds I.B-12.X-26.A-1 to I.B-12.X- 26.A-3600; compounds I.C-12.X-26.A-1 to I.C-12.X-26.A-3600; compounds I.D-12.X-26.A-1 to I.D-12.X-26.A-3600; compounds I.E-12.X-26.A-1 to I.E-12.X-26.A-3600; compounds I.F-12.X-

26. A-1 to I.F-12.X-26.A-3600; compounds I.G-12.X-26.A-1 to I.G-12.X-26.A-3600).

Table 27a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-27 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-27.A-1 to I.A-2.X-27.A-3600; compounds I.B-2.X-27.A-1 to I.B-2.X-27.A- 3600; compounds I.C-2.X-27.A-1 to I.C-2.X-27.A-3600; compounds I.D-2.X-27.A-1 to I.D-2.X-

27. A-3600; compounds I.E-2.X-27.A-1 to I.E-2. X-27. A-3600; compounds I.F-2.X-27.A-1 to I.F-

2. X-27.A-3600; compounds I.G-2.X-27.A-1 to I.G-2.X-27.A-3600;

compounds I.A-3.X-27.A-1 to I.A-3.X-27.A-3600; compounds I.B-3.X-27.A-1 to I.B-3.X-27.A- 3600; compounds I.C-3.X-27.A-1 to I.C-3.X-27.A-3600; compounds I.D-3.X-27.A-1 to I.D-3.X- 27.A-3600; compounds I.E-3.X-27.A-1 to I.E-3.X-27.A-3600; compounds I.F-3.X-27.A-1 to I.F-

3. X-27.A-3600; compounds I.G-3.X-27.A-1 to I.G-3.X-27.A-3600; compounds I.A-4.X-27.A-1 to I.A-4.X-27.A-3600; compounds I.B-4.X-27.A-1 to I.B-4.X-27.A- 3600; compounds I.C-4.X-27.A-1 to I.C-4.X-27.A-3600; compounds I.D-4.X-27.A-1 to I.D-4.X- 27.A-3600; compounds I.E-4.X-27.A-1 to I.E-4.X-27.A-3600; compounds I.F-4.X-27.A-1 to I.F-

4. X-27.A-3600; compounds I.G-4.X-27.A-1 to I.G-4.X-27.A-3600;

compounds I.A-5.X-27.A-1 to I.A-5.X-27.A-3600; compounds I.B-5.X-27.A-1 to I.B-5.X-27.A- 3600; compounds I.C-5.X-27.A-1 to I.C-5.X-27.A-3600; compounds I.D-5.X-27.A-1 to I.D-5.X- 27.A-3600; compounds I.E-5.X-27.A-1 to I.E-5.X-27.A-3600; compounds I.F-5.X-27.A-1 to I.F-

5. X-27.A-3600; compounds I.G-5.X-27.A-1 to I.G-5.X-27.A-3600;

compounds I.A-6.X-27.A-1 to I.A-6.X-27.A-3600; compounds I.B-6.X-27.A-1 to I.B-6.X-27.A- 3600; compounds I.C-6.X-27.A-1 to I.C-6.X-27.A-3600; compounds I.D-6.X-27.A-1 to I.D-6.X- 27.A-3600; compounds I.E-6.X-27.A-1 to I.E-6.X-27.A-3600; compounds I.F-6.X-27.A-1 to I.F-

6. X-27.A-3600; compounds I.G-6.X-27.A-1 to I.G-6.X-27.A-3600;

compounds I.A-7.X-27.A-1 to I.A-7.X-27.A-3600; compounds I.B-7.X-27.A-1 to I.B-7.X-27.A- 3600; compounds I.C-7.X-27.A-1 to I.C-7.X-27.A-3600; compounds I.D-7.X-27.A-1 to I.D-7.X- 27.A-3600; compounds I.E-7.X-27.A-1 to I.E-7.X-27.A-3600; compounds I.F-7.X-27.A-1 to I.F-

7. X-27.A-3600; compounds I.G-7.X-27.A-1 to I.G-7.X-27.A-3600;

compounds I.A-8.X-27.A-1 to I.A-8.X-27.A-3600; compounds I.B-8.X-27.A-1 to I.B-8.X-27.A- 3600; compounds I.C-8.X-27.A-1 to I.C-8.X-27.A-3600; compounds I.D-8.X-27.A-1 to I.D-8.X- 27.A-3600; compounds I.E-8.X-27.A-1 to I.E-8.X-27.A-3600; compounds I.F-8.X-27.A-1 to I.F- 8.X-27.A-3600; compounds I.G-8.X-27.A-1 to I.G-8.X-27.A-3600;

compounds I.A-9.X-27.A-1 to I.A-9.X-27.A-3600; compounds I.B-9.X-27.A-1 to I.B-9.X-27.A- 3600; compounds I.C-9.X-27.A-1 to I.C-9.X-27.A-3600; compounds I.D-9.X-27.A-1 to I.D-9.X- 27.A-3600; compounds I.E-9.X-27.A-1 to I.E-9.X-27.A-3600; compounds I.F-9.X-27.A-1 to I.F- 9.X-27.A-3600; compounds I.G-9.X-27.A-1 to I.G-9.X-27.A-3600;

compounds I.A-10.X-27.A-1 to I.A-10.X-27.A-3600; compounds I.B-10.X-27.A-1 to I.B-10.X- 27.A-3600; compounds I.C-10.X-27.A-1 to I.C-10.X-27.A-3600; compounds I.D-10.X-27.A-1 to I.D-10.X-27.A-3600; compounds I.E-10.X-27.A-1 to I.E-10.X-27.A-3600; compounds I.F-10.X- 27.A-1 to I.F-10.X-27.A-3600; compounds I.G-10.X-27.A-1 to I.G-10.X-27.A-3600;

compounds I.A-1 1.X-27.A-1 to I.A-1 1.X-27.A-3600; compounds I.B-1 1.X-27.A-1 to I.B-1 1.X- 27.A-3600; compounds I.C-1 1.X-27.A-1 to I.C-1 1 .X-27.A-3600; compounds I.D-1 1.X-27.A-1 to I.D-1 1.X-27.A-3600; compounds I.E-1 1 .X-27.A-1 to I.E-1 1.X-27.A-3600; compounds I.F-1 1.X- 27.A-1 to I.F-1 1.X-27.A-3600; compounds I.G-1 1.X-27.A-1 to I.G-1 1.X-27.A-3600;

compounds I.A-12.X-27.A-1 to I.A-12.X-27.A-3600; compounds I.B-12.X-27.A-1 to I.B-12.X- 27.A-3600; compounds I.C-12.X-27.A-1 to I.C-12.X-27.A-3600; compounds I.D-12.X-27.A-1 to I.D-12.X-27.A-3600; compounds I.E-12.X-27.A-1 to I.E-12.X-27.A-3600; compounds I.F-12.X- 27.A-1 to I.F-12.X-27.A-3600; compounds I.G-12.X-27.A-1 to I.G-12.X-27.A-3600).

Table 28a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A-

8. I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-28 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (compounds I.A-2.X-28.A-1 to I.A-2.X-28.A-3600; compounds I.B-2.X-28.A-1 to I.B-2.X-28.A- 3600; compounds I.C-2.X-28.A-1 to I.C-2.X-28.A-3600; compounds I.D-2.X-28.A-1 to I.D-2.X- 28.A-3600; compounds I.E-2.X-28.A-1 to I.E-2.X-28.A-3600; compounds I.F-2.X-28.A-1 to I.F-

2. X-28.A-3600; compounds I.G-2.X-28.A-1 to I.G-2.X-28.A-3600;

compounds I.A-3.X-28.A-1 to I.A-3.X-28.A-3600; compounds I.B-3.X-28.A-1 to I.B-3.X-28.A- 3600; compounds I.C-3.X-28.A-1 to I.C-3.X-28.A-3600; compounds I.D-3.X-28.A-1 to I.D-3.X- 28.A-3600; compounds I.E-3.X-28.A-1 to I.E-3.X-28.A-3600; compounds I.F-3.X-28.A-1 to I.F-

3. X-28.A-3600; compounds I.G-3.X-28.A-1 to I.G-3.X-28.A-3600;

compounds I.A-4.X-28.A-1 to I.A-4.X-28.A-3600; compounds I.B-4.X-28.A-1 to I.B-4.X-28.A- 3600; compounds I.C-4.X-28.A-1 to I.C-4.X-28.A-3600; compounds I.D-4.X-28.A-1 to I.D-4.X- 28.A-3600; compounds I.E-4.X-28.A-1 to I.E-4.X-28.A-3600; compounds I.F-4.X-28.A-1 to I.F-

4. X-28.A-3600; compounds I.G-4.X-28.A-1 to I.G-4.X-28.A-3600;

compounds I.A-5.X-28.A-1 to I.A-5.X-28.A-3600; compounds I.B-5.X-28.A-1 to I.B-5.X-28.A- 3600; compounds I.C-5.X-28.A-1 to I.C-5.X-28.A-3600; compounds I.D-5.X-28.A-1 to I.D-5.X- 28.A-3600; compounds I.E-5.X-28.A-1 to I.E-5.X-28.A-3600; compounds I.F-5.X-28.A-1 to I.F- 5.X-28.A-3600; compounds I.G-5.X-28.A-1 to I.G-5.X-28.A-3600;

compounds I.A-6.X-28.A-1 to I.A-6.X-28.A-3600; compounds I.B-6.X-28.A-1 to I.B-6.X-28.A- 3600; compounds I.C-6.X-28.A-1 to I.C-6.X-28.A-3600; compounds I.D-6.X-28.A-1 to I.D-6.X- 28.A-3600; compounds I.E-6.X-28.A-1 to I.E-6.X-28.A-3600; compounds I.F-6.X-28.A-1 to I.F-

6. X-28.A-3600; compounds I.G-6.X-28.A-1 to I.G-6.X-28.A-3600;

compounds I.A-7.X-28.A-1 to I.A-7.X-28.A-3600; compounds I.B-7.X-28.A-1 to I.B-7.X-28.A- 3600; compounds I.C-7.X-28.A-1 to I.C-7.X-28.A-3600; compounds I.D-7.X-28.A-1 to I.D-7.X- 28.A-3600; compounds I.E-7.X-28.A-1 to I.E-7.X-28.A-3600; compounds I.F-7.X-28.A-1 to I.F-

7. X-28.A-3600; compounds I.G-7.X-28.A-1 to I.G-7.X-28.A-3600;

compounds I.A-8.X-28.A-1 to I.A-8.X-28.A-3600; compounds I.B-8.X-28.A-1 to I.B-8.X-28.A- 3600; compounds I.C-8.X-28.A-1 to I.C-8.X-28.A-3600; compounds I.D-8.X-28.A-1 to I.D-8.X- 28.A-3600; compounds I.E-8.X-28.A-1 to I.E-8.X-28.A-3600; compounds I.F-8.X-28.A-1 to I.F-

8. X-28.A-3600; compounds I.G-8.X-28.A-1 to I.G-8.X-28.A-3600;

compounds I.A-9.X-28.A-1 to I.A-9.X-28.A-3600; compounds I.B-9.X-28.A-1 to I.B-9.X-28.A- 3600; compounds I.C-9.X-28.A-1 to I.C-9.X-28.A-3600; compounds I.D-9.X-28.A-1 to I.D-9.X- 28.A-3600; compounds I.E-9.X-28.A-1 to I.E-9.X-28.A-3600; compounds I.F-9.X-28.A-1 to I.F-

9. X-28.A-3600; compounds I.G-9.X-28.A-1 to I.G-9.X-28.A-3600;

compounds I.A-10.X-28.A-1 to I.A-10.X-28.A-3600; compounds I.B-10.X-28.A-1 to I.B-10.X- 28.A-3600; compounds I.C-10.X-28.A-1 to I.C-10.X-28.A-3600; compounds I.D-10.X-28.A-1 to I.D-10.X-28.A-3600; compounds I.E-10.X-28.A-1 to I.E-10.X-28.A-3600; compounds I.F-10.X- 28.A-1 to I.F-10.X-28.A-3600; compounds I.G-10.X-28.A-1 to I.G-10.X-28.A-3600; compounds I.A-1 1.X-28.A-1 to I.A-1 1.X-28.A-3600; compounds I.B-1 1.X-28.A-1 to I.B-1 1.X- 28.A-3600; compounds I.C-1 1.X-28.A-1 to I.C-1 1 .X-28.A-3600; compounds I.D-1 1.X-28.A-1 to I.D-1 1.X-28.A-3600; compounds I.E-1 1 .X-28.A-1 to I.E-1 1.X-28.A-3600; compounds I.F-1 1.X- 28.A-1 to I.F-1 1.X-28.A-3600; compounds I.G-1 1.X-28.A-1 to I.G-1 1.X-28.A-3600;

compounds I.A-12.X-28.A-1 to I.A-12.X-28.A-3600; compounds I.B-12.X-28.A-1 to I.B-12.X- 28.A-3600; compounds I.C-12.X-28.A-1 to I.C-12.X-28.A-3600; compounds I.D-12.X-28.A-1 to I.D-12.X-28.A-3600; compounds I.E-12.X-28.A-1 to I.E-12.X-28.A-3600; compounds I.F-12.X-

28. A-1 to I.F-12.X-28.A-3600; compounds I.G-12.X-28.A-1 to I.G-12.X-28.A-3600).

Table 29a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10,

1. C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-29 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-29.A-1 to I.A-2.X-29.A-3600; compounds I.B-2.X-29.A-1 to I.B-2.X-29.A- 3600; compounds I.C-2.X-29.A-1 to I.C-2.X-29.A-3600; compounds I.D-2.X-29.A-1 to I.D-2.X- 29.A-3600; compounds I.E-2.X-29.A-1 to I.E-2.X-29.A-3600; compounds I.F-2.X-29.A-1 to I.F-

2. X-29.A-3600; compounds I.G-2.X-29.A-1 to I.G-2.X-29.A-3600;

compounds I.A-3.X-29.A-1 to I.A-3.X-29.A-3600; compounds I.B-3.X-29.A-1 to I.B-3.X-29.A- 3600; compounds I.C-3.X-29.A-1 to I.C-3.X-29.A-3600; compounds I.D-3.X-29.A-1 to I.D-3.X-

29. A-3600; compounds I.E-3.X-29.A-1 to I.E-3.X-29.A-3600; compounds I.F-3.X-29.A-1 to I.F- 3.X-29.A-3600; compounds I.G-3.X-29.A-1 to I.G-3.X-29.A-3600;

compounds I.A-4.X-29.A-1 to I.A-4.X-29.A-3600; compounds I.B-4.X-29.A-1 to I.B-4.X-29.A- 3600; compounds I.C-4.X-29.A-1 to I.C-4.X-29.A-3600; compounds I.D-4.X-29.A-1 to I.D-4.X- 29.A-3600; compounds I.E-4.X-29.A-1 to I.E-4.X-29.A-3600; compounds I.F-4.X-29.A-1 to I.F-

4. X-29.A-3600; compounds I.G-4.X-29.A-1 to I.G-4.X-29.A-3600;

compounds I.A-5.X-29.A-1 to I.A-5.X-29.A-3600; compounds I.B-5.X-29.A-1 to I.B-5.X-29.A- 3600; compounds I.C-5.X-29.A-1 to I.C-5.X-29.A-3600; compounds I.D-5.X-29.A-1 to I.D-5.X- 29.A-3600; compounds I.E-5.X-29.A-1 to I.E-5.X-29.A-3600; compounds I.F-5.X-29.A-1 to I.F-

5. X-29.A-3600; compounds I.G-5.X-29.A-1 to I.G-5.X-29.A-3600;

compounds I.A-6.X-29.A-1 to I.A-6.X-29.A-3600; compounds I.B-6.X-29.A-1 to I.B-6.X-29.A- 3600; compounds I.C-6.X-29.A-1 to I.C-6.X-29.A-3600; compounds I.D-6.X-29.A-1 to I.D-6.X- 29.A-3600; compounds I.E-6.X-29.A-1 to I.E-6.X-29.A-3600; compounds I.F-6.X-29.A-1 to I.F-

6. X-29.A-3600; compounds I.G-6.X-29.A-1 to I.G-6.X-29.A-3600;

compounds I.A-7.X-29.A-1 to I.A-7.X-29.A-3600; compounds I.B-7.X-29.A-1 to I.B-7.X-29.A- 3600; compounds I.C-7.X-29.A-1 to I.C-7.X-29.A-3600; compounds I.D-7.X-29.A-1 to I.D-7.X- 29.A-3600; compounds I.E-7.X-29.A-1 to I.E-7.X-29.A-3600; compounds I.F-7.X-29.A-1 to I.F-

7. X-29.A-3600; compounds I.G-7.X-29.A-1 to I.G-7.X-29.A-3600; compounds I.A-8.X-29.A-1 to I.A-8.X-29.A-3600; compounds I.B-8.X-29.A-1 to I.B-8.X-29.A- 3600; compounds I.C-8.X-29.A-1 to I.C-8.X-29.A-3600; compounds I.D-8.X-29.A-1 to I.D-8.X- 29.A-3600; compounds I.E-8.X-29.A-1 to I.E-8.X-29.A-3600; compounds I.F-8.X-29.A-1 to I.F-

8. X-29.A-3600; compounds I.G-8.X-29.A-1 to I.G-8.X-29.A-3600;

compounds I.A-9.X-29.A-1 to I.A-9.X-29.A-3600; compounds I.B-9.X-29.A-1 to I.B-9.X-29.A- 3600; compounds I.C-9.X-29.A-1 to I.C-9.X-29.A-3600; compounds I.D-9.X-29.A-1 to I.D-9.X- 29.A-3600; compounds I.E-9.X-29.A-1 to I.E-9.X-29.A-3600; compounds I.F-9.X-29.A-1 to I.F-

9. X-29.A-3600; compounds I.G-9.X-29.A-1 to I.G-9.X-29.A-3600;

compounds I.A-10.X-29.A-1 to I.A-10.X-29.A-3600; compounds I.B-10.X-29.A-1 to I.B-10.X- 29.A-3600; compounds I.C-10.X-29.A-1 to I.C-10.X-29.A-3600; compounds I.D-10.X-29.A-1 to I.D-10.X-29.A-3600; compounds I.E-10.X-29.A-1 to I.E-10.X-29.A-3600; compounds I.F-10.X- 29.A-1 to I.F-10.X-29.A-3600; compounds I.G-10.X-29.A-1 to I.G-10.X-29.A-3600;

compounds I.A-1 1.X-29.A-1 to I.A-1 1.X-29.A-3600; compounds I.B-1 1.X-29.A-1 to I.B-1 1.X- 29.A-3600; compounds I.C-1 1.X-29.A-1 to I.C-1 1 .X-29.A-3600; compounds I.D-1 1.X-29.A-1 to I.D-1 1.X-29.A-3600; compounds I.E-1 1 .X-29.A-1 to I.E-1 1.X-29.A-3600; compounds I.F-1 1.X- 29.A-1 to I.F-1 1.X-29.A-3600; compounds I.G-1 1.X-29.A-1 to I.G-1 1.X-29.A-3600;

compounds I.A-12.X-29.A-1 to I.A-12.X-29.A-3600; compounds I.B-12.X-29.A-1 to I.B-12.X-

29. A-3600; compounds I.C-12.X-29.A-1 to I.C-12.X-29.A-3600; compounds I.D-12.X-29.A-1 to I.D-12.X-29.A-3600; compounds I.E-12.X-29.A-1 to I.E-12.X-29.A-3600; compounds I.F-12.X- 29.A-1 to I.F-12.X-29.A-3600; compounds I.G-12.X-29.A-1 to I.G-12.X-29.A-3600).

Table 30a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-30 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (compounds I.A-2.X-30.A-1 to I.A-2.X-30.A-3600; compounds I.B-2.X-30.A-1 to I.B-2.X-30.A- 3600; compounds I.C-2.X-30.A-1 to I.C-2.X-30.A-3600; compounds I.D-2.X-30.A-1 to I.D-2.X-

30. A-3600; compounds I.E-2.X-30.A-1 to I.E-2.X-30.A-3600; compounds I.F-2.X-30.A-1 to I.F-

2. X-30.A-3600; compounds I.G-2.X-30.A-1 to I.G-2.X-30.A-3600;

compounds I.A-3.X-30.A-1 to I.A-3.X-30.A-3600; compounds I.B-3.X-30.A-1 to I.B-3.X-30.A- 3600; compounds I.C-3.X-30.A-1 to I.C-3.X-30.A-3600; compounds I.D-3.X-30.A-1 to I.D-3.X- 30.A-3600; compounds I.E-3.X-30.A-1 to I.E-3.X-30.A-3600; compounds I.F-3.X-30.A-1 to I.F-

3. X-30.A-3600; compounds I.G-3.X-30.A-1 to I.G-3.X-30.A-3600;

compounds I.A-4.X-30.A-1 to I.A-4.X-30.A-3600; compounds I.B-4.X-30.A-1 to I.B-4.X-30.A- 3600; compounds I.C-4.X-30.A-1 to I.C-4.X-30.A-3600; compounds I.D-4.X-30.A-1 to I.D-4.X- 30.A-3600; compounds I.E-4.X-30.A-1 to I.E-4.X-30.A-3600; compounds I.F-4.X-30.A-1 to I.F-

4. X-30.A-3600; compounds I.G-4.X-30.A-1 to I.G-4.X-30.A-3600; compounds I.A-5.X-30.A-1 to I.A-5.X-30.A-3600; compounds I.B-5.X-30.A-1 to I.B-5.X-30.A- 3600; compounds I.C-5.X-30.A-1 to I.C-5.X-30.A-3600; compounds I.D-5.X-30.A-1 to I.D-5.X- 30.A-3600; compounds I.E-5.X-30.A-1 to I.E-5.X-30.A-3600; compounds I.F-5.X-30.A-1 to I.F-

5. X-30.A-3600; compounds I.G-5.X-30.A-1 to I.G-5.X-30.A-3600;

compounds I.A-6.X-30.A-1 to I.A-6.X-30.A-3600; compounds I.B-6.X-30.A-1 to I.B-6.X-30.A- 3600; compounds I.C-6.X-30.A-1 to I.C-6.X-30.A-3600; compounds I.D-6.X-30.A-1 to I.D-6.X- 30.A-3600; compounds I.E-6.X-30.A-1 to I.E-6.X-30.A-3600; compounds I.F-6.X-30.A-1 to I.F-

6. X-30.A-3600; compounds I.G-6.X-30.A-1 to I.G-6.X-30.A-3600;

compounds I.A-7.X-30.A-1 to I.A-7.X-30.A-3600; compounds I.B-7.X-30.A-1 to I.B-7.X-30.A- 3600; compounds I.C-7.X-30.A-1 to I.C-7.X-30.A-3600; compounds I.D-7.X-30.A-1 to I.D-7.X- 30.A-3600; compounds I.E-7.X-30.A-1 to I.E-7.X-30.A-3600; compounds I.F-7.X-30.A-1 to I.F-

7. X-30.A-3600; compounds I.G-7.X-30.A-1 to I.G-7.X-30.A-3600;

compounds I.A-8.X-30.A-1 to I.A-8.X-30.A-3600; compounds I.B-8.X-30.A-1 to I.B-8.X-30.A- 3600; compounds I.C-8.X-30.A-1 to I.C-8.X-30.A-3600; compounds I.D-8.X-30.A-1 to I.D-8.X- 30.A-3600; compounds I.E-8.X-30.A-1 to I.E-8.X-30.A-3600; compounds I.F-8.X-30.A-1 to I.F-

8. X-30.A-3600; compounds I.G-8.X-30.A-1 to I.G-8.X-30.A-3600;

compounds I.A-9.X-30.A-1 to I.A-9.X-30.A-3600; compounds I.B-9.X-30.A-1 to I.B-9.X-30.A- 3600; compounds I.C-9.X-30.A-1 to I.C-9.X-30.A-3600; compounds I.D-9.X-30.A-1 to I.D-9.X- 30.A-3600; compounds I.E-9.X-30.A-1 to I.E-9.X-30.A-3600; compounds I.F-9.X-30.A-1 to I.F- 9.X-30.A-3600; compounds I.G-9.X-30.A-1 to I.G-9.X-30.A-3600;

compounds I.A-10.X-30.A-1 to I.A-10.X-30.A-3600; compounds I.B-10.X-30.A-1 to I.B-10.X- 30.A-3600; compounds I.C-10.X-30.A-1 to I.C-10.X-30.A-3600; compounds I.D-10.X-30.A-1 to I.D-10.X-30.A-3600; compounds I.E-10.X-30.A-1 to I.E-10.X-30.A-3600; compounds I.F-10.X- 30.A-1 to I.F-10.X-30.A-3600; compounds I.G-10.X-30.A-1 to I.G-10.X-30.A-3600;

compounds I.A-1 1.X-30.A-1 to I.A-1 1.X-30.A-3600; compounds I.B-1 1.X-30.A-1 to I.B-1 1.X- 30.A-3600; compounds I.C-1 1.X-30.A-1 to I.C-1 1 .X-30.A-3600; compounds I.D-1 1.X-30.A-1 to I.D-1 1.X-30.A-3600; compounds I.E-1 1 .X-30.A-1 to I.E-1 1.X-30.A-3600; compounds I.F-1 1.X- 30.A-1 to I.F-1 1.X-30.A-3600; compounds I.G-1 1.X-30.A-1 to I.G-1 1.X-30.A-3600;

compounds I.A-12.X-30.A-1 to I.A-12.X-30.A-3600; compounds I.B-12.X-30.A-1 to I.B-12.X- 30.A-3600; compounds I.C-12.X-30.A-1 to I.C-12.X-30.A-3600; compounds I.D-12.X-30.A-1 to I.D-12.X-30.A-3600; compounds I.E-12.X-30.A-1 to I.E-12.X-30.A-3600; compounds I.F-12.X- 30.A-1 to I.F-12.X-30.A-3600; compounds I.G-12.X-30.A-1 to I.G-12.X-30.A-3600).

Table 31 a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-31 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (

compounds I.A-2.X-31.A-1 to I.A-2.X-31 .A-3600; compounds I.B-2.X-31 .A-1 to I.B-2.X-31 .A- 3600; compounds I.C-2.X-31.A-1 to I. C-2.X-31. A-3600; compounds I.D-2.X-31.A-1 to I.D-2.X- 31. A-3600; compounds I.E-2.X-31.A-1 to I. E-2.X-31. A-3600; compounds I.F-2.X-31.A-1 to I.F- 2.X-31 .A-3600; compounds I.G-2.X-31 .A-1 to I.G-2.X-31 .A-3600;

compounds I.A-3.X-31.A-1 to I. A-3.X-31 .A-3600; compounds I.B-3.X-31 .A-1 to I.B-3.X-31 .A- 3600; compounds I.C-3.X-31.A-1 to I. C-3.X-31. A-3600; compounds I.D-3.X-31.A-1 to I.D-3.X- 31. A-3600; compounds I.E-3.X-31.A-1 to I. E-3.X-31. A-3600; compounds I.F-3.X-31.A-1 to I.F-

3. X-31 . A-3600; compounds I.G-3.X-31 .A-1 to I. G-3.X-31 .A-3600;

compounds I.A-4.X-31.A-1 to I. A-4.X-31 .A-3600; compounds I.B-4.X-31 .A-1 to I.B-4.X-31 .A- 3600; compounds I.C-4.X-31.A-1 to I. C-4.X-31. A-3600; compounds I.D-4.X-31.A-1 to I.D-4.X- 31. A-3600; compounds I.E-4.X-31.A-1 to I. E-4.X-31. A-3600; compounds I.F-4.X-31.A-1 to I.F-

4. X-31 . A-3600; compounds I.G-4.X-31 .A-1 to I. G-4.X-31 .A-3600;

compounds I.A-5.X-31.A-1 to I. A-5.X-31 .A-3600; compounds I.B-5.X-31 .A-1 to I.B-5.X-31 .A- 3600; compounds I.C-5.X-31.A-1 to I. C-5.X-31. A-3600; compounds I.D-5.X-31.A-1 to I.D-5.X- 31. A-3600; compounds I.E-5.X-31.A-1 to I. E-5.X-31. A-3600; compounds I.F-5.X-31.A-1 to I.F-

5. X-31 . A-3600; compounds I.G-5.X-31 .A-1 to I. G-5.X-31 .A-3600;

compounds I.A-6.X-31.A-1 to I. A-6.X-31 .A-3600; compounds I.B-6.X-31 .A-1 to I.B-6.X-31 .A- 3600; compounds I.C-6.X-31.A-1 to I. C-6.X-31. A-3600; compounds I.D-6.X-31.A-1 to I.D-6.X- 31. A-3600; compounds I.E-6.X-31.A-1 to I. E-6.X-31. A-3600; compounds I.F-6.X-31.A-1 to I.F-

6. X-31 . A-3600; compounds I.G-6.X-31 .A-1 to I. G-6.X-31 .A-3600;

compounds I.A-7.X-31.A-1 to I. A-7.X-31 .A-3600; compounds I.B-7.X-31 .A-1 to I.B-7.X-31 .A- 3600; compounds I.C-7.X-31.A-1 to I. C-7.X-31. A-3600; compounds I.D-7.X-31.A-1 to I.D-7.X- 31. A-3600; compounds I.E-7.X-31.A-1 to I. E-7.X-31. A-3600; compounds I.F-7.X-31.A-1 to I.F- 7.X-31 .A-3600; compounds I.G-7.X-31 .A-1 to I.G-7.X-31 .A-3600;

compounds I.A-8.X-31.A-1 to I. A-8.X-31 .A-3600; compounds I.B-8.X-31 .A-1 to I.B-8.X-31 .A- 3600; compounds I.C-8.X-31.A-1 to I. C-8.X-31. A-3600; compounds I.D-8.X-31.A-1 to I.D-8.X- 31. A-3600; compounds I.E-8.X-31.A-1 to I. E-8.X-31. A-3600; compounds I.F-8.X-31.A-1 to I.F-

8. X-31 . A-3600; compounds I.G-8.X-31 .A-1 to I. G-8.X-31 .A-3600;

compounds I.A-9.X-31.A-1 to I. A-9.X-31 .A-3600; compounds I.B-9.X-31 .A-1 to I.B-9.X-31 .A- 3600; compounds I.C-9.X-31.A-1 to I. C-9.X-31. A-3600; compounds I.D-9.X-31.A-1 to I.D-9.X- 31. A-3600; compounds I.E-9.X-31.A-1 to I. E-9.X-31. A-3600; compounds I.F-9.X-31.A-1 to I.F-

9. X-31 . A-3600; compounds I.G-9.X-31 .A-1 to I. G-9.X-31 .A-3600;

compounds I.A-10.X-31.A-1 to I.A-10.X-31. A-3600; compounds I.B-10.X-31.A-1 to I.B-10.X- 31.A-3600; compounds I.C-10.X-31. A-1 to I.C-10.X-31. A-3600; compounds I.D-10.X-31.A-1 to I. D-10.X-31. A-3600; compounds I.E-10.X-31.A-1 to I.E-10.X-31 .A-3600; compounds I.F-10.X- 31. A-1 to I. F-10.X-31. A-3600; compounds I.G-10.X-31.A-1 to I.G-10.X-31. A-3600;

compounds I.A-1 1.X-31.A-1 to I .A-1 1.X-31. A-3600; compounds I.B-1 1.X-31.A-1 to I.B-1 1.X- 31. A-3600; compounds I.C-1 1.X-31. A-1 to I. C-1 1 .X-31. A-3600; compounds I.D-1 1.X-31. A-1 to I.D-1 1.X-31. A-3600; compounds I.E-1 1 .X-31.A-1 to I. E-1 1.X-31 . A-3600; compounds I.F-1 1.X- 31 . A-1 to I. F-1 1.X-31. A-3600; compounds I.G-1 1.X-31.A-1 to I.G-1 1.X-31. A-3600; compounds I.A-12.X-31.A-1 to I.A-12.X-31.A-3600; compounds I.B-12.X-31.A-1 to I.B-12.X- 31.A-3600; compounds I.C-12.X-31.A-1 to I.C-12.X-31.A-3600; compounds I.D-12.X-31.A-1 to I.D-12.X-31.A-3600; compounds I.E-12.X-31.A-1 to I.E-12.X-31 .A-3600; compounds I.F-12.X-

31. A-1 to I. F-12.X-31. A-3600; compounds I.G-12.X-31.A-1 to I.G-12.X-31. A-3600).

Table 32a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-32 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-32.A-1 to I.A-2.X-32.A-3600; compounds I.B-2.X-32.A-1 to I.B-2.X-32.A- 3600; compounds I.C-2.X-32.A-1 to I.C-2.X-32.A-3600; compounds I.D-2.X-32.A-1 to I.D-2.X-

32. A-3600; compounds I.E-2.X-32.A-1 to I.E-2.X-32.A-3600; compounds I.F-2.X-32.A-1 to I.F-

2. X-32.A-3600; compounds I.G-2.X-32.A-1 to I.G-2.X-32.A-3600;

compounds I.A-3.X-32.A-1 to I.A-3.X-32.A-3600; compounds I.B-3.X-32.A-1 to I.B-3.X-32.A- 3600; compounds I.C-3.X-32.A-1 to I.C-3.X-32.A-3600; compounds I.D-3.X-32.A-1 to I.D-3.X- 32.A-3600; compounds I.E-3.X-32.A-1 to I.E-3.X-32.A-3600; compounds I.F-3.X-32.A-1 to I.F-

3. X-32.A-3600; compounds I.G-3.X-32.A-1 to I.G-3.X-32.A-3600;

compounds I.A-4.X-32.A-1 to I.A-4.X-32.A-3600; compounds I.B-4.X-32.A-1 to I.B-4.X-32.A- 3600; compounds I.C-4.X-32.A-1 to I.C-4.X-32.A-3600; compounds I.D-4.X-32.A-1 to I.D-4.X- 32.A-3600; compounds I.E-4.X-32.A-1 to I.E-4.X-32.A-3600; compounds I.F-4.X-32.A-1 to I.F- 4.X-32.A-3600; compounds I.G-4.X-32.A-1 to I.G-4.X-32.A-3600;

compounds I.A-5.X-32.A-1 to I.A-5.X-32.A-3600; compounds I.B-5.X-32.A-1 to I.B-5.X-32.A- 3600; compounds I.C-5.X-32.A-1 to I.C-5.X-32.A-3600; compounds I.D-5.X-32.A-1 to I.D-5.X- 32.A-3600; compounds I.E-5.X-32.A-1 to I.E-5.X-32.A-3600; compounds I.F-5.X-32.A-1 to I.F-

5. X-32.A-3600; compounds I.G-5.X-32.A-1 to I.G-5.X-32.A-3600;

compounds I.A-6.X-32.A-1 to I.A-6.X-32.A-3600; compounds I.B-6.X-32.A-1 to I.B-6.X-32.A- 3600; compounds I.C-6.X-32.A-1 to I.C-6.X-32.A-3600; compounds I.D-6.X-32.A-1 to I.D-6.X- 32.A-3600; compounds I.E-6.X-32.A-1 to I.E-6.X-32.A-3600; compounds I.F-6.X-32.A-1 to I.F-

6. X-32.A-3600; compounds I.G-6.X-32.A-1 to I.G-6.X-32.A-3600;

compounds I.A-7.X-32.A-1 to I.A-7.X-32.A-3600; compounds I.B-7.X-32.A-1 to I.B-7.X-32.A- 3600; compounds I.C-7.X-32.A-1 to I.C-7.X-32.A-3600; compounds I.D-7.X-32.A-1 to I.D-7.X- 32.A-3600; compounds I.E-7.X-32.A-1 to I.E-7.X-32.A-3600; compounds I.F-7.X-32.A-1 to I.F-

7. X-32.A-3600; compounds I.G-7.X-32.A-1 to I.G-7.X-32.A-3600;

compounds I.A-8.X-32.A-1 to I.A-8.X-32.A-3600; compounds I.B-8.X-32.A-1 to I.B-8.X-32.A- 3600; compounds I.C-8.X-32.A-1 to I.C-8.X-32.A-3600; compounds I.D-8.X-32.A-1 to I.D-8.X- 32.A-3600; compounds I.E-8.X-32.A-1 to I.E-8.X-32.A-3600; compounds I.F-8.X-32.A-1 to I.F-

8. X-32.A-3600; compounds I.G-8.X-32.A-1 to I.G-8.X-32.A-3600; compounds I.A-9.X-32.A-1 to I.A-9.X-32.A-3600; compounds I.B-9.X-32.A-1 to I.B-9.X-32.A- 3600; compounds I.C-9.X-32.A-1 to I.C-9.X-32.A-3600; compounds I.D-9.X-32.A-1 to I.D-9.X- 32.A-3600; compounds I.E-9.X-32.A-1 to I.E-9.X-32.A-3600; compounds I.F-9.X-32.A-1 to I.F- 9.X-32.A-3600; compounds I.G-9.X-32.A-1 to I.G-9.X-32.A-3600;

compounds I.A-10.X-32.A-1 to I.A-10.X-32.A-3600; compounds I.B-10.X-32.A-1 to I.B-10.X- 32.A-3600; compounds I.C-10.X-32.A-1 to I.C-10.X-32.A-3600; compounds I.D-10.X-32.A-1 to I.D-10.X-32.A-3600; compounds I.E-10.X-32.A-1 to I.E-10.X-32.A-3600; compounds I.F-10.X- 32.A-1 to I.F-10.X-32.A-3600; compounds I.G-10.X-32.A-1 to I.G-10.X-32.A-3600;

compounds I.A-1 1.X-32.A-1 to I.A-1 1.X-32.A-3600; compounds I.B-1 1.X-32.A-1 to I.B-1 1.X- 32.A-3600; compounds I.C-1 1.X-32.A-1 to I.C-1 1 .X-32.A-3600; compounds I.D-1 1.X-32.A-1 to I.D-1 1.X-32.A-3600; compounds I.E-1 1 .X-32.A-1 to I.E-1 1.X-32.A-3600; compounds I.F-1 1.X- 32.A-1 to I.F-1 1.X-32.A-3600; compounds I.G-1 1.X-32.A-1 to I.G-1 1.X-32.A-3600;

compounds I.A-12.X-32.A-1 to I.A-12.X-32.A-3600; compounds I.B-12.X-32.A-1 to I.B-12.X- 32.A-3600; compounds I.C-12.X-32.A-1 to I.C-12.X-32.A-3600; compounds I.D-12.X-32.A-1 to I.D-12.X-32.A-3600; compounds I.E-12.X-32.A-1 to I.E-12.X-32.A-3600; compounds I.F-12.X-

32. A-1 to I.F-12.X-32.A-3600; compounds I.G-12.X-32.A-1 to I.G-12.X-32.A-3600).

Table 33a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-33 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-33.A-1 to I.A-2.X-33.A-3600; compounds I.B-2.X-33.A-1 to I.B-2.X-33.A- 3600; compounds I.C-2.X-33.A-1 to I.C-2.X-33.A-3600; compounds I.D-2.X-33.A-1 to I.D-2.X-

33. A-3600; compounds I.E-2.X-33.A-1 to I.E-2.X-33.A-3600; compounds I.F-2.X-33.A-1 to I.F-

2. X-33.A-3600; compounds I.G-2.X-33.A-1 to I.G-2.X-33.A-3600;

compounds I.A-3.X-33.A-1 to I.A-3.X-33.A-3600; compounds I.B-3.X-33.A-1 to I.B-3.X-33.A- 3600; compounds I.C-3.X-33.A-1 to I.C-3.X-33.A-3600; compounds I.D-3.X-33.A-1 to I.D-3.X- 33.A-3600; compounds I.E-3.X-33.A-1 to I.E-3.X-33.A-3600; compounds I.F-3.X-33.A-1 to I.F-

3. X-33.A-3600; compounds I.G-3.X-33.A-1 to I.G-3.X-33.A-3600;

compounds I.A-4.X-33.A-1 to I.A-4.X-33.A-3600; compounds I.B-4.X-33.A-1 to I.B-4.X-33.A- 3600; compounds I.C-4.X-33.A-1 to I.C-4.X-33.A-3600; compounds I.D-4.X-33.A-1 to I.D-4.X- 33.A-3600; compounds I.E-4.X-33.A-1 to I.E-4.X-33.A-3600; compounds I.F-4.X-33.A-1 to I.F-

4. X-33.A-3600; compounds I.G-4.X-33.A-1 to I.G-4.X-33.A-3600;

compounds I.A-5.X-33.A-1 to I.A-5.X-33.A-3600; compounds I.B-5.X-33.A-1 to I.B-5.X-33.A- 3600; compounds I.C-5.X-33.A-1 to I.C-5.X-33.A-3600; compounds I.D-5.X-33.A-1 to I.D-5.X- 33.A-3600; compounds I.E-5.X-33.A-1 to I.E-5.X-33.A-3600; compounds I.F-5.X-33.A-1 to I.F-

5. X-33.A-3600; compounds I.G-5.X-33.A-1 to I.G-5.X-33.A-3600; compounds I.A-6.X-33.A-1 to I.A-6.X-33.A-3600; compounds I.B-6.X-33.A-1 to I.B-6.X-33.A- 3600; compounds I.C-6.X-33.A-1 to I.C-6.X-33.A-3600; compounds I.D-6.X-33.A-1 to I.D-6.X- 33.A-3600; compounds I.E-6.X-33.A-1 to I.E-6.X-33.A-3600; compounds I.F-6.X-33.A-1 to I.F-

6. X-33.A-3600; compounds I.G-6.X-33.A-1 to I.G-6.X-33.A-3600;

compounds I.A-7.X-33.A-1 to I.A-7.X-33.A-3600; compounds I.B-7.X-33.A-1 to I.B-7.X-33.A- 3600; compounds I.C-7.X-33.A-1 to I.C-7.X-33.A-3600; compounds I.D-7.X-33.A-1 to I.D-7.X- 33.A-3600; compounds I.E-7.X-33.A-1 to I.E-7.X-33.A-3600; compounds I.F-7.X-33.A-1 to I.F-

7. X-33.A-3600; compounds I.G-7.X-33.A-1 to I.G-7.X-33.A-3600;

compounds I.A-8.X-33.A-1 to I.A-8.X-33.A-3600; compounds I.B-8.X-33.A-1 to I.B-8.X-33.A- 3600; compounds I.C-8.X-33.A-1 to I.C-8.X-33.A-3600; compounds I.D-8.X-33.A-1 to I.D-8.X- 33.A-3600; compounds I.E-8.X-33.A-1 to I.E-8.X-33.A-3600; compounds I.F-8.X-33.A-1 to I.F-

8. X-33.A-3600; compounds I.G-8.X-33.A-1 to I.G-8.X-33.A-3600;

compounds I.A-9.X-33.A-1 to I.A-9.X-33.A-3600; compounds I.B-9.X-33.A-1 to I.B-9.X-33.A- 3600; compounds I.C-9.X-33.A-1 to I.C-9.X-33.A-3600; compounds I.D-9.X-33.A-1 to I.D-9.X- 33.A-3600; compounds I.E-9.X-33.A-1 to I.E-9.X-33.A-3600; compounds I.F-9.X-33.A-1 to I.F-

9. X-33.A-3600; compounds I.G-9.X-33.A-1 to I.G-9.X-33.A-3600;

compounds I.A-10.X-33.A-1 to I.A-10.X-33.A-3600; compounds I.B-10.X-33.A-1 to I.B-10.X- 33.A-3600; compounds I.C-10.X-33.A-1 to I.C-10.X-33.A-3600; compounds I.D-10.X-33.A-1 to I.D-10.X-33.A-3600; compounds I.E-10.X-33.A-1 to I.E-10.X-33.A-3600; compounds I.F-10.X- 33.A-1 to I.F-10.X-33.A-3600; compounds I.G-10.X-33.A-1 to I.G-10.X-33.A-3600;

compounds I.A-1 1.X-33.A-1 to I.A-1 1.X-33.A-3600; compounds I.B-1 1.X-33.A-1 to I.B-1 1.X- 33.A-3600; compounds I.C-1 1.X-33.A-1 to I.C-1 1 .X-33.A-3600; compounds I.D-1 1.X-33.A-1 to I.D-1 1.X-33.A-3600; compounds I.E-1 1 .X-33.A-1 to I.E-1 1.X-33.A-3600; compounds I.F-1 1.X- 33.A-1 to I.F-1 1.X-33.A-3600; compounds I.G-1 1.X-33.A-1 to I.G-1 1.X-33.A-3600;

compounds I.A-12.X-33.A-1 to I.A-12.X-33.A-3600; compounds I.B-12.X-33.A-1 to I.B-12.X- 33.A-3600; compounds I.C-12.X-33.A-1 to I.C-12.X-33.A-3600; compounds I.D-12.X-33.A-1 to I.D-12.X-33.A-3600; compounds I.E-12.X-33.A-1 to I.E-12.X-33.A-3600; compounds I.F-12.X- 33.A-1 to I.F-12.X-33.A-3600; compounds I.G-12.X-33.A-1 to I.G-12.X-33.A-3600).

Table 34a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10,

1. C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-34 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-34.A-1 to I.A-2.X-34.A-3600; compounds I.B-2.X-34.A-1 to I.B-2.X-34.A- 3600; compounds I.C-2.X-34.A-1 to I.C-2.X-34.A-3600; compounds I.D-2.X-34.A-1 to I.D-2.X- 34.A-3600; compounds I.E-2.X-34.A-1 to I.E-2.X-34.A-3600; compounds I.F-2.X-34.A-1 to I.F-

2. X-34.A-3600; compounds I.G-2.X-34.A-1 to I.G-2.X-34.A-3600; compounds I.A-3.X-34.A-1 to I.A-3.X-34.A-3600; compounds I.B-3.X-34.A-1 to I.B-3.X-34.A- 3600; compounds I.C-3.X-34.A-1 to I.C-3.X-34.A-3600; compounds I.D-3.X-34.A-1 to I.D-3.X- 34.A-3600; compounds I.E-3.X-34.A-1 to I.E-3.X-34.A-3600; compounds I.F-3.X-34.A-1 to I.F-

3. X-34.A-3600; compounds I.G-3.X-34.A-1 to I.G-3.X-34.A-3600;

compounds I.A-4.X-34.A-1 to I.A-4.X-34.A-3600; compounds I.B-4.X-34.A-1 to I.B-4.X-34.A- 3600; compounds I.C-4.X-34.A-1 to I.C-4.X-34.A-3600; compounds I.D-4.X-34.A-1 to I.D-4.X- 34.A-3600; compounds I.E-4.X-34.A-1 to I.E-4.X-34.A-3600; compounds I.F-4.X-34.A-1 to I.F-

4. X-34.A-3600; compounds I.G-4.X-34.A-1 to I.G-4.X-34.A-3600;

compounds I.A-5.X-34.A-1 to I.A-5.X-34.A-3600; compounds I.B-5.X-34.A-1 to I.B-5.X-34.A- 3600; compounds I.C-5.X-34.A-1 to I.C-5.X-34.A-3600; compounds I.D-5.X-34.A-1 to I.D-5.X- 34.A-3600; compounds I.E-5.X-34.A-1 to I.E-5.X-34.A-3600; compounds I.F-5.X-34.A-1 to I.F-

5. X-34.A-3600; compounds I.G-5.X-34.A-1 to I.G-5.X-34.A-3600;

compounds I.A-6.X-34.A-1 to I.A-6.X-34.A-3600; compounds I.B-6.X-34.A-1 to I.B-6.X-34.A- 3600; compounds I.C-6.X-34.A-1 to I.C-6.X-34.A-3600; compounds I.D-6.X-34.A-1 to I.D-6.X- 34.A-3600; compounds I.E-6.X-34.A-1 to I.E-6.X-34.A-3600; compounds I.F-6.X-34.A-1 to I.F-

6. X-34.A-3600; compounds I.G-6.X-34.A-1 to I.G-6.X-34.A-3600;

compounds I.A-7.X-34.A-1 to I.A-7.X-34.A-3600; compounds I.B-7.X-34.A-1 to I.B-7.X-34.A- 3600; compounds I.C-7.X-34.A-1 to I.C-7.X-34.A-3600; compounds I.D-7.X-34.A-1 to I.D-7.X- 34.A-3600; compounds I.E-7.X-34.A-1 to I.E-7.X-34.A-3600; compounds I.F-7.X-34.A-1 to I.F- 7.X-34.A-3600; compounds I.G-7.X-34.A-1 to I.G-7.X-34.A-3600;

compounds I.A-8.X-34.A-1 to I.A-8.X-34.A-3600; compounds I.B-8.X-34.A-1 to I.B-8.X-34.A- 3600; compounds I.C-8.X-34.A-1 to I.C-8.X-34.A-3600; compounds I.D-8.X-34.A-1 to I.D-8.X- 34.A-3600; compounds I.E-8.X-34.A-1 to I.E-8.X-34.A-3600; compounds I.F-8.X-34.A-1 to I.F-

8. X-34.A-3600; compounds I.G-8.X-34.A-1 to I.G-8.X-34.A-3600;

compounds I.A-9.X-34.A-1 to I.A-9.X-34.A-3600; compounds I.B-9.X-34.A-1 to I.B-9.X-34.A- 3600; compounds I.C-9.X-34.A-1 to I.C-9.X-34.A-3600; compounds I.D-9.X-34.A-1 to I.D-9.X- 34.A-3600; compounds I.E-9.X-34.A-1 to I.E-9.X-34.A-3600; compounds I.F-9.X-34.A-1 to I.F-

9. X-34.A-3600; compounds I.G-9.X-34.A-1 to I.G-9.X-34.A-3600;

compounds I.A-10.X-34.A-1 to I.A-10.X-34.A-3600; compounds I.B-10.X-34.A-1 to I.B-10.X- 34.A-3600; compounds I.C-10.X-34.A-1 to I.C-10.X-34.A-3600; compounds I.D-10.X-34.A-1 to I.D-10.X-34.A-3600; compounds I.E-10.X-34.A-1 to I.E-10.X-34.A-3600; compounds I.F-10.X- 34.A-1 to I.F-10.X-34.A-3600; compounds I.G-10.X-34.A-1 to I.G-10.X-34.A-3600;

compounds I.A-1 1.X-34.A-1 to I.A-1 1.X-34.A-3600; compounds I.B-1 1.X-34.A-1 to I.B-1 1.X- 34.A-3600; compounds I.C-1 1.X-34.A-1 to I.C-1 1 .X-34.A-3600; compounds I.D-1 1.X-34.A-1 to I.D-1 1.X-34.A-3600; compounds I.E-1 1 .X-34.A-1 to I.E-1 1.X-34.A-3600; compounds I.F-1 1.X- 34.A-1 to I.F-1 1 .X-34.A-3600; compounds I.G-1 1.X-34.A-1 to I.G-1 1.X-34.A-3600;

compounds I.A-12.X-34.A-1 to I.A-12.X-34.A-3600; compounds I.B-12.X-34.A-1 to I.B-12.X- 34.A-3600; compounds I.C-12.X-34.A-1 to I.C-12.X-34.A-3600; compounds I.D-12.X-34.A-1 to I.D-12.X-34.A-3600; compounds I.E-12.X-34.A-1 to I.E-12.X-34.A-3600; compounds I.F-12.X- 34.A-1 to I.F-12.X-34.A-3600; compounds I.G-12.X-34.A-1 to I.G-12.X-34.A-3600).

Table 35a Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-35 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(

compounds I.A-2.X-35.A-1 to I.A-2.X-35.A-3600; compounds I.B-2.X-35.A-1 to I.B-2.X-35.A- 3600; compounds I.C-2.X-35.A-1 to I.C-2.X-35.A-3600; compounds I.D-2.X-35.A-1 to I.D-2.X- 35.A-3600; compounds I.E-2.X-35.A-1 to I.E-2.X-35.A-3600; compounds I.F-2.X-35.A-1 to I.F-

2. X-35.A-3600; compounds I.G-2.X-35.A-1 to I.G-2.X-35.A-3600;

compounds I.A-3.X-35.A-1 to I.A-3.X-35.A-3600; compounds I.B-3.X-35.A-1 to I.B-3.X-35.A- 3600; compounds I.C-3.X-35.A-1 to I.C-3.X-35.A-3600; compounds I.D-3.X-35.A-1 to I.D-3.X- 35.A-3600; compounds I.E-3.X-35.A-1 to I.E-3.X-35.A-3600; compounds I.F-3.X-35.A-1 to I.F-

3. X-35.A-3600; compounds I.G-3.X-35.A-1 to I.G-3.X-35.A-3600;

compounds I.A-4.X-35.A-1 to I.A-4.X-35.A-3600; compounds I.B-4.X-35.A-1 to I.B-4.X-35.A- 3600; compounds I.C-4.X-35.A-1 to I.C-4.X-35.A-3600; compounds I.D-4.X-35.A-1 to I.D-4.X- 35.A-3600; compounds I.E-4.X-35.A-1 to I.E-4.X-35.A-3600; compounds I.F-4.X-35.A-1 to I.F-

4. X-35.A-3600; compounds I.G-4.X-35.A-1 to I.G-4.X-35.A-3600;

compounds I.A-5.X-35.A-1 to I.A-5.X-35.A-3600; compounds I.B-5.X-35.A-1 to I.B-5.X-35.A- 3600; compounds I.C-5.X-35.A-1 to I.C-5.X-35.A-3600; compounds I.D-5.X-35.A-1 to I.D-5.X- 35.A-3600; compounds I.E-5.X-35.A-1 to I.E-5.X-35.A-3600; compounds I.F-5.X-35.A-1 to I.F- 5.X-35.A-3600; compounds I.G-5.X-35.A-1 to I.G-5.X-35.A-3600;

compounds I.A-6.X-35.A-1 to I.A-6.X-35.A-3600; compounds I.B-6.X-35.A-1 to I.B-6.X-35.A- 3600; compounds I.C-6.X-35.A-1 to I.C-6.X-35.A-3600; compounds I.D-6.X-35.A-1 to I.D-6.X- 35.A-3600; compounds I.E-6.X-35.A-1 to I.E-6.X-35.A-3600; compounds I.F-6.X-35.A-1 to I.F-

6. X-35.A-3600; compounds I.G-6.X-35.A-1 to I.G-6.X-35.A-3600;

compounds I.A-7.X-35.A-1 to I.A-7.X-35.A-3600; compounds I.B-7.X-35.A-1 to I.B-7.X-35.A- 3600; compounds I.C-7.X-35.A-1 to I.C-7.X-35.A-3600; compounds I.D-7.X-35.A-1 to I.D-7.X- 35.A-3600; compounds I.E-7.X-35.A-1 to I.E-7.X-35.A-3600; compounds I.F-7.X-35.A-1 to I.F-

7. X-35.A-3600; compounds I.G-7.X-35.A-1 to I.G-7.X-35.A-3600;

compounds I.A-8.X-35.A-1 to I.A-8.X-35.A-3600; compounds I.B-8.X-35.A-1 to I.B-8.X-35.A- 3600; compounds I.C-8.X-35.A-1 to I.C-8.X-35.A-3600; compounds I.D-8.X-35.A-1 to I.D-8.X- 35.A-3600; compounds I.E-8.X-35.A-1 to I.E-8.X-35.A-3600; compounds I.F-8.X-35.A-1 to I.F-

8. X-35.A-3600; compounds I.G-8.X-35.A-1 to I.G-8.X-35.A-3600;

compounds I.A-9.X-35.A-1 to I.A-9.X-35.A-3600; compounds I.B-9.X-35.A-1 to I.B-9.X-35.A- 3600; compounds I.C-9.X-35.A-1 to I.C-9.X-35.A-3600; compounds I.D-9.X-35.A-1 to I.D-9.X- 35.A-3600; compounds I.E-9.X-35.A-1 to I.E-9.X-35.A-3600; compounds I.F-9.X-35.A-1 to I.F-

9. X-35.A-3600; compounds I.G-9.X-35.A-1 to I.G-9.X-35.A-3600; compounds I.A-10.X-35.A-1 to I.A-10.X-35.A-3600; compounds I.B-10.X-35.A-1 to I.B-10.X- 35.A-3600; compounds I.C-10.X-35.A-1 to I.C-10.X-35.A-3600; compounds I.D-10.X-35.A-1 to I.D-10.X-35.A-3600; compounds I.E-10.X-35.A-1 to I.E-10.X-35.A-3600; compounds I.F-10.X- 35.A-1 to I.F-10.X-35.A-3600; compounds I.G-10.X-35.A-1 to I.G-10.X-35.A-3600;

compounds I.A-1 1.X-35.A-1 to I.A-1 1.X-35.A-3600; compounds I.B-1 1.X-35.A-1 to I.B-1 1.X- 35.A-3600; compounds I.C-1 1.X-35.A-1 to I.C-1 1 .X-35.A-3600; compounds I.D-1 1.X-35.A-1 to I.D-1 1.X-35.A-3600; compounds I.E-1 1 .X-35.A-1 to I.E-1 1.X-35.A-3600; compounds I.F-1 1.X- 35.A-1 to I.F-1 1.X-35.A-3600; compounds I.G-1 1.X-35.A-1 to I.G-1 1.X-35.A-3600;

compounds I.A-12.X-35.A-1 to I.A-12.X-35.A-3600; compounds I.B-12.X-35.A-1 to I.B-12.X- 35.A-3600; compounds I.C-12.X-35.A-1 to I.C-12.X-35.A-3600; compounds I.D-12.X-35.A-1 to I.D-12.X-35.A-3600; compounds I.E-12.X-35.A-1 to I.E-12.X-35.A-3600; compounds I.F-12.X-

35. A-1 to I.F-12.X-35.A-3600; compounds I.G-12.X-35.A-1 to I.G-12.X-35.A-3600).

Table 36a

Compounds of the formula II.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-36 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-36.A-1 to I.A-2.X-36.A-3600; compounds I.B-2.X-36.A-1 to I.B-2.X-36.A- 3600; compounds I.C-2.X-36.A-1 to I.C-2.X-36.A-3600; compounds I.D-2.X-36.A-1 to I.D-2.X-

36. A-3600; compounds I.E-2.X-36.A-1 to I.E-2.X-36.A-3600; compounds I.F-2.X-36.A-1 to I.F- 2.X-36.A-3600; compounds I.G-2.X-36.A-1 to I.G-2.X-36.A-3600;

compounds I.A-3.X-36.A-1 to I.A-3.X-36.A-3600; compounds I.B-3.X-36.A-1 to I.B-3.X-36.A- 3600; compounds I.C-3.X-36.A-1 to I.C-3.X-36.A-3600; compounds I.D-3.X-36.A-1 to I.D-3.X- 36.A-3600; compounds I.E-3.X-36.A-1 to I.E-3.X-36.A-3600; compounds I.F-3.X-36.A-1 to I.F-

3. X-36.A-3600; compounds I.G-3.X-36.A-1 to I.G-3.X-36.A-3600;

compounds I.A-4.X-36.A-1 to I.A-4.X-36.A-3600; compounds I.B-4.X-36.A-1 to I.B-4.X-36.A- 3600; compounds I.C-4.X-36.A-1 to I.C-4.X-36.A-3600; compounds I.D-4.X-36.A-1 to I.D-4.X- 36.A-3600; compounds I.E-4.X-36.A-1 to I.E-4.X-36.A-3600; compounds I.F-4.X-36.A-1 to I.F-

4. X-36.A-3600; compounds I.G-4.X-36.A-1 to I.G-4.X-36.A-3600;

compounds I.A-5.X-36.A-1 to I.A-5.X-36.A-3600; compounds I.B-5.X-36.A-1 to I.B-5.X-36.A- 3600; compounds I.C-5.X-36.A-1 to I.C-5.X-36.A-3600; compounds I.D-5.X-36.A-1 to I.D-5.X- 36.A-3600; compounds I.E-5.X-36.A-1 to I.E-5.X-36.A-3600; compounds I.F-5.X-36.A-1 to I.F-

5. X-36.A-3600; compounds I.G-5.X-36.A-1 to I.G-5.X-36.A-3600;

compounds I.A-6.X-36.A-1 to I.A-6.X-36.A-3600; compounds I.B-6.X-36.A-1 to I.B-6.X-36.A- 3600; compounds I.C-6.X-36.A-1 to I.C-6.X-36.A-3600; compounds I.D-6.X-36.A-1 to I.D-6.X- 36.A-3600; compounds I.E-6.X-36.A-1 to I.E-6.X-36.A-3600; compounds I.F-6.X-36.A-1 to I.F-

6. X-36.A-3600; compounds I.G-6.X-36.A-1 to I.G-6.X-36.A-3600; compounds I.A-7.X-36.A-1 to I.A-7.X-36.A-3600; compounds I.B-7.X-36.A-1 to I.B-7.X-36.A- 3600; compounds I.C-7.X-36.A-1 to I.C-7.X-36.A-3600; compounds I.D-7.X-36.A-1 to I.D-7.X- 36.A-3600; compounds I.E-7.X-36.A-1 to I.E-7.X-36.A-3600; compounds I.F-7.X-36.A-1 to I.F-

7. X-36.A-3600; compounds I.G-7.X-36.A-1 to I.G-7.X-36.A-3600;

compounds I.A-8.X-36.A-1 to I.A-8.X-36.A-3600; compounds I.B-8.X-36.A-1 to I.B-8.X-36.A- 3600; compounds I.C-8.X-36.A-1 to I.C-8.X-36.A-3600; compounds I.D-8.X-36.A-1 to I.D-8.X- 36.A-3600; compounds I.E-8.X-36.A-1 to I.E-8.X-36.A-3600; compounds I.F-8.X-36.A-1 to I.F-

8. X-36.A-3600; compounds I.G-8.X-36.A-1 to I.G-8.X-36.A-3600;

compounds I.A-9.X-36.A-1 to I.A-9.X-36.A-3600; compounds I.B-9.X-36.A-1 to I.B-9.X-36.A- 3600; compounds I.C-9.X-36.A-1 to I.C-9.X-36.A-3600; compounds I.D-9.X-36.A-1 to I.D-9.X- 36.A-3600; compounds I.E-9.X-36.A-1 to I.E-9.X-36.A-3600; compounds I.F-9.X-36.A-1 to I.F-

9. X-36.A-3600; compounds I.G-9.X-36.A-1 to I.G-9.X-36.A-3600;

compounds I.A-10.X-36.A-1 to I.A-10.X-36.A-3600; compounds I.B-10.X-36.A-1 to I.B-10.X- 36.A-3600; compounds I.C-10.X-36.A-1 to I.C-10.X-36.A-3600; compounds I.D-10.X-36.A-1 to I.D-10.X-36.A-3600; compounds I.E-10.X-36.A-1 to I.E-10.X-36.A-3600; compounds I.F-10.X- 36.A-1 to I.F-10.X-36.A-3600; compounds I.G-10.X-36.A-1 to I.G-10.X-36.A-3600;

compounds I.A-1 1.X-36.A-1 to I.A-1 1.X-36.A-3600; compounds I.B-1 1.X-36.A-1 to I.B-1 1.X- 36.A-3600; compounds I.C-1 1.X-36.A-1 to I.C-1 1 .X-36.A-3600; compounds I.D-1 1.X-36.A-1 to I.D-1 1.X-36.A-3600; compounds I.E-1 1 .X-36.A-1 to I.E-1 1.X-36.A-3600; compounds I.F-1 1.X- 36.A-1 to I.F-1 1.X-36.A-3600; compounds I.G-1 1.X-36.A-1 to I.G-1 1.X-36.A-3600;

compounds I.A-12.X-36.A-1 to I.A-12.X-36.A-3600; compounds I.B-12.X-36.A-1 to I.B-12.X- 36.A-3600; compounds I.C-12.X-36.A-1 to I.C-12.X-36.A-3600; compounds I.D-12.X-36.A-1 to I.D-12.X-36.A-3600; compounds I.E-12.X-36.A-1 to I.E-12.X-36.A-3600; compounds I.F-12.X-

36. A-1 to I.F-12.X-36.A-3600; compounds I.G-12.X-36.A-1 to I.G-12.X-36.A-3600).

Table 37a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-37 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-37.A-1 to I.A-2.X-37.A-3600; compounds I.B-2.X-37.A-1 to I.B-2.X-37.A- 3600; compounds I.C-2.X-37.A-1 to I.C-2.X-37.A-3600; compounds I.D-2.X-37.A-1 to I.D-2.X-

37. A-3600; compounds I.E-2.X-37.A-1 to I.E-2.X-37.A-3600; compounds I.F-2.X-37.A-1 to I.F-

2. X-37.A-3600; compounds I.G-2.X-37.A-1 to I.G-2.X-37.A-3600;

compounds I.A-3.X-37.A-1 to I.A-3.X-37.A-3600; compounds I.B-3.X-37.A-1 to I.B-3.X-37.A- 3600; compounds I.C-3.X-37.A-1 to I.C-3.X-37.A-3600; compounds I.D-3.X-37.A-1 to I.D-3.X- 37.A-3600; compounds I.E-3.X-37.A-1 to I.E-3.X-37.A-3600; compounds I.F-3.X-37.A-1 to I.F-

3. X-37.A-3600; compounds I.G-3.X-37.A-1 to I.G-3.X-37.A-3600; compounds I.A-4.X-37.A-1 to I.A-4.X-37.A-3600; compounds I.B-4.X-37.A-1 to I.B-4.X-37.A- 3600; compounds I.C-4.X-37.A-1 to I.C-4.X-37.A-3600; compounds I.D-4.X-37.A-1 to I.D-4.X- 37.A-3600; compounds I.E-4.X-37.A-1 to I.E-4.X-37.A-3600; compounds I.F-4.X-37.A-1 to I.F-

4. X-37.A-3600; compounds I.G-4.X-37.A-1 to I.G-4.X-37.A-3600;

compounds I.A-5.X-37.A-1 to I.A-5.X-37.A-3600; compounds I.B-5.X-37.A-1 to I.B-5.X-37.A- 3600; compounds I.C-5.X-37.A-1 to I.C-5.X-37.A-3600; compounds I.D-5.X-37.A-1 to I.D-5.X- 37.A-3600; compounds I.E-5.X-37.A-1 to I.E-5.X-37.A-3600; compounds I.F-5.X-37.A-1 to I.F-

5. X-37.A-3600; compounds I.G-5.X-37.A-1 to I.G-5.X-37.A-3600;

compounds I.A-6.X-37.A-1 to I.A-6.X-37.A-3600; compounds I.B-6.X-37.A-1 to I.B-6.X-37.A- 3600; compounds I.C-6.X-37.A-1 to I.C-6.X-37.A-3600; compounds I.D-6.X-37.A-1 to I.D-6.X- 37.A-3600; compounds I.E-6.X-37.A-1 to I.E-6.X-37.A-3600; compounds I.F-6.X-37.A-1 to I.F-

6. X-37.A-3600; compounds I.G-6.X-37.A-1 to I.G-6.X-37.A-3600;

compounds I.A-7.X-37.A-1 to I.A-7.X-37.A-3600; compounds I.B-7.X-37.A-1 to I.B-7.X-37.A- 3600; compounds I.C-7.X-37.A-1 to I.C-7.X-37.A-3600; compounds I.D-7.X-37.A-1 to I.D-7.X- 37.A-3600; compounds I.E-7.X-37.A-1 to I.E-7.X-37.A-3600; compounds I.F-7.X-37.A-1 to I.F-

7. X-37.A-3600; compounds I.G-7.X-37.A-1 to I.G-7.X-37.A-3600;

compounds I.A-8.X-37.A-1 to I.A-8.X-37.A-3600; compounds I.B-8.X-37.A-1 to I.B-8.X-37.A- 3600; compounds I.C-8.X-37.A-1 to I.C-8.X-37.A-3600; compounds I.D-8.X-37.A-1 to I.D-8.X- 37.A-3600; compounds I.E-8.X-37.A-1 to I.E-8.X-37.A-3600; compounds I.F-8.X-37.A-1 to I.F- 8.X-37.A-3600; compounds I.G-8.X-37.A-1 to I.G-8.X-37.A-3600;

compounds I.A-9.X-37.A-1 to I.A-9.X-37.A-3600; compounds I.B-9.X-37.A-1 to I.B-9.X-37.A- 3600; compounds I.C-9.X-37.A-1 to I.C-9.X-37.A-3600; compounds I.D-9.X-37.A-1 to I.D-9.X- 37.A-3600; compounds I.E-9.X-37.A-1 to I.E-9.X-37.A-3600; compounds I.F-9.X-37.A-1 to I.F- 9.X-37.A-3600; compounds I.G-9.X-37.A-1 to I.G-9.X-37.A-3600;

compounds I.A-10.X-37.A-1 to I.A-10.X-37.A-3600; compounds I.B-10.X-37.A-1 to I.B-10.X- 37.A-3600; compounds I.C-10.X-37.A-1 to I.C-10.X-37.A-3600; compounds I.D-10.X-37.A-1 to I.D-10.X-37.A-3600; compounds I.E-10.X-37.A-1 to I.E-10.X-37.A-3600; compounds I.F-10.X- 37.A-1 to I.F-10.X-37.A-3600; compounds I.G-10.X-37.A-1 to I.G-10.X-37.A-3600;

compounds I.A-1 1.X-37.A-1 to I.A-1 1 .X-37.A-3600; compounds I.B-1 1.X-37.A-1 to I.B-1 1.X- 37.A-3600; compounds I.C-1 1.X-37.A-1 to I.C-1 1 .X-37.A-3600; compounds I.D-1 1.X-37.A-1 to I.D-1 1.X-37.A-3600; compounds I.E-1 1 .X-37.A-1 to I.E-1 1.X-37.A-3600; compounds I.F-1 1.X- 37.A-1 to I.F-1 1.X-37.A-3600; compounds I.G-1 1.X-37.A-1 to I.G-1 1.X-37.A-3600;

compounds I.A-12.X-37.A-1 to I.A-12.X-37.A-3600; compounds I.B-12.X-37.A-1 to I.B-12.X- 37.A-3600; compounds I.C-12.X-37.A-1 to I.C-12.X-37.A-3600; compounds I.D-12.X-37.A-1 to I.D-12.X-37.A-3600; compounds I.E-12.X-37.A-1 to I.E-12.X-37.A-3600; compounds I.F-12.X- 37.A-1 to I.F-12.X-37.A-3600; compounds I.G-12.X-37.A-1 to I.G-12.X-37.A-3600).

Table 38a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A-

8. I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-38 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (compounds I.A-2.X-38.A-1 to I.A-2.X-38.A-3600; compounds I.B-2.X-38.A-1 to I.B-2.X-38.A- 3600; compounds I.C-2.X-38.A-1 to I.C-2.X-38.A-3600; compounds I.D-2.X-38.A-1 to I.D-2.X- 38.A-3600; compounds I.E-2.X-38.A-1 to I.E-2.X-38.A-3600; compounds I.F-2.X-38.A-1 to I.F-

2. X-38.A-3600; compounds I.G-2.X-38.A-1 to I.G-2.X-38.A-3600;

compounds I.A-3.X-38.A-1 to I.A-3.X-38.A-3600; compounds I.B-3.X-38.A-1 to I.B-3.X-38.A- 3600; compounds I.C-3.X-38.A-1 to I.C-3.X-38.A-3600; compounds I.D-3.X-38.A-1 to I.D-3.X- 38.A-3600; compounds I.E-3.X-38.A-1 to I.E-3.X-38.A-3600; compounds I.F-3.X-38.A-1 to I.F-

3. X-38.A-3600; compounds I.G-3.X-38.A-1 to I.G-3.X-38.A-3600;

compounds I.A-4.X-38.A-1 to I.A-4.X-38.A-3600; compounds I.B-4.X-38.A-1 to I.B-4.X-38.A- 3600; compounds I.C-4.X-38.A-1 to I.C-4.X-38.A-3600; compounds I.D-4.X-38.A-1 to I.D-4.X- 38.A-3600; compounds I.E-4.X-38.A-1 to I.E-4.X-38.A-3600; compounds I.F-4.X-38.A-1 to I.F-

4. X-38.A-3600; compounds I.G-4.X-38.A-1 to I.G-4.X-38.A-3600;

compounds I.A-5.X-38.A-1 to I.A-5.X-38.A-3600; compounds I.B-5.X-38.A-1 to I.B-5.X-38.A- 3600; compounds I.C-5.X-38.A-1 to I.C-5.X-38.A-3600; compounds I.D-5.X-38.A-1 to I.D-5.X- 38.A-3600; compounds I.E-5.X-38.A-1 to I.E-5.X-38.A-3600; compounds I.F-5.X-38.A-1 to I.F- 5.X-38.A-3600; compounds I.G-5.X-38.A-1 to I.G-5.X-38.A-3600;

compounds I.A-6.X-38.A-1 to I.A-6.X-38.A-3600; compounds I.B-6.X-38.A-1 to I.B-6.X-38.A- 3600; compounds I.C-6.X-38.A-1 to I.C-6.X-38.A-3600; compounds I.D-6.X-38.A-1 to I.D-6.X- 38.A-3600; compounds I.E-6.X-38.A-1 to I.E-6.X-38.A-3600; compounds I.F-6.X-38.A-1 to I.F-

6. X-38.A-3600; compounds I.G-6.X-38.A-1 to I.G-6.X-38.A-3600;

compounds I.A-7.X-38.A-1 to I.A-7.X-38.A-3600; compounds I.B-7.X-38.A-1 to I.B-7.X-38.A- 3600; compounds I.C-7.X-38.A-1 to I.C-7.X-38.A-3600; compounds I.D-7.X-38.A-1 to I.D-7.X- 38.A-3600; compounds I.E-7.X-38.A-1 to I.E-7.X-38.A-3600; compounds I.F-7.X-38.A-1 to I.F-

7. X-38.A-3600; compounds I.G-7.X-38.A-1 to I.G-7.X-38.A-3600;

compounds I.A-8.X-38.A-1 to I.A-8.X-38.A-3600; compounds I.B-8.X-38.A-1 to I.B-8.X-38.A- 3600; compounds I.C-8.X-38.A-1 to I.C-8.X-38.A-3600; compounds I.D-8.X-38.A-1 to I.D-8.X- 38.A-3600; compounds I.E-8.X-38.A-1 to I.E-8.X-38.A-3600; compounds I.F-8.X-38.A-1 to I.F-

8. X-38.A-3600; compounds I.G-8.X-38.A-1 to I.G-8.X-38.A-3600;

compounds I.A-9.X-38.A-1 to I.A-9.X-38.A-3600; compounds I.B-9.X-38.A-1 to I.B-9.X-38.A- 3600; compounds I.C-9.X-38.A-1 to I.C-9.X-38.A-3600; compounds I.D-9.X-38.A-1 to I.D-9.X- 38.A-3600; compounds I.E-9.X-38.A-1 to I.E-9.X-38.A-3600; compounds I.F-9.X-38.A-1 to I.F-

9. X-38.A-3600; compounds I.G-9.X-38.A-1 to I.G-9.X-38.A-3600;

compounds I.A-10.X-38.A-1 to I.A-10.X-38.A-3600; compounds I.B-10.X-38.A-1 to I.B-10.X- 38.A-3600; compounds I.C-10.X-38.A-1 to I.C-10.X-38.A-3600; compounds I.D-10.X-38.A-1 to I.D-10.X-38.A-3600; compounds I.E-10.X-38.A-1 to I.E-10.X-38.A-3600; compounds I.F-10.X- 38.A-1 to I.F-10.X-38.A-3600; compounds I.G-10.X-38.A-1 to I.G-10.X-38.A-3600; compounds I.A-1 1.X-38.A-1 to I.A-1 1.X-38.A-3600; compounds I.B-1 1.X-38.A-1 to I.B-1 1.X- 38.A-3600; compounds I.C-1 1.X-38.A-1 to I.C-1 1 .X-38.A-3600; compounds I.D-1 1.X-38.A-1 to I.D-1 1.X-38.A-3600; compounds I.E-1 1 .X-38.A-1 to I.E-1 1.X-38.A-3600; compounds I.F-1 1.X- 38.A-1 to I.F-1 1.X-38.A-3600; compounds I.G-1 1.X-38.A-1 to I.G-1 1.X-38.A-3600;

compounds I.A-12.X-38.A-1 to I.A-12.X-38.A-3600; compounds I.B-12.X-38.A-1 to I.B-12.X- 38.A-3600; compounds I.C-12.X-38.A-1 to I.C-12.X-38.A-3600; compounds I.D-12.X-38.A-1 to I.D-12.X-38.A-3600; compounds I.E-12.X-38.A-1 to I.E-12.X-38.A-3600; compounds I.F-12.X-

38. A-1 to I.F-12.X-38.A-3600; compounds I.G-12.X-38.A-1 to I.G-12.X-38.A-3600).

Table 39a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10,

1. C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12, I.B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-39 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A

(compounds I.A-2.X-39.A-1 to I.A-2.X-39.A-3600; compounds I.B-2.X-39.A-1 to I.B-2.X-39.A- 3600; compounds I.C-2.X-39.A-1 to I.C-2.X-39.A-3600; compounds I.D-2.X-39.A-1 to I.D-2.X- 39.A-3600; compounds I.E-2.X-39.A-1 to I.E-2.X-39.A-3600; compounds I.F-2.X-39.A-1 to I.F-

2. X-39.A-3600; compounds I.G-2.X-39.A-1 to I.G-2.X-39.A-3600;

compounds I.A-3.X-39.A-1 to I.A-3.X-39.A-3600; compounds I.B-3.X-39.A-1 to I.B-3.X-39.A- 3600; compounds I.C-3.X-39.A-1 to I.C-3.X-39.A-3600; compounds I.D-3.X-39.A-1 to I.D-3.X-

39. A-3600; compounds I.E-3.X-39.A-1 to I.E-3.X-39.A-3600; compounds I.F-3.X-39.A-1 to I.F- 3.X-39.A-3600; compounds I.G-3.X-39.A-1 to I.G-3.X-39.A-3600;

compounds I.A-4.X-39.A-1 to I.A-4.X-39.A-3600; compounds I.B-4.X-39.A-1 to I.B-4.X-39.A- 3600; compounds I.C-4.X-39.A-1 to I.C-4.X-39.A-3600; compounds I.D-4.X-39.A-1 to I.D-4.X- 39.A-3600; compounds I.E-4.X-39.A-1 to I.E-4.X-39.A-3600; compounds I.F-4.X-39.A-1 to I.F-

4. X-39.A-3600; compounds I.G-4.X-39.A-1 to I.G-4.X-39.A-3600;

compounds I.A-5.X-39.A-1 to I.A-5.X-39.A-3600; compounds I.B-5.X-39.A-1 to I.B-5.X-39.A- 3600; compounds I.C-5.X-39.A-1 to I.C-5.X-39.A-3600; compounds I.D-5.X-39.A-1 to I.D-5.X- 39.A-3600; compounds I.E-5.X-39.A-1 to I.E-5.X-39.A-3600; compounds I.F-5.X-39.A-1 to I.F-

5. X-39.A-3600; compounds I.G-5.X-39.A-1 to I.G-5.X-39.A-3600;

compounds I.A-6.X-39.A-1 to I.A-6.X-39.A-3600; compounds I.B-6.X-39.A-1 to I.B-6.X-39.A- 3600; compounds I.C-6.X-39.A-1 to I.C-6.X-39.A-3600; compounds I.D-6.X-39.A-1 to I.D-6.X- 39.A-3600; compounds I.E-6.X-39.A-1 to I.E-6.X-39.A-3600; compounds I.F-6.X-39.A-1 to I.F-

6. X-39.A-3600; compounds I.G-6.X-39.A-1 to I.G-6.X-39.A-3600;

compounds I.A-7.X-39.A-1 to I.A-7.X-39.A-3600; compounds I.B-7.X-39.A-1 to I.B-7.X-39.A- 3600; compounds I.C-7.X-39.A-1 to I.C-7.X-39.A-3600; compounds I.D-7.X-39.A-1 to I.D-7.X- 39.A-3600; compounds I.E-7.X-39.A-1 to I.E-7.X-39.A-3600; compounds I.F-7.X-39.A-1 to I.F-

7. X-39.A-3600; compounds I.G-7.X-39.A-1 to I.G-7.X-39.A-3600; compounds I.A-8.X-39.A-1 to I.A-8.X-39.A-3600; compounds I.B-8.X-39.A-1 to I.B-8.X-39.A- 3600; compounds I.C-8.X-39.A-1 to I.C-8.X-39.A-3600; compounds I.D-8.X-39.A-1 to I.D-8.X- 39.A-3600; compounds I.E-8.X-39.A-1 to I.E-8.X-39.A-3600; compounds I.F-8.X-39.A-1 to I.F-

8. X-39.A-3600; compounds I.G-8.X-39.A-1 to I.G-8.X-39.A-3600;

compounds I.A-9.X-39.A-1 to I.A-9.X-39.A-3600; compounds I.B-9.X-39.A-1 to I.B-9.X-39.A- 3600; compounds I.C-9.X-39.A-1 to I.C-9.X-39.A-3600; compounds I.D-9.X-39.A-1 to I.D-9.X- 39.A-3600; compounds I.E-9.X-39.A-1 to I.E-9.X-39.A-3600; compounds I.F-9.X-39.A-1 to I.F-

9. X-39.A-3600; compounds I.G-9.X-39.A-1 to I.G-9.X-39.A-3600;

compounds I.A-10.X-39.A-1 to I.A-10.X-39.A-3600; compounds I.B-10.X-39.A-1 to I.B-10.X- 39.A-3600; compounds I.C-10.X-39.A-1 to I.C-10.X-39.A-3600; compounds I.D-10.X-39.A-1 to I.D-10.X-39.A-3600; compounds I.E-10.X-39.A-1 to I.E-10.X-39.A-3600; compounds I.F-10.X- 39.A-1 to I.F-10.X-39.A-3600; compounds I.G-10.X-39.A-1 to I.G-10.X-39.A-3600;

compounds I.A-1 1.X-39.A-1 to I.A-1 1.X-39.A-3600; compounds I.B-1 1.X-39.A-1 to I.B-1 1.X- 39.A-3600; compounds I.C-1 1.X-39.A-1 to I.C-1 1 .X-39.A-3600; compounds I.D-1 1.X-39.A-1 to I.D-1 1.X-39.A-3600; compounds I.E-1 1 .X-39.A-1 to I.E-1 1.X-39.A-3600; compounds I.F-1 1.X- 39.A-1 to I.F-1 1.X-39.A-3600; compounds I.G-1 1.X-39.A-1 to I.G-1 1.X-39.A-3600;

compounds I.A-12.X-39.A-1 to I.A-12.X-39.A-3600; compounds I.B-12.X-39.A-1 to I.B-12.X-

39. A-3600; compounds I.C-12.X-39.A-1 to I.C-12.X-39.A-3600; compounds I.D-12.X-39.A-1 to I.D-12.X-39.A-3600; compounds I.E-12.X-39.A-1 to I.E-12.X-39.A-3600; compounds I.F-12.X- 39.A-1 to I.F-12.X-39.A-3600; compounds I.G-12.X-39.A-1 to I.G-12.X-39.A-3600).

Table 40a

Compounds of the formula I.A-2, I.B-2, I.C-2, I.D-2, I.E-2, I.F-2, I.G-2; I.A-3, I.B-3, I.C-3, I.D-3, I.E-3, I.F-3, I.G-3;I.A-4, I.B-4, I.C-4, I.D-4, I.E-4, I.F-4, I.G-4; I.A-5, I.B-5, I.C-5, I.D-5, I.E-5, I.F-5, I.G-5; I.A-6, I.B-6, I.C-6, I.D-6, I.E-6, I.F-6, I.G-6; I.A-7, I.B-7, I.C-7, I.D-7, I.E-7, I.F-7, I.G-7; I.A- 8, I.B-8, I.C-8, I.D-8, I.E-8, I.F-8, I.G-8; I.A-9, I.B-9, I.C-9, I.D-9, I.E-9, I.F-9, I.G-9; I.A-10, I.B-10, I.C-10, I.D-10, I.E-10, I.F-10, I.G-10; I.A-1 1 , I.B-1 1 , I.C-1 1 , I.D-1 1 , I.E-1 1 , I.F-1 1 , I.G-1 1 ; I.A-12,

1. B-12, I.C-12, I.D-12, I.E-12, I.F-12, I.G-12;

in which X _n is as defined in line X-40 of Table X and the meaning for the combination of R ¹ , R ² , R ³ and R ⁴ for each individual compound corresponds in each case to one line of Table A (compounds I.A-2.X-40.A-1 to I.A-2.X-40.A-3600; compounds I.B-2.X-40.A-1 to I.B-2.X-40.A- 3600; compounds I.C-2.X-40.A-1 to I.C-2.X-40.A-3600; compounds I.D-2.X-40.A-1 to I.D-2.X-

40. A-3600; compounds I.E-2.X-40.A-1 to I.E-2.X-40.A-3600; compounds I.F-2.X-40.A-1 to I.F-

2. X-40.A-3600; compounds I.G-2.X-40.A-1 to I.G-2.X-40.A-3600;

compounds I.A-3.X-40.A-1 to I.A-3.X-40.A-3600; compounds I.B-3.X-40.A-1 to I.B-3.X-40.A- 3600; compounds I.C-3.X-40.A-1 to I.C-3.X-40.A-3600; compounds I.D-3.X-40.A-1 to I.D-3.X- 40.A-3600; compounds I.E-3.X-40.A-1 to I.E-3.X-40.A-3600; compounds I.F-3.X-40.A-1 to I.F-

3. X-40.A-3600; compounds I.G-3.X-40.A-1 to I.G-3.X-40.A-3600;

compounds I.A-4.X-40.A-1 to I.A-4.X-40.A-3600; compounds I.B-4.X-40.A-1 to I.B-4.X-40.A- 3600; compounds I.C-4.X-40.A-1 to I.C-4.X-40.A-3600; compounds I.D-4.X-40.A-1 to I.D-4.X- 40.A-3600; compounds I.E-4.X-40.A-1 to I.E-4.X-40.A-3600; compounds I.F-4.X-40.A-1 to I.F-

4. X-40.A-3600; compounds I.G-4.X-40.A-1 to I.G-4.X-40.A-3600; compounds I.A-5.X-40.A-1 to I.A-5.X-40.A-3600; compounds I.B-5.X-40.A-1 to I.B-5.X-40.A- 3600; compounds I.C-5.X-40.A-1 to I.C-5.X-40.A-3600; compounds I.D-5.X-40.A-1 to I.D-5.X- 40.A-3600; compounds I.E-5.X-40.A-1 to I.E-5.X-40.A-3600; compounds I.F-5.X-40.A-1 to I.F-

5. X-40.A-3600; compounds I.G-5.X-40.A-1 to I.G-5.X-40.A-3600;

compounds I.A-6.X-40.A-1 to I.A-6.X-40.A-3600; compounds I.B-6.X-40.A-1 to I.B-6.X-40.A- 3600; compounds I.C-6.X-40.A-1 to I.C-6.X-40.A-3600; compounds I.D-6.X-40.A-1 to I.D-6.X- 40.A-3600; compounds I.E-6.X-40.A-1 to I.E-6.X-40.A-3600; compounds I.F-6.X-40.A-1 to I.F-

6. X-40.A-3600; compounds I.G-6.X-40.A-1 to I.G-6.X-40.A-3600;

compounds I.A-7.X-40.A-1 to I.A-7.X-40.A-3600; compounds I.B-7.X-40.A-1 to I.B-7.X-40.A- 3600; compounds I.C-7.X-40.A-1 to I.C-7.X-40.A-3600; compounds I.D-7.X-40.A-1 to I.D-7.X- 40.A-3600; compounds I.E-7.X-40.A-1 to I.E-7.X-40.A-3600; compounds I.F-7.X-40.A-1 to I.F-

7. X-40.A-3600; compounds I.G-7.X-40.A-1 to I.G-7.X-40.A-3600;

compounds I.A-8.X-40.A-1 to I.A-8.X-40.A-3600; compounds I.B-8.X-40.A-1 to I.B-8.X-40.A- 3600; compounds I.C-8.X-40.A-1 to I.C-8.X-40.A-3600; compounds I.D-8.X-40.A-1 to I.D-8.X- 40.A-3600; compounds I.E-8.X-40.A-1 to I.E-8.X-40.A-3600; compounds I.F-8.X-40.A-1 to I.F-

8. X-40.A-3600; compounds I.G-8.X-40.A-1 to I.G-8.X-40.A-3600;

compounds I.A-9.X-40.A-1 to I.A-9.X-40.A-3600; compounds I.B-9.X-40.A-1 to I.B-9.X-40.A- 3600; compounds I.C-9.X-40.A-1 to I.C-9.X-40.A-3600; compounds I.D-9.X-40.A-1 to I.D-9.X- 40.A-3600; compounds I.E-9.X-40.A-1 to I.E-9.X-40.A-3600; compounds I.F-9.X-40.A-1 to I.F- 9.X-40.A-3600; compounds I.G-9.X-40.A-1 to I.G-9.X-40.A-3600;

compounds I.A-10.X-40.A-1 to I.A-10.X-40.A-3600; compounds I.B-10.X-40.A-1 to I.B-10.X- 40.A-3600; compounds I.C-10.X-40.A-1 to I.C-10.X-40.A-3600; compounds I.D-10.X-40.A-1 to I.D-10.X-40.A-3600; compounds I.E-10.X-40.A-1 to I.E-10.X-40.A-3600; compounds I.F-10.X- 40.A-1 to I.F-10.X-40.A-3600; compounds I.G-10.X-40.A-1 to I.G-10.X-40.A-3600;

compounds I.A-1 1.X-40.A-1 to I.A-1 1.X-40.A-3600; compounds I.B-1 1.X-40.A-1 to I.B-1 1.X- 40.A-3600; compounds I.C-1 1.X-40.A-1 to I.C-1 1 .X-40.A-3600; compounds I.D-1 1.X-40.A-1 to I.D-1 1.X-40.A-3600; compounds I.E-1 1 .X-40.A-1 to I.E-1 1.X-40.A-3600; compounds I.F-1 1.X- 40.A-1 to I.F-1 1.X-40.A-3600; compounds I.G-1 1.X-40.A-1 to I.G-1 1.X-40.A-3600;

compounds I.A-12.X-40.A-1 to I.A-12.X-40.A-3600; compounds I.B-12.X-40.A-1 to I.B-12.X- 40.A-3600; compounds I.C-12.X-40.A-1 to I.C-12.X-40.A-3600; compounds I.D-12.X-40.A-1 to I.D-12.X-40.A-3600; compounds I.E-12.X-40.A-1 to I.E-12.X-40.A-3600; compounds I.F-12.X- 40.A-1 to I.F-12.X-40.A-3600; compounds I.G-12.X-40.A-1 to I.G-12.X-40.A-3600).

I

line 1 2 3 4

X-1 CI H H H

X-2 H CI H H

X-3 H H CI H

X-4 H H H CI

X-5 F H H H

X-6 H F H H

X-7 H H F H

X-8 H H H F

X-9 CI CI H H

X-10 CI H CI H

X-1 1 CI H H CI

X-12 H CI CI H

X-13 H CI H CI

X-14 H H CI CI

X-15 F F H H

X-16 F H F H

X-17 F H H F

X-18 H F F H

X-19 H F H F

X-20 H H F F

X-21 CI F H H

X-22 F CI H H

X-23 CI H F H

X-24 F H CI H

X-25 CI H H F

X-26 F H H CI

X-27 H CI F H

X-28 H F CI H

X-29 H CI H F

X-30 H F H CI

X-31 H H CI F

X-32 H H F CI X-33 CN H H H

X-34 H CN H H

X-35 H H CN H

X-36 H H H CN

X-37 CHs H H H

X-38 H CHs H H

X-39 H H CHs H

X-40 H H H CHs

Table A line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1 CI CI H H A-30 CFs Br H H

A-2 F CI H H A-31 CHF ₂ Br H H

A-3 Br CI H H A-32 C3H7 Br H H

A-4 CN CI H H A-33 CONH2 Br H H

A-5 CHs CI H H A-34 SCHs Br H H

A-6 CFs CI H H A-35 SOCHs Br H H

A-7 CHF ₂ CI H H A-36 OCHs Br H H

A-8 CsH ₇ CI H H A-37 CI CN H H

A-9 CONH2 CI H H A-38 F CN H H

A-10 SCHs CI H H A-39 Br CN H H

A-1 1 SOCHs CI H H A-40 CN CN H H

A-12 OCHs CI H H A-41 CHs CN H H

A-13 CI F H H A-42 CFs CN H H

A-14 F F H H A-43 CHF ₂ CN H H

A-15 Br F H H A-44 C3H7 CN H H

A-16 CN F H H A-45 CONH2 CN H H

A-17 CHs F H H A-46 SCHs CN H H

A-18 CFs F H H A-47 SOCHs CN H H

A-19 CHF ₂ F H H A-48 OCHs CN H H

A-20 C3H7 F H H A-49 CI CHs H H

A-21 CONH2 F H H A-50 F CHs H H

A-22 SCHs F H H A-51 Br CHs H H

A-23 SOCHs F H H A-52 CN CHs H H

A-24 OCHs F H H A-53 CHs CHs H H

A-25 CI Br H H A-54 CFs CHs H H

A-26 F Br H H A-55 CHF ₂ CHs H H

A-27 Br Br H H A-56 C3H7 CHs H H

A-28 CN Br H H A-57 CONH2 CHs H H

A-29 CHs Br H H A-58 SCHs CHs H H line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-59 SOCHs CHs H H A-100 CN CONH2 H H

A-60 OCH3 CHs H H A-101 CHs CONH2 H H

A-61 CI CFs H H A-102 CFs CONH2 H H

A-62 F CFs H H A-103 CHF ₂ CONH2 H H

A-63 Br CFs H H A-104 C3H7 CONH2 H H

A-64 CN CFs H H A-105 CONH2 CONH2 H H

A-65 CHs CFs H H A-106 SCHs CONH2 H H

A-66 CFs CFs H H A-107 SOCHs CONH2 H H

A-67 CHF ₂ CFs H H A-108 OCHs CONH2 H H

A-68 C3H7 CFs H H A-109 CI SCHs H H

A-69 CONH2 CFs H H A-1 10 F SCHs H H

A-70 SCHs CFs H H A-1 1 1 Br SCHs H H

A-71 SOCHs CFs H H A-1 12 CN SCHs H H

A-72 OCHs CFs H H A-1 13 CHs SCHs H H

A-73 CI CHF ₂ H H A-1 14 CFs SCHs H H

A-74 F CHF ₂ H H A-1 15 CHF ₂ SCHs H H

A-75 Br CHF ₂ H H A-1 16 C3H7 SCHs H H

A-76 CN CHF ₂ H H A-1 17 CONH2 SCHs H H

A-77 CHs CHF ₂ H H A-1 18 SCHs SCHs H H

A-78 CFs CHF ₂ H H A-1 19 SOCHs SCHs H H

A-79 CHF ₂ CHF ₂ H H A-120 OCHs SCHs H H

A-80 C3H7 CHF ₂ H H A-121 CI SOCHs H H

A-81 CONH2 CHF ₂ H H A-122 F SOCHs H H

A-82 SCHs CHF ₂ H H A-123 Br SOCHs H H

A-83 SOCHs CHF ₂ H H A-124 CN SOCHs H H

A-84 OCHs CHF ₂ H H A-125 CHs SOCHs H H

A-85 CI C3H7 H H A-126 CFs SOCHs H H

A-86 F C3H7 H H A-127 CHF ₂ SOCHs H H

A-87 Br C3H7 H H A-128 C3H7 SOCHs H H

A-88 CN C3H7 H H A-129 CONH2 SOCHs H H

A-89 CHs C3H7 H H A-130 SCHs SOCHs H H

A-90 CFs C3H7 H H A-131 SOCHs SOCHs H H

A-91 CHF ₂ C3H7 H H A-132 OCHs SOCHs H H

A-92 C3H7 C3H7 H H A-133 CI OCHs H H

A-93 CONH2 C3H7 H H A-134 F OCHs H H

A-94 SCHs C3H7 H H A-135 Br OCHs H H

A-95 SOCHs C3H7 H H A-136 CN OCHs H H

A-96 OCHs C3H7 H H A-137 CHs OCHs H H

A-97 CI CONH2 H H A-138 CFs OCHs H H

A-98 F CONH2 H H A-139 CHF ₂ OCHs H H

A-99 Br CONH2 H H A-140 C3H7 OCHs H H line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-141 CONH ₂ OCHs H H A-182 F CN F H

A-142 SCHs OCHs H H A-183 Br CN F H

A-143 SOCH3 OCHs H H A-184 CN CN F H

A-144 OCH3 OCHs H H A-185 CHs CN F H

A-145 CI CI F H A-186 CFs CN F H

A-146 F CI F H A-187 CHF ₂ CN F H

A-147 Br CI F H A-188 C3H7 CN F H

A-148 CN CI F H A-189 CONH2 CN F H

A-149 CHs CI F H A-190 SCHs CN F H

A-150 CFs CI F H A-191 SOCHs CN F H

A-151 CHF ₂ CI F H A-192 OCHs CN F H

A-152 C3H7 CI F H A-193 CI CHs F H

A-153 CONH2 CI F H A-194 F CHs F H

A-154 SCHs CI F H A-195 Br CHs F H

A-155 SOCHs CI F H A-196 CN CHs F H

A-156 OCHs CI F H A-197 CHs CHs F H

A-157 CI F F H A-198 CFs CHs F H

A-158 F F F H A-199 CHF ₂ CHs F H

A-159 Br F F H A-200 C3H7 CHs F H

A-160 CN F F H A-201 CONH2 CHs F H

A-161 CHs F F H A-202 SCHs CHs F H

A-162 CFs F F H A-203 SOCHs CHs F H

A-163 CHF ₂ F F H A-204 OCHs CHs F H

A-164 C3H7 F F H A-205 CI CFs F H

A-165 CONH2 F F H A-206 F CFs F H

A-166 SCHs F F H A-207 Br CFs F H

A-167 SOCHs F F H A-208 CN CFs F H

A-168 OCHs F F H A-209 CHs CFs F H

A-169 CI Br F H A-210 CFs CFs F H

A-170 F Br F H A-21 1 CHF ₂ CFs F H

A-171 Br Br F H A-212 C3H7 CFs F H

A-172 CN Br F H A-213 CONH2 CFs F H

A-173 CHs Br F H A-214 SCHs CFs F H

A-174 CFs Br F H A-215 SOCHs CFs F H

A-175 CHF ₂ Br F H A-216 OCHs CFs F H

A-176 C3H7 Br F H A-217 CI CHF ₂ F H

A-177 CONH2 Br F H A-218 F CHF ₂ F H

A-178 SCHs Br F H A-219 Br CHF ₂ F H

A-179 SOCHs Br F H A-220 CN CHF ₂ F H

A-180 OCHs Br F H A-221 CHs CHF ₂ F H

A-181 CI CN F H A-222 CFs CHF ₂ F H line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-223 CHF ₂ CHF2 F H A-264 OCHs SCHs F H

A-224 C3H7 CHF2 F H A-265 CI SOCHs F H

A-225 CONH2 CHF2 F H A-266 F SOCHs F H

A-226 SCHs CHF2 F H A-267 Br SOCHs F H

A-227 SOCH3 CHF2 F H A-268 CN SOCHs F H

A-228 OCH3 CHF2 F H A-269 CHs SOCHs F H

A-229 CI C3H7 F H A-270 CFs SOCHs F H

A-230 F C3H7 F H A-271 CHF ₂ SOCHs F H

A-231 Br C3H7 F H A-272 C3H7 SOCHs F H

A-232 CN C3H7 F H A-273 CONH2 SOCHs F H

A-233 CHs C3H7 F H A-274 SCHs SOCHs F H

A-234 CFs C3H7 F H A-275 SOCHs SOCHs F H

A-235 CHF ₂ C3H7 F H A-276 OCHs SOCHs F H

A-236 C3H7 C3H7 F H A-277 CI OCHs F H

A-237 CONH2 C3H7 F H A-278 F OCHs F H

A-238 SCHs C3H7 F H A-279 Br OCHs F H

A-239 SOCHs C3H7 F H A-280 CN OCHs F H

A-240 OCHs C3H7 F H A-281 CHs OCHs F H

A-241 CI CONH2 F H A-282 CFs OCHs F H

A-242 F CONH2 F H A-283 CHF ₂ OCHs F H

A-243 Br CONH2 F H A-284 C3H7 OCHs F H

A-244 CN CONH2 F H A-285 CONH2 OCHs F H

A-245 CHs CONH2 F H A-286 SCHs OCHs F H

A-246 CFs CONH2 F H A-287 SOCHs OCHs F H

A-247 CHF ₂ CONH2 F H A-288 OCHs OCHs F H

A-248 C3H7 CONH2 F H A-289 CI CI CI H

A-249 CONH2 CONH2 F H A-290 F CI CI H

A-250 SCHs CONH2 F H A-291 Br CI CI H

A-251 SOCHs CONH2 F H A-292 CN CI CI H

A-252 OCHs CONH2 F H A-293 CHs CI CI H

A-253 CI SCHs F H A-294 CFs CI CI H

A-254 F SCHs F H A-295 CHF ₂ CI CI H

A-255 Br SCHs F H A-296 C3H7 CI CI H

A-256 CN SCHs F H A-297 CONH2 CI CI H

A-257 CHs SCHs F H A-298 SCHs CI CI H

A-258 CFs SCHs F H A-299 SOCHs CI CI H

A-259 CHF ₂ SCHs F H A-300 OCHs CI CI H

A-260 C3H7 SCHs F H A-301 CI F CI H

A-261 CONH2 SCHs F H A-302 F F CI H

A-262 SCHs SCHs F H A-303 Br F CI H

A-263 SOCHs SCHs F H A-304 CN F CI H line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-305 CHs F CI H A-346 SCHs CHs CI H

A-306 CFs F CI H A-347 SOCHs CHs CI H

A-307 CHF ₂ F CI H A-348 OCHs CHs CI H

A-308 C3H7 F CI H A-349 CI CFs CI H

A-309 CONH2 F CI H A-350 F CFs CI H

A-310 SCHs F CI H A-351 Br CFs CI H

A-31 1 SOCHs F CI H A-352 CN CFs CI H

A-312 OCHs F CI H A-353 CHs CFs CI H

A-313 CI Br CI H A-354 CFs CFs CI H

A-314 F Br CI H A-355 CHF ₂ CFs CI H

A-315 Br Br CI H A-356 C3H7 CFs CI H

A-316 CN Br CI H A-357 CONH2 CFs CI H

A-317 CHs Br CI H A-358 SCHs CFs CI H

A-318 CFs Br CI H A-359 SOCHs CFs CI H

A-319 CHF ₂ Br CI H A-360 OCHs CFs CI H

A-320 C3H7 Br CI H A-361 CI CHF ₂ CI H

A-321 CONH2 Br CI H A-362 F CHF ₂ CI H

A-322 SCHs Br CI H A-363 Br CHF ₂ CI H

A-323 SOCHs Br CI H A-364 CN CHF ₂ CI H

A-324 OCHs Br CI H A-365 CHs CHF ₂ CI H

A-325 CI CN CI H A-366 CFs CHF ₂ CI H

A-326 F CN CI H A-367 CHF ₂ CHF ₂ CI H

A-327 Br CN CI H A-368 C3H7 CHF ₂ CI H

A-328 CN CN CI H A-369 CONH2 CHF ₂ CI H

A-329 CHs CN CI H A-370 SCHs CHF ₂ CI H

A-330 CFs CN CI H A-371 SOCHs CHF ₂ CI H

A-331 CHF ₂ CN CI H A-372 OCHs CHF ₂ CI H

A-332 C3H7 CN CI H A-373 CI C3H7 CI H

A-333 CONH2 CN CI H A-374 F C3H7 CI H

A-334 SCHs CN CI H A-375 Br C3H7 CI H

A-335 SOCHs CN CI H A-376 CN C3H7 CI H

A-336 OCHs CN CI H A-377 CHs C3H7 CI H

A-337 CI CHs CI H A-378 CFs C3H7 CI H

A-338 F CHs CI H A-379 CHF ₂ C3H7 CI H

A-339 Br CHs CI H A-380 C3H7 C3H7 CI H

A-340 CN CHs CI H A-381 CONH2 C3H7 CI H

A-341 CHs CHs CI H A-382 SCHs C3H7 CI H

A-342 CFs CHs CI H A-383 SOCHs C3H7 CI H

A-343 CHF ₂ CHs CI H A-384 OCHs C3H7 CI H

A-344 C3H7 CHs CI H A-385 CI CONH2 CI H

A-345 CONH2 CHs CI H A-386 F CONH2 CI H line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-387 Br CONH2 CI H A-428 C3H7 OCHs CI H

A-388 CN CONH2 CI H A-429 CONH2 OCHs CI H

A-389 CHs CONH2 CI H A-430 SCHs OCHs CI H

A-390 CFs CONH2 CI H A-431 SOCHs OCHs CI H

A-391 CHF ₂ CONH2 CI H A-432 OCHs OCHs CI H

A-392 C3H7 CONH2 CI H A-433 CI CI CN H

A-393 CONH2 CONH2 CI H A-434 F CI CN H

A-394 SCHs CONH2 CI H A-435 Br CI CN H

A-395 SOCHs CONH2 CI H A-436 CN CI CN H

A-396 OCHs CONH2 CI H A-437 CHs CI CN H

A-397 CI SCHs CI H A-438 CFs CI CN H

A-398 F SCHs CI H A-439 CHF ₂ CI CN H

A-399 Br SCHs CI H A-440 C3H7 CI CN H

A-400 CN SCHs CI H A-441 CONH2 CI CN H

A-401 CHs SCHs CI H A-442 SCHs CI CN H

A-402 CFs SCHs CI H A-443 SOCHs CI CN H

A-403 CHF ₂ SCHs CI H A-444 OCHs CI CN H

A-404 C3H7 SCHs CI H A-445 CI F CN H

A-405 CONH2 SCHs CI H A-446 F F CN H

A-406 SCHs SCHs CI H A-447 Br F CN H

A-407 SOCHs SCHs CI H A-448 CN F CN H

A-408 OCHs SCHs CI H A-449 CHs F CN H

A-409 CI SOCHs CI H A-450 CFs F CN H

A-410 F SOCHs CI H A-451 CHF ₂ F CN H

A-41 1 Br SOCHs CI H A-452 C3H7 F CN H

A-412 CN SOCHs CI H A-453 CONH2 F CN H

A-413 CHs SOCHs CI H A-454 SCHs F CN H

A-414 CFs SOCHs CI H A-455 SOCHs F CN H

A-415 CHF ₂ SOCHs CI H A-456 OCHs F CN H

A-416 C3H7 SOCHs CI H A-457 CI Br CN H

A-417 CONH2 SOCHs CI H A-458 F Br CN H

A-418 SCHs SOCHs CI H A-459 Br Br CN H

A-419 SOCHs SOCHs CI H A-460 CN Br CN H

A-420 OCHs SOCHs CI H A-461 CHs Br CN H

A-421 CI OCHs CI H A-462 CFs Br CN H

A-422 F OCHs CI H A-463 CHF ₂ Br CN H

A-423 Br OCHs CI H A-464 C3H7 Br CN H

A-424 CN OCHs CI H A-465 CONH2 Br CN H

A-425 CHs OCHs CI H A-466 SCHs Br CN H

A-426 CFs OCHs CI H A-467 SOCHs Br CN H

A-427 CHF ₂ OCHs CI H A-468 OCHs Br CN H line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-469 CI CN CN H A-510 CFs CHF ₂ CN H

A-470 F CN CN H A-51 1 CHF ₂ CHF ₂ CN H

A-471 Br CN CN H A-512 C3H7 CHF ₂ CN H

A-472 CN CN CN H A-513 CONH2 CHF ₂ CN H

A-473 CHs CN CN H A-514 SCHs CHF ₂ CN H

A-474 CFs CN CN H A-515 SOCHs CHF ₂ CN H

A-475 CHF ₂ CN CN H A-516 OCHs CHF ₂ CN H

A-476 C3H7 CN CN H A-517 CI C3H7 CN H

A-477 CONH2 CN CN H A-518 F C3H7 CN H

A-478 SCHs CN CN H A-519 Br C3H7 CN H

A-479 SOCHs CN CN H A-520 CN C3H7 CN H

A-480 OCHs CN CN H A-521 CHs C3H7 CN H

A-481 CI CHs CN H A-522 CFs C3H7 CN H

A-482 F CHs CN H A-523 CHF ₂ C3H7 CN H

A-483 Br CHs CN H A-524 C3H7 C3H7 CN H

A-484 CN CHs CN H A-525 CONH2 C3H7 CN H

A-485 CHs CHs CN H A-526 SCHs C3H7 CN H

A-486 CFs CHs CN H A-527 SOCHs C3H7 CN H

A-487 CHF ₂ CHs CN H A-528 OCHs C3H7 CN H

A-488 C3H7 CHs CN H A-529 CI CONH2 CN H

A-489 CONH2 CHs CN H A-530 F CONH2 CN H

A-490 SCHs CHs CN H A-531 Br CONH2 CN H

A-491 SOCHs CHs CN H A-532 CN CONH2 CN H

A-492 OCHs CHs CN H A-533 CHs CONH2 CN H

A-493 CI CFs CN H A-534 CFs CONH2 CN H

A-494 F CFs CN H A-535 CHF ₂ CONH2 CN H

A-495 Br CFs CN H A-536 C3H7 CONH2 CN H

A-496 CN CFs CN H A-537 CONH2 CONH2 CN H

A-497 CHs CFs CN H A-538 SCHs CONH2 CN H

A-498 CFs CFs CN H A-539 SOCHs CONH2 CN H

A-499 CHF ₂ CFs CN H A-540 OCHs CONH2 CN H

A-500 C3H7 CFs CN H A-541 CI SCHs CN H

A-501 CONH2 CFs CN H A-542 F SCHs CN H

A-502 SCHs CFs CN H A-543 Br SCHs CN H

A-503 SOCHs CFs CN H A-544 CN SCHs CN H

A-504 OCHs CFs CN H A-545 CHs SCHs CN H

A-505 CI CHF ₂ CN H A-546 CFs SCHs CN H

A-506 F CHF ₂ CN H A-547 CHF ₂ SCHs CN H

A-507 Br CHF ₂ CN H A-548 C3H7 SCHs CN H

A-508 CN CHF ₂ CN H A-549 CONH2 SCHs CN H

A-509 CHs CHF ₂ CN H A-550 SCHs SCHs CN H line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-551 SOCHs SCHs CN H A-592 CN F CHs H

A-552 OCH3 SCHs CN H A-593 CHs F CHs H

A-553 CI SOCHs CN H A-594 CFs F CHs H

A-554 F SOCHs CN H A-595 CHF ₂ F CHs H

A-555 Br SOCHs CN H A-596 C3H7 F CHs H

A-556 CN SOCHs CN H A-597 CONH2 F CHs H

A-557 CHs SOCHs CN H A-598 SCHs F CHs H

A-558 CF ₃ SOCHs CN H A-599 SOCHs F CHs H

A-559 CHF ₂ SOCHs CN H A-600 OCHs F CHs H

A-560 C3H7 SOCHs CN H A-601 CI Br CHs H

A-561 CONH2 SOCHs CN H A-602 F Br CHs H

A-562 SCHs SOCHs CN H A-603 Br Br CHs H

A-563 SOCHs SOCHs CN H A-604 CN Br CHs H

A-564 OCH3 SOCHs CN H A-605 CHs Br CHs H

A-565 CI OCHs CN H A-606 CFs Br CHs H

A-566 F OCHs CN H A-607 CHF ₂ Br CHs H

A-567 Br OCHs CN H A-608 C3H7 Br CHs H

A-568 CN OCHs CN H A-609 CONH2 Br CHs H

A-569 CHs OCHs CN H A-610 SCHs Br CHs H

A-570 CF ₃ OCHs CN H A-61 1 SOCHs Br CHs H

A-571 CHF ₂ OCHs CN H A-612 OCHs Br CHs H

A-572 C3H7 OCHs CN H A-613 CI CN CHs H

A-573 CONH2 OCHs CN H A-614 F CN CHs H

A-574 SCHs OCHs CN H A-615 Br CN CHs H

A-575 SOCHs OCHs CN H A-616 CN CN CHs H

A-576 OCHs OCHs CN H A-617 CHs CN CHs H

A-577 CI CI CHs H A-618 CFs CN CHs H

A-578 F CI CHs H A-619 CHF ₂ CN CHs H

A-579 Br CI CHs H A-620 C3H7 CN CHs H

A-580 CN CI CHs H A-621 CONH2 CN CHs H

A-581 CHs CI CHs H A-622 SCHs CN CHs H

A-582 CFs CI CHs H A-623 SOCHs CN CHs H

A-583 CHF ₂ CI CHs H A-624 OCHs CN CHs H

A-584 C3H7 CI CHs H A-625 CI CHs CHs H

A-585 CONH2 CI CHs H A-626 F CHs CHs H

A-586 SCHs CI CHs H A-627 Br CHs CHs H

A-587 SOCHs CI CHs H A-628 CN CHs CHs H

A-588 OCHs CI CHs H A-629 CHs CHs CHs H

A-589 CI F CHs H A-630 CFs CHs CHs H

A-590 F F CHs H A-631 CHF ₂ CHs CHs H

A-591 Br F CHs H A-632 C3H7 CHs CHs H line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-633 CONH ₂ CHs CHs H A-674 F CONH2 CHs H

A-634 SCHs CHs CHs H A-675 Br CONH2 CHs H

A-635 SOCH3 CHs CHs H A-676 CN CONH2 CHs H

A-636 OCH3 CHs CHs H A-677 CHs CONH2 CHs H

A-637 CI CFs CHs H A-678 CFs CONH2 CHs H

A-638 F CFs CHs H A-679 CHF ₂ CONH2 CHs H

A-639 Br CFs CHs H A-680 C3H7 CONH2 CHs H

A-640 CN CFs CHs H A-681 CONH2 CONH2 CHs H

A-641 CHs CFs CHs H A-682 SCHs CONH2 CHs H

A-642 CFs CFs CHs H A-683 SOCHs CONH2 CHs H

A-643 CHF ₂ CFs CHs H A-684 OCHs CONH2 CHs H

A-644 C3H7 CFs CHs H A-685 CI SCHs CHs H

A-645 CONH2 CFs CHs H A-686 F SCHs CHs H

A-646 SCHs CFs CHs H A-687 Br SCHs CHs H

A-647 SOCHs CFs CHs H A-688 CN SCHs CHs H

A-648 OCHs CFs CHs H A-689 CHs SCHs CHs H

A-649 CI CHF ₂ CHs H A-690 CFs SCHs CHs H

A-650 F CHF ₂ CHs H A-691 CHF ₂ SCHs CHs H

A-651 Br CHF ₂ CHs H A-692 C3H7 SCHs CHs H

A-652 CN CHF ₂ CHs H A-693 CONH2 SCHs CHs H

A-653 CHs CHF ₂ CHs H A-694 SCHs SCHs CHs H

A-654 CFs CHF ₂ CHs H A-695 SOCHs SCHs CHs H

A-655 CHF ₂ CHF ₂ CHs H A-696 OCHs SCHs CHs H

A-656 C3H7 CHF ₂ CHs H A-697 CI SOCHs CHs H

A-657 CONH2 CHF ₂ CHs H A-698 F SOCHs CHs H

A-658 SCHs CHF ₂ CHs H A-699 Br SOCHs CHs H

A-659 SOCHs CHF ₂ CHs H A-700 CN SOCHs CHs H

A-660 OCHs CHF ₂ CHs H A-701 CHs SOCHs CHs H

A-661 CI C3H7 CHs H A-702 CFs SOCHs CHs H

A-662 F C3H7 CHs H A-703 CHF ₂ SOCHs CHs H

A-663 Br C3H7 CHs H A-704 C3H7 SOCHs CHs H

A-664 CN C3H7 CHs H A-705 CONH2 SOCHs CHs H

A-665 CHs C3H7 CHs H A-706 SCHs SOCHs CHs H

A-666 CFs C3H7 CHs H A-707 SOCHs SOCHs CHs H

A-667 CHF ₂ C3H7 CHs H A-708 OCHs SOCHs CHs H

A-668 C3H7 C3H7 CHs H A-709 CI OCHs CHs H

A-669 CONH2 C3H7 CHs H A-710 F OCHs CHs H

A-670 SCHs C3H7 CHs H A-71 1 Br OCHs CHs H

A-671 SOCHs C3H7 CHs H A-712 CN OCHs CHs H

A-672 OCHs C3H7 CHs H A-713 CHs OCHs CHs H

A-673 CI CONH2 CHs H A-714 CFs OCHs CHs H line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-715 CHF ₂ OCHs CHs H A-756 OCHs Br H F

A-716 C3H7 OCHs CHs H A-757 CI CN H F

A-717 CONH2 OCHs CHs H A-758 F CN H F

A-718 SCHs OCHs CHs H A-759 Br CN H F

A-719 SOCH3 OCHs CHs H A-760 CN CN H F

A-720 OCH3 OCHs CHs H A-761 CHs CN H F

A-721 CI CI H F A-762 CFs CN H F

A-722 F CI H F A-763 CHF ₂ CN H F

A-723 Br CI H F A-764 C3H7 CN H F

A-724 CN CI H F A-765 CONH2 CN H F

A-725 CHs CI H F A-766 SCHs CN H F

A-726 CFs CI H F A-767 SOCHs CN H F

A-727 CHF ₂ CI H F A-768 OCHs CN H F

A-728 C3H7 CI H F A-769 CI CHs H F

A-729 CONH2 CI H F A-770 F CHs H F

A-730 SCHs CI H F A-771 Br CHs H F

A-731 SOCHs CI H F A-772 CN CHs H F

A-732 OCHs CI H F A-773 CHs CHs H F

A-733 CI F H F A-774 CFs CHs H F

A-734 F F H F A-775 CHF ₂ CHs H F

A-735 Br F H F A-776 C3H7 CHs H F

A-736 CN F H F A-777 CONH2 CHs H F

A-737 CHs F H F A-778 SCHs CHs H F

A-738 CFs F H F A-779 SOCHs CHs H F

A-739 CHF ₂ F H F A-780 OCHs CHs H F

A-740 C3H7 F H F A-781 CI CFs H F

A-741 CONH2 F H F A-782 F CFs H F

A-742 SCHs F H F A-783 Br CFs H F

A-743 SOCHs F H F A-784 CN CFs H F

A-744 OCHs F H F A-785 CHs CFs H F

A-745 CI Br H F A-786 CFs CFs H F

A-746 F Br H F A-787 CHF ₂ CFs H F

A-747 Br Br H F A-788 C3H7 CFs H F

A-748 CN Br H F A-789 CONH2 CFs H F

A-749 CHs Br H F A-790 SCHs CFs H F

A-750 CFs Br H F A-791 SOCHs CFs H F

A-751 CHF ₂ Br H F A-792 OCHs CFs H F

A-752 C3H7 Br H F A-793 CI CHF ₂ H F

A-753 CONH2 Br H F A-794 F CHF ₂ H F

A-754 SCHs Br H F A-795 Br CHF ₂ H F

A-755 SOCHs Br H F A-796 CN CHF ₂ H F line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-797 CHs CHF ₂ H F A-838 SCHs SCHs H F

A-798 CFs CHF ₂ H F A-839 SOCHs SCHs H F

A-799 CHF ₂ CHF ₂ H F A-840 OCHs SCHs H F

A-800 C3H7 CHF ₂ H F A-841 CI SOCHs H F

A-801 CONH2 CHF ₂ H F A-842 F SOCHs H F

A-802 SCHs CHF ₂ H F A-843 Br SOCHs H F

A-803 SOCHs CHF ₂ H F A-844 CN SOCHs H F

A-804 OCHs CHF ₂ H F A-845 CHs SOCHs H F

A-805 CI C3H7 H F A-846 CFs SOCHs H F

A-806 F C3H7 H F A-847 CHF ₂ SOCHs H F

A-807 Br C3H7 H F A-848 C3H7 SOCHs H F

A-808 CN C3H7 H F A-849 CONH2 SOCHs H F

A-809 CHs C3H7 H F A-850 SCHs SOCHs H F

A-810 CFs C3H7 H F A-851 SOCHs SOCHs H F

A-81 1 CHF ₂ C3H7 H F A-852 OCHs SOCHs H F

A-812 C3H7 C3H7 H F A-853 CI OCHs H F

A-813 CONH2 C3H7 H F A-854 F OCHs H F

A-814 SCHs C3H7 H F A-855 Br OCHs H F

A-815 SOCHs C3H7 H F A-856 CN OCHs H F

A-816 OCHs C3H7 H F A-857 CHs OCHs H F

A-817 CI CONH2 H F A-858 CFs OCHs H F

A-818 F CONH2 H F A-859 CHF ₂ OCHs H F

A-819 Br CONH2 H F A-860 C3H7 OCHs H F

A-820 CN CONH2 H F A-861 CONH2 OCHs H F

A-821 CHs CONH2 H F A-862 SCHs OCHs H F

A-822 CFs CONH2 H F A-863 SOCHs OCHs H F

A-823 CHF ₂ CONH2 H F A-864 OCHs OCHs H F

A-824 C3H7 CONH2 H F A-865 CI CI F F

A-825 CONH2 CONH2 H F A-866 F CI F F

A-826 SCHs CONH2 H F A-867 Br CI F F

A-827 SOCHs CONH2 H F A-868 CN CI F F

A-828 OCHs CONH2 H F A-869 CHs CI F F

A-829 CI SCHs H F A-870 CFs CI F F

A-830 F SCHs H F A-871 CHF ₂ CI F F

A-831 Br SCHs H F A-872 C3H7 CI F F

A-832 CN SCHs H F A-873 CONH2 CI F F

A-833 CHs SCHs H F A-874 SCHs CI F F

A-834 CFs SCHs H F A-875 SOCHs CI F F

A-835 CHF ₂ SCHs H F A-876 OCHs CI F F

A-836 C3H7 SCHs H F A-877 CI F F F

A-837 CONH2 SCHs H F A-878 F F F F line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-879 Br F F F A-920 C3H7 CHs F F

A-880 CN F F F A-921 CONH2 CHs F F

A-881 CHs F F F A-922 SCHs CHs F F

A-882 CFs F F F A-923 SOCHs CHs F F

A-883 CHF ₂ F F F A-924 OCHs CHs F F

A-884 C3H7 F F F A-925 CI CFs F F

A-885 CONH2 F F F A-926 F CFs F F

A-886 SCHs F F F A-927 Br CFs F F

A-887 SOCHs F F F A-928 CN CFs F F

A-888 OCHs F F F A-929 CHs CFs F F

A-889 CI Br F F A-930 CFs CFs F F

A-890 F Br F F A-931 CHF ₂ CFs F F

A-891 Br Br F F A-932 C3H7 CFs F F

A-892 CN Br F F A-933 CONH2 CFs F F

A-893 CHs Br F F A-934 SCHs CFs F F

A-894 CFs Br F F A-935 SOCHs CFs F F

A-895 CHF ₂ Br F F A-936 OCHs CFs F F

A-896 C3H7 Br F F A-937 CI CHF ₂ F F

A-897 CONH2 Br F F A-938 F CHF ₂ F F

A-898 SCHs Br F F A-939 Br CHF ₂ F F

A-899 SOCHs Br F F A-940 CN CHF ₂ F F

A-900 OCHs Br F F A-941 CHs CHF ₂ F F

A-901 CI CN F F A-942 CFs CHF ₂ F F

A-902 F CN F F A-943 CHF ₂ CHF ₂ F F

A-903 Br CN F F A-944 C3H7 CHF ₂ F F

A-904 CN CN F F A-945 CONH2 CHF ₂ F F

A-905 CHs CN F F A-946 SCHs CHF ₂ F F

A-906 CFs CN F F A-947 SOCHs CHF ₂ F F

A-907 CHF ₂ CN F F A-948 OCHs CHF ₂ F F

A-908 C3H7 CN F F A-949 CI C3H7 F F

A-909 CONH2 CN F F A-950 F C3H7 F F

A-910 SCHs CN F F A-951 Br C3H7 F F

A-91 1 SOCHs CN F F A-952 CN C3H7 F F

A-912 OCHs CN F F A-953 CHs C3H7 F F

A-913 CI CHs F F A-954 CFs C3H7 F F

A-914 F CHs F F A-955 CHF ₂ C3H7 F F

A-915 Br CHs F F A-956 C3H7 C3H7 F F

A-916 CN CHs F F A-957 CONH2 C3H7 F F

A-917 CHs CHs F F A-958 SCHs C3H7 F F

A-918 CFs CHs F F A-959 SOCHs C3H7 F F

A-919 CHF ₂ CHs F F A-960 OCHs C3H7 F F line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-961 CI CONH2 F F A-1002 CFs OCHs F F

A-962 F CONH2 F F A-1003 CHF ₂ OCHs F F

A-963 Br CONH2 F F A-1004 C3H7 OCHs F F

A-964 CN CONH2 F F A-1005 CONH2 OCHs F F

A-965 CHs CONH2 F F A-1006 SCHs OCHs F F

A-966 CFs CONH2 F F A-1007 SOCHs OCHs F F

A-967 CHF ₂ CONH2 F F A-1008 OCHs OCHs F F

A-968 C3H7 CONH2 F F A-1009 CI CI CI F

A-969 CONH2 CONH2 F F A-1010 F CI CI F

A-970 SCHs CONH2 F F A-101 1 Br CI CI F

A-971 SOCHs CONH2 F F A-1012 CN CI CI F

A-972 OCHs CONH2 F F A-1013 CHs CI CI F

A-973 CI SCHs F F A-1014 CFs CI CI F

A-974 F SCHs F F A-1015 CHF ₂ CI CI F

A-975 Br SCHs F F A-1016 C3H7 CI CI F

A-976 CN SCHs F F A-1017 CONH2 CI CI F

A-977 CHs SCHs F F A-1018 SCHs CI CI F

A-978 CFs SCHs F F A-1019 SOCHs CI CI F

A-979 CHF ₂ SCHs F F A-1020 OCHs CI CI F

A-980 C3H7 SCHs F F A-1021 CI F CI F

A-981 CONH2 SCHs F F A-1022 F F CI F

A-982 SCHs SCHs F F A-1023 Br F CI F

A-983 SOCHs SCHs F F A-1024 CN F CI F

A-984 OCHs SCHs F F A-1025 CHs F CI F

A-985 CI SOCHs F F A-1026 CFs F CI F

A-986 F SOCHs F F A-1027 CHF ₂ F CI F

A-987 Br SOCHs F F A-1028 C3H7 F CI F

A-988 CN SOCHs F F A-1029 CONH2 F CI F

A-989 CHs SOCHs F F A-1030 SCHs F CI F

A-990 CFs SOCHs F F A-1031 SOCHs F CI F

A-991 CHF ₂ SOCHs F F A-1032 OCHs F CI F

A-992 C3H7 SOCHs F F A-1033 CI Br CI F

A-993 CONH2 SOCHs F F A-1034 F Br CI F

A-994 SCHs SOCHs F F A-1035 Br Br CI F

A-995 SOCHs SOCHs F F A-1036 CN Br CI F

A-996 OCHs SOCHs F F A-1037 CHs Br CI F

A-997 CI OCHs F F A-1038 CFs Br CI F

A-998 F OCHs F F A-1039 CHF ₂ Br CI F

A-999 Br OCHs F F A-1040 C3H7 Br CI F

A-1000 CN OCHs F F A-1041 CONH2 Br CI F

A-1001 CHs OCHs F F A-1042 SCHs Br CI F line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1043 SOCHs Br CI F A-1084 CN CHF ₂ CI F

A-1044 OCH3 Br CI F A-1085 CHs CHF ₂ CI F

A-1045 CI CN CI F A-1086 CFs CHF ₂ CI F

A-1046 F CN CI F A-1087 CHF ₂ CHF ₂ CI F

A-1047 Br CN CI F A-1088 C3H7 CHF ₂ CI F

A-1048 CN CN CI F A-1089 CONH2 CHF ₂ CI F

A-1049 CHs CN CI F A-1090 SCHs CHF ₂ CI F

A-1050 CFs CN CI F A-1091 SOCHs CHF ₂ CI F

A-1051 CHF ₂ CN CI F A-1092 OCHs CHF ₂ CI F

A-1052 C3H7 CN CI F A-1093 CI C3H7 CI F

A-1053 CONH2 CN CI F A-1094 F C3H7 CI F

A-1054 SCHs CN CI F A-1095 Br C3H7 CI F

A-1055 SOCHs CN CI F A-1096 CN C3H7 CI F

A-1056 OCHs CN CI F A-1097 CHs C3H7 CI F

A-1057 CI CHs CI F A-1098 CFs C3H7 CI F

A-1058 F CHs CI F A-1099 CHF ₂ C3H7 CI F

A-1059 Br CHs CI F A-1 100 C3H7 C3H7 CI F

A-1060 CN CHs CI F A-1 101 CONH2 C3H7 CI F

A-1061 CHs CHs CI F A-1 102 SCHs C3H7 CI F

A-1062 CFs CHs CI F A-1 103 SOCHs C3H7 CI F

A-1063 CHF ₂ CHs CI F A-1 104 OCHs C3H7 CI F

A-1064 C3H7 CHs CI F A-1 105 CI CONH2 CI F

A-1065 CONH2 CHs CI F A-1 106 F CONH2 CI F

A-1066 SCHs CHs CI F A-1 107 Br CONH2 CI F

A-1067 SOCHs CHs CI F A-1 108 CN CONH2 CI F

A-1068 OCHs CHs CI F A-1 109 CHs CONH2 CI F

A-1069 CI CFs CI F A-1 1 10 CFs CONH2 CI F

A-1070 F CFs CI F A-1 1 1 1 CHF ₂ CONH2 CI F

A-1071 Br CFs CI F A-1 1 12 C3H7 CONH2 CI F

A-1072 CN CFs CI F A-1 1 13 CONH2 CONH2 CI F

A-1073 CHs CFs CI F A-1 1 14 SCHs CONH2 CI F

A-1074 CFs CFs CI F A-1 1 15 SOCHs CONH2 CI F

A-1075 CHF ₂ CFs CI F A-1 1 16 OCHs CONH2 CI F

A-1076 C3H7 CFs CI F A-1 1 17 CI SCHs CI F

A-1077 CONH2 CFs CI F A-1 1 18 F SCHs CI F

A-1078 SCHs CFs CI F A-1 1 19 Br SCHs CI F

A-1079 SOCHs CFs CI F A-1 120 CN SCHs CI F

A-1080 OCHs CFs CI F A-1 121 CHs SCHs CI F

A-1081 CI CHF ₂ CI F A-1 122 CFs SCHs CI F

A-1082 F CHF ₂ CI F A-1 123 CHF ₂ SCHs CI F

A-1083 Br CHF ₂ CI F A-1 124 C3H7 SCHs CI F line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1125 CONH ₂ SCHs CI F A-1166 F F CN F

A-1126 SCHs SCHs CI F A-1167 Br F CN F

A-1127 SOCH3 SCHs CI F A-1168 CN F CN F

A-1128 OCH3 SCHs CI F A-1169 CHs F CN F

A-1129 CI SOCHs CI F A-1170 CFs F CN F

A-1130 F SOCHs CI F A-1171 CHF ₂ F CN F

A-1131 Br SOCHs CI F A-1172 C3H7 F CN F

A-1132 CN SOCHs CI F A-1173 CONH2 F CN F

A-1133 CHs SOCHs CI F A-1174 SCHs F CN F

A-1134 CFs SOCHs CI F A-1175 SOCHs F CN F

A-1135 CHF ₂ SOCHs CI F A-1176 OCHs F CN F

A-1136 C3H7 SOCHs CI F A-1177 CI Br CN F

A-1137 CONH2 SOCHs CI F A-1178 F Br CN F

A-1138 SCHs SOCHs CI F A-1179 Br Br CN F

A-1139 SOCHs SOCHs CI F A-1180 CN Br CN F

A-1140 OCHs SOCHs CI F A-1181 CHs Br CN F

A-1141 CI OCHs CI F A-1182 CFs Br CN F

A-1142 F OCHs CI F A-1183 CHF ₂ Br CN F

A-1143 Br OCHs CI F A-1184 C3H7 Br CN F

A-1144 CN OCHs CI F A-1185 CONH2 Br CN F

A-1145 CHs OCHs CI F A-1186 SCHs Br CN F

A-1146 CFs OCHs CI F A-1187 SOCHs Br CN F

A-1147 CHF ₂ OCHs CI F A-1188 OCHs Br CN F

A-1148 C3H7 OCHs CI F A-1189 CI CN CN F

A-1149 CONH2 OCHs CI F A-1190 F CN CN F

A-1150 SCHs OCHs CI F A-1191 Br CN CN F

A-1151 SOCHs OCHs CI F A-1192 CN CN CN F

A-1152 OCHs OCHs CI F A-1193 CHs CN CN F

A-1153 CI CI CN F A-1194 CFs CN CN F

A-1154 F CI CN F A-1195 CHF ₂ CN CN F

A-1155 Br CI CN F A-1196 C3H7 CN CN F

A-1156 CN CI CN F A-1197 CONH2 CN CN F

A-1157 CHs CI CN F A-1198 SCHs CN CN F

A-1158 CFs CI CN F A-1199 SOCHs CN CN F

A-1159 CHF ₂ CI CN F A-1200 OCHs CN CN F

A-1160 C3H7 CI CN F A-1201 CI CHs CN F

A-1161 CONH2 CI CN F A-1202 F CHs CN F

A-1162 SCHs CI CN F A-1203 Br CHs CN F

A-1163 SOCHs CI CN F A-1204 CN CHs CN F

A-1164 OCHs CI CN F A-1205 CHs CHs CN F

A-1165 CI F CN F A-1206 CFs CHs CN F line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1207 CHF ₂ CHs CN F A-1248 OCHs C3H7 CN F

A-1208 C3H7 CHs CN F A-1249 CI CONH2 CN F

A-1209 CONH2 CHs CN F A-1250 F CONH2 CN F

A-1210 SCHs CHs CN F A-1251 Br CONH2 CN F

A-121 1 SOCH3 CHs CN F A-1252 CN CONH2 CN F

A-1212 OCH3 CHs CN F A-1253 CHs CONH2 CN F

A-1213 CI CFs CN F A-1254 CFs CONH2 CN F

A-1214 F CFs CN F A-1255 CHF ₂ CONH2 CN F

A-1215 Br CFs CN F A-1256 C3H7 CONH2 CN F

A-1216 CN CFs CN F A-1257 CONH2 CONH2 CN F

A-1217 CHs CFs CN F A-1258 SCHs CONH2 CN F

A-1218 CFs CFs CN F A-1259 SOCHs CONH2 CN F

A-1219 CHF ₂ CFs CN F A-1260 OCHs CONH2 CN F

A-1220 C3H7 CFs CN F A-1261 CI SCHs CN F

A-1221 CONH2 CFs CN F A-1262 F SCHs CN F

A-1222 SCHs CFs CN F A-1263 Br SCHs CN F

A-1223 SOCHs CFs CN F A-1264 CN SCHs CN F

A-1224 OCHs CFs CN F A-1265 CHs SCHs CN F

A-1225 CI CHF ₂ CN F A-1266 CFs SCHs CN F

A-1226 F CHF ₂ CN F A-1267 CHF ₂ SCHs CN F

A-1227 Br CHF ₂ CN F A-1268 C3H7 SCHs CN F

A-1228 CN CHF ₂ CN F A-1269 CONH2 SCHs CN F

A-1229 CHs CHF ₂ CN F A-1270 SCHs SCHs CN F

A-1230 CFs CHF ₂ CN F A-1271 SOCHs SCHs CN F

A-1231 CHF ₂ CHF ₂ CN F A-1272 OCHs SCHs CN F

A-1232 C3H7 CHF ₂ CN F A-1273 CI SOCHs CN F

A-1233 CONH2 CHF ₂ CN F A-1274 F SOCHs CN F

A-1234 SCHs CHF ₂ CN F A-1275 Br SOCHs CN F

A-1235 SOCHs CHF ₂ CN F A-1276 CN SOCHs CN F

A-1236 OCHs CHF ₂ CN F A-1277 CHs SOCHs CN F

A-1237 CI C3H7 CN F A-1278 CFs SOCHs CN F

A-1238 F C3H7 CN F A-1279 CHF ₂ SOCHs CN F

A-1239 Br C3H7 CN F A-1280 C3H7 SOCHs CN F

A-1240 CN C3H7 CN F A-1281 CONH2 SOCHs CN F

A-1241 CHs C3H7 CN F A-1282 SCHs SOCHs CN F

A-1242 CFs C3H7 CN F A-1283 SOCHs SOCHs CN F

A-1243 CHF ₂ C3H7 CN F A-1284 OCHs SOCHs CN F

A-1244 C3H7 C3H7 CN F A-1285 CI OCHs CN F

A-1245 CONH2 C3H7 CN F A-1286 F OCHs CN F

A-1246 SCHs C3H7 CN F A-1287 Br OCHs CN F

A-1247 SOCHs C3H7 CN F A-1288 CN OCHs CN F line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1289 CHs OCHs CN F A-1330 SCHs Br CHs F

A-1290 CFs OCHs CN F A-1331 SOCHs Br CHs F

A-1291 CHF ₂ OCHs CN F A-1332 OCHs Br CHs F

A-1292 C3H7 OCHs CN F A-1333 CI CN CHs F

A-1293 CONH2 OCHs CN F A-1334 F CN CHs F

A-1294 SCHs OCHs CN F A-1335 Br CN CHs F

A-1295 SOCHs OCHs CN F A-1336 CN CN CHs F

A-1296 OCHs OCHs CN F A-1337 CHs CN CHs F

A-1297 CI CI CHs F A-1338 CFs CN CHs F

A-1298 F CI CHs F A-1339 CHF ₂ CN CHs F

A-1299 Br CI CHs F A-1340 C3H7 CN CHs F

A-1300 CN CI CHs F A-1341 CONH2 CN CHs F

A-1301 CHs CI CHs F A-1342 SCHs CN CHs F

A-1302 CFs CI CHs F A-1343 SOCHs CN CHs F

A-1303 CHF ₂ CI CHs F A-1344 OCHs CN CHs F

A-1304 C3H7 CI CHs F A-1345 CI CHs CHs F

A-1305 CONH2 CI CHs F A-1346 F CHs CHs F

A-1306 SCHs CI CHs F A-1347 Br CHs CHs F

A-1307 SOCHs CI CHs F A-1348 CN CHs CHs F

A-1308 OCHs CI CHs F A-1349 CHs CHs CHs F

A-1309 CI F CHs F A-1350 CFs CHs CHs F

A-1310 F F CHs F A-1351 CHF ₂ CHs CHs F

A-131 1 Br F CHs F A-1352 C3H7 CHs CHs F

A-1312 CN F CHs F A-1353 CONH2 CHs CHs F

A-1313 CHs F CHs F A-1354 SCHs CHs CHs F

A-1314 CFs F CHs F A-1355 SOCHs CHs CHs F

A-1315 CHF ₂ F CHs F A-1356 OCHs CHs CHs F

A-1316 C3H7 F CHs F A-1357 CI CFs CHs F

A-1317 CONH2 F CHs F A-1358 F CFs CHs F

A-1318 SCHs F CHs F A-1359 Br CFs CHs F

A-1319 SOCHs F CHs F A-1360 CN CFs CHs F

A-1320 OCHs F CHs F A-1361 CHs CFs CHs F

A-1321 CI Br CHs F A-1362 CFs CFs CHs F

A-1322 F Br CHs F A-1363 CHF ₂ CFs CHs F

A-1323 Br Br CHs F A-1364 C3H7 CFs CHs F

A-1324 CN Br CHs F A-1365 CONH2 CFs CHs F

A-1325 CHs Br CHs F A-1366 SCHs CFs CHs F

A-1326 CFs Br CHs F A-1367 SOCHs CFs CHs F

A-1327 CHF ₂ Br CHs F A-1368 OCHs CFs CHs F

A-1328 C3H7 Br CHs F A-1369 CI CHF ₂ CHs F

A-1329 CONH2 Br CHs F A-1370 F CHF ₂ CHs F line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1371 Br CHF ₂ CHs F A-1412 C3H7 SCHs CHs F

A-1372 CN CHF ₂ CHs F A-1413 CONH2 SCHs CHs F

A-1373 CHs CHF ₂ CHs F A-1414 SCHs SCHs CHs F

A-1374 CFs CHF ₂ CHs F A-1415 SOCHs SCHs CHs F

A-1375 CHF ₂ CHF ₂ CHs F A-1416 OCHs SCHs CHs F

A-1376 C3H7 CHF ₂ CHs F A-1417 CI SOCHs CHs F

A-1377 CONH2 CHF ₂ CHs F A-1418 F SOCHs CHs F

A-1378 SCHs CHF ₂ CHs F A-1419 Br SOCHs CHs F

A-1379 SOCHs CHF ₂ CHs F A-1420 CN SOCHs CHs F

A-1380 OCHs CHF ₂ CHs F A-1421 CHs SOCHs CHs F

A-1381 CI C3H7 CHs F A-1422 CFs SOCHs CHs F

A-1382 F C3H7 CHs F A-1423 CHF ₂ SOCHs CHs F

A-1383 Br C3H7 CHs F A-1424 C3H7 SOCHs CHs F

A-1384 CN C3H7 CHs F A-1425 CONH2 SOCHs CHs F

A-1385 CHs C3H7 CHs F A-1426 SCHs SOCHs CHs F

A-1386 CFs C3H7 CHs F A-1427 SOCHs SOCHs CHs F

A-1387 CHF ₂ C3H7 CHs F A-1428 OCHs SOCHs CHs F

A-1388 C3H7 C3H7 CHs F A-1429 CI OCHs CHs F

A-1389 CONH2 C3H7 CHs F A-1430 F OCHs CHs F

A-1390 SCHs C3H7 CHs F A-1431 Br OCHs CHs F

A-1391 SOCHs C3H7 CHs F A-1432 CN OCHs CHs F

A-1392 OCHs C3H7 CHs F A-1433 CHs OCHs CHs F

A-1393 CI CONH2 CHs F A-1434 CFs OCHs CHs F

A-1394 F CONH2 CHs F A-1435 CHF ₂ OCHs CHs F

A-1395 Br CONH2 CHs F A-1436 C3H7 OCHs CHs F

A-1396 CN CONH2 CHs F A-1437 CONH2 OCHs CHs F

A-1397 CHs CONH2 CHs F A-1438 SCHs OCHs CHs F

A-1398 CFs CONH2 CHs F A-1439 SOCHs OCHs CHs F

A-1399 CHF ₂ CONH2 CHs F A-1440 OCHs OCHs CHs F

A-1400 C3H7 CONH2 CHs F A-1441 CI CI H CI

A-1401 CONH2 CONH2 CHs F A-1442 F CI H CI

A-1402 SCHs CONH2 CHs F A-1443 Br CI H CI

A-1403 SOCHs CONH2 CHs F A-1444 CN CI H CI

A-1404 OCHs CONH2 CHs F A-1445 CHs CI H CI

A-1405 CI SCHs CHs F A-1446 CFs CI H CI

A-1406 F SCHs CHs F A-1447 CHF ₂ CI H CI

A-1407 Br SCHs CHs F A-1448 C3H7 CI H CI

A-1408 CN SCHs CHs F A-1449 CONH2 CI H CI

A-1409 CHs SCHs CHs F A-1450 SCHs CI H CI

A-1410 CFs SCHs CHs F A-1451 SOCHs CI H CI

A-141 1 CHF ₂ SCHs CHs F A-1452 OCHs CI H CI line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1453 CI F H CI A-1494 CFs CHs H CI

A-1454 F F H CI A-1495 CHF ₂ CHs H CI

A- 1455 Br F H CI A-1496 C3H7 CHs H CI

A-1456 CN F H CI A-1497 CONH2 CHs H CI

A-1457 CHs F H CI A-1498 SCHs CHs H CI

A-1458 CFs F H CI A-1499 SOCHs CHs H CI

A-1459 CHF ₂ F H CI A-1500 OCHs CHs H CI

A-1460 CsH ₇ F H CI A-1501 CI CFs H CI

A-1461 CONH2 F H CI A-1502 F CFs H CI

A-1462 SCHs F H CI A-1503 Br CFs H CI

A-1463 SOCHs F H CI A-1504 CN CFs H CI

A-1464 OCHs F H CI A-1505 CHs CFs H CI

A-1465 CI Br H CI A-1506 CFs CFs H CI

A-1466 F Br H CI A-1507 CHF ₂ CFs H CI

A-1467 Br Br H CI A-1508 C3H7 CFs H CI

A-1468 CN Br H CI A-1509 CONH2 CFs H CI

A-1469 CHs Br H CI A-1510 SCHs CFs H CI

A-1470 CFs Br H CI A-151 1 SOCHs CFs H CI

A-1471 CHF ₂ Br H CI A-1512 OCHs CFs H CI

A-1472 C3H7 Br H CI A-1513 CI CHF ₂ H CI

A-1473 CONH2 Br H CI A-1514 F CHF ₂ H CI

A-1474 SCHs Br H CI A-1515 Br CHF ₂ H CI

A-1475 SOCHs Br H CI A-1516 CN CHF ₂ H CI

A-1476 OCHs Br H CI A-1517 CHs CHF ₂ H CI

A-1477 CI CN H CI A-1518 CFs CHF ₂ H CI

A-1478 F CN H CI A-1519 CHF ₂ CHF ₂ H CI

A-1479 Br CN H CI A-1520 C3H7 CHF ₂ H CI

A-1480 CN CN H CI A-1521 CONH2 CHF ₂ H CI

A-1481 CHs CN H CI A-1522 SCHs CHF ₂ H CI

A-1482 CFs CN H CI A-1523 SOCHs CHF ₂ H CI

A-1483 CHF ₂ CN H CI A-1524 OCHs CHF ₂ H CI

A-1484 C3H7 CN H CI A-1525 CI C3H7 H CI

A-1485 CONH2 CN H CI A-1526 F C3H7 H CI

A-1486 SCHs CN H CI A-1527 Br C3H7 H CI

A-1487 SOCHs CN H CI A-1528 CN C3H7 H CI

A-1488 OCHs CN H CI A-1529 CHs C3H7 H CI

A-1489 CI CHs H CI A-1530 CFs C3H7 H CI

A-1490 F CHs H CI A-1531 CHF ₂ C3H7 H CI

A-1491 Br CHs H CI A-1532 C3H7 C3H7 H CI

A-1492 CN CHs H CI A-1533 CONH2 C3H7 H CI

A-1493 CHs CHs H CI A-1534 SCHs C3H7 H CI line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1535 SOCHs C3H7 H CI A-1576 CN OCHs H CI

A-1536 OCHs C3H7 H CI A- 1577 CHs OCHs H CI

A-1537 CI CONH2 H CI A-1578 CFs OCHs H CI

A-1538 F CONH2 H CI A-1579 CHF ₂ OCHs H CI

A-1539 Br CONH2 H CI A-1580 C3H7 OCHs H CI

A-1540 CN CONH2 H CI A-1581 CONH2 OCHs H CI

A-1541 CHs CONH2 H CI A-1582 SCHs OCHs H CI

A-1542 CFs CONH2 H CI A-1583 SOCHs OCHs H CI

A-1543 CHF ₂ CONH2 H CI A-1584 OCHs OCHs H CI

A-1544 CsH ₇ CONH2 H CI A-1585 CI CI F CI

A-1545 CONH2 CONH2 H CI A-1586 F CI F CI

A-1546 SCHs CONH2 H CI A-1587 Br CI F CI

A-1547 SOCHs CONH2 H CI A-1588 CN CI F CI

A-1548 OCHs CONH2 H CI A-1589 CHs CI F CI

A-1549 CI SCHs H CI A-1590 CFs CI F CI

A-1550 F SCHs H CI A-1591 CHF ₂ CI F CI

A-1551 Br SCHs H CI A-1592 C3H7 CI F CI

A-1552 CN SCHs H CI A-1593 CONH2 CI F CI

A-1553 CHs SCHs H CI A-1594 SCHs CI F CI

A- 1554 CFs SCHs H CI A-1595 SOCHs CI F CI

A-1555 CHF ₂ SCHs H CI A-1596 OCHs CI F CI

A-1556 C3H7 SCHs H CI A-1597 CI F F CI

A- 1557 CONH2 SCHs H CI A-1598 F F F CI

A-1558 SCHs SCHs H CI A-1599 Br F F CI

A-1559 SOCHs SCHs H CI A-1600 CN F F CI

A-1560 OCHs SCHs H CI A-1601 CHs F F CI

A-1561 CI SOCHs H CI A-1602 CFs F F CI

A-1562 F SOCHs H CI A-1603 CHF ₂ F F CI

A-1563 Br SOCHs H CI A-1604 C3H7 F F CI

A-1564 CN SOCHs H CI A-1605 CONH2 F F CI

A-1565 CHs SOCHs H CI A-1606 SCHs F F CI

A-1566 CFs SOCHs H CI A-1607 SOCHs F F CI

A-1567 CHF ₂ SOCHs H CI A-1608 OCHs F F CI

A-1568 C3H7 SOCHs H CI A-1609 CI Br F CI

A-1569 CONH2 SOCHs H CI A-1610 F Br F CI

A-1570 SCHs SOCHs H CI A-161 1 Br Br F CI

A-1571 SOCHs SOCHs H CI A-1612 CN Br F CI

A-1572 OCHs SOCHs H CI A-1613 CHs Br F CI

A-1573 CI OCHs H CI A-1614 CFs Br F CI

A-1574 F OCHs H CI A-1615 CHF ₂ Br F CI

A- 1575 Br OCHs H CI A-1616 C3H7 Br F CI line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1617 CONH ₂ Br F CI A-1658 F CHF ₂ F CI

A-1618 SCHs Br F CI A-1659 Br CHF ₂ F CI

A-1619 SOCH3 Br F CI A-1660 CN CHF ₂ F CI

A-1620 OCH3 Br F CI A-1661 CHs CHF ₂ F CI

A-1621 CI CN F CI A-1662 CFs CHF ₂ F CI

A-1622 F CN F CI A-1663 CHF ₂ CHF ₂ F CI

A-1623 Br CN F CI A-1664 C3H7 CHF ₂ F CI

A-1624 CN CN F CI A-1665 CONH2 CHF ₂ F CI

A-1625 CHs CN F CI A-1666 SCHs CHF ₂ F CI

A-1626 CFs CN F CI A-1667 SOCHs CHF ₂ F CI

A-1627 CHF ₂ CN F CI A-1668 OCHs CHF ₂ F CI

A-1628 C3H7 CN F CI A-1669 CI C3H7 F CI

A-1629 CONH2 CN F CI A-1670 F C3H7 F CI

A-1630 SCHs CN F CI A-1671 Br C3H7 F CI

A-1631 SOCHs CN F CI A-1672 CN C3H7 F CI

A-1632 OCHs CN F CI A-1673 CHs C3H7 F CI

A-1633 CI CHs F CI A-1674 CFs C3H7 F CI

A-1634 F CHs F CI A-1675 CHF ₂ C3H7 F CI

A-1635 Br CHs F CI A-1676 C3H7 C3H7 F CI

A-1636 CN CHs F CI A-1677 CONH2 C3H7 F CI

A-1637 CHs CHs F CI A-1678 SCHs C3H7 F CI

A-1638 CFs CHs F CI A-1679 SOCHs C3H7 F CI

A-1639 CHF ₂ CHs F CI A-1680 OCHs C3H7 F CI

A-1640 C3H7 CHs F CI A-1681 CI CONH2 F CI

A-1641 CONH2 CHs F CI A-1682 F CONH2 F CI

A-1642 SCHs CHs F CI A-1683 Br CONH2 F CI

A-1643 SOCHs CHs F CI A-1684 CN CONH2 F CI

A-1644 OCHs CHs F CI A-1685 CHs CONH2 F CI

A-1645 CI CFs F CI A-1686 CFs CONH2 F CI

A-1646 F CFs F CI A-1687 CHF ₂ CONH2 F CI

A-1647 Br CFs F CI A-1688 C3H7 CONH2 F CI

A-1648 CN CFs F CI A-1689 CONH2 CONH2 F CI

A-1649 CHs CFs F CI A-1690 SCHs CONH2 F CI

A-1650 CFs CFs F CI A-1691 SOCHs CONH2 F CI

A-1651 CHF ₂ CFs F CI A-1692 OCHs CONH2 F CI

A-1652 C3H7 CFs F CI A-1693 CI SCHs F CI

A-1653 CONH2 CFs F CI A-1694 F SCHs F CI

A-1654 SCHs CFs F CI A-1695 Br SCHs F CI

A-1655 SOCHs CFs F CI A-1696 CN SCHs F CI

A-1656 OCHs CFs F CI A-1697 CHs SCHs F CI

A-1657 CI CHF ₂ F CI A-1698 CFs SCHs F CI line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1699 CHF ₂ SCHs F CI A-1740 OCHs CI CI CI

A-1700 C3H7 SCHs F CI A-1741 CI F CI CI

A-1701 CONH2 SCHs F CI A-1742 F F CI CI

A-1702 SCHs SCHs F CI A-1743 Br F CI CI

A-1703 SOCH3 SCHs F CI A-1744 CN F CI CI

A-1704 OCH3 SCHs F CI A-1745 CHs F CI CI

A-1705 CI SOCHs F CI A-1746 CFs F CI CI

A-1706 F SOCHs F CI A-1747 CHF ₂ F CI CI

A-1707 Br SOCHs F CI A-1748 C3H7 F CI CI

A-1708 CN SOCHs F CI A-1749 CONH2 F CI CI

A-1709 CHs SOCHs F CI A-1750 SCHs F CI CI

A-1710 CFs SOCHs F CI A-1751 SOCHs F CI CI

A-171 1 CHF ₂ SOCHs F CI A-1752 OCHs F CI CI

A-1712 C3H7 SOCHs F CI A-1753 CI Br CI CI

A-1713 CONH2 SOCHs F CI A-1754 F Br CI CI

A-1714 SCHs SOCHs F CI A- 1755 Br Br CI CI

A-1715 SOCHs SOCHs F CI A-1756 CN Br CI CI

A-1716 OCHs SOCHs F CI A- 1757 CHs Br CI CI

A-1717 CI OCHs F CI A-1758 CFs Br CI CI

A-1718 F OCHs F CI A-1759 CHF ₂ Br CI CI

A-1719 Br OCHs F CI A-1760 C3H7 Br CI CI

A-1720 CN OCHs F CI A-1761 CONH2 Br CI CI

A-1721 CHs OCHs F CI A-1762 SCHs Br CI CI

A-1722 CFs OCHs F CI A-1763 SOCHs Br CI CI

A-1723 CHF ₂ OCHs F CI A-1764 OCHs Br CI CI

A-1724 C3H7 OCHs F CI A-1765 CI CN CI CI

A-1725 CONH2 OCHs F CI A-1766 F CN CI CI

A-1726 SCHs OCHs F CI A-1767 Br CN CI CI

A-1727 SOCHs OCHs F CI A-1768 CN CN CI CI

A-1728 OCHs OCHs F CI A-1769 CHs CN CI CI

A-1729 CI CI CI CI A-1770 CFs CN CI CI

A-1730 F CI CI CI A-1771 CHF ₂ CN CI CI

A-1731 Br CI CI CI A-1772 C3H7 CN CI CI

A-1732 CN CI CI CI A-1773 CONH2 CN CI CI

A-1733 CHs CI CI CI A-1774 SCHs CN CI CI

A-1734 CFs CI CI CI A- 1775 SOCHs CN CI CI

A-1735 CHF ₂ CI CI CI A-1776 OCHs CN CI CI

A-1736 C3H7 CI CI CI A- 1777 CI CHs CI CI

A-1737 CONH2 CI CI CI A-1778 F CHs CI CI

A-1738 SCHs CI CI CI A-1779 Br CHs CI CI

A-1739 SOCHs CI CI CI A-1780 CN CHs CI CI line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1781 CHs CHs CI CI A-1822 SCHs C3H7 CI CI

A-1782 CFs CHs CI CI A-1823 SOCHs C3H7 CI CI

A-1783 CHF ₂ CHs CI CI A-1824 OCHs C3H7 CI CI

A-1784 C3H7 CHs CI CI A-1825 CI CONH2 CI CI

A-1785 CONH2 CHs CI CI A-1826 F CONH2 CI CI

A-1786 SCHs CHs CI CI A-1827 Br CONH2 CI CI

A-1787 SOCHs CHs CI CI A-1828 CN CONH2 CI CI

A-1788 OCHs CHs CI CI A-1829 CHs CONH2 CI CI

A-1789 CI CFs CI CI A-1830 CFs CONH2 CI CI

A-1790 F CFs CI CI A-1831 CHF ₂ CONH2 CI CI

A-1791 Br CFs CI CI A-1832 C3H7 CONH2 CI CI

A-1792 CN CFs CI CI A-1833 CONH2 CONH2 CI CI

A-1793 CHs CFs CI CI A-1834 SCHs CONH2 CI CI

A-1794 CFs CFs CI CI A-1835 SOCHs CONH2 CI CI

A-1795 CHF ₂ CFs CI CI A-1836 OCHs CONH2 CI CI

A-1796 C3H7 CFs CI CI A-1837 CI SCHs CI CI

A-1797 CONH2 CFs CI CI A-1838 F SCHs CI CI

A-1798 SCHs CFs CI CI A-1839 Br SCHs CI CI

A-1799 SOCHs CFs CI CI A-1840 CN SCHs CI CI

A-1800 OCHs CFs CI CI A-1841 CHs SCHs CI CI

A-1801 CI CHF ₂ CI CI A-1842 CFs SCHs CI CI

A-1802 F CHF ₂ CI CI A-1843 CHF ₂ SCHs CI CI

A-1803 Br CHF ₂ CI CI A-1844 C3H7 SCHs CI CI

A-1804 CN CHF ₂ CI CI A-1845 CONH2 SCHs CI CI

A-1805 CHs CHF ₂ CI CI A-1846 SCHs SCHs CI CI

A-1806 CFs CHF ₂ CI CI A-1847 SOCHs SCHs CI CI

A-1807 CHF ₂ CHF ₂ CI CI A-1848 OCHs SCHs CI CI

A-1808 C3H7 CHF ₂ CI CI A-1849 CI SOCHs CI CI

A-1809 CONH2 CHF ₂ CI CI A-1850 F SOCHs CI CI

A-1810 SCHs CHF ₂ CI CI A-1851 Br SOCHs CI CI

A-181 1 SOCHs CHF ₂ CI CI A-1852 CN SOCHs CI CI

A-1812 OCHs CHF ₂ CI CI A-1853 CHs SOCHs CI CI

A-1813 CI C3H7 CI CI A-1854 CFs SOCHs CI CI

A-1814 F C3H7 CI CI A-1855 CHF ₂ SOCHs CI CI

A-1815 Br C3H7 CI CI A-1856 C3H7 SOCHs CI CI

A-1816 CN C3H7 CI CI A-1857 CONH2 SOCHs CI CI

A-1817 CHs C3H7 CI CI A-1858 SCHs SOCHs CI CI

A-1818 CFs C3H7 CI CI A-1859 SOCHs SOCHs CI CI

A-1819 CHF ₂ C3H7 CI CI A-1860 OCHs SOCHs CI CI

A-1820 C3H7 C3H7 CI CI A-1861 CI OCHs CI CI

A-1821 CONH2 C3H7 CI CI A-1862 F OCHs CI CI line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1863 Br OCHs CI CI A-1904 C3H7 Br CN CI

A-1864 CN OCHs CI CI A-1905 CONH2 Br CN CI

A-1865 CHs OCHs CI CI A-1906 SCHs Br CN CI

A-1866 CFs OCHs CI CI A-1907 SOCHs Br CN CI

A-1867 CHF ₂ OCHs CI CI A-1908 OCHs Br CN CI

A-1868 C3H7 OCHs CI CI A-1909 CI CN CN CI

A-1869 CONH2 OCHs CI CI A-1910 F CN CN CI

A-1870 SCHs OCHs CI CI A-191 1 Br CN CN CI

A-1871 SOCHs OCHs CI CI A-1912 CN CN CN CI

A-1872 OCHs OCHs CI CI A-1913 CHs CN CN CI

A-1873 CI CI CN CI A-1914 CFs CN CN CI

A-1874 F CI CN CI A-1915 CHF ₂ CN CN CI

A-1875 Br CI CN CI A-1916 C3H7 CN CN CI

A-1876 CN CI CN CI A-1917 CONH2 CN CN CI

A-1877 CHs CI CN CI A-1918 SCHs CN CN CI

A-1878 CFs CI CN CI A-1919 SOCHs CN CN CI

A-1879 CHF ₂ CI CN CI A-1920 OCHs CN CN CI

A-1880 C3H7 CI CN CI A-1921 CI CHs CN CI

A-1881 CONH2 CI CN CI A-1922 F CHs CN CI

A-1882 SCHs CI CN CI A-1923 Br CHs CN CI

A-1883 SOCHs CI CN CI A-1924 CN CHs CN CI

A-1884 OCHs CI CN CI A-1925 CHs CHs CN CI

A-1885 CI F CN CI A-1926 CFs CHs CN CI

A-1886 F F CN CI A-1927 CHF ₂ CHs CN CI

A-1887 Br F CN CI A-1928 C3H7 CHs CN CI

A-1888 CN F CN CI A-1929 CONH2 CHs CN CI

A-1889 CHs F CN CI A-1930 SCHs CHs CN CI

A-1890 CFs F CN CI A-1931 SOCHs CHs CN CI

A-1891 CHF ₂ F CN CI A-1932 OCHs CHs CN CI

A-1892 C3H7 F CN CI A-1933 CI CFs CN CI

A-1893 CONH2 F CN CI A-1934 F CFs CN CI

A-1894 SCHs F CN CI A-1935 Br CFs CN CI

A-1895 SOCHs F CN CI A-1936 CN CFs CN CI

A-1896 OCHs F CN CI A-1937 CHs CFs CN CI

A-1897 CI Br CN CI A-1938 CFs CFs CN CI

A-1898 F Br CN CI A-1939 CHF ₂ CFs CN CI

A-1899 Br Br CN CI A-1940 C3H7 CFs CN CI

A-1900 CN Br CN CI A-1941 CONH2 CFs CN CI

A-1901 CHs Br CN CI A-1942 SCHs CFs CN CI

A-1902 CFs Br CN CI A-1943 SOCHs CFs CN CI

A-1903 CHF ₂ Br CN CI A-1944 OCHs CFs CN CI line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-1945 CI CHF ₂ CN CI A-1986 CFs SCHs CN CI

A-1946 F CHF ₂ CN CI A-1987 CHF ₂ SCHs CN CI

A-1947 Br CHF ₂ CN CI A-1988 C3H7 SCHs CN CI

A-1948 CN CHF ₂ CN CI A-1989 CONH2 SCHs CN CI

A-1949 CHs CHF ₂ CN CI A-1990 SCHs SCHs CN CI

A-1950 CFs CHF ₂ CN CI A-1991 SOCHs SCHs CN CI

A-1951 CHF ₂ CHF ₂ CN CI A-1992 OCHs SCHs CN CI

A-1952 C3H7 CHF ₂ CN CI A-1993 CI SOCHs CN CI

A-1953 CONH2 CHF ₂ CN CI A-1994 F SOCHs CN CI

A-1954 SCHs CHF ₂ CN CI A-1995 Br SOCHs CN CI

A-1955 SOCHs CHF ₂ CN CI A-1996 CN SOCHs CN CI

A-1956 OCHs CHF ₂ CN CI A-1997 CHs SOCHs CN CI

A-1957 CI C3H7 CN CI A-1998 CFs SOCHs CN CI

A-1958 F C3H7 CN CI A-1999 CHF ₂ SOCHs CN CI

A-1959 Br C3H7 CN CI A-2000 C3H7 SOCHs CN CI

A-1960 CN C3H7 CN CI A-2001 CONH2 SOCHs CN CI

A-1961 CHs C3H7 CN CI A-2002 SCHs SOCHs CN CI

A-1962 CFs C3H7 CN CI A-2003 SOCHs SOCHs CN CI

A-1963 CHF ₂ C3H7 CN CI A-2004 OCHs SOCHs CN CI

A-1964 C3H7 C3H7 CN CI A-2005 CI OCHs CN CI

A-1965 CONH2 C3H7 CN CI A-2006 F OCHs CN CI

A-1966 SCHs C3H7 CN CI A-2007 Br OCHs CN CI

A-1967 SOCHs C3H7 CN CI A-2008 CN OCHs CN CI

A-1968 OCHs C3H7 CN CI A-2009 CHs OCHs CN CI

A-1969 CI CONH2 CN CI A-2010 CFs OCHs CN CI

A-1970 F CONH2 CN CI A-201 1 CHF ₂ OCHs CN CI

A-1971 Br CONH2 CN CI A-2012 C3H7 OCHs CN CI

A-1972 CN CONH2 CN CI A-2013 CONH2 OCHs CN CI

A-1973 CHs CONH2 CN CI A-2014 SCHs OCHs CN CI

A-1974 CFs CONH2 CN CI A-2015 SOCHs OCHs CN CI

A-1975 CHF ₂ CONH2 CN CI A-2016 OCHs OCHs CN CI

A-1976 C3H7 CONH2 CN CI A-2017 CI CI CHs CI

A-1977 CONH2 CONH2 CN CI A-2018 F CI CHs CI

A-1978 SCHs CONH2 CN CI A-2019 Br CI CHs CI

A-1979 SOCHs CONH2 CN CI A-2020 CN CI CHs CI

A-1980 OCHs CONH2 CN CI A-2021 CHs CI CHs CI

A-1981 CI SCHs CN CI A-2022 CFs CI CHs CI

A-1982 F SCHs CN CI A-2023 CHF ₂ CI CHs CI

A-1983 Br SCHs CN CI A-2024 C3H7 CI CHs CI

A-1984 CN SCHs CN CI A-2025 CONH2 CI CHs CI

A-1985 CHs SCHs CN CI A-2026 SCHs CI CHs CI line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-2027 SOCHs CI CHs CI A-2068 CN CHs CHs CI

A-2028 OCH3 CI CHs CI A-2069 CHs CHs CHs CI

A-2029 CI F CHs CI A-2070 CFs CHs CHs CI

A-2030 F F CHs CI A-2071 CHF ₂ CHs CHs CI

A-2031 Br F CHs CI A-2072 C3H7 CHs CHs CI

A-2032 CN F CHs CI A-2073 CONH2 CHs CHs CI

A-2033 CHs F CHs CI A-2074 SCHs CHs CHs CI

A-2034 CFs F CHs CI A-2075 SOCHs CHs CHs CI

A-2035 CHF ₂ F CHs CI A-2076 OCHs CHs CHs CI

A-2036 C3H7 F CHs CI A-2077 CI CFs CHs CI

A-2037 CONH2 F CHs CI A-2078 F CFs CHs CI

A-2038 SCHs F CHs CI A-2079 Br CFs CHs CI

A-2039 SOCHs F CHs CI A-2080 CN CFs CHs CI

A-2040 OCHs F CHs CI A-2081 CHs CFs CHs CI

A-2041 CI Br CHs CI A-2082 CFs CFs CHs CI

A-2042 F Br CHs CI A-2083 CHF ₂ CFs CHs CI

A-2043 Br Br CHs CI A-2084 C3H7 CFs CHs CI

A-2044 CN Br CHs CI A-2085 CONH2 CFs CHs CI

A-2045 CHs Br CHs CI A-2086 SCHs CFs CHs CI

A-2046 CFs Br CHs CI A-2087 SOCHs CFs CHs CI

A-2047 CHF ₂ Br CHs CI A-2088 OCHs CFs CHs CI

A-2048 C3H7 Br CHs CI A-2089 CI CHF ₂ CHs CI

A-2049 CONH2 Br CHs CI A-2090 F CHF ₂ CHs CI

A-2050 SCHs Br CHs CI A-2091 Br CHF ₂ CHs CI

A-2051 SOCHs Br CHs CI A-2092 CN CHF ₂ CHs CI

A-2052 OCHs Br CHs CI A-2093 CHs CHF ₂ CHs CI

A-2053 CI CN CHs CI A-2094 CFs CHF ₂ CHs CI

A-2054 F CN CHs CI A-2095 CHF ₂ CHF ₂ CHs CI

A-2055 Br CN CHs CI A-2096 C3H7 CHF ₂ CHs CI

A-2056 CN CN CHs CI A-2097 CONH2 CHF ₂ CHs CI

A-2057 CHs CN CHs CI A-2098 SCHs CHF ₂ CHs CI

A-2058 CFs CN CHs CI A-2099 SOCHs CHF ₂ CHs CI

A-2059 CHF ₂ CN CHs CI A-2100 OCHs CHF ₂ CHs CI

A-2060 C3H7 CN CHs CI A-2101 CI C3H7 CHs CI

A-2061 CONH2 CN CHs CI A-2102 F C3H7 CHs CI

A-2062 SCHs CN CHs CI A-2103 Br C3H7 CHs CI

A-2063 SOCHs CN CHs CI A-2104 CN C3H7 CHs CI

A-2064 OCHs CN CHs CI A-2105 CHs C3H7 CHs CI

A-2065 CI CHs CHs CI A-2106 CFs C3H7 CHs CI

A-2066 F CHs CHs CI A-2107 CHF ₂ C3H7 CHs CI

A-2067 Br CHs CHs CI A-2108 C3H7 C3H7 CHs CI line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-2109 CONH ₂ C3H7 CHs CI A-2150 F OCHs CHs CI

A-21 10 SCHs C3H7 CHs CI A-2151 Br OCHs CHs CI

A-21 1 1 SOCH3 C3H7 CHs CI A-2152 CN OCHs CHs CI

A-21 12 OCH3 C3H7 CHs CI A-2153 CHs OCHs CHs CI

A-21 13 CI CONH2 CHs CI A-2154 CFs OCHs CHs CI

A-21 14 F CONH2 CHs CI A-2155 CHF ₂ OCHs CHs CI

A-21 15 Br CONH2 CHs CI A-2156 C3H7 OCHs CHs CI

A-21 16 CN CONH2 CHs CI A-2157 CONH2 OCHs CHs CI

A-21 17 CHs CONH2 CHs CI A-2158 SCHs OCHs CHs CI

A-21 18 CFs CONH2 CHs CI A-2159 SOCHs OCHs CHs CI

A-21 19 CHF ₂ CONH2 CHs CI A-2160 OCHs OCHs CHs CI

A-2120 C3H7 CONH2 CHs CI A-2161 CI CI H CN

A-2121 CONH2 CONH2 CHs CI A-2162 F CI H CN

A-2122 SCHs CONH2 CHs CI A-2163 Br CI H CN

A-2123 SOCHs CONH2 CHs CI A-2164 CN CI H CN

A-2124 OCHs CONH2 CHs CI A-2165 CHs CI H CN

A-2125 CI SCHs CHs CI A-2166 CFs CI H CN

A-2126 F SCHs CHs CI A-2167 CHF ₂ CI H CN

A-2127 Br SCHs CHs CI A-2168 C3H7 CI H CN

A-2128 CN SCHs CHs CI A-2169 CONH2 CI H CN

A-2129 CHs SCHs CHs CI A-2170 SCHs CI H CN

A-2130 CFs SCHs CHs CI A-2171 SOCHs CI H CN

A-2131 CHF ₂ SCHs CHs CI A-2172 OCHs CI H CN

A-2132 C3H7 SCHs CHs CI A-2173 CI F H CN

A-2133 CONH2 SCHs CHs CI A-2174 F F H CN

A-2134 SCHs SCHs CHs CI A-2175 Br F H CN

A-2135 SOCHs SCHs CHs CI A-2176 CN F H CN

A-2136 OCHs SCHs CHs CI A-2177 CHs F H CN

A-2137 CI SOCHs CHs CI A-2178 CFs F H CN

A-2138 F SOCHs CHs CI A-2179 CHF ₂ F H CN

A-2139 Br SOCHs CHs CI A-2180 C3H7 F H CN

A-2140 CN SOCHs CHs CI A-2181 CONH2 F H CN

A-2141 CHs SOCHs CHs CI A-2182 SCHs F H CN

A-2142 CFs SOCHs CHs CI A-2183 SOCHs F H CN

A-2143 CHF ₂ SOCHs CHs CI A-2184 OCHs F H CN

A-2144 C3H7 SOCHs CHs CI A-2185 CI Br H CN

A-2145 CONH2 SOCHs CHs CI A-2186 F Br H CN

A-2146 SCHs SOCHs CHs CI A-2187 Br Br H CN

A-2147 SOCHs SOCHs CHs CI A-2188 CN Br H CN

A-2148 OCHs SOCHs CHs CI A-2189 CHs Br H CN

A-2149 CI OCHs CHs CI A-2190 CFs Br H CN line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-2191 CHF ₂ Br H CN A-2232 OCHs CFs H CN

A-2192 C ₃ H ₇ Br H CN A-2233 CI CHF ₂ H CN

A-2193 CONH2 Br H CN A-2234 F CHF ₂ H CN

A-2194 SCHs Br H CN A-2235 Br CHF ₂ H CN

A-2195 SOCH3 Br H CN A-2236 CN CHF ₂ H CN

A-2196 OCH3 Br H CN A-2237 CHs CHF ₂ H CN

A-2197 CI CN H CN A-2238 CFs CHF ₂ H CN

A-2198 F CN H CN A-2239 CHF ₂ CHF ₂ H CN

A-2199 Br CN H CN A-2240 C3H7 CHF ₂ H CN

A-2200 CN CN H CN A-2241 CONH2 CHF ₂ H CN

A-2201 CHs CN H CN A-2242 SCHs CHF ₂ H CN

A-2202 CFs CN H CN A-2243 SOCHs CHF ₂ H CN

A-2203 CHF ₂ CN H CN A-2244 OCHs CHF ₂ H CN

A-2204 C3H7 CN H CN A-2245 CI C3H7 H CN

A-2205 CONH2 CN H CN A-2246 F C3H7 H CN

A-2206 SCHs CN H CN A-2247 Br C3H7 H CN

A-2207 SOCHs CN H CN A-2248 CN C3H7 H CN

A-2208 OCHs CN H CN A-2249 CHs C3H7 H CN

A-2209 CI CHs H CN A-2250 CFs C3H7 H CN

A-2210 F CHs H CN A-2251 CHF ₂ C3H7 H CN

A-221 1 Br CHs H CN A-2252 C3H7 C3H7 H CN

A-2212 CN CHs H CN A-2253 CONH2 C3H7 H CN

A-2213 CHs CHs H CN A-2254 SCHs C3H7 H CN

A-2214 CFs CHs H CN A-2255 SOCHs C3H7 H CN

A-2215 CHF ₂ CHs H CN A-2256 OCHs C3H7 H CN

A-2216 C3H7 CHs H CN A-2257 CI CONH2 H CN

A-2217 CONH2 CHs H CN A-2258 F CONH2 H CN

A-2218 SCHs CHs H CN A-2259 Br CONH2 H CN

A-2219 SOCHs CHs H CN A-2260 CN CONH2 H CN

A-2220 OCHs CHs H CN A-2261 CHs CONH2 H CN

A-2221 CI CFs H CN A-2262 CFs CONH2 H CN

A-2222 F CFs H CN A-2263 CHF ₂ CONH2 H CN

A-2223 Br CFs H CN A-2264 C3H7 CONH2 H CN

A-2224 CN CFs H CN A-2265 CONH2 CONH2 H CN

A-2225 CHs CFs H CN A-2266 SCHs CONH2 H CN

A-2226 CFs CFs H CN A-2267 SOCHs CONH2 H CN

A-2227 CHF ₂ CFs H CN A-2268 OCHs CONH2 H CN

A-2228 C3H7 CFs H CN A-2269 CI SCHs H CN

A-2229 CONH2 CFs H CN A-2270 F SCHs H CN

A-2230 SCHs CFs H CN A-2271 Br SCHs H CN

A-2231 SOCHs CFs H CN A-2272 CN SCHs H CN line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-2273 CHs SCHs H CN A-2314 SCHs CI F CN

A-2274 CFs SCHs H CN A-2315 SOCHs CI F CN

A-2275 CHF ₂ SCHs H CN A-2316 OCHs CI F CN

A-2276 CsH ₇ SCHs H CN A-2317 CI F F CN

A-2277 CONH2 SCHs H CN A-2318 F F F CN

A-2278 SCHs SCHs H CN A-2319 Br F F CN

A-2279 SOCHs SCHs H CN A-2320 CN F F CN

A-2280 OCHs SCHs H CN A-2321 CHs F F CN

A-2281 CI SOCHs H CN A-2322 CFs F F CN

A-2282 F SOCHs H CN A-2323 CHF ₂ F F CN

A-2283 Br SOCHs H CN A-2324 C3H7 F F CN

A-2284 CN SOCHs H CN A-2325 CONH2 F F CN

A-2285 CHs SOCHs H CN A-2326 SCHs F F CN

A-2286 CFs SOCHs H CN A-2327 SOCHs F F CN

A-2287 CHF ₂ SOCHs H CN A-2328 OCHs F F CN

A-2288 C3H7 SOCHs H CN A-2329 CI Br F CN

A-2289 CONH2 SOCHs H CN A-2330 F Br F CN

A-2290 SCHs SOCHs H CN A-2331 Br Br F CN

A-2291 SOCHs SOCHs H CN A-2332 CN Br F CN

A-2292 OCHs SOCHs H CN A-2333 CHs Br F CN

A-2293 CI OCHs H CN A-2334 CFs Br F CN

A-2294 F OCHs H CN A-2335 CHF ₂ Br F CN

A-2295 Br OCHs H CN A-2336 C3H7 Br F CN

A-2296 CN OCHs H CN A-2337 CONH2 Br F CN

A-2297 CHs OCHs H CN A-2338 SCHs Br F CN

A-2298 CFs OCHs H CN A-2339 SOCHs Br F CN

A-2299 CHF ₂ OCHs H CN A-2340 OCHs Br F CN

A-2300 C3H7 OCHs H CN A-2341 CI CN F CN

A-2301 CONH2 OCHs H CN A-2342 F CN F CN

A-2302 SCHs OCHs H CN A-2343 Br CN F CN

A-2303 SOCHs OCHs H CN A-2344 CN CN F CN

A-2304 OCHs OCHs H CN A-2345 CHs CN F CN

A-2305 CI CI F CN A-2346 CFs CN F CN

A-2306 F CI F CN A-2347 CHF ₂ CN F CN

A-2307 Br CI F CN A-2348 C3H7 CN F CN

A-2308 CN CI F CN A-2349 CONH2 CN F CN

A-2309 CHs CI F CN A-2350 SCHs CN F CN

A-2310 CFs CI F CN A-2351 SOCHs CN F CN

A-231 1 CHF ₂ CI F CN A-2352 OCHs CN F CN

A-2312 C3H7 CI F CN A-2353 CI CHs F CN

A-2313 CONH2 CI F CN A-2354 F CHs F CN line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-2355 Br CHs F CN A-2396 C3H7 C3H7 F CN

A-2356 CN CHs F CN A-2397 CONH2 C3H7 F CN

A-2357 CHs CHs F CN A-2398 SCHs C3H7 F CN

A-2358 CFs CHs F CN A-2399 SOCHs C3H7 F CN

A-2359 CHF ₂ CHs F CN A-2400 OCHs C3H7 F CN

A-2360 C3H7 CHs F CN A-2401 CI CONH2 F CN

A-2361 CONH2 CHs F CN A-2402 F CONH2 F CN

A-2362 SCHs CHs F CN A-2403 Br CONH2 F CN

A-2363 SOCHs CHs F CN A-2404 CN CONH2 F CN

A-2364 OCHs CHs F CN A-2405 CHs CONH2 F CN

A-2365 CI CFs F CN A-2406 CFs CONH2 F CN

A-2366 F CFs F CN A-2407 CHF ₂ CONH2 F CN

A-2367 Br CFs F CN A-2408 C3H7 CONH2 F CN

A-2368 CN CFs F CN A-2409 CONH2 CONH2 F CN

A-2369 CHs CFs F CN A-2410 SCHs CONH2 F CN

A-2370 CFs CFs F CN A-241 1 SOCHs CONH2 F CN

A-2371 CHF ₂ CFs F CN A-2412 OCHs CONH2 F CN

A-2372 C3H7 CFs F CN A-2413 CI SCHs F CN

A-2373 CONH2 CFs F CN A-2414 F SCHs F CN

A-2374 SCHs CFs F CN A-2415 Br SCHs F CN

A-2375 SOCHs CFs F CN A-2416 CN SCHs F CN

A-2376 OCHs CFs F CN A-2417 CHs SCHs F CN

A-2377 CI CHF ₂ F CN A-2418 CFs SCHs F CN

A-2378 F CHF ₂ F CN A-2419 CHF ₂ SCHs F CN

A-2379 Br CHF ₂ F CN A-2420 C3H7 SCHs F CN

A-2380 CN CHF ₂ F CN A-2421 CONH2 SCHs F CN

A-2381 CHs CHF ₂ F CN A-2422 SCHs SCHs F CN

A-2382 CFs CHF ₂ F CN A-2423 SOCHs SCHs F CN

A-2383 CHF ₂ CHF ₂ F CN A-2424 OCHs SCHs F CN

A-2384 C3H7 CHF ₂ F CN A-2425 CI SOCHs F CN

A-2385 CONH2 CHF ₂ F CN A-2426 F SOCHs F CN

A-2386 SCHs CHF ₂ F CN A-2427 Br SOCHs F CN

A-2387 SOCHs CHF ₂ F CN A-2428 CN SOCHs F CN

A-2388 OCHs CHF ₂ F CN A-2429 CHs SOCHs F CN

A-2389 CI C3H7 F CN A-2430 CFs SOCHs F CN

A-2390 F C3H7 F CN A-2431 CHF ₂ SOCHs F CN

A-2391 Br C3H7 F CN A-2432 C3H7 SOCHs F CN

A-2392 CN C3H7 F CN A-2433 CONH2 SOCHs F CN

A-2393 CHs C3H7 F CN A-2434 SCHs SOCHs F CN

A-2394 CFs C3H7 F CN A-2435 SOCHs SOCHs F CN

A-2395 CHF ₂ C3H7 F CN A-2436 OCHs SOCHs F CN line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-2437 CI OCHs F CN A-2478 CFs Br CI CN

A-2438 F OCHs F CN A-2479 CHF ₂ Br CI CN

A-2439 Br OCHs F CN A-2480 C3H7 Br CI CN

A-2440 CN OCHs F CN A-2481 CONH2 Br CI CN

A-2441 CHs OCHs F CN A-2482 SCHs Br CI CN

A-2442 CFs OCHs F CN A-2483 SOCHs Br CI CN

A-2443 CHF ₂ OCHs F CN A-2484 OCHs Br CI CN

A-2444 C3H7 OCHs F CN A-2485 CI CN CI CN

A-2445 CONH2 OCHs F CN A-2486 F CN CI CN

A-2446 SCHs OCHs F CN A-2487 Br CN CI CN

A-2447 SOCHs OCHs F CN A-2488 CN CN CI CN

A-2448 OCHs OCHs F CN A-2489 CHs CN CI CN

A-2449 CI CI CI CN A-2490 CFs CN CI CN

A-2450 F CI CI CN A-2491 CHF ₂ CN CI CN

A-2451 Br CI CI CN A-2492 C3H7 CN CI CN

A-2452 CN CI CI CN A-2493 CONH2 CN CI CN

A-2453 CHs CI CI CN A-2494 SCHs CN CI CN

A-2454 CFs CI CI CN A-2495 SOCHs CN CI CN

A-2455 CHF ₂ CI CI CN A-2496 OCHs CN CI CN

A-2456 C3H7 CI CI CN A-2497 CI CHs CI CN

A-2457 CONH2 CI CI CN A-2498 F CHs CI CN

A-2458 SCHs CI CI CN A-2499 Br CHs CI CN

A-2459 SOCHs CI CI CN A-2500 CN CHs CI CN

A-2460 OCHs CI CI CN A-2501 CHs CHs CI CN

A-2461 CI F CI CN A-2502 CFs CHs CI CN

A-2462 F F CI CN A-2503 CHF ₂ CHs CI CN

A-2463 Br F CI CN A-2504 C3H7 CHs CI CN

A-2464 CN F CI CN A-2505 CONH2 CHs CI CN

A-2465 CHs F CI CN A-2506 SCHs CHs CI CN

A-2466 CFs F CI CN A-2507 SOCHs CHs CI CN

A-2467 CHF ₂ F CI CN A-2508 OCHs CHs CI CN

A-2468 C3H7 F CI CN A-2509 CI CFs CI CN

A-2469 CONH2 F CI CN A-2510 F CFs CI CN

A-2470 SCHs F CI CN A-251 1 Br CFs CI CN

A-2471 SOCHs F CI CN A-2512 CN CFs CI CN

A-2472 OCHs F CI CN A-2513 CHs CFs CI CN

A-2473 CI Br CI CN A-2514 CFs CFs CI CN

A-2474 F Br CI CN A-2515 CHF ₂ CFs CI CN

A-2475 Br Br CI CN A-2516 C3H7 CFs CI CN

A-2476 CN Br CI CN A-2517 CONH2 CFs CI CN

A-2477 CHs Br CI CN A-2518 SCHs CFs CI CN line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-2519 SOCHs CFs CI CN A-2560 CN SCHs CI CN

A-2520 OCH3 CFs CI CN A-2561 CHs SCHs CI CN

A-2521 CI CHF ₂ CI CN A-2562 CFs SCHs CI CN

A-2522 F CHF ₂ CI CN A-2563 CHF ₂ SCHs CI CN

A-2523 Br CHF ₂ CI CN A-2564 C3H7 SCHs CI CN

A-2524 CN CHF ₂ CI CN A-2565 CONH2 SCHs CI CN

A-2525 CHs CHF ₂ CI CN A-2566 SCHs SCHs CI CN

A-2526 CFs CHF ₂ CI CN A-2567 SOCHs SCHs CI CN

A-2527 CHF ₂ CHF ₂ CI CN A-2568 OCHs SCHs CI CN

A-2528 C3H7 CHF ₂ CI CN A-2569 CI SOCHs CI CN

A-2529 CONH2 CHF ₂ CI CN A-2570 F SOCHs CI CN

A-2530 SCHs CHF ₂ CI CN A-2571 Br SOCHs CI CN

A-2531 SOCHs CHF ₂ CI CN A-2572 CN SOCHs CI CN

A-2532 OCHs CHF ₂ CI CN A-2573 CHs SOCHs CI CN

A-2533 CI C3H7 CI CN A-2574 CFs SOCHs CI CN

A-2534 F C3H7 CI CN A-2575 CHF ₂ SOCHs CI CN

A-2535 Br C3H7 CI CN A-2576 C3H7 SOCHs CI CN

A-2536 CN C3H7 CI CN A-2577 CONH2 SOCHs CI CN

A-2537 CHs C3H7 CI CN A-2578 SCHs SOCHs CI CN

A-2538 CFs C3H7 CI CN A-2579 SOCHs SOCHs CI CN

A-2539 CHF ₂ C3H7 CI CN A-2580 OCHs SOCHs CI CN

A-2540 C3H7 C3H7 CI CN A-2581 CI OCHs CI CN

A-2541 CONH2 C3H7 CI CN A-2582 F OCHs CI CN

A-2542 SCHs C3H7 CI CN A-2583 Br OCHs CI CN

A-2543 SOCHs C3H7 CI CN A-2584 CN OCHs CI CN

A-2544 OCHs C3H7 CI CN A-2585 CHs OCHs CI CN

A-2545 CI CONH2 CI CN A-2586 CFs OCHs CI CN

A-2546 F CONH2 CI CN A-2587 CHF ₂ OCHs CI CN

A-2547 Br CONH2 CI CN A-2588 C3H7 OCHs CI CN

A-2548 CN CONH2 CI CN A-2589 CONH2 OCHs CI CN

A-2549 CHs CONH2 CI CN A-2590 SCHs OCHs CI CN

A-2550 CFs CONH2 CI CN A-2591 SOCHs OCHs CI CN

A-2551 CHF ₂ CONH2 CI CN A-2592 OCHs OCHs CI CN

A-2552 C3H7 CONH2 CI CN A-2593 CI CI CN CN

A-2553 CONH2 CONH2 CI CN A-2594 F CI CN CN

A-2554 SCHs CONH2 CI CN A-2595 Br CI CN CN

A-2555 SOCHs CONH2 CI CN A-2596 CN CI CN CN

A-2556 OCHs CONH2 CI CN A-2597 CHs CI CN CN

A-2557 CI SCHs CI CN A-2598 CFs CI CN CN

A-2558 F SCHs CI CN A-2599 CHF ₂ CI CN CN

A-2559 Br SCHs CI CN A-2600 C3H7 CI CN CN line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-2601 CONH ₂ CI CN CN A-2642 F CHs CN CN

A-2602 SCHs CI CN CN A-2643 Br CHs CN CN

A-2603 SOCH3 CI CN CN A-2644 CN CHs CN CN

A-2604 OCH3 CI CN CN A-2645 CHs CHs CN CN

A-2605 CI F CN CN A-2646 CFs CHs CN CN

A-2606 F F CN CN A-2647 CHF ₂ CHs CN CN

A-2607 Br F CN CN A-2648 C3H7 CHs CN CN

A-2608 CN F CN CN A-2649 CONH2 CHs CN CN

A-2609 CHs F CN CN A-2650 SCHs CHs CN CN

A-2610 CFs F CN CN A-2651 SOCHs CHs CN CN

A-261 1 CHF ₂ F CN CN A-2652 OCHs CHs CN CN

A-2612 C3H7 F CN CN A-2653 CI CFs CN CN

A-2613 CONH2 F CN CN A-2654 F CFs CN CN

A-2614 SCHs F CN CN A-2655 Br CFs CN CN

A-2615 SOCHs F CN CN A-2656 CN CFs CN CN

A-2616 OCHs F CN CN A-2657 CHs CFs CN CN

A-2617 CI Br CN CN A-2658 CFs CFs CN CN

A-2618 F Br CN CN A-2659 CHF ₂ CFs CN CN

A-2619 Br Br CN CN A-2660 C3H7 CFs CN CN

A-2620 CN Br CN CN A-2661 CONH2 CFs CN CN

A-2621 CHs Br CN CN A-2662 SCHs CFs CN CN

A-2622 CFs Br CN CN A-2663 SOCHs CFs CN CN

A-2623 CHF ₂ Br CN CN A-2664 OCHs CFs CN CN

A-2624 C3H7 Br CN CN A-2665 CI CHF ₂ CN CN

A-2625 CONH2 Br CN CN A-2666 F CHF ₂ CN CN

A-2626 SCHs Br CN CN A-2667 Br CHF ₂ CN CN

A-2627 SOCHs Br CN CN A-2668 CN CHF ₂ CN CN

A-2628 OCHs Br CN CN A-2669 CHs CHF ₂ CN CN

A-2629 CI CN CN CN A-2670 CFs CHF ₂ CN CN

A-2630 F CN CN CN A-2671 CHF ₂ CHF ₂ CN CN

A-2631 Br CN CN CN A-2672 C3H7 CHF ₂ CN CN

A-2632 CN CN CN CN A-2673 CONH2 CHF ₂ CN CN

A-2633 CHs CN CN CN A-2674 SCHs CHF ₂ CN CN

A-2634 CFs CN CN CN A-2675 SOCHs CHF ₂ CN CN

A-2635 CHF ₂ CN CN CN A-2676 OCHs CHF ₂ CN CN

A-2636 C3H7 CN CN CN A-2677 CI C3H7 CN CN

A-2637 CONH2 CN CN CN A-2678 F C3H7 CN CN

A-2638 SCHs CN CN CN A-2679 Br C3H7 CN CN

A-2639 SOCHs CN CN CN A-2680 CN C3H7 CN CN

A-2640 OCHs CN CN CN A-2681 CHs C3H7 CN CN

A-2641 CI CHs CN CN A-2682 CFs C3H7 CN CN line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-2683 CHF ₂ C3H7 CN CN A-2724 OCHs SOCHs CN CN

A-2684 C ₃ H ₇ C3H7 CN CN A-2725 CI OCHs CN CN

A-2685 CONH2 C3H7 CN CN A-2726 F OCHs CN CN

A-2686 SCHs C3H7 CN CN A-2727 Br OCHs CN CN

A-2687 SOCH3 C3H7 CN CN A-2728 CN OCHs CN CN

A-2688 OCH3 C3H7 CN CN A-2729 CHs OCHs CN CN

A-2689 CI CONH2 CN CN A-2730 CFs OCHs CN CN

A-2690 F CONH2 CN CN A-2731 CHF ₂ OCHs CN CN

A-2691 Br CONH2 CN CN A-2732 C3H7 OCHs CN CN

A-2692 CN CONH2 CN CN A-2733 CONH2 OCHs CN CN

A-2693 CHs CONH2 CN CN A-2734 SCHs OCHs CN CN

A-2694 CFs CONH2 CN CN A-2735 SOCHs OCHs CN CN

A-2695 CHF ₂ CONH2 CN CN A-2736 OCHs OCHs CN CN

A-2696 C3H7 CONH2 CN CN A-2737 CI CI CHs CN

A-2697 CONH2 CONH2 CN CN A-2738 F CI CHs CN

A-2698 SCHs CONH2 CN CN A-2739 Br CI CHs CN

A-2699 SOCHs CONH2 CN CN A-2740 CN CI CHs CN

A-2700 OCHs CONH2 CN CN A-2741 CHs CI CHs CN

A-2701 CI SCHs CN CN A-2742 CFs CI CHs CN

A-2702 F SCHs CN CN A-2743 CHF ₂ CI CHs CN

A-2703 Br SCHs CN CN A-2744 C3H7 CI CHs CN

A-2704 CN SCHs CN CN A-2745 CONH2 CI CHs CN

A-2705 CHs SCHs CN CN A-2746 SCHs CI CHs CN

A-2706 CFs SCHs CN CN A-2747 SOCHs CI CHs CN

A-2707 CHF ₂ SCHs CN CN A-2748 OCHs CI CHs CN

A-2708 C3H7 SCHs CN CN A-2749 CI F CHs CN

A-2709 CONH2 SCHs CN CN A-2750 F F CHs CN

A-2710 SCHs SCHs CN CN A-2751 Br F CHs CN

A-271 1 SOCHs SCHs CN CN A-2752 CN F CHs CN

A-2712 OCHs SCHs CN CN A-2753 CHs F CHs CN

A-2713 CI SOCHs CN CN A-2754 CFs F CHs CN

A-2714 F SOCHs CN CN A-2755 CHF ₂ F CHs CN

A-2715 Br SOCHs CN CN A-2756 C3H7 F CHs CN

A-2716 CN SOCHs CN CN A-2757 CONH2 F CHs CN

A-2717 CHs SOCHs CN CN A-2758 SCHs F CHs CN

A-2718 CFs SOCHs CN CN A-2759 SOCHs F CHs CN

A-2719 CHF ₂ SOCHs CN CN A-2760 OCHs F CHs CN

A-2720 C3H7 SOCHs CN CN A-2761 CI Br CHs CN

A-2721 CONH2 SOCHs CN CN A-2762 F Br CHs CN

A-2722 SCHs SOCHs CN CN A-2763 Br Br CHs CN

A-2723 SOCHs SOCHs CN CN A-2764 CN Br CHs CN line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-2765 CHs Br CHs CN A-2806 SCHs CFs CHs CN

A-2766 CFs Br CHs CN A-2807 SOCHs CFs CHs CN

A-2767 CHF ₂ Br CHs CN A-2808 OCHs CFs CHs CN

A-2768 C3H7 Br CHs CN A-2809 CI CHF ₂ CHs CN

A-2769 CONH2 Br CHs CN A-2810 F CHF ₂ CHs CN

A-2770 SCHs Br CHs CN A-281 1 Br CHF ₂ CHs CN

A-2771 SOCHs Br CHs CN A-2812 CN CHF ₂ CHs CN

A-2772 OCHs Br CHs CN A-2813 CHs CHF ₂ CHs CN

A-2773 CI CN CHs CN A-2814 CFs CHF ₂ CHs CN

A-2774 F CN CHs CN A-2815 CHF ₂ CHF ₂ CHs CN

A-2775 Br CN CHs CN A-2816 C3H7 CHF ₂ CHs CN

A-2776 CN CN CHs CN A-2817 CONH2 CHF ₂ CHs CN

A-2777 CHs CN CHs CN A-2818 SCHs CHF ₂ CHs CN

A-2778 CFs CN CHs CN A-2819 SOCHs CHF ₂ CHs CN

A-2779 CHF ₂ CN CHs CN A-2820 OCHs CHF ₂ CHs CN

A-2780 C3H7 CN CHs CN A-2821 CI C3H7 CHs CN

A-2781 CONH2 CN CHs CN A-2822 F C3H7 CHs CN

A-2782 SCHs CN CHs CN A-2823 Br C3H7 CHs CN

A-2783 SOCHs CN CHs CN A-2824 CN C3H7 CHs CN

A-2784 OCHs CN CHs CN A-2825 CHs C3H7 CHs CN

A-2785 CI CHs CHs CN A-2826 CFs C3H7 CHs CN

A-2786 F CHs CHs CN A-2827 CHF ₂ C3H7 CHs CN

A-2787 Br CHs CHs CN A-2828 C3H7 C3H7 CHs CN

A-2788 CN CHs CHs CN A-2829 CONH2 C3H7 CHs CN

A-2789 CHs CHs CHs CN A-2830 SCHs C3H7 CHs CN

A-2790 CFs CHs CHs CN A-2831 SOCHs C3H7 CHs CN

A-2791 CHF ₂ CHs CHs CN A-2832 OCHs C3H7 CHs CN

A-2792 C3H7 CHs CHs CN A-2833 CI CONH2 CHs CN

A-2793 CONH2 CHs CHs CN A-2834 F CONH2 CHs CN

A-2794 SCHs CHs CHs CN A-2835 Br CONH2 CHs CN

A-2795 SOCHs CHs CHs CN A-2836 CN CONH2 CHs CN

A-2796 OCHs CHs CHs CN A-2837 CHs CONH2 CHs CN

A-2797 CI CFs CHs CN A-2838 CFs CONH2 CHs CN

A-2798 F CFs CHs CN A-2839 CHF ₂ CONH2 CHs CN

A-2799 Br CFs CHs CN A-2840 C3H7 CONH2 CHs CN

A-2800 CN CFs CHs CN A-2841 CONH2 CONH2 CHs CN

A-2801 CHs CFs CHs CN A-2842 SCHs CONH2 CHs CN

A-2802 CFs CFs CHs CN A-2843 SOCHs CONH2 CHs CN

A-2803 CHF ₂ CFs CHs CN A-2844 OCHs CONH2 CHs CN

A-2804 C3H7 CFs CHs CN A-2845 CI SCHs CHs CN

A-2805 CONH2 CFs CHs CN A-2846 F SCHs CHs CN line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-2847 Br SCHs CHs CN A-2888 C3H7 CI H CHs

A-2848 CN SCHs CHs CN A-2889 CONH2 CI H CHs

A-2849 CHs SCHs CHs CN A-2890 SCHs CI H CHs

A-2850 CFs SCHs CHs CN A-2891 SOCHs CI H CHs

A-2851 CHF ₂ SCHs CHs CN A-2892 OCHs CI H CHs

A-2852 C3H7 SCHs CHs CN A-2893 CI F H CHs

A-2853 CONH2 SCHs CHs CN A-2894 F F H CHs

A-2854 SCHs SCHs CHs CN A-2895 Br F H CHs

A-2855 SOCHs SCHs CHs CN A-2896 CN F H CHs

A-2856 OCHs SCHs CHs CN A-2897 CHs F H CHs

A-2857 CI SOCHs CHs CN A-2898 CFs F H CHs

A-2858 F SOCHs CHs CN A-2899 CHF ₂ F H CHs

A-2859 Br SOCHs CHs CN A-2900 C3H7 F H CHs

A-2860 CN SOCHs CHs CN A-2901 CONH2 F H CHs

A-2861 CHs SOCHs CHs CN A-2902 SCHs F H CHs

A-2862 CFs SOCHs CHs CN A-2903 SOCHs F H CHs

A-2863 CHF ₂ SOCHs CHs CN A-2904 OCHs F H CHs

A-2864 C3H7 SOCHs CHs CN A-2905 CI Br H CHs

A-2865 CONH2 SOCHs CHs CN A-2906 F Br H CHs

A-2866 SCHs SOCHs CHs CN A-2907 Br Br H CHs

A-2867 SOCHs SOCHs CHs CN A-2908 CN Br H CHs

A-2868 OCHs SOCHs CHs CN A-2909 CHs Br H CHs

A-2869 CI OCHs CHs CN A-2910 CFs Br H CHs

A-2870 F OCHs CHs CN A-291 1 CHF ₂ Br H CHs

A-2871 Br OCHs CHs CN A-2912 C3H7 Br H CHs

A-2872 CN OCHs CHs CN A-2913 CONH2 Br H CHs

A-2873 CHs OCHs CHs CN A-2914 SCHs Br H CHs

A-2874 CFs OCHs CHs CN A-2915 SOCHs Br H CHs

A-2875 CHF ₂ OCHs CHs CN A-2916 OCHs Br H CHs

A-2876 C3H7 OCHs CHs CN A-2917 CI CN H CHs

A-2877 CONH2 OCHs CHs CN A-2918 F CN H CHs

A-2878 SCHs OCHs CHs CN A-2919 Br CN H CHs

A-2879 SOCHs OCHs CHs CN A-2920 CN CN H CHs

A-2880 OCHs OCHs CHs CN A-2921 CHs CN H CHs

A-2881 CI CI H CHs A-2922 CFs CN H CHs

A-2882 F CI H CHs A-2923 CHF ₂ CN H CHs

A-2883 Br CI H CHs A-2924 C3H7 CN H CHs

A-2884 CN CI H CHs A-2925 CONH2 CN H CHs

A-2885 CHs CI H CHs A-2926 SCHs CN H CHs

A-2886 CFs CI H CHs A-2927 SOCHs CN H CHs

A-2887 CHF ₂ CI H CHs A-2928 OCHs CN H CHs line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-2929 CI CHs H CHs A-2970 CFs C3H7 H CHs

A-2930 F CHs H CHs A-2971 CHF ₂ C3H7 H CHs

A-2931 Br CHs H CHs A-2972 C3H7 C3H7 H CHs

A-2932 CN CHs H CHs A-2973 CONH2 C3H7 H CHs

A-2933 CHs CHs H CHs A-2974 SCHs C3H7 H CHs

A-2934 CFs CHs H CHs A-2975 SOCHs C3H7 H CHs

A-2935 CHF ₂ CHs H CHs A-2976 OCHs C3H7 H CHs

A-2936 C3H7 CHs H CHs A-2977 CI CONH2 H CHs

A-2937 CONH2 CHs H CHs A-2978 F CONH2 H CHs

A-2938 SCHs CHs H CHs A-2979 Br CONH2 H CHs

A-2939 SOCHs CHs H CHs A-2980 CN CONH2 H CHs

A-2940 OCHs CHs H CHs A-2981 CHs CONH2 H CHs

A-2941 CI CFs H CHs A-2982 CFs CONH2 H CHs

A-2942 F CFs H CHs A-2983 CHF ₂ CONH2 H CHs

A-2943 Br CFs H CHs A-2984 C3H7 CONH2 H CHs

A-2944 CN CFs H CHs A-2985 CONH2 CONH2 H CHs

A-2945 CHs CFs H CHs A-2986 SCHs CONH2 H CHs

A-2946 CFs CFs H CHs A-2987 SOCHs CONH2 H CHs

A-2947 CHF ₂ CFs H CHs A-2988 OCHs CONH2 H CHs

A-2948 C3H7 CFs H CHs A-2989 CI SCHs H CHs

A-2949 CONH2 CFs H CHs A-2990 F SCHs H CHs

A-2950 SCHs CFs H CHs A-2991 Br SCHs H CHs

A-2951 SOCHs CFs H CHs A-2992 CN SCHs H CHs

A-2952 OCHs CFs H CHs A-2993 CHs SCHs H CHs

A-2953 CI CHF ₂ H CHs A-2994 CFs SCHs H CHs

A-2954 F CHF ₂ H CHs A-2995 CHF ₂ SCHs H CHs

A-2955 Br CHF ₂ H CHs A-2996 C3H7 SCHs H CHs

A-2956 CN CHF ₂ H CHs A-2997 CONH2 SCHs H CHs

A-2957 CHs CHF ₂ H CHs A-2998 SCHs SCHs H CHs

A-2958 CFs CHF ₂ H CHs A-2999 SOCHs SCHs H CHs

A-2959 CHF ₂ CHF ₂ H CHs A-3000 OCHs SCHs H CHs

A-2960 C3H7 CHF ₂ H CHs A-3001 CI SOCHs H CHs

A-2961 CONH2 CHF ₂ H CHs A-3002 F SOCHs H CHs

A-2962 SCHs CHF ₂ H CHs A-3003 Br SOCHs H CHs

A-2963 SOCHs CHF ₂ H CHs A-3004 CN SOCHs H CHs

A-2964 OCHs CHF ₂ H CHs A-3005 CHs SOCHs H CHs

A-2965 CI C3H7 H CHs A-3006 CFs SOCHs H CHs

A-2966 F C3H7 H CHs A-3007 CHF ₂ SOCHs H CHs

A-2967 Br C3H7 H CHs A-3008 C3H7 SOCHs H CHs

A-2968 CN C3H7 H CHs A-3009 CONH2 SOCHs H CHs

A-2969 CHs C3H7 H CHs A-3010 SCHs SOCHs H CHs line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-301 1 SOCHs SOCHs H CHs A-3052 CN Br F CHs

A-3012 OCHs SOCHs H CHs A-3053 CHs Br F CHs

A-3013 CI OCHs H CHs A-3054 CFs Br F CHs

A-3014 F OCHs H CHs A-3055 CHF ₂ Br F CHs

A-3015 Br OCHs H CHs A-3056 C3H7 Br F CHs

A-3016 CN OCHs H CHs A-3057 CONH2 Br F CHs

A-3017 CHs OCHs H CHs A-3058 SCHs Br F CHs

A-3018 CFs OCHs H CHs A-3059 SOCHs Br F CHs

A-3019 CHF ₂ OCHs H CHs A-3060 OCHs Br F CHs

A-3020 CsH ₇ OCHs H CHs A-3061 CI CN F CHs

A-3021 CONH2 OCHs H CHs A-3062 F CN F CHs

A-3022 SCHs OCHs H CHs A-3063 Br CN F CHs

A-3023 SOCHs OCHs H CHs A-3064 CN CN F CHs

A-3024 OCHs OCHs H CHs A-3065 CHs CN F CHs

A-3025 CI CI F CHs A-3066 CFs CN F CHs

A-3026 F CI F CHs A-3067 CHF ₂ CN F CHs

A-3027 Br CI F CHs A-3068 C3H7 CN F CHs

A-3028 CN CI F CHs A-3069 CONH2 CN F CHs

A-3029 CHs CI F CHs A-3070 SCHs CN F CHs

A-3030 CFs CI F CHs A-3071 SOCHs CN F CHs

A-3031 CHF ₂ CI F CHs A-3072 OCHs CN F CHs

A-3032 C3H7 CI F CHs A-3073 CI CHs F CHs

A-3033 CONH2 CI F CHs A-3074 F CHs F CHs

A-3034 SCHs CI F CHs A-3075 Br CHs F CHs

A-3035 SOCHs CI F CHs A-3076 CN CHs F CHs

A-3036 OCHs CI F CHs A-3077 CHs CHs F CHs

A-3037 CI F F CHs A-3078 CFs CHs F CHs

A-3038 F F F CHs A-3079 CHF ₂ CHs F CHs

A-3039 Br F F CHs A-3080 C3H7 CHs F CHs

A-3040 CN F F CHs A-3081 CONH2 CHs F CHs

A-3041 CHs F F CHs A-3082 SCHs CHs F CHs

A-3042 CFs F F CHs A-3083 SOCHs CHs F CHs

A-3043 CHF ₂ F F CHs A-3084 OCHs CHs F CHs

A-3044 C3H7 F F CHs A-3085 CI CFs F CHs

A-3045 CONH2 F F CHs A-3086 F CFs F CHs

A-3046 SCHs F F CHs A-3087 Br CFs F CHs

A-3047 SOCHs F F CHs A-3088 CN CFs F CHs

A-3048 OCHs F F CHs A-3089 CHs CFs F CHs

A-3049 CI Br F CHs A-3090 CFs CFs F CHs

A-3050 F Br F CHs A-3091 CHF ₂ CFs F CHs

A-3051 Br Br F CHs A-3092 C3H7 CFs F CHs line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-3093 CONH ₂ CFs F CHs A-3134 F SCHs F CHs

A-3094 SCHs CFs F CHs A-3135 Br SCHs F CHs

A-3095 SOCH3 CFs F CHs A-3136 CN SCHs F CHs

A-3096 OCH3 CFs F CHs A-3137 CHs SCHs F CHs

A-3097 CI CHF ₂ F CHs A-3138 CFs SCHs F CHs

A-3098 F CHF ₂ F CHs A-3139 CHF ₂ SCHs F CHs

A-3099 Br CHF ₂ F CHs A-3140 C3H7 SCHs F CHs

A-3100 CN CHF ₂ F CHs A-3141 CONH2 SCHs F CHs

A-3101 CHs CHF ₂ F CHs A-3142 SCHs SCHs F CHs

A-3102 CFs CHF ₂ F CHs A-3143 SOCHs SCHs F CHs

A-3103 CHF ₂ CHF ₂ F CHs A-3144 OCHs SCHs F CHs

A-3104 C3H7 CHF ₂ F CHs A-3145 CI SOCHs F CHs

A-3105 CONH2 CHF ₂ F CHs A-3146 F SOCHs F CHs

A-3106 SCHs CHF ₂ F CHs A-3147 Br SOCHs F CHs

A-3107 SOCHs CHF ₂ F CHs A-3148 CN SOCHs F CHs

A-3108 OCHs CHF ₂ F CHs A-3149 CHs SOCHs F CHs

A-3109 CI C3H7 F CHs A-3150 CFs SOCHs F CHs

A-31 10 F C3H7 F CHs A-3151 CHF ₂ SOCHs F CHs

A-31 1 1 Br C3H7 F CHs A-3152 C3H7 SOCHs F CHs

A-31 12 CN C3H7 F CHs A-3153 CONH2 SOCHs F CHs

A-31 13 CHs C3H7 F CHs A-3154 SCHs SOCHs F CHs

A-31 14 CFs C3H7 F CHs A-3155 SOCHs SOCHs F CHs

A-31 15 CHF ₂ C3H7 F CHs A-3156 OCHs SOCHs F CHs

A-31 16 C3H7 C3H7 F CHs A-3157 CI OCHs F CHs

A-31 17 CONH2 C3H7 F CHs A-3158 F OCHs F CHs

A-31 18 SCHs C3H7 F CHs A-3159 Br OCHs F CHs

A-31 19 SOCHs C3H7 F CHs A-3160 CN OCHs F CHs

A-3120 OCHs C3H7 F CHs A-3161 CHs OCHs F CHs

A-3121 CI CONH2 F CHs A-3162 CFs OCHs F CHs

A-3122 F CONH2 F CHs A-3163 CHF ₂ OCHs F CHs

A-3123 Br CONH2 F CHs A-3164 C3H7 OCHs F CHs

A-3124 CN CONH2 F CHs A-3165 CONH2 OCHs F CHs

A-3125 CHs CONH2 F CHs A-3166 SCHs OCHs F CHs

A-3126 CFs CONH2 F CHs A-3167 SOCHs OCHs F CHs

A-3127 CHF ₂ CONH2 F CHs A-3168 OCHs OCHs F CHs

A-3128 C3H7 CONH2 F CHs A-3169 CI CI CI CHs

A-3129 CONH2 CONH2 F CHs A-3170 F CI CI CHs

A-3130 SCHs CONH2 F CHs A-3171 Br CI CI CHs

A-3131 SOCHs CONH2 F CHs A-3172 CN CI CI CHs

A-3132 OCHs CONH2 F CHs A-3173 CHs CI CI CHs

A-3133 CI SCHs F CHs A-3174 CFs CI CI CHs line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-3175 CHF ₂ CI CI CHs A-3216 OCHs CN CI CHs

A-3176 C ₃ H ₇ CI CI CHs A-3217 CI CHs CI CHs

A-3177 CONH2 CI CI CHs A-3218 F CHs CI CHs

A-3178 SCHs CI CI CHs A-3219 Br CHs CI CHs

A-3179 SOCH3 CI CI CHs A-3220 CN CHs CI CHs

A-3180 OCH3 CI CI CHs A-3221 CHs CHs CI CHs

A-3181 CI F CI CHs A-3222 CFs CHs CI CHs

A-3182 F F CI CHs A-3223 CHF ₂ CHs CI CHs

A-3183 Br F CI CHs A-3224 C3H7 CHs CI CHs

A-3184 CN F CI CHs A-3225 CONH2 CHs CI CHs

A-3185 CHs F CI CHs A-3226 SCHs CHs CI CHs

A-3186 CFs F CI CHs A-3227 SOCHs CHs CI CHs

A-3187 CHF ₂ F CI CHs A-3228 OCHs CHs CI CHs

A-3188 C3H7 F CI CHs A-3229 CI CFs CI CHs

A-3189 CONH2 F CI CHs A-3230 F CFs CI CHs

A-3190 SCHs F CI CHs A-3231 Br CFs CI CHs

A-3191 SOCHs F CI CHs A-3232 CN CFs CI CHs

A-3192 OCHs F CI CHs A-3233 CHs CFs CI CHs

A-3193 CI Br CI CHs A-3234 CFs CFs CI CHs

A-3194 F Br CI CHs A-3235 CHF ₂ CFs CI CHs

A-3195 Br Br CI CHs A-3236 C3H7 CFs CI CHs

A-3196 CN Br CI CHs A-3237 CONH2 CFs CI CHs

A-3197 CHs Br CI CHs A-3238 SCHs CFs CI CHs

A-3198 CFs Br CI CHs A-3239 SOCHs CFs CI CHs

A-3199 CHF ₂ Br CI CHs A-3240 OCHs CFs CI CHs

A-3200 C3H7 Br CI CHs A-3241 CI CHF ₂ CI CHs

A-3201 CONH2 Br CI CHs A-3242 F CHF ₂ CI CHs

A-3202 SCHs Br CI CHs A-3243 Br CHF ₂ CI CHs

A-3203 SOCHs Br CI CHs A-3244 CN CHF ₂ CI CHs

A-3204 OCHs Br CI CHs A-3245 CHs CHF ₂ CI CHs

A-3205 CI CN CI CHs A-3246 CFs CHF ₂ CI CHs

A-3206 F CN CI CHs A-3247 CHF ₂ CHF ₂ CI CHs

A-3207 Br CN CI CHs A-3248 C3H7 CHF ₂ CI CHs

A-3208 CN CN CI CHs A-3249 CONH2 CHF ₂ CI CHs

A-3209 CHs CN CI CHs A-3250 SCHs CHF ₂ CI CHs

A-3210 CFs CN CI CHs A-3251 SOCHs CHF ₂ CI CHs

A-321 1 CHF ₂ CN CI CHs A-3252 OCHs CHF ₂ CI CHs

A-3212 C3H7 CN CI CHs A-3253 CI C3H7 CI CHs

A-3213 CONH2 CN CI CHs A-3254 F C3H7 CI CHs

A-3214 SCHs CN CI CHs A-3255 Br C3H7 CI CHs

A-3215 SOCHs CN CI CHs A-3256 CN C3H7 CI CHs line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-3257 CHs C3H7 CI CHs A-3298 SCHs SOCHs CI CHs

A-3258 CFs C3H7 CI CHs A-3299 SOCHs SOCHs CI CHs

A-3259 CHF ₂ C3H7 CI CHs A-3300 OCHs SOCHs CI CHs

A-3260 C3H7 C3H7 CI CHs A-3301 CI OCHs CI CHs

A-3261 CONH2 C3H7 CI CHs A-3302 F OCHs CI CHs

A-3262 SCHs C3H7 CI CHs A-3303 Br OCHs CI CHs

A-3263 SOCHs C3H7 CI CHs A-3304 CN OCHs CI CHs

A-3264 OCHs C3H7 CI CHs A-3305 CHs OCHs CI CHs

A-3265 CI CONH2 CI CHs A-3306 CFs OCHs CI CHs

A-3266 F CONH2 CI CHs A-3307 CHF ₂ OCHs CI CHs

A-3267 Br CONH2 CI CHs A-3308 C3H7 OCHs CI CHs

A-3268 CN CONH2 CI CHs A-3309 CONH2 OCHs CI CHs

A-3269 CHs CONH2 CI CHs A-3310 SCHs OCHs CI CHs

A-3270 CFs CONH2 CI CHs A-331 1 SOCHs OCHs CI CHs

A-3271 CHF ₂ CONH2 CI CHs A-3312 OCHs OCHs CI CHs

A-3272 C3H7 CONH2 CI CHs A-3313 CI CI CN CHs

A-3273 CONH2 CONH2 CI CHs A-3314 F CI CN CHs

A-3274 SCHs CONH2 CI CHs A-3315 Br CI CN CHs

A-3275 SOCHs CONH2 CI CHs A-3316 CN CI CN CHs

A-3276 OCHs CONH2 CI CHs A-3317 CHs CI CN CHs

A-3277 CI SCHs CI CHs A-3318 CFs CI CN CHs

A-3278 F SCHs CI CHs A-3319 CHF ₂ CI CN CHs

A-3279 Br SCHs CI CHs A-3320 C3H7 CI CN CHs

A-3280 CN SCHs CI CHs A-3321 CONH2 CI CN CHs

A-3281 CHs SCHs CI CHs A-3322 SCHs CI CN CHs

A-3282 CFs SCHs CI CHs A-3323 SOCHs CI CN CHs

A-3283 CHF ₂ SCHs CI CHs A-3324 OCHs CI CN CHs

A-3284 C3H7 SCHs CI CHs A-3325 CI F CN CHs

A-3285 CONH2 SCHs CI CHs A-3326 F F CN CHs

A-3286 SCHs SCHs CI CHs A-3327 Br F CN CHs

A-3287 SOCHs SCHs CI CHs A-3328 CN F CN CHs

A-3288 OCHs SCHs CI CHs A-3329 CHs F CN CHs

A-3289 CI SOCHs CI CHs A-3330 CFs F CN CHs

A-3290 F SOCHs CI CHs A-3331 CHF ₂ F CN CHs

A-3291 Br SOCHs CI CHs A-3332 C3H7 F CN CHs

A-3292 CN SOCHs CI CHs A-3333 CONH2 F CN CHs

A-3293 CHs SOCHs CI CHs A-3334 SCHs F CN CHs

A-3294 CFs SOCHs CI CHs A-3335 SOCHs F CN CHs

A-3295 CHF ₂ SOCHs CI CHs A-3336 OCHs F CN CHs

A-3296 C3H7 SOCHs CI CHs A-3337 CI Br CN CHs

A-3297 CONH2 SOCHs CI CHs A-3338 F Br CN CHs line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-3339 Br Br CN CHs A-3380 C3H7 CFs CN CHs

A-3340 CN Br CN CHs A-3381 CONH2 CFs CN CHs

A-3341 CHs Br CN CHs A-3382 SCHs CFs CN CHs

A-3342 CFs Br CN CHs A-3383 SOCHs CFs CN CHs

A-3343 CHF ₂ Br CN CHs A-3384 OCHs CFs CN CHs

A-3344 C3H7 Br CN CHs A-3385 CI CHF ₂ CN CHs

A-3345 CONH2 Br CN CHs A-3386 F CHF ₂ CN CHs

A-3346 SCHs Br CN CHs A-3387 Br CHF ₂ CN CHs

A-3347 SOCH3 Br CN CHs A-3388 CN CHF ₂ CN CHs

A-3348 OCH3 Br CN CHs A-3389 CHs CHF ₂ CN CHs

A-3349 CI CN CN CHs A-3390 CFs CHF ₂ CN CHs

A-3350 F CN CN CHs A-3391 CHF ₂ CHF ₂ CN CHs

A-3351 Br CN CN CHs A-3392 C3H7 CHF ₂ CN CHs

A-3352 CN CN CN CHs A-3393 CONH2 CHF ₂ CN CHs

A-3353 CHs CN CN CHs A-3394 SCHs CHF ₂ CN CHs

A-3354 CFs CN CN CHs A-3395 SOCHs CHF ₂ CN CHs

A-3355 CHF ₂ CN CN CHs A-3396 OCHs CHF ₂ CN CHs

A-3356 C3H7 CN CN CHs A-3397 CI C3H7 CN CHs

A-3357 CONH2 CN CN CHs A-3398 F C3H7 CN CHs

A-3358 SCHs CN CN CHs A-3399 Br C3H7 CN CHs

A-3359 SOCHs CN CN CHs A-3400 CN C3H7 CN CHs

A-3360 OCHs CN CN CHs A-3401 CHs C3H7 CN CHs

A-3361 CI CHs CN CHs A-3402 CFs C3H7 CN CHs

A-3362 F CHs CN CHs A-3403 CHF ₂ C3H7 CN CHs

A-3363 Br CHs CN CHs A-3404 C3H7 C3H7 CN CHs

A-3364 CN CHs CN CHs A-3405 CONH2 C3H7 CN CHs

A-3365 CHs CHs CN CHs A-3406 SCHs C3H7 CN CHs

A-3366 CFs CHs CN CHs A-3407 SOCHs C3H7 CN CHs

A-3367 CHF ₂ CHs CN CHs A-3408 OCHs C3H7 CN CHs

A-3368 C3H7 CHs CN CHs A-3409 CI CONH2 CN CHs

A-3369 CONH2 CHs CN CHs A-3410 F CONH2 CN CHs

A-3370 SCHs CHs CN CHs A-341 1 Br CONH2 CN CHs

A-3371 SOCHs CHs CN CHs A-3412 CN CONH2 CN CHs

A-3372 OCHs CHs CN CHs A-3413 CHs CONH2 CN CHs

A-3373 CI CFs CN CHs A-3414 CFs CONH2 CN CHs

A-3374 F CFs CN CHs A-3415 CHF ₂ CONH2 CN CHs

A-3375 Br CFs CN CHs A-3416 C3H7 CONH2 CN CHs

A-3376 CN CFs CN CHs A-3417 CONH2 CONH2 CN CHs

A-3377 CHs CFs CN CHs A-3418 SCHs CONH2 CN CHs

A-3378 CFs CFs CN CHs A-3419 SOCHs CONH2 CN CHs

A-3379 CHF ₂ CFs CN CHs A-3420 OCHs CONH2 CN CHs line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-3421 CI SCHs CN CHs A-3462 CFs CI CHs CHs

A-3422 F SCHs CN CHs A-3463 CHF ₂ CI CHs CHs

A-3423 Br SCHs CN CHs A-3464 C3H7 CI CHs CHs

A-3424 CN SCHs CN CHs A-3465 CONH2 CI CHs CHs

A-3425 CHs SCHs CN CHs A-3466 SCHs CI CHs CHs

A-3426 CFs SCHs CN CHs A-3467 SOCHs CI CHs CHs

A-3427 CHF ₂ SCHs CN CHs A-3468 OCHs CI CHs CHs

A-3428 C3H7 SCHs CN CHs A-3469 CI F CHs CHs

A-3429 CONH2 SCHs CN CHs A-3470 F F CHs CHs

A-3430 SCHs SCHs CN CHs A-3471 Br F CHs CHs

A-3431 SOCHs SCHs CN CHs A-3472 CN F CHs CHs

A-3432 OCHs SCHs CN CHs A-3473 CHs F CHs CHs

A-3433 CI SOCHs CN CHs A-3474 CFs F CHs CHs

A-3434 F SOCHs CN CHs A-3475 CHF ₂ F CHs CHs

A-3435 Br SOCHs CN CHs A-3476 C3H7 F CHs CHs

A-3436 CN SOCHs CN CHs A-3477 CONH2 F CHs CHs

A-3437 CHs SOCHs CN CHs A-3478 SCHs F CHs CHs

A-3438 CFs SOCHs CN CHs A-3479 SOCHs F CHs CHs

A-3439 CHF ₂ SOCHs CN CHs A-3480 OCHs F CHs CHs

A-3440 C3H7 SOCHs CN CHs A-3481 CI Br CHs CHs

A-3441 CONH2 SOCHs CN CHs A-3482 F Br CHs CHs

A-3442 SCHs SOCHs CN CHs A-3483 Br Br CHs CHs

A-3443 SOCHs SOCHs CN CHs A-3484 CN Br CHs CHs

A-3444 OCHs SOCHs CN CHs A-3485 CHs Br CHs CHs

A-3445 CI OCHs CN CHs A-3486 CFs Br CHs CHs

A-3446 F OCHs CN CHs A-3487 CHF ₂ Br CHs CHs

A-3447 Br OCHs CN CHs A-3488 C3H7 Br CHs CHs

A-3448 CN OCHs CN CHs A-3489 CONH2 Br CHs CHs

A-3449 CHs OCHs CN CHs A-3490 SCHs Br CHs CHs

A-3450 CFs OCHs CN CHs A-3491 SOCHs Br CHs CHs

A-3451 CHF ₂ OCHs CN CHs A-3492 OCHs Br CHs CHs

A-3452 C3H7 OCHs CN CHs A-3493 CI CN CHs CHs

A-3453 CONH2 OCHs CN CHs A-3494 F CN CHs CHs

A-3454 SCHs OCHs CN CHs A-3495 Br CN CHs CHs

A-3455 SOCHs OCHs CN CHs A-3496 CN CN CHs CHs

A-3456 OCHs OCHs CN CHs A-3497 CHs CN CHs CHs

A-3457 CI CI CHs CHs A-3498 CFs CN CHs CHs

A-3458 F CI CHs CHs A-3499 CHF ₂ CN CHs CHs

A-3459 Br CI CHs CHs A-3500 C3H7 CN CHs CHs

A-3460 CN CI CHs CHs A-3501 CONH2 CN CHs CHs

A-3461 CHs CI CHs CHs A-3502 SCHs CN CHs CHs line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-3503 SOCHs CN CHs CHs A-3544 CN C3H7 CHs CHs

A-3504 OCHs CN CHs CHs A-3545 CHs C3H7 CHs CHs

A-3505 CI CHs CHs CHs A-3546 CFs C3H7 CHs CHs

A-3506 F CHs CHs CHs A-3547 CHF ₂ C3H7 CHs CHs

A-3507 Br CHs CHs CHs A-3548 C3H7 C3H7 CHs CHs

A-3508 CN CHs CHs CHs A-3549 CONH2 C3H7 CHs CHs

A-3509 CHs CHs CHs CHs A-3550 SCHs C3H7 CHs CHs

A-3510 CFs CHs CHs CHs A-3551 SOCHs C3H7 CHs CHs

A-351 1 CHF ₂ CHs CHs CHs A-3552 OCHs C3H7 CHs CHs

A-3512 CsH ₇ CHs CHs CHs A-3553 CI CONH2 CHs CHs

A-3513 CONH2 CHs CHs CHs A-3554 F CONH2 CHs CHs

A-3514 SCHs CHs CHs CHs A-3555 Br CONH2 CHs CHs

A-3515 SOCHs CHs CHs CHs A-3556 CN CONH2 CHs CHs

A-3516 OCHs CHs CHs CHs A-3557 CHs CONH2 CHs CHs

A-3517 CI CFs CHs CHs A-3558 CFs CONH2 CHs CHs

A-3518 F CFs CHs CHs A-3559 CHF ₂ CONH2 CHs CHs

A-3519 Br CFs CHs CHs A-3560 C3H7 CONH2 CHs CHs

A-3520 CN CFs CHs CHs A-3561 CONH2 CONH2 CHs CHs

A-3521 CHs CFs CHs CHs A-3562 SCHs CONH2 CHs CHs

A-3522 CFs CFs CHs CHs A-3563 SOCHs CONH2 CHs CHs

A-3523 CHF ₂ CFs CHs CHs A-3564 OCHs CONH2 CHs CHs

A-3524 C3H7 CFs CHs CHs A-3565 CI SCHs CHs CHs

A-3525 CONH2 CFs CHs CHs A-3566 F SCHs CHs CHs

A-3526 SCHs CFs CHs CHs A-3567 Br SCHs CHs CHs

A-3527 SOCHs CFs CHs CHs A-3568 CN SCHs CHs CHs

A-3528 OCHs CFs CHs CHs A-3569 CHs SCHs CHs CHs

A-3529 CI CHF ₂ CHs CHs A-3570 CFs SCHs CHs CHs

A-3530 F CHF ₂ CHs CHs A-3571 CHF ₂ SCHs CHs CHs

A-3531 Br CHF ₂ CHs CHs A-3572 C3H7 SCHs CHs CHs

A-3532 CN CHF ₂ CHs CHs A-3573 CONH2 SCHs CHs CHs

A-3533 CHs CHF ₂ CHs CHs A-3574 SCHs SCHs CHs CHs

A-3534 CFs CHF ₂ CHs CHs A-3575 SOCHs SCHs CHs CHs

A-3535 CHF ₂ CHF ₂ CHs CHs A-3576 OCHs SCHs CHs CHs

A-3536 C3H7 CHF ₂ CHs CHs A-3577 CI SOCHs CHs CHs

A-3537 CONH2 CHF ₂ CHs CHs A-3578 F SOCHs CHs CHs

A-3538 SCHs CHF ₂ CHs CHs A-3579 Br SOCHs CHs CHs

A-3539 SOCHs CHF ₂ CHs CHs A-3580 CN SOCHs CHs CHs

A-3540 OCHs CHF ₂ CHs CHs A-3581 CHs SOCHs CHs CHs

A-3541 CI C3H7 CHs CHs A-3582 CFs SOCHs CHs CHs

A-3542 F C3H7 CHs CHs A-3583 CHF ₂ SOCHs CHs CHs

A-3543 Br C3H7 CHs CHs A-3584 C3H7 SOCHs CHs CHs line R ¹ R2 R ³ R ⁴ line R ¹ R2 R ³ R ⁴

A-3585 CONH ₂ SOCH3 CH ₃ CH ₃ A-3593 CH ₃ OCH3 CH ₃ CH ₃

A-3586 SCHs SOCH3 CH ₃ CH ₃ A-3594 CF ₃ OCH3 CH ₃ CH ₃

A-3587 SOCH3 SOCH3 CH ₃ CH ₃ A-3595 CHF ₂ OCH3 CH ₃ CH ₃

A-3588 OCH3 SOCH3 CH ₃ CH ₃ A-3596 C3H7 OCH3 CH ₃ CH ₃

A-3589 CI OCH3 CH ₃ CH ₃ A-3597 CONH2 OCH3 CH ₃ CH ₃

A-3590 F OCH3 CH ₃ CH ₃ A-3598 SCH ₃ OCH3 CH ₃ CH ₃

A-3591 Br OCH3 CH ₃ CH ₃ A-3599 SOCH3 OCH3 CH ₃ CH ₃

A-3592 CN OCH3 CH ₃ CH ₃ A-3600 OCH3 OCH3 CH ₃ CH ₃

The compounds of the formula I and the compositions according to the invention, respectively, are suitable as fungicides. They are distinguished by an outstanding effectiveness against a broad spectrum of phytopathogenic fungi, including soil-borne fungi, which derive especially from the following classes or are closely related to any of them: Ascomycota (Ascomycetes), for example, but not limited to the genus Cocholiobolus, Colletotrichum, Fusarium, Microdochium, Penicillium, Phoma, Magnaporte, Zymoseptoria, and Pseudocercosporella; Basdiomycota (Ba- sidiomycetes), for example, but not limited to the genus Phakospora, Puccinia, Rhizoctonia, Sphacelotheca, Tilletia, Typhula, and Ustilago; Chytridiomycota (Chytridiomycetes), for exam- pie, but not limited to the genus Chytridiales, and Synchytrium; Deuteromycetes (syn. Fungi imperfecti), for example, but not limited to the genus Ascochyta, Diplodia, Erysiphe, Fusarium, Phomopsis, and Pyrenophora; Peronosporomycetes (syn. Oomycetes), for example but not limited to the genus Peronospora, Pythium, Phytophthora; Plasmodiophoromycetes, for example but not limited to the genus Plasmodiophora; Zygomycetes, for example, but not limited to the genus Rhizopus.

The compounds I and the compositions according to the invention are particularly important in the control of a multitude of phytopathogenic fungi on various cultivated plants, such as cereals, e. g. wheat, rye, barley, triticale, oats or rice; beet, e. g. sugar beet or fodder beet; fruits, such as pomes, stone fruits or soft fruits, e. g. apples, pears, plums, peaches, almonds, cherries, strawberries, raspberries, blackberries or gooseberries; leguminous plants, such as lentils, peas, alfalfa or soybeans; oil plants, such as rape, mustard, olives, sunflowers, coconut, cocoa beans, castor oil plants, oil palms, ground nuts or soybeans; cucurbits, such as squashes, cucumber or melons; fiber plants, such as cotton, flax, hemp or jute; citrus fruit, such as oranges, lemons, grapefruits or mandarins; vegetables, such as spinach, lettuce, asparagus, cabbages, carrots, onions, tomatoes, potatoes, cucurbits or paprika; lauraceous plants, such as avocados, cinnamon or camphor; energy and raw material plants, such as corn, soybean, rape, sugar cane or oil palm; corn; tobacco; nuts; coffee; tea; bananas; vines (table grapes and grape juice grape vines); hop; turf; sweet leaf (also called Stevia); natural rubber plants or ornamental and forestry plants, such as flowers, shrubs, broad-leaved trees or evergreens, e. g. conifers; and on the plant propagation material, such as seeds, and the crop material of these plants; Preferably, compounds of the formula I and compositions thereof, respectively, are used for controlling a multitude of fungi on field crops, such as potatoes, sugar beets, tobacco, wheat, rye, barley, oats, rice, corn, cotton, soybeans, rape, legumes, sunflowers, coffee or sugar cane; fruits; vines; ornamentals; or vegetables, such as cucumbers, tomatoes, beans, carots or squashes. Particularly the compounds of the formula I and the compositions according to the invention are important in the control of phytopathogenic fungi on soybeans, cereals and corn and on the plant propagation material, such as seeds, and the crop material of these crops.

The term "plant propagation material" is to be understood to denote all the generative parts of the plant such as seeds and vegetative plant material such as cuttings and tubers (e. g. potatoes), which can be used for the multiplication of the plant. This includes seeds, roots, fruits, tubers, bulbs, rhizomes, shoots, sprouts and other parts of plants, including seedlings and young plants, which are to be transplanted after germination or after emergence from soil.

These young plants may also be protected before transplantation by a total or partial treatment by immersion or pouring.

Preferably, treatment of plant propagation materials with compounds I and compositions thereof, respectively, is used for controlling a multitude of fungi on cereals, such as wheat, rye, barley and oats; rice, corn, cotton and soybeans.

The term "cultivated plants" is to be understood as including plants which have been modified by breeding, mutagenesis or genetic engineering including but not limiting to agricultural biotech products on the market or in development (cf. http://cera-gmc.org/, see GM crop database therein). Genetically modified plants are plants, which genetic material has been so modified by the use of recombinant DNA techniques that under natural circumstances cannot readily be obtained by cross breeding, mutations or natural recombination. Typically, one or more genes have been integrated into the genetic material of a genetically modified plant in order to improve certain properties of the plant. Such genetic modifications also include but are not limited to targeted post-translational modification of protein(s), oligo- or polypeptides e. g. by glycosylation or polymer additions such as prenylated, acetylated or farnesylated moieties or PEG moieties.

Plants that have been modified by breeding, mutagenesis or genetic engineering, e. g. have been rendered tolerant to applications of specific classes of herbicides, such as auxin herbicides such as dicamba or 2,4-D; bleacher herbicides such as hydroxylphenylpyruvate dioxy- genase (HPPD) inhibitors or phytoene desaturase (PDS) inhibitors; acetolactate synthase (ALS) inhibitors such as sulfonyl ureas or imidazolinones; enolpyruvylshikimate-3-phosphate synthase (EPSPS) inhibitors, such as glyphosate; glutamine synthetase (GS) inhibitors such as glufosinate; protoporphyrinogen-IX oxidase inhibitors; lipid biosynthesis inhibitors such as acetyl CoA carboxylase (ACCase) inhibitors; or oxynil (i. e. bromoxynil or ioxynil) herbicides as a result of conventional methods of breeding or genetic engineering. Furthermore, plants have been made resistant to multiple classes of herbicides through multiple genetic modifications, such as resistance to both glyphosate and glufosinate or to both glyphosate and a herbicide from anoth- er class such as ALS inhibitors, HPPD inhibitors, auxin herbicides, or ACCase inhibitors. These herbicide resistance technologies are e. g. described in Pest Managem. Sci. 61 , 2005, 246; 61 , 2005, 258; 61 , 2005, 277; 61 , 2005, 269; 61 , 2005, 286; 64, 2008, 326; 64, 2008, 332; Weed Sci. 57, 2009, 108; Austral. J. Agricult. Res. 58, 2007, 708; Science 316, 2007, 1 185; and references quoted therein. Several cultivated plants have been rendered tolerant to herbicides by conventional methods of breeding (mutagenesis), e. g. Clearfield ^® summer rape (Canola, BASF SE, Germany) being tolerant to imidazolinones, e. g. imazamox, or ExpressSun ^® sunflowers (DuPont, USA) being tolerant to sulfonyl ureas, e. g. tribenuron. Genetic engineering methods have been used to render cultivated plants such as soybean, cotton, corn, beets and rape, tol- erant to herbicides such as glyphosate and glufosinate, some of which are commercially available under the trade names RoundupReady ^® (glyphosate-tolerant, Monsanto, U.S.A.), Cul- tivance ^® (imidazolinone tolerant, BASF SE, Germany) and LibertyLink ^® (glufosinate-tolerant, Bayer CropScience, Germany).

Furthermore, plants are also covered that are by the use of recombinant DNA techniques capable to synthesize one or more insecticidal proteins, especially those known from the bacterial genus Bacillus, particularly from Bacillus thuringiensis, such as δ-endotoxins, e. g. CrylA(b), CrylA(c), CrylF, CrylF(a2), CryllA(b), CrylllA, CrylllB(bl ) or Cry9c; vegetative insecticidal proteins (VIP), e. g. VIP1 , VIP2, VIP3 or VIP3A; insecticidal proteins of bacteria colonizing nema- todes, e. g. Photorhabdus spp. or Xenorhabdus spp.; toxins produced by animals, such as scorpion toxins, arachnid toxins, wasp toxins, or other insect-specific neurotoxins; toxins produced by fungi, such Streptomycetes toxins, plant lectins, such as pea or barley lectins; agglutinins; proteinase inhibitors, such as trypsin inhibitors, serine protease inhibitors, patatin, cystatin or papain inhibitors; ribosome-inactivating proteins (RIP), such as ricin, maize-RIP, abrin, luffin, saporin or bryodin; steroid metabolism enzymes, such as 3-hydroxysteroid oxidase, ecdyster- oid-IDP-glycosyl-transferase, cholesterol oxidases, ecdysone inhibitors or HMG-CoA-reductase; ion channel blockers, such as blockers of sodium or calcium channels; juvenile hormone esterase; diuretic hormone receptors (helicokinin receptors); stilbene synthase, bibenzyl synthase, chitinases or glucanases. In the context of the present invention these insecticidal proteins or toxins are to be understood expressly also as pre-toxins, hybrid proteins, truncated or otherwise modified proteins. Hybrid proteins are characterized by a new combination of protein domains, (see, e. g. WO 02/015701 ). Further examples of such toxins or genetically modified plants capable of synthesizing such toxins are disclosed, e. g., in EP-A 374 753, WO 93/007278, WO 95/34656, EP-A 427 529, EP-A 451 878, WO 03/18810 und WO 03/52073. The methods for producing such genetically modified plants are generally known to the person skilled in the art and are described, e. g. in the publications mentioned above. These insecticidal proteins contained in the genetically modified plants impart to the plants producing these proteins tolerance to harmful pests from all taxonomic groups of arthropods, especially to beetles (Coelop- tera), two-winged insects (Diptera), and moths (Lepidoptera) and to nematodes (Nematoda). Genetically modified plants capable to synthesize one or more insecticidal proteins are, e. g., described in the publications mentioned above, and some of which are commercially available such as YieldGard ^® (corn cultivars producing the CrylAb toxin), YieldGard ^® Plus (corn cultivars producing CrylAb and Cry3Bb1 toxins), Starlink ^® (corn cultivars producing the Cry9c toxin), Herculex ^® RW (corn cultivars producing Cry34Ab1 , Cry35Ab1 and the enzyme phosphinothri- cin-N-acetyltransferase [PAT]); NuCOTN ^® 33B (cotton cultivars producing the Cry1 Ac toxin), Bollgard ^® I (cotton cultivars producing the CrylAc toxin), Bollgard ^® II (cotton cultivars producing CrylAc and Cry2Ab2 toxins); VIPCOT ^® (cotton cultivars producing a VIP-toxin); NewLeaf ^® (potato cultivars producing the Cry3A toxin); Bt-Xtra ^® , NatureGard ^® , KnockOut ^® , BiteGard ^® , Pro- tecta ^® , Bt1 1 (e. g. Agrisure ^® CB) and Bt176 from Syngenta Seeds SAS, France, (corn cultivars producing the CrylAb toxin and PAT enyzme), MIR604 from Syngenta Seeds SAS, France (corn cultivars producing a modified version of the Cry3A toxin, c.f. WO 03/018810), MON 863 from Monsanto Europe S.A., Belgium (corn cultivars producing the Cry3Bb1 toxin), IPC 531 from Monsanto Europe S.A., Belgium (cotton cultivars producing a modified version of the CrylAc toxin) and 1507 from Pioneer Overseas Corporation, Belgium (corn cultivars producing the Cry1 F toxin and PAT enzyme).

Furthermore, plants are also covered that are by the use of recombinant DNA techniques capable to synthesize one or more proteins to increase the resistance or tolerance of those plants to bacterial, viral or fungal pathogens. Examples of such proteins are the so-called "pathogene- sis-related proteins" (PR proteins, see, e. g. EP-A 392 225), plant disease resistance genes (e. g. potato cultivars, which express resistance genes acting against Phytophthora infestans derived from the Mexican wild potato Solanum bulbocastanum) or T4-lysozym (e. g. potato cultivars capable of synthesizing these proteins with increased resistance against bacteria such as Erwinia amylvora). The methods for producing such genetically modified plants are generally known to the person skilled in the art and are described, e. g. in the publications mentioned above.

Furthermore, plants are also covered that are by the use of recombinant DNA techniques capable to synthesize one or more proteins to increase the productivity (e. g. bio mass production, grain yield, starch content, oil content or protein content), tolerance to drought, salinity or other growth-limiting environmental factors or tolerance to pests and fungal, bacterial or viral pathogens of those plants.

Furthermore, plants are also covered that contain by the use of recombinant DNA techniques a modified amount of substances of content or new substances of content, specifically to improve human or animal nutrition, e. g. oil crops that produce health-promoting long-chain ome- ga-3 fatty acids or unsaturated omega-9 fatty acids (e. g. Nexera ^® rape, DOW Agro Sciences, Canada).

Furthermore, plants are also covered that contain by the use of recombinant DNA techniques a modified amount of substances of content or new substances of content, specifically to improve raw material production, e. g. potatoes that produce increased amounts of amylopectin (e. g. Amflora ^® potato, BASF SE, Germany).

The compounds I and compositions thereof, respectively, are particularly suitable for controlling the following plant diseases:

Albugo spp. (white rust) on ornamentals, vegetables (e. g. A. Candida) and sunflowers (e. g. A. tragopogonis); Alternaria spp. (Alternaria leaf spot) on vegetables, rape (A. brassicola or brassi- cae), sugar beets (A. tenuis), fruits, rice, soybeans, potatoes (e. g. A. solani or A. alternata), tomatoes (e. g. A. solani or A. alternata) and wheat; Aphanomyces spp. on sugar beets and vegetables; Ascochyta spp. on cereals and vegetables, e. g. A. tritici (anthracnose) on wheat and A. hordei on barley; Bipolaris and Drechslera spp. (teleomorph: Cochliobolus spp.), e. g. Southern leaf blight (D. maydis) or Northern leaf blight (B. zeicola) on corn, e. g. spot blotch (B. sorokiniana) on cereals and e. g. B. oryzae on rice and turfs; Blumeria (formerly Erysiphe) graminis (powdery mildew) on cereals (e. g. on wheat or barley); Botrytis cinerea (teleomorph: Botryotinia fuckeliana: grey mold) on fruits and berries (e. g. strawberries), vegetables (e. g. lettuce, carrots, celery and cabbages), rape, flowers, vines, forestry plants and wheat; Bremia lactucae (downy mildew) on lettuce; Ceratocystis (syn. Ophiostoma) spp. (rot or wilt) on broad- leaved trees and evergreens, e. g. C. ulmi (Dutch elm disease) on elms; Cercospora spp. (Cer- cospora leaf spots) on corn (e. g. Gray leaf spot: C. zeae-maydis), rice, sugar beets (e. g. C. beticola), sugar cane, vegetables, coffee, soybeans (e. g. C. sojina or C. kikuchii) and rice; Cladosporium spp. on tomatoes (e. g. C. fulvum: leaf mold) and cereals, e. g. C. herbarum (black ear) on wheat; Claviceps purpurea (ergot) on cereals; Cochliobolus (anamorph: Helmin- thosporium of Bipolaris) spp. (leaf spots) on corn (C. carbonum), cereals (e. g. C. sativus, anamorph: B. sorokiniana) and rice (e. g. C. miyabeanus, anamorph: H. oryzae); Colletotrichum (teleomorph: Glomerella) spp. (anthracnose) on cotton (e. g. C. gossypii), corn (e. g. C. gramini- cola: Anthracnose stalk rot), soft fruits, potatoes (e. g. C. coccodes: black dot), beans (e. g. C. lindemuthianum) and soybeans (e. g. C. truncatum or C. gloeosporioides); Corticium spp., e. g. C. sasakii (sheath blight) on rice; Corynespora cassiicola (leaf spots) on soybeans and ornamentals; Cycloconium spp., e. g. C. oleaginum on olive trees; Cylindrocarpon spp. (e. g. fruit tree canker or young vine decline, teleomorph: Nectria or Neonectria spp.) on fruit trees, vines (e. g. C. liriodendri, teleomorph: Neonectria liriodendri: Black Foot Disease) and ornamentals; Dematophora (teleomorph: Rosellinia) necatrix (root and stem rot) on soybeans; Diaporthe spp., e. g. D. phaseolorum (damping off) on soybeans; Drechslera (syn. Helminthosporium, teleomorph: Pyrenophora) spp. on corn, cereals, such as barley (e. g. D. teres, net blotch) and wheat (e. g. D. tritici-repentis: tan spot), rice and turf; Esca (dieback, apoplexy) on vines, caused by Formitiporia (syn. Phellinus) punctata, F. mediterranea, Phaeomoniella chlamydospora (earlier Phaeoacremonium chlamydosporum), Phaeoacremonium aleophilum and/or Botryosphaeria obtusa; Elsinoe spp. on pome fruits (£. pyri), soft fruits (£. veneta: anthracnose) and vines (£. ampelina: anthracnose); Entyloma oryzae (leaf smut) on rice; Epicoccum spp. (black mold) on wheat; Erysiphe spp. (powdery mildew) on sugar beets (£. betae), vegetables (e. g. E. pisi), such as cucurbits (e. g. E. cichoracearum), cabbages, rape (e. g. E. cruciferarum); Eutypa lata (Eutypa canker or dieback, anamorph: Cytosporina lata, syn. Libertella blepharis) on fruit trees, vines and ornamental woods; Exserohilum (syn. Helminthosporium) spp. on corn (e. g. E. turci- cum); Fusarium (teleomorph: Gibberella) spp. (wilt, root or stem rot) on various plants, such as F. graminearum or F. culmorum (root rot, scab or head blight) on cereals (e. g. wheat or barley), F. oxysporum on tomatoes, F. solani (f. sp. glycines now syn. F. virguliforme ) and F. tucumani- ae and F. brasiliense each causing sudden death syndrome on soybeans, and F. verticillioides on corn; Gaeumannomyces graminis (take-all) on cereals (e. g. wheat or barley) and corn; Gibberella spp. on cereals (e. g. G. zeae) and rice (e. g. G. fujikuroi: Bakanae disease); Glomerella cingulata on vines, pome fruits and other plants and G. gossypii on cotton; Grainstaining complex on rice; Guignardia bidwellii (black rot) on vines; Gymnosporangium spp. on rosaceous plants and junipers, e. g. G. sabinae (rust) on pears; Helminthosporium spp. (syn. Drechslera, teleomorph: Cochliobolus) on corn, cereals and rice; Hemileia spp., e. g. H. vastatrix (coffee leaf rust) on coffee; Isariopsis clavispora (syn. Cladosporium vitis) on vines; Macrophomina phaseolina (syn. phaseoli) (root and stem rot) on soybeans and cotton; Microdochium (syn. Fusarium) nivale (pink snow mold) on cereals (e. g. wheat or barley); Microsphaera diffusa (powdery mildew) on soybeans; Monilinia spp., e. g. M. laxa, M. fructicola and M. fructigena (bloom and twig blight, brown rot) on stone fruits and other rosaceous plants; Mycosphaerella spp. on cereals, bananas, soft fruits and ground nuts, such as e. g. M. graminicola (anamorph: Septoria tritici, Septoria blotch) on wheat or M. fijiensis (black Sigatoka disease) on bananas; Peronospora spp. (downy mildew) on cabbage (e. g. P. brassicae), rape (e. g. P. parasitica), onions (e. g. P. destructor), tobacco (P. tabacina) and soybeans (e. g. P. manshurica);

Phakopsora pachyrhizi and P. meibomiae (soybean rust) on soybeans; Phialophora spp. e. g. on vines (e. g. P. tracheiphila and P. tetraspora) and soybeans (e. g. P. gregata: stem rot); Phoma lingam (root and stem rot) on rape and cabbage and P. betae (root rot, leaf spot and damping-off) on sugar beets; Phomopsis spp. on sunflowers, vines (e. g. P. viticola: can and leaf spot) and soybeans (e. g. stem rot: P. phaseoli, teleomorph: Diaporthe phaseolorum); Phy- soderma maydis (brown spots) on corn; Phytophthora spp. (wilt, root, leaf, fruit and stem root) on various plants, such as paprika and cucurbits (e. g. P. capsici), soybeans (e. g. P.

megasperma, syn. P. sojae), potatoes and tomatoes (e. g. P. infestans: late blight) and broad- leaved trees (e. g. P. ramorum: sudden oak death); Plasmodiophora brassicae (club root) on cabbage, rape, radish and other plants; Plasmopara spp., e. g. P. viticola (grapevine downy mildew) on vines and P. halstedii on sunflowers; Podosphaera spp. (powdery mildew) on rosa- ceous plants, hop, pome and soft fruits, e. g. P. leucotricha on apples; Polymyxa spp., e. g. on cereals, such as barley and wheat (P. graminis) and sugar beets (P. betae) and thereby transmitted viral diseases; Pseudocercosporella herpotrichoides (eyespot, teleomorph: Tapesia yal- lundae) on cereals, e. g. wheat or barley; Pseudoperonospora (downy mildew) on various plants, e. g. P. cubensis on cucurbits or P. humili on hop; Pseudopezicula tracheiphila (red fire disease or .rotbrenner', anamorph: Phialophora) on vines; Puccinia spp. (rusts) on various plants, e. g. P. triticina (brown or leaf rust), P. striiformis (stripe or yellow rust), P. hordei (dwarf rust), P. graminis (stem or black rust) or P. recondita (brown or leaf rust) on cereals, such as e. g. wheat, barley or rye, P. kuehnii (orange rust) on sugar cane and P. asparagi on asparagus; Pyrenophora (anamorph: Drechslera) tritici-repentis (tan spot) on wheat or P. feres (net blotch) on barley; Pyricularia spp., e. g. P. oryzae (teleomorph: Magnaporthe grisea, rice blast) on rice and P. grisea on turf and cereals; Pythium spp. (damping-off) on turf, rice, corn, wheat, cotton, rape, sunflowers, soybeans, sugar beets, vegetables and various other plants (e. g. P. ultimum or P. aphanidermatum); Ramularia spp., e. g. R. collo-cygni (Ramularia leaf spots, Physiological leaf spots) on barley and R. beticola on sugar beets; Rhizoctonia spp. on cotton, rice, potatoes, turf, corn, rape, potatoes, sugar beets, vegetables and various other plants, e. g. R. solani (root and stem rot) on soybeans, R. solani (sheath blight) on rice or R. cerealis (Rhizoctonia spring blight) on wheat or barley; Rhizopus stolonifer (black mold, soft rot) on strawberries, carrots, cabbage, vines and tomatoes; Rhynchosporium secalis (scald) on barley, rye and triticale; Sa- rocladium oryzae and S. attenuatum (sheath rot) on rice; Sclerotinia spp. (stem rot or white mold) on vegetables and field crops, such as rape, sunflowers (e. g. S. sclerotiorum) and soybeans (e. g. S. rolfsii or S. sclerotiorum); Septoria spp. on various plants, e. g. S. glycines (brown spot) on soybeans, S. tritici (Septoria blotch) on wheat and S. (syn. Stagonospora) no- dorum (Stagonospora blotch) on cereals; Uncinula (syn. Erysiphe) necator (powdery mildew, anamorph: Oidium tuckeri) on vines; Setospaeria spp. (leaf blight) on corn (e. g. S. turcicum, syn. Helminthosporium turcicum) and turf; Sphacelotheca spp. (smut) on corn, (e. g. S. reiliana: head smut), sorghum und sugar cane; Sphaerotheca fuliginea (powdery mildew) on cucurbits; Spongospora subterranea (powdery scab) on potatoes and thereby transmitted viral diseases; Stagonospora spp. on cereals, e. g. S. nodorum (Stagonospora blotch, teleomorph: Lepto- sphaeria [syn. Phaeosphaeria] nodorum) on wheat; Synchytrium endobioticum on potatoes (po- tato wart disease); Taphrina spp., e. g. T. deformans (leaf curl disease) on peaches and T. pruni (plum pocket) on plums; Thielaviopsis spp. (black root rot) on tobacco, pome fruits, vegetables, soybeans and cotton, e. g. T. basicola (syn. Chalara elegans); Tilletia spp. (common bunt or stinking smut) on cereals, such as e. g. T. tritici (syn. T. caries, wheat bunt) and T. controversa (dwarf bunt) on wheat; Typhula incarnata (grey snow mold) on barley or wheat; Urocystis spp., e. g. U. occulta (stem smut) on rye; Uromyces spp. (rust) on vegetables, such as beans (e. g. U. appendiculatus, syn. U. phaseoli) and sugar beets (e. g. U. betae); Ustilago spp. (loose smut) on cereals (e. g. U. nuda and U. avaenae), corn (e. g. U. maydis: corn smut) and sugar cane; Venturia spp. (scab) on apples (e. g. V. inaequalis) and pears; and Verticillium spp. (wilt) on various plants, such as fruits and ornamentals, vines, soft fruits, vegetables and field crops, e. g. V. dahliae on strawberries, rape, potatoes and tomatoes.

The compounds I and compositions thereof, respectively, are also suitable for controlling harmful fungi in the protection of stored products or harvest and in the protection of materials.

The term "protection of materials" is to be understood to denote the protection of technical and non-living materials, such as adhesives, glues, wood, paper and paperboard, textiles, leather, paint dispersions, plastics, cooling lubricants, fiber or fabrics, against the infestation and destruction by harmful microorganisms, such as fungi and bacteria. As to the protection of wood and other materials, the particular attention is paid to the following harmful fungi: Ascomycetes such as Ophiostoma spp., Ceratocystis spp., Aureobasidium pullulans, Sclerophoma spp., Chaetomium spp., Humicola spp., Petriella spp., Trichurus spp.; Basidiomycetes such as Coni- ophora spp., Coriolus spp., Gloeophyllum spp., Lentinus spp., Pleurotus spp., Poria spp., Ser- pula spp. and Tyromyces spp., Deuteromycetes such as Aspergillus spp., Cladosporium spp., Penicillium spp., Trichoderma spp., Alternaria spp., Paecilomyces spp. and Zygomycetes such as Mucor spp., and in addition in the protection of stored products and harvest the following yeast fungi are worthy of note: Candida spp. and Saccharomyces cerevisae.

The method of treatment according to the invention can also be used in the field of protecting stored products or harvest against attack of fungi and microorganisms. According to the present invention, the term "stored products" is understood to denote natural substances of plant or animal origin and their processed forms, which have been taken from the natural life cycle and for which long-term protection is desired. Stored products of crop plant origin, such as plants or parts thereof, for example stalks, leafs, tubers, seeds, fruits or grains, can be protected in the freshly harvested state or in processed form, such as pre-dried, moistened, comminuted, ground, pressed or roasted, which process is also known as post-harvest treatment. Also falling under the definition of stored products is timber, whether in the form of crude timber, such as construction timber, electricity pylons and barriers, or in the form of finished articles, such as furniture or objects made from wood. Stored products of animal origin are hides, leather, furs, hairs and the like. The combinations according the present invention can prevent disadvantageous effects such as decay, discoloration or mold. Preferably "stored products" is understood to denote natural substances of plant origin and their processed forms, more preferably fruits and their processed forms, such as pomes, stone fruits, soft fruits and citrus fruits and their processed forms.

The compounds I and compositions thereof, respectively, may be used for improving the health of a plant. The invention also relates to a method for improving plant health by treating a plant, its propagation material and/or the locus where the plant is growing or is to grow with an effective amount of compounds I and compositions thereof, respectively.

The term "plant health" is to be understood to denote a condition of the plant and/or its products which is determined by several indicators alone or in combination with each other such as yield (e. g. increased biomass and/or increased content of valuable ingredients), plant vigor (e. g. improved plant growth and/or greener leaves ("greening effect")), quality (e. g. improved content or composition of certain ingredients) and tolerance to abiotic and/or biotic stress. The above identified indicators for the health condition of a plant may be interdependent or may re- suit from each other.

The compounds of formula I can be present in different crystal modifications whose biological activity may differ. They are likewise subject matter of the present invention.

The compounds I are employed as such or in form of compositions by treating the fungi or the plants, plant propagation materials, such as seeds, soil, surfaces, materials or rooms to be pro- tected from fungal attack with a fungicidally effective amount of the active substances. The application can be carried out both before and after the infection of the plants, plant propagation materials, such as seeds, soil, surfaces, materials or rooms by the fungi.

Plant propagation materials may be treated with compounds I as such or a composition comprising at least one compound I prophylactically either at or before planting or transplanting. The invention also relates to agrochemical compositions comprising an auxiliary and at least one compound I according to the invention.

An agrochemical composition comprises a fungicidally effective amount of a compound I. The term "effective amount" denotes an amount of the composition or of the compounds I, which is sufficient for controlling harmful fungi on cultivated plants or in the protection of materials and which does not result in a substantial damage to the treated plants. Such an amount can vary in a broad range and is dependent on various factors, such as the fungal species to be controlled, the treated cultivated plant or material, the climatic conditions and the specific compound I used.

The compounds I, their N-oxides and salts can be converted into customary types of agro- chemical compositions, e. g. solutions, emulsions, suspensions, dusts, powders, pastes, granules, pressings, capsules, and mixtures thereof. Examples for composition types are suspensions (e. g. SC, OD, FS), emulsifiable concentrates (e. g. EC), emulsions (e. g. EW, EO, ES, ME), capsules (e. g. CS, ZC), pastes, pastilles, wettable powders or dusts (e. g. WP, SP, WS, DP, DS), pressings (e. g. BR, TB, DT), granules (e. g. WG, SG, GR, FG, GG, MG), insecticidal articles (e. g. LN), as well as gel formulations for the treatment of plant propagation materials such as seeds (e. g. GF). These and further compositions types are defined in the "Catalogue of pesticide formulation types and international coding system", Technical Monograph No. 2, 6 ^th Ed. May 2008, CropLife International.

The compositions are prepared in a known manner, such as described by Mollet and Grube- mann, Formulation technology, Wiley VCH, Weinheim, 2001 ; or Knowles, New developments in crop protection product formulation, Agrow Reports DS243, T&F Informa, London, 2005.

Suitable auxiliaries are solvents, liquid carriers, solid carriers or fillers, surfactants, disper- sants, emulsifiers, wetters, adjuvants, solubilizers, penetration enhancers, protective colloids, adhesion agents, thickeners, humectants, repellents, attractants, feeding stimulants, compatibil- izers, bactericides, anti-freezing agents, anti-foaming agents, colorants, tackifiers and binders.

Suitable solvents and liquid carriers are water and organic solvents, such as mineral oil frac- tions of medium to high boiling point, e. g. kerosene, diesel oil; oils of vegetable or animal origin; aliphatic, cyclic and aromatic hydrocarbons, e. g. toluene, paraffin, tetrahydronaphthalene, alkylated naphthalenes; alcohols, e. g. ethanol, propanol, butanol, benzyl alcohol, cyclohexanol; glycols; DMSO; ketones, e. g. cyclohexanone; esters, e. g. lactates, carbonates, fatty acid es- ters, gamma-butyrolactone; fatty acids; phosphonates; amines; amides, e. g. N-methyl pyrroli- done, fatty acid dimethyl amides; and mixtures thereof.

Suitable solid carriers or fillers are mineral earths, e. g. silicates, silica gels, talc, kaolins, limestone, lime, chalk, clays, dolomite, diatomaceous earth, bentonite, calcium sulfate, magnesium sulfate, magnesium oxide; polysaccharides, e. g. cellulose, starch; fertilizers, e. g. ammonium sulfate, ammonium phosphate, ammonium nitrate, ureas; products of vegetable origin, e. g. cereal meal, tree bark meal, wood meal, nutshell meal, and mixtures thereof.

Suitable surfactants are surface-active compounds, such as anionic, cationic, nonionic and amphoteric surfactants, block polymers, polyelectrolytes, and mixtures thereof. Such surfactants can be used as emulsifier, dispersant, solubilizer, wetter, penetration enhancer, protective col- loid, or adjuvant. Examples of surfactants are listed in McCutcheon's, Vol.1 : Emulsifiers & Detergents, McCutcheon's Directories, Glen Rock, USA, 2008 (International Ed. or North American Ed.).

Suitable anionic surfactants are alkali, alkaline earth or ammonium salts of sulfonates, sulfates, phosphates, carboxylates, and mixtures thereof. Examples of sulfonates are alkylaryl sul- fonates, diphenyl sulfonates, alpha-olefin sulfonates, lignin sulfonates, sulfonates of fatty acids and oils, sulfonates of ethoxylated alkylphenols, sulfonates of alkoxylated arylphenols, sulfonates of condensed naphthalenes, sulfonates of dodecyl- and tridecylbenzenes, sulfonates of naphthalenes and alkyl naphthalenes, sulfosuccinates or sulfosuccinamates. Examples of sulfates are sulfates of fatty acids and oils, of ethoxylated alkylphenols, of alcohols, of ethoxylated alcohols, or of fatty acid esters. Examples of phosphates are phosphate esters. Examples of carboxylates are alkyl carboxylates, and carboxylated alcohol or alkylphenol ethoxylates.

Suitable nonionic surfactants are alkoxylates, N-substituted fatty acid amides, amine oxides, esters, sugar-based surfactants, polymeric surfactants, and mixtures thereof. Examples of alkoxylates are compounds such as alcohols, alkylphenols, amines, amides, arylphenols, fatty acids or fatty acid esters which have been alkoxylated with 1 to 50 equivalents. Ethylene oxide and/or propylene oxide may be employed for the alkoxylation, preferably ethylene oxide. Examples of N-substituted fatty acid amides are fatty acid glucamides or fatty acid alkanolamides. Examples of esters are fatty acid esters, glycerol esters or monoglycerides. Examples of sugar- based surfactants are sorbitans, ethoxylated sorbitans, sucrose and glucose esters or al- kylpolyglucosides. Examples of polymeric surfactants are home- or copolymers of vinyl pyrroli- done, vinyl alcohols, or vinyl acetate.

Suitable cationic surfactants are quaternary surfactants, for example quaternary ammonium compounds with one or two hydrophobic groups, or salts of long-chain primary amines. Suitable amphoteric surfactants are alkylbetains and imidazolines. Suitable block polymers are block polymers of the A-B or A-B-A type comprising blocks of polyethylene oxide and polypropylene oxide, or of the A-B-C type comprising alkanol, polyethylene oxide and polypropylene oxide. Suitable polyelectrolytes are polyacids or polybases. Examples of polyacids are alkali salts of polyacrylic acid or polyacid comb polymers. Examples of polybases are polyvinyl amines or polyethylene amines.

Suitable adjuvants are compounds, which have a negligible or even no pesticidal activity themselves, and which improve the biological performance of the compound I on the target. Examples are surfactants, mineral or vegetable oils, and other auxiliaries. Further examples are listed by Knowles, Adjuvants and additives, Agrow Reports DS256, T&F Informa UK, 2006, chapter 5.

Suitable thickeners are polysaccharides (e. g. xanthan gum, carboxymethyl cellulose), inorganic clays (organically modified or unmodified), polycarboxylates, and silicates.

Suitable bactericides are bronopol and isothiazolinone derivatives such as alkyliso- thiazolinones and benzisothiazolinones.

Suitable anti-freezing agents are ethylene glycol, propylene glycol, urea and glycerin.

Suitable anti-foaming agents are silicones, long chain alcohols, and salts of fatty acids.

Suitable colorants (e. g. in red, blue, or green) are pigments of low water solubility and water- soluble dyes. Examples are inorganic colorants (e. g. iron oxide, titan oxide, iron hexacyanofer- rate) and organic colorants (e. g. alizarin-, azo- and phthalocyanine colorants).

Suitable tackifiers or binders are polyvinyl pyrrolidones, polyvinyl acetates, polyvinyl alcohols, polyacrylates, biological or synthetic waxes, and cellulose ethers. Examples for composition types and their preparation are:

i) Water-soluble concentrates (SL, LS)

10-60 wt% of a compound I and 5-15 wt% wetting agent (e. g. alcohol alkoxylates) are dissolved in water and/or in a water-soluble solvent (e. g. alcohols) ad 100 wt%. The active substance dissolves upon dilution with water.

ii) Dispersible concentrates (DC)

5-25 wt% of a compound I and 1 -10 wt% dispersant (e. g. polyvinyl pyrrolidone) are dissolved in organic solvent (e. g. cyclohexanone) ad 100 wt%. Dilution with water gives a dispersion. iii) Emulsifiable concentrates (EC)

15-70 wt% of a compound I and 5-10 wt% emulsifiers (e. g. calcium dodecylbenzenesulfonate and castor oil ethoxylate) are dissolved in water-insoluble organic solvent (e. g. aromatic hydrocarbon) ad 100 wt%. Dilution with water gives an emulsion.

iv) Emulsions (EW, EO, ES)

5-40 wt% of a compound I and 1 -10 wt% emulsifiers (e. g. calcium dodecylbenzenesulfonate and castor oil ethoxylate) are dissolved in 20-40 wt% water-insoluble organic solvent (e. g. aro- matic hydrocarbon). This mixture is introduced into water ad 100 wt% by means of an emulsifying machine and made into a homogeneous emulsion. Dilution with water gives an emulsion. v) Suspensions (SC, OD, FS) In an agitated ball mill, 20-60 wt% of a compound I are comminuted with addition of 2-10 wt% dispersants and wetting agents (e. g. sodium lignosulfonate and alcohol ethoxylate), 0.1 -2 wt% thickener (e. g. xanthan gum) and water ad 100 wt% to give a fine active substance suspension. Dilution with water gives a stable suspension of the active substance. For FS type composition up to 40 wt% binder (e. g. polyvinyl alcohol) is added.

vi) Water-dispersible granules and water-soluble granules (WG, SG)

50-80 wt% of a compound I are ground finely with addition of dispersants and wetting agents (e. g. sodium lignosulfonate and alcohol ethoxylate) ad 100 wt% and prepared as water- dispersible or water-soluble granules by means of technical appliances (e. g. extrusion, spray tower, fluidized bed). Dilution with water gives a stable dispersion or solution of the active substance.

vii) Water-dispersible powders and water-soluble powders (WP, SP, WS)

50-80 wt% of a compound I are ground in a rotor-stator mill with addition of 1 -5 wt% dispersants (e. g. sodium lignosulfonate), 1 -3 wt% wetting agents (e. g. alcohol ethoxylate) and solid carrier (e. g. silica gel) ad 100 wt%. Dilution with water gives a stable dispersion or solution of the active substance.

viii) Gel (GW, GF)

In an agitated ball mill, 5-25 wt% of a compound I are comminuted with addition of 3-10 wt% dispersants (e. g. sodium lignosulfonate), 1 -5 wt% thickener (e. g. carboxymethyl cellulose) and water ad 100 wt% to give a fine suspension of the active substance. Dilution with water gives a stable suspension of the active substance.

ix) Microemulsion (ME)

5-20 wt% of a compound I are added to 5-30 wt% organic solvent blend (e. g. fatty acid dimethyl amide and cyclohexanone), 10-25 wt% surfactant blend (e. g. alcohol ethoxylate and ar- ylphenol ethoxylate), and water ad 100 %. This mixture is stirred for 1 h to produce spontaneously a thermodynamically stable microemulsion.

x) Microcapsules (CS)

An oil phase comprising 5-50 wt% of a compound I, 0-40 wt% water insoluble organic solvent (e. g. aromatic hydrocarbon), 2-15 wt% acrylic monomers (e. g. methylmethacrylate, methacrylic acid and a di- or triacrylate) are dispersed into an aqueous solution of a protective colloid (e. g. polyvinyl alcohol). Radical polymerization results in the formation of poly(meth)acrylate microcapsules. Alternatively, an oil phase comprising 5-50 wt% of a compound I according to the invention, 0-40 wt% water insoluble organic solvent (e. g. aromatic hydrocarbon), and an isocya- nate monomer (e. g. diphenylmethene-4,4'-diisocyanatae) are dispersed into an aqueous solu- tion of a protective colloid (e. g. polyvinyl alcohol). The addition of a polyamine (e. g. hexameth- ylenediamine) results in the formation of polyurea microcapsules. The monomers amount to 1 - 10 wt%. The wt% relate to the total CS composition.

xi) Dustable powders (DP, DS)

1 -10 wt% of a compound I are ground finely and mixed intimately with solid carrier (e. g. finely divided kaolin) ad 100 wt%. xii) Granules (GR, FG)

0.5-30 wt% of a compound I is ground finely and associated with solid carrier (e. g. silicate) ad 100 wt%. Granulation is achieved by extrusion, spray-drying or fluidized bed.

xiii) Ultra-low volume liquids (UL)

1 -50 wt% of a compound I are dissolved in organic solvent (e. g. aromatic hydrocarbon) ad 100 wt%.

The compositions types i) to xiii) may optionally comprise further auxiliaries, such as 0.1 -1 wt% bactericides, 5-15 wt% anti-freezing agents, 0.1 -1 wt% anti-foaming agents, and 0.1 -1 wt% colorants.

The agrochemical compositions generally comprise between 0.01 and 95%, preferably between 0.1 and 90%, and in particular between 0.5 and 75%, by weight of active substance. The active substances are employed in a purity of from 90% to 100%, preferably from 95% to 100% (according to NMR spectrum).

For the purposes of treatment of plant propagation materials, particularly seeds, solutions for seed treatment (LS), Suspoemulsions (SE), flowable concentrates (FS), powders for dry treatment (DS), water-dispersible powders for slurry treatment (WS), water-soluble powders (SS), emulsions (ES), emulsifiable concentrates (EC), and gels (GF) are usually employed. The compositions in question give, after two-to-tenfold dilution, active substance concentrations of from 0.01 to 60% by weight, preferably from 0.1 to 40%, in the ready-to-use preparations. Application can be carried out before or during sowing. Methods for applying compound I and compositions thereof, respectively, onto plant propagation material, especially seeds, include dressing, coating, pelleting, dusting, and soaking as well as in-furrow application methods. Preferably, compound I or the compositions thereof, respectively, are applied on to the plant propagation mate- rial by a method such that germination is not induced, e. g. by seed dressing, pelleting, coating and dusting.

When employed in plant protection, the amounts of active substances applied are, depending on the kind of effect desired, from 0.001 to 2 kg per ha, preferably from 0.005 to 2 kg per ha, more preferably from 0.05 to 0.9 kg per ha, and in particular from 0.1 to 0.75 kg per ha.

In treatment of plant propagation materials such as seeds, e. g. by dusting, coating or drenching seed, amounts of active substance of from 0.1 to 1000 g, preferably from 1 to 1000 g, more preferably from 1 to 100 g and most preferably from 5 to 100 g, per 100 kilogram of plant propagation material (preferably seeds) are generally required.

When used in the protection of materials or stored products, the amount of active substance applied depends on the kind of application area and on the desired effect. Amounts customarily applied in the protection of materials are 0.001 g to 2 kg, preferably 0.005 g to 1 kg, of active substance per cubic meter of treated material.

Various types of oils, wetters, adjuvants, fertilizer, or micronutrients, and further pesticides (e. g. herbicides, insecticides, fungicides, growth regulators, safeners, biopesticides) may be added to the active substances or the compositions comprising them as premix or, if appropriate not until immediately prior to use (tank mix). These agents can be admixed with the compositions according to the invention in a weight ratio of 1 :100 to 100:1 , preferably 1 :10 to 10:1.

A pesticide is generally a chemical or biological agent (such as pestidal active ingredient, compound, composition, virus, bacterium, antimicrobial or disinfectant) that through its effect deters, incapacitates, kills or otherwise discourages pests. Target pests can include insects, plant pathogens, weeds, mollusks, birds, mammals, fish, nematodes (roundworms), and microbes that destroy property, cause nuisance, spread disease or are vectors for disease. The term "pesticide" includes also plant growth regulators that alter the expected growth, flowering, or reproduction rate of plants; defoliants that cause leaves or other foliage to drop from a plant, usually to facilitate harvest; desiccants that promote drying of living tissues, such as unwanted plant tops; plant activators that activate plant physiology for defense of against certain pests; safeners that reduce unwanted herbicidal action of pesticides on crop plants; and plant growth promoters that affect plant physiology e.g. to increase plant growth, biomass, yield or any other quality parameter of the harvestable goods of a crop plant.

The user applies the composition according to the invention usually from a predosage device, a knapsack sprayer, a spray tank, a spray plane, or an irrigation system. Usually, the agrochemical composition is made up with water, buffer, and/or further auxiliaries to the desired application concentration and the ready-to-use spray liquor or the agrochemical composition according to the invention is thus obtained. Usually, 20 to 2000 liters, preferably 50 to 400 liters, of the ready-to-use spray liquor are applied per hectare of agricultural useful area.

According to one embodiment, individual components of the composition according to the invention such as parts of a kit or parts of a binary or ternary mixture may be mixed by the user himself in a spray tank or any other kind of vessel used for applications (e. g. seed treater drums, seed pelleting machinery, knapsack sprayer) and further auxiliaries may be added, if appropriate.

Consequently, one embodiment of the invention is a kit for preparing a usable pesticidal composition, the kit comprising a) a composition comprising component 1 ) as defined herein and at least one auxiliary; and b) a composition comprising component 2) as defined herein and at least one auxiliary; and optionally c) a composition comprising at least one auxiliary and optionally a further active component 3) as defined herein.

Mixing the compounds I or the compositions comprising them in the use form as fungicides with other fungicides results in many cases in an expansion of the fungicidal spectrum of activity being obtained or in a prevention of fungicide resistance development. Furthermore, in many cases, synergistic effects are obtained.

The following list of pesticides II, or component 2) (e. g. pesticidally-active substances), in conjunction with which the compounds I can be used, is intended to illustrate the possible combinations but does not limit them:

A) Respiration inhibitors

- Inhibitors of complex III at Q ₀ site (e. g. strobilurins): azoxystrobin (A.1 .1 ), coumeth- oxystrobin (A.1 .2), coumoxystrobin (A.1.3), dimoxystrobin (A.1.4), enestroburin (A.1 .5), fenaminstrobin (A.1 .6), fenoxystrobin/flufenoxystrobin (A.1 .7), fluoxastrobin (A.1.8), kresox- im-methyl (A.1.9), mandestrobin (A.1.10), metominostrobin (A.1.1 1 ), orysastrobin (A.1.12), picoxystrobin (A.1.13), pyraclostrobin (A.1.14), pyrametostrobin (A.1.15), pyraoxystrobin (A.1.16), trifloxystrobin (A.1 .17), 2-(2-(3-(2,6-dichlorophenyl)-1 -methyl-allylideneaminooxy- methyl)-phenyl)-2-methoxyimino-N-methyl-acetamide (A.1 .18), pyribencarb (A.1.19), triclopyricarb/chlorodincarb (A.1.20), famoxadone (A.1.21 ), fenamidone (A.1 .21 ), methyl-/V- [2-[(1 ,4-dimethyl-5-phenyl-pyrazol-3-yl)oxylmethyl]phenyl]-N-metho xy-carbamate (A.1.22), 1 -[3-chloro-2-[[1 -(4-chlorophenyl)pyrazol-3-yl]oxymethyl]phenyl]-4-methyl-tet razol-5-one instead of 1 -[3-chloro-2-[[[1 -(4-chlorophenyl)-1 H-pyrazol-3-yl]oxy]methyl]phenyl]-1 ,4-dihydro- 4-methyl-5H-tetrazol-5-one (A.1.23), (Z,2E)-5-[1 -(2,4-dichlorophenyl)-1 H-pyrazo!-3-yl]oxy-2-

(methoxyimino)-N,3-dimethyl-pent-3-enamide (A.1 .24), (Z,2E)-5-[1 -(4-chlorophenyl)-1 H- pyrazol-3-yl]oxy-2-(methoxyimino)-N,3-dirnethyl-pent-3-enami de (A.1.25), (Z,2E)-5-[1 -(4- chloro-2-fluoro-phenyl)pyrazol-3-yl]oxy-2-methoxyimino-N,3-d imethyl-pent-3-enamide (A.1.26), 1 -[3-bromo-2-[[1 -(4-chlorophenyl)pyrazol-3-yl]oxymethyl]phenyl]-4-methyl-tet razol- 5-one (A.1 .27),

1 -[2-[[1 -(4-chlorophenyl)pyrazol-3-yl]oxymethyl]-3-methyl-phenyl]-4- methyl-tetrazol-5-one (A.1.28). 1 -f2-[[1 -(4-chlorophenyl)pyrazol-3-yl]oxymethyl]-3-fluoro-phenyl]-4- methyl-tetrazol- 5-one (A.1 .29). 1 -[2-[[1 -(2,4-dichlorophenyl)pyrazol-3-yl]oxymethyl]-3-fluoro-phenyl ]-4- methyl-tetrazol-5-one (A.1.30), 1 -[2-[[4-(4-chlorophenyl)thiazol-2-yl]oxymethyl]-3-methyl- phenyl]-4-rnethyl-tetrazol-5-one (A.1 .31 ), 1 -[3-chloro-2-[[4-(p-tolyl)thiazol-2- yl]oxymethyl]phenyl]-4-methyl-tetrazol-5-one (A.1 .32), 1 -[3-cyclopropyl-2-[[2-methyl-4-(1 - methylpyrazol-3-yl)phenoxy]methyl]pheny!]-4-methyl-tetrazol- 5-one (A.1.33);

inhibitors of complex III at Q, site: cyazofamid (A.2.1 ), amisulbrom (A.2.2),

[(3S,6S,7R,8R)-8-benzyl-3-[(3-acetoxy-4-methoxy-pyridine- 2-carbonyl)amino]-6-methyl-4,9- dioxo-1 ,5-dioxonan-7-yl] 2-methylpropanoate (A.2.3), [(3S,6S,7R,8R)-8-benzyl-3-[[3-(acet- oxymethoxy)-4-methoxy-pyridine-2-carbonyl]amino]-6-methyl-4, 9-dioxo-1 ,5-dioxonan-7-yl] 2-methylpropanoate (A.2.4), [(3S,6S,7R,8R)-8-benzyl-3-[(3-isobutoxycarbonyloxy-4-meth- oxy-pyridine-2-carbonyl)amino]-6-methyl-4,9-dioxo-1 ,5-dioxonan-7-yl] 2-methylpropanoate (A.2.5), [(3S,6S,7R,8R)-8-benzyl-3-[[3-(1 ,3-benzodioxol-5-ylmethoxy)-4-methoxy-pyridine-2- carbonyl]amino]-6-methyl-4,9-dioxo-1 ,5-dioxonan-7-yl] 2-methylpropanoate (A.2.6);

(3S,6S,7R,8R)-3-[[(3-hydroxy-4-methoxy-2-pyridinyl)carbonyl] amino]-6-methyl-4,9-dioxo-8- (phenylmethyl)-1 ,5-dioxonan-7-yl 2-methylpropanoate (A.2.7), (3S,6S,7R,8R)-8-benzyl-3-[3- [(isobutyryloxy)methoxy]-4-methoxypicolinamido]-6-methyl-4,9 -dioxo-1 ,5-dioxonan-7-yl iso- butyrate (A.2.8);

- inhibitors of complex II (e. g. carboxamides): benodanil (A.3.1 ), benzovindiflupyr

(A.3.2), bixafen (A.3.3), boscalid (A.3.4), carboxin (A.3.5), fenfuram (A.3.6), fluopyram (A.3.7), flutolanil (A.3.8), fluxapyroxad (A.3.9), furametpyr (A.3.10), isofetamid (A.3.1 1 ), iso- pyrazam (A.3.12), mepronil (A.3.13), oxycarboxin (A.3.14), penflufen (A.3.14), penthiopyrad (A.3.15), sedaxane (A.3.16), tecloftalam (A.3.17), thifluzamide (A.3.18), N-(4'- trifluoromethylthiobiphenyl-2-yl)-3-difluoromethyl-1-methyl- 1 H-pyrazole-4-carboxamide (A.3.19), N-(2-(1 ,3,3-trimethyl-butyl)-phenyl)-1 ,3-dimethyl-5-fluoro-1 H-pyrazole- 4-carboxamide (A.3.20), 3-(difluoromethyl)-1 -methyl-N-(1 ,1 ,3-trimethylindan-4-yl)pyrazole-4- carboxamide (A.3.21 ), 3-(trifluoromethyl)-1 -methyl-N-(1 ,1 ,3-trimethylindan-4-yl)pyrazole-4- carboxamide (A.3.22), 1 ,3-dimethyl-N-(1 ,1 ,3-trimethylindan-4-yl)pyrazole-4-carboxamide (A.3.23), 3-(trifluoromethyl)-1 ,5-dimethyl-N-(1 ,1 ,3-trimethylindan-4-yl)pyrazole-4- carboxamide (A.3.24), 1 ,3,5-trimethyl-N-(1 ,1 ,3-trimethylindan-4-yl)pyrazole-4-carboxamide (A.3.25), N-(7-fluoro-1 ,1 ,3-trimethyl-indan-4-yl)-1 ,3-dimethyl-pyrazole-4-carboxamide (A.3.26), N-[2-(2,4-dichlorophenyl)-2-methoxy-1 -methyl-ethyl]-3-(difluoromethyl)-1 -methyl- pyrazole-4-carboxamide (A.3.27);

other respiration inhibitors (e. g. complex I, uncouplers): diflumetorim (A.4.1 ), (5,8- difluoroquinazolin-4-yl)-{2-[2-fluoro-4-(4-trifluoromethylpy ridin-2-yloxy)-phenyl]-ethyl}-amine (A.4.2); nitrophenyl derivates: binapacryl (A.4.3), dinobuton (A.4.4), dinocap (A.4.5), fluazi- nam (A.4.6); ferimzone (A.4.7); organometal compounds: fentin salts, such as fentin-acetate (A.4.8), fentin chloride (A.4.9) or fentin hydroxide (A.4.10); ametoctradin (A.4.1 1 ); and silthi- ofam (A.4.12);

B) Sterol biosynthesis inhibitors (SBI fungicides)

C14 demethylase inhibitors (DMI fungicides): triazoles: azaconazole (B.1 .1 ), biterta- nol (B.1.2), bromuconazole (B.1 .3), cyproconazole (B.1.4), difenoconazole (B.1.5), dinicona- zole (B.1.6), diniconazole-M (B.1 .7), epoxiconazole (B.1.8), fenbuconazole (B.1.9), fluquin- conazole (B.1 .10), flusilazole (B.1.1 1 ), flutriafol (B.1.12), hexaconazole (B.1 .13), imiben- conazole (B.1.14), ipconazole (B.1.15), metconazole (B.1.17), myclobutanil (B.1.18), oxpoconazole (B.1 .19), paclobutrazole (B.1 .20), penconazole (B.1 .21 ), propiconazole (B.1.22), prothioconazole (B.1.23), simeconazole (B.1 .24), tebuconazole (B.1 .25), tetracon- azole (B.1 .26), triadimefon (B.1.27), triadimenol (B.1.28), triticonazole (B.1 .29), uniconazole (B.1.30), 1 -[re/-(2S;3R)-3-(2-chlorophenyl)-2-(2,4-difluorophenyl)-oxir anylmethyl]-5-thio- cyanato-1 H-[1 ,2,4]triazolo (B.1.31 ), 2-[re/-(2S;3R)-3-(2-chlorophenyl)-2-(2,4-difluorophenyl)- oxiranylmethyl]-2H-[1 ,2,4]triazole-3-thiol (B.1 .32), 2-[2-chloro-4-(4-chlorophenoxy)phenyl]- 1 -(1 ,2,4-triazol-1 -yl)pentan-2-ol (B.1.33), 1 -[4-(4-chlorophenoxy)-2-(trifluoromethyl)phenyl]- 1 -cyclopropyl-2-(1 ,2,4-triazol-1 -yl)ethanol (B.1.34), 2-[4-(4-chlorophenoxy)-2-(trifluorometh- yl)phenyl]-1 -(1 ,2,4-triazol-1 -yl)butan-2-ol (B.1.35), 2-[2-chloro-4-(4-chlorophenoxy)phenyl]-1 - (1 ,2,4-triazol-1 -yl)butan-2-ol (B.1.36), 2-[4-(4-chlorophenoxy)-2-(trifluoromethyl)phenyl]-3- methyl-1 -(1 ,2,4-triazol-1 -yl)butan-2-ol (B.1.37), 2-[4-(4-chlorophenoxy)-2-(trifluoromethyl)- phenyl]-1 -(1 ,2,4-triazol-1 -yl)propan-2-ol (B.1.38), 2-[2-chloro-4-(4-chlorophenoxy)phenyl]-3- methyl-1 -(1 ,2,4-triazol-1 -yl)butan-2-ol (B.1.39), 2-[4-(4-chlorophenoxy)-2-(trifluoromethyl)- phenyl]-1 -(1 ,2,4-triazol-1 -yl)pentan-2-ol (B.1.40), 2-[4-(4-fluorophenoxy)-2-(trifluoromethyl)- phenyl]-1 -(1 ,2,4-triazol-1 -yl)propan-2-ol (B.1.41 ), 2-[2-chloro-4-(4-chlorophenoxy)phenyl]-1 - (1 ,2,4-triazol-1 -yl)pent-3-yn-2-ol (B.1 .51 ); imidazoles: imazalil (B.1 .42), pefurazoate (B.1.43), prochloraz (B.1.44), triflumizol (B.1 .45); pyrimidines, pyridines and piperazines: fenarimol (B.1.46), nuarimol (B.1 .47), pyrifenox (B.1.48), triforine (B.1 .49), [3-(4-chloro-2-fluoro- phenyl)-5-(2,4-difluorophenyl)isoxazol-4-yl]-(3-pyridyl)meth anol (B.1 .50);

Delta14-reductase inhibitors: aldimorph (B.2.1 ), dodemorph (B.2.2), dodemorph- acetate (B.2.3), fenpropimorph (B.2.4), tridemorph (B.2.5), fenpropidin (B.2.6), piperalin (B.2.7), spiroxamine (B.2.8);

Inhibitors of 3-keto reductase: fenhexamid (B.3.1 );

C) Nucleic acid synthesis inhibitors phenylamides or acyl amino acid fungicides: benalaxyl (C.1.1 ), benalaxyl-M (C.1 .2), kiralaxyl (C.1.3), metalaxyl (C.1.4), metalaxyl-M (mefenoxam, C.1 .5), ofurace (C.1.6), oxa- dixyl (C.1 .7);

others: hymexazole (C.2.1 ), octhilinone (C.2.2), oxolinic acid (C.2.3), bupirimate (C.2.4), 5-fluorocytosine (C.2.5), 5-fluoro-2-(p-tolylmethoxy)pyrimidin-4-amine (C.2.6), 5- fluoro-2-(4-fluorophenylmethoxy)pyrimidin-4-amine (C.2.7);

D) Inhibitors of cell division and cytoskeleton

tubulin inhibitors, such as benzimidazoles, thiophanates: benomyl (D1.1 ), car- bendazim (D1.2), fuberidazole (D1 .3), thiabendazole (D1 .4), thiophanate-methyl (D1.5); tria- zolopyrimidines: 5-chloro-7-(4-methylpiperidin-1 -yl)-6-(2,4,6-trifluorophenyl)-[1 ,2,4]tri- azolo[1 ,5-a]pyrimidine (D1 .6);

other cell division inhibitors: diethofencarb (D2.1 ), ethaboxam (D2.2), pencycuron (D2.3), fluopicolide (D2.4), zoxamide (D2.5), metrafenone (D2.6), pyriofenone (D2.7);

E) Inhibitors of amino acid and protein synthesis

- methionine synthesis inhibitors (anilino-pyrimidines): cyprodinil (E.1 .1 ), mepanipyrim

(E.1.2), pyrimethanil (E.1 .3);

protein synthesis inhibitors: blasticidin-S (E.2.1 ), kasugamycin (E.2.2), kasugamycin hydrochloride-hydrate (E.2.3), mildiomycin (E.2.4), streptomycin (E.2.5), oxytetracyclin (E.2.6), polyoxine (E.2.7), validamycin A (E.2.8);

F) Signal transduction inhibitors

MAP / histidine kinase inhibitors: fluoroimid (F.1 .1 ), iprodione (F.1 .2), procymidone (F.1 .3), vinclozolin (F.1.4), fenpiclonil (F.1 .5), fludioxonil (F.1.6);

G protein inhibitors: quinoxyfen (F.2.1 );

G) Lipid and membrane synthesis inhibitors

- Phospholipid biosynthesis inhibitors: edifenphos (G.1.1 ), iprobenfos (G.1 .2), pyrazo- phos (G.1 .3), isoprothiolane (G.1 .4);

lipid peroxidation: dicloran (G.2.1 ), quintozene (G.2.2), tecnazene (G.2.3), tolclofos- methyl (G.2.4), biphenyl (G.2.5), chloroneb (G.2.6), etridiazole (G.2.7);

phospholipid biosynthesis and cell wall deposition: dimethomorph (G.3.1 ), flumorph (G.3.2), mandipropamid (G.3.3), pyrimorph (G.3.4), benthiavalicarb (G.3.5), iprovalicarb

(G.3.6), valifenalate (G.3.7) and N-(1 -(1 -(4-cyano-phenyl)ethanesulfonyl)-but-2-yl) carbamic acid-(4-fluorophenyl) ester (G.3.8);

compounds affecting cell membrane permeability and fatty acides: propamocarb

(G.4.1 );

- fatty acid amide hydrolase inhibitors: oxathiapiprolin (G.5.1 ), 2-{3-[2-(1 -{[3,5-bis(di- fluoromethyl-1 H-pyrazol-1 -yl]acetyl}piperidin-4-yl)-1 ,3-thiazol-4-yl]-4,5-dihydro-1 ,2-oxazol-5- yl}phenyl methanesulfonate (G.5.2), 2-{3-[2-(1 -{[3, 5-bis(difluoromethyl)-1 H-pyrazol-1 - yl]acetyl}piperidin-4-yl) 1 ,3-thiazol-4-yl]-4,5-dihydro-1 ,2-oxazol-5-yl}-3-chlorophenyl me- thanesulfonate (G.5.3);

H) Inhibitors with Multi Site Action

inorganic active substances: Bordeaux mixture (H.1 .1 ), copper acetate (H.1.2), copper hydroxide (H.1.3), copper oxychloride (H.1.4), basic copper sulfate (H.1 .5), sulfur (H.1 .6);

thio- and dithiocarbamates: ferbam (H.2.1 ), mancozeb (H.2.2), maneb (H.2.3), metam (H.2.4), metiram (H.2.5), propineb (H.2.6), thiram (H.2.7), zineb (H.2.8), ziram (H.2.9);

organochlorine compounds (e. g. phthalimides, sulfamides, chloronitriles): anilazine (H.3.1 ), chlorothalonil (H.3.2), captafol (H.3.3), captan (H.3.4), folpet (H.3.5), dichlofluanid

(H.3.6), dichlorophen (H.3.7), hexachlorobenzene (H.3.8), pentachlorphenole (H.3.9) and its salts, phthalide (H.3.10), tolylfluanid (H.3.1 1 ), N-(4-chloro-2-nitro-phenyl)-N-ethyl-4-methyl- benzenesulfonamide (H.3.12);

guanidines and others: guanidine (H.4.1 ), dodine (H.4.2), dodine free base (H.4.3), guazatine (H.4.4), guazatine-acetate (H.4.5), iminoctadine (H.4.6), iminoctadine-triacetate (H.4.7), iminoctadine-tris(albesilate) (H.4.8), dithianon (H.4.9), 2,6-dimethyl-1 H,5H- [1 ,4]dithiino[2,3-c:5,6-c']dipyrrole-1 ,3,5,7(2H,6H)-tetraone (H.4.10);

I) Cell wall synthesis inhibitors

inhibitors of glucan synthesis: validamycin (1.1.1 ), polyoxin B (1.1 .2);

- melanin synthesis inhibitors: pyroquilon (1.2.1 ), tricyclazole (1.2.2), carpropamid

(I.2.3), dicyclomet (I.2.4), fenoxanil (I.2.5);

J) Plant defence inducers

acibenzolar-S-methyl (J.1.1 ), probenazole (J.1 .2), isotianil (J.1 .3), tiadinil (J.1.4), prohexadione-calcium (J.1.5); phosphonates: fosetyl (J.1 .6), fosetyl-aluminum (J.1.7), phos- phorous acid and its salts (J.1 .8), potassium or sodium bicarbonate (J.1 .9);

K) Unknown mode of action

bronopol (K.1.1 ), chinomethionat (K.1 .2), cyflufenamid (K.1.3), cymoxanil (K.1 .4), dazomet (K.1 .5), debacarb (K.1.6), diclomezine (K.1 .7), difenzoquat (K.1.8), difenzoquat- methylsulfate (K.1 .9), diphenylamin (K.1 .10), fenpyrazamine (K.1 .1 1 ), flumetover (K.1.12), flusulfamide (K.1 .13), flutianil (K.1 .14), methasulfocarb (K.1 .15), nitrapyrin (K.1 .16), nitrothal- isopropyl (K.1.18), oxathiapiprolin (K.1.19), tolprocarb (K.1 .20), oxin-copper (K.1 .21 ), pro- quinazid (K.1 .22), tebufloquin (K.1.23), tecloftalam (K.1 .24), triazoxide (K.1.25), 2-butoxy-6- iodo-3-propylchromen-4-one (K.1.26), 2-[3,5-bis(difluoromethyl)-1 H-pyrazol-1 -yl]-1 -[4-(4-{5- [2-(prop-2-yn-1 -yloxy)phenyl]-4,5-dihydro-1 ,2-oxazol-3-yl}-1 ,3-thiazol-2-yl)piperidin-1 -yljetha- none (K.1 .27), 2-[3,5-bis(difluoromethyl)-1 H-pyrazol-1 -yl]-1 -[4-(4-{5-[2-fluoro-6-(prop-2-yn-1 - yloxy)phenyl]-4,5-dihydro-1 ,2-oxazol-3-yl}-1 ,3-thiazol-2-yl)piperidin-1 -yl]ethanone (K.1.28), 2-[3,5-bis(difluoromethyl)-1 H-pyrazol-1 -yl]-1 -[4-(4-{5-[2-chloro-6-(prop-2-yn-1 -yloxy)phenyl]- 4,5-dihydro-1 ,2-oxazol-3-yl}-1 ,3-thiazol-2-yl)piperidin-1 -yl]ethanone (K.1.29), N-(cyclo- propylmethoxyimino-(6-difluoro-methoxy-2,3-difluoro-phenyl)- methyl)-2-phenyl acetamide (K.1.30), N'-(4-(4-chloro-3-trifluoromethyl-phenoxy)-2,5-dimethyl-phen yl)-N-ethyl-N-methyl formamidine (K.1.31 ), N'-(4-(4-fluoro-3-trifluoromethyl-phenoxy)-2,5-dimethyl-phen yl)-N- ethyl-N-methyl formamidine (K.1 .32), N'-(2-methyl-5-trifluoromethyl-4-(3-trimethylsilanyl- propoxy)-phenyl)-N-ethyl-N-methyl formamidine (K.1.33), N'-(5-difluoromethyl-2-methyl-4-(3- trimethylsilanyl-propoxy)-phenyl)-N-ethyl-N-methyl formamidine (K.1.34), methoxy-acetic ac- id 6-tert-butyl-8-fluoro-2,3-dimethyl-quinolin-4-yl ester (K.1 .35), 3-[5-(4-methylphenyl)-2,3- dimethyl-isoxazolidin-3-yl]-pyridine (K.1 .36), 3-[5-(4-chloro-phenyl)-2,3-dimethyl-isoxazolidin- 3-yl]-pyridine (pyrisoxazole) (K.1 .37), N-(6-methoxy-pyridin-3-yl) cyclopropanecarboxylic acid amide (K.1 .38), 5-chloro-1 -(4,6-dimethoxy-pyrimidin-2-yl)-2-methyl-1 H-benzoimidazole (K.1.39), 2-(4-chloro-phenyl)-N-[4-(3,4-dimethoxy-phenyl)-isoxazol-5-y l]-2-prop-2-ynyloxy- acetamide, ethyl (Z)-3-amino-2-cyano-3-phenyl-prop-2-enoate (K.1.40), picarbutrazox

(K.1 .41 ), pentyl N-[6-[[(Z)-[(1 -methyltetrazol-5-yl)-phenyl-methylene]amino]oxymethyl]-2- pyridyl]carbamate (K.1 .42), 2-[2-[(7,8-difluoro-2-methyl-3-quinolyl)oxy]-6-fluoro- phenyl]propan-2-ol (K.1 .43), 2-[2-fluoro-6-[(8-fluoro-2-methyl-3-quinolyl)oxy]phen-yl]pro pan- 2-ol (K.1 .44), 3-(5-fluoro-3,3,4,4-tetramethyl-3,4-dihydroisoquinolin-1 -yl)quinoline (K.1 .45), 3- (4,4-difluoro-3,3-dimethyl-3,4-dihydroisoquinolin-1-yl)quino line (K.1.46), 3-(4,4,5-trifluoro- 3,3-dimethyl-3,4-dihydroisoquinolin-1 -yl)quinoline (K.1 .47), 9-fluoro-2,2-dimethyl-5-(3- quinolyl)-3H-1 ,4-benzoxazepine (K.1.48);

M) Growth regulators

abscisic acid (M.1.1 ), amidochlor, ancymidol, 6-benzylaminopurine, brassinolide, butralin, chlormequat, chlormequat chloride, choline chloride, cyclanilide, daminozide, dikegulac, dime- thipin, 2,6-dimethylpuridine, ethephon, flumetralin, flurprimidol, fluthiacet, forchlorfenuron, gib- berellic acid, inabenfide, indole-3-acetic acid , maleic hydrazide, mefluidide, mepiquat, mepiquat chloride, naphthaleneacetic acid, N-6-benzyladenine, paclobutrazol, prohexadione, prohexadi- one-calcium, prohydrojasmon, thidiazuron, triapenthenol, tributyl phosphorotrithioate,

2,3,5-tri-iodobenzoic acid , trinexapac-ethyl and uniconazole;

N) Herbicides

acetamides: acetochlor (N.1 .1 ), alachlor, butachlor, dimethachlor, dimethenamid (N.1 .2), flufenacet (N.1 .3), mefenacet (N.1.4), metolachlor (N.1 .5), metazachlor (N.1 .6), napropamide, naproanilide, pethoxamid, pretilachlor, propachlor, thenylchlor;

- amino acid derivatives: bilanafos, glyphosate (N.2.1 ), glufosinate (N.2.2), sulfosate

(N.2.3);

aryloxyphenoxypropionates: clodinafop (N.3.1 ), cyhalofop-butyl, fenoxaprop (N.3.2), fluazifop (N.3.3), haloxyfop (N.3.4), metamifop, propaquizafop, quizalofop, quizalofop-P- tefuryl;

- Bipyridyls: diquat, paraquat (N.4.1 );

(thio)carbamates: asulam, butylate, carbetamide, desmedipham, dimepiperate, ep- tam (EPTC), esprocarb, molinate, orbencarb, phenmedipham (N.5.1 ), prosulfocarb, pyributi- carb, thiobencarb, triallate;

cyclohexanediones: butroxydim, clethodim (N.6.1 ), cycloxydim (N.6.2), profoxydim (N.6.3), sethoxydim (N.6.4), tepraloxydim (N.6.5), tralkoxydim;

dinitroanilines: benfluralin, ethalfluralin, oryzalin, pendimethalin (N.7.1 ), prodiamine (N.7.2), trifluralin (N.7.3);

diphenyl ethers: acifluorfen (N.8.1 ), aclonifen, bifenox, diclofop, ethoxyfen, fomesafen, lactofen, oxyfluorfen;

hydroxybenzonitriles: bomoxynil (N.9.1 ), dichlobenil, ioxynil;

- imidazolinones: imazamethabenz, imazamox (N.10.1 ), imazapic (N.10.2), imazapyr

(N.10.3), imazaquin (N.10.4), imazethapyr (N.10.5);

phenoxy acetic acids: clomeprop, 2,4-dichlorophenoxyacetic acid (2,4-D) (N.1 1 .1 ), 2,4-DB, dichlorprop, MCPA, MCPA-thioethyl, MCPB, Mecoprop;

pyrazines: chloridazon (N.1 1.1 ), flufenpyr-ethyl, fluthiacet, norflurazon, pyridate; - pyridines: aminopyralid, clopyralid (N.12.1 ), diflufenican, dithiopyr, fluridone, fluroxy- pyr (N.12.2), picloram (N.12.3), picolinafen (N.12.4), thiazopyr;

sulfonyl ureas: amidosulfuron, azimsulfuron, bensulfuron (N.13.1 ), chlorimuron-ethyl (N.13.2), chlorsulfuron, cinosulfuron, cyclosulfamuron (N.13.3), ethoxysulfuron, flazasulfu- ron, flucetosulfuron, flupyrsulfuron, foramsulfuron, halosulfuron, imazosulfuron, iodosulfuron (N.13.4), mesosulfuron (N.13.5), metazosulfuron, metsulfuron-methyl (N.13.6), nicosulfuron (N.13.7), oxasulfuron, primisulfuron, prosulfuron, pyrazosulfuron, rimsulfuron (N.13.8), sul- fometuron, sulfosulfuron, thifensulfuron, triasulfuron, tribenuron, trifloxysulfuron, triflusulfuron (N.13.9), tritosulfuron, 1 -((2-chloro-6-propyl-imidazo[1 ,2-b]pyridazin-3-yl)sulfonyl)-3-(4,6- d i methoxy-pyri m id i n-2-yl) u rea ;

- triazines: ametryn, atrazine (N.14.1 ), cyanazine, dimethametryn, ethiozin, hexazi- none (N.14.2), metamitron, metribuzin, prometryn, simazine, terbuthylazine, terbutryn, tria- ziflam, trifludimoxazin (N14.3);

ureas: chlorotoluron, daimuron, diuron (N.15.1 ), fluometuron, isoproturon, linuron, methabenzthiazuron, tebuthiuron;

- other acetolactate synthase inhibitors: bispyribac-sodium, cloransulam-methyl, di- closulam, florasulam (N.16.1 ), flucarbazone, flumetsulam, metosulam, ortho-sulfamuron, pe- noxsulam, propoxycarbazone, pyribambenz-propyl, pyribenzoxim, pyriftalid, pyriminobac- methyl, pyrimisulfan, pyrithiobac, pyroxasulfone (N.16.2), pyroxsulam;

others: amicarbazone, aminotriazole, anilofos, beflubutamid, benazolin, bencarba- zone,benfluresate, benzofenap, bentazone (N.17.1 ), benzobicyclon, bicyclopyrone, broma- cil, bromobutide, butafenacil, butamifos, cafenstrole, carfentrazone, cinidon-ethyl (N.17.2), chlorthal, cinmethylin (N.17.3), clomazone (N.17.4), cumyluron, cyprosulfamide, dicamba (N.17.5), difenzoquat, diflufenzopyr (N.17.6), Drechslera monoceras, endothal,

ethofumesate, etobenzanid, fenoxasulfone, fentrazamide, flumiclorac-pentyl, flumioxazin, flupoxam, flurochloridone, flurtamone, indanofan, isoxaben, isoxaflutole, lenacil, propanil, propyzamide, quinclorac (N.17.7), quinmerac (N.17.8), mesotrione (N.17.9), methyl arsonic acid, naptalam, oxadiargyl, oxadiazon, oxazidomefone, pentoxazone, pinoxaden, pyraclonil, pyraf I uf en-ethyl, pyrasulfotole, pyrazoxyfen, pyrazolynate, quinoclamine, saflufenacil (N.17.10), sulcotrione (N.17.1 1 ), sulfentrazone, terbacil, tefuryltrione, tembotrione, thien- carbazone, topramezone (N.17.12), (3-[2-chloro-4-fluoro-5-(3-methyl-2,6-dioxo-4- trifluoromethyl-3,6-dihydro-2H-pyrimidin-1 -yl)-phenoxy]-pyridin-2-yloxy^ acid ethyl ester, 6-amino-5-chloro-2-cyclopropyl-pyrimidine-4-carboxylic acid methyl ester, 6-chloro-3-(2- cyclopropyl-6-methyl-phenoxy)-pyridazin-4-ol, 4-amino-3-chloro-6-(4-chloro-phenyl)-5-fluoro- pyridine-2-carboxylic acid, 4-amino-3-chloro-6-(4-chloro-2-fluoro-3-methoxy-phenyl)- pyridine-2-carboxylic acid methyl ester, and 4-amino-3-chloro-6-(4-chloro-3-dimethylamino- 2-fluoro-phenyl)-pyridine-2-carboxylic acid methyl ester;

O) Insecticides

organo(thio)phosphates: acephate (0.1.1 ), azamethiphos (0.1.2), azinphos-methyl (0.1.3), chlorpyrifos (0.1 .4), chlorpyrifos-methyl (0.1.5), chlorfenvinphos (0.1.6), diazinon (0.1.7), dichlorvos (0.1 .8), dicrotophos (0.1.9), dimethoate (0.1.10), disulfoton (0.1.1 1 ), ethion (0.1 .12), fenitrothion (0.1.13), fenthion (0.1 .14), isoxathion (0.1 .15), malathion (0.1.16), methamidophos (0.1.17), methidathion (0.1 .18), methyl-parathion (0.1.19), mevinphos (0.1.20), monocrotophos (0.1.21 ), oxydemeton-methyl (0.1.22), paraoxon (0.1.23), parathion (0.1 .24), phenthoate (0.1 .25), phosalone (0.1 .26), phosmet (0.1.27), phosphamidon (0.1 .28), phorate (0.1 .29), phoxim (O.1 .30), pirimiphos-methyl (0.1.31 ), profenofos (0.1.32), prothiofos (0.1 .33), sulprophos (0.1.34), tetrachlorvinphos (0.1.35), terbufos (0.1 .36), triazophos (0.1 .37), trichlorfon (0.1 .38);

carbamates: alanycarb (0.2.1 ), aldicarb (0.2.2), bendiocarb (0.2.3), benfuracarb (0.2.4), carbaryl (0.2.5), carbofuran (0.2.6), carbosulfan (0.2.7), fenoxycarb (0.2.8), furathiocarb (0.2.9), methiocarb (0.2.10), methomyl (0.2.1 1 ), oxamyl (0.2.12), pirimicarb (0.2.13), propoxur (0.2.14), thiodicarb (0.2.15), triazamate (0.2.16);

pyrethroids: allethrin (0.3.1 ), bifenthrin (0.3.2), cyfluthrin (0.3.3), cyhalothrin (0.3.4), cyphenothrin (0.3.5), cypermethrin (0.3.6), alpha-cypermethrin (0.3.7), beta- cypermethrin (0.3.8), zeta-cypermethrin (0.3.9), deltamethrin (0.3.10), esfenvalerate (0.3.1 1 ), etofenprox (0.3.1 1 ), fenpropathrin (0.3.12), fenvalerate (0.3.13), imiprothrin

(0.3.14), lambda-cyhalothrin (0.3.15), permethrin (0.3.16), prallethrin (0.3.17), pyrethrin I and II (0.3.18), resmethrin (0.3.19), silafluofen (O.3.20), tau-fluvalinate (0.3.21 ), tefluthrin (0.3.22), tetramethrin (0.3.23), tralomethrin (0.3.24), transfluthrin (0.3.25), profluthrin (0.3.26), dimefluthrin (0.3.27);

- insect growth regulators: a) chitin synthesis inhibitors: benzoylureas: chlorfluazuron

(0.4.1 ), cyramazin (0.4.2), diflubenzuron (0.4.3), flucycloxuron (0.4.4), flufenoxuron (0.4.5), hexaflumuron (0.4.6), lufenuron (0.4.7), novaluron (0.4.8), teflubenzuron (0.4.9), triflumuron (0.4.10); buprofezin (0.4.1 1 ), diofenolan (0.4.12), hexythiazox (0.4.13), etox- azole (0.4.14), clofentazine (0.4.15); b) ecdysone antagonists: halofenozide (0.4.16), methoxyfenozide (0.4.17), tebufenozide (0.4.18), azadirachtin (0.4.19); c) juvenoids:

pyriproxyfen (0.4.20), methoprene (0.4.21 ), fenoxycarb (0.4.22); d) lipid biosynthesis inhibitors: spirodiclofen (0.4.23), spiromesifen (0.4.24), spirotetramat (0.4.24);

nicotinic receptor agonists/antagonists compounds: clothianidin (0.5.1 ), dinotefuran (0.5.2), flupyradifurone (0.5.3), imidacloprid (0.5.4), thiamethoxam (0.5.5), nitenpyram (0.5.6), acetamiprid (0.5.7), thiacloprid (0.5.8), 1 -2-chloro-thiazol-5-ylmethyl)-2-nitrimino- 3,5-dimethyl-[1 ,3,5]triazinane (0.5.9);

GABA antagonist compounds: endosulfan (0.6.19, ethiprole (0.6.2), fipronil (0.6.3), vaniliprole (0.6.4), pyrafluprole (0.6.5), pyriprole (0.6.6), 5-amino-1 -(2,6-dichloro-4-methyl- phenyl)-4-sulfinamoyl-1 H-pyrazole-3-carbothioic acid amide (0.6.7);

macrocyclic lactone insecticides: abamectin (0.7.1 ), emamectin (0.7.2), milbemec- tin (0.7.3), lepimectin (0.7.4), spinosad (0.7.5), spinetoram (0.7.6);

- mitochondrial electron transport inhibitor (METI) I acaricides: fenazaquin (0.8.1 ), pyridaben (0.8.2), tebufenpyrad (0.8.3), tolfenpyrad (0.8.4), flufenerim (0.8.5);

METI II and III compounds: acequinocyl (0.9.1 ), fluacyprim (0.9.2), hydramethylnon

(0.9.3);

Uncouplers: chlorfenapyr (0.10.1 );

- oxidative phosphorylation inhibitors: cyhexatin (0.1 1.1 ), diafenthiuron (0.1 1 .2), fenbutatin oxide (0.1 1 .3), propargite (0.1 1 .4);

moulting disruptor compounds: cryomazine (0.12.1 );

mixed function oxidase inhibitors: piperonyl butoxide (0.13.1 );

sodium channel blockers: indoxacarb (0.14.1 ), metaflumizone (0.14.2); - ryanodine receptor inhibitors: chlorantraniliprole (0.15.1 ), cyantraniliprole (0.15.2), flubendiamide (0.15.3), N-[4,6-dichloro-2-[(diethyl-lambda-4-sulfanylidene)carbamoyl ]- phenyl]-2-(3-chloro-2-pyridyl)-5-(trifluoromethyl)pyrazole-3 -carboxamide (0.15.4); N-[4- chloro-2-[(diethyl-lambda-4-sulfanylidene)carbamoyl]-6-methy l-phenyl]-2-(3-chloro-2-pyridyl)- 5-(trifluoromethyl)pyrazole-3-carboxamide (0.15.5); N-[4-chloro-2-[(di-2-propyl-lambda-4- sulfanylidene)carbamoyl]-6-methyl-phenyl]-2-(3-chloro-2-pyri dyl)-5-(trifluoromethyl)pyrazole- 3-carboxamide (0.15.6); N-[4,6-dichloro-2-[(di-2-propyl-lambda-4-sulfanylidene)carba moyl]- phenyl]-2-(3-chloro-2-pyridyl)-5-(trifluoromethyl)pyrazole-3 -carboxamide (0.15.7); N-[4,6-di- chloro-2-[(diethyl-lambda-4-sulfanylidene)carbamoyl]-phenyl] -2-(3-chloro-2-pyridyl)-5-(di- fluoromethyl)pyrazole-3-carboxamide (0.15.8); N-[4,6-dibromo-2-[(di-2-propyl-lambda-4-sul- fanylidene)carbamoyl]-phenyl]-2-(3-chloro-2-pyridyl)-5-(trif luoromethyl)pyrazole-3-carbox- amide (0.15.9); N-[4-chloro-2-[(di-2-propyl-lambda-4-sulfanylidene)carbamoyl ]-6-cyano- phenyl]-2-(3-chloro-2-pyridyl)-5-(trifluoromethyl)pyrazole-3 -carboxamide (0.15.10); N-[4,6- dibromo-2-[(diethyl-lambda-4-sulfanylidene)carbamoyl]-phenyl ]-2-(3-chloro-2-pyridyl)-5-(tri- fluoromethyl)pyrazole-3-carboxamide (0.15.1 1 );

- others: benclothiaz (0.16.1 ), bifenazate (0.16.2), artap (0.16.3), flonicamid

(0.16.4), pyridalyl (0.16.5), pymetrozine (0.16.6), sulfur (0.16.7), thiocyclam (0.16.8), cye- nopyrafen (0.16.9), flupyrazofos (0.16.10), cyflumetofen (0.16.1 1 ), amidoflumet (0.16.12), imicyafos (0.16.13), bistrifluron (0.16.14), pyrifluquinazon (0.16.15) and

1 , 1 '-[(3S,4R,4aR,6S,6aS, 12R, 12aS, 12bS)-4-[[(2-cyclopropylacetyl)oxy]methyl]- 1 ,3,4,4a,5,6,6a,12,12a,12b-decahydro-12-hydroxy-4,6a,12b-trim ethyl-1 1 -oxo-9-(3-pyridinyl)- 21-1,1 1 H-naphtho[2,1 -b]pyrano[3,4-e]pyran-3,6-diyl] cyclopropaneacetic acid ester (0.16.16).

The active substances referred to as component 2, their preparation and their activity e. g. against harmful fungi is known (cf.: http://www.alanwood.net/pesticides/); these substances are commercially available. The compounds described by lUPAC nomenclature, their preparation and their pesticidal activity are also known (cf. Can. J. Plant Sci. 48(6), 587-94, 1968; EP-A 141 317; EP-A 152 031 ; EP-A 226 917; EP-A 243 970; EP-A 256 503; EP-A 428 941 ; EP- A 532 022; EP-A 1 028 125; EP-A 1 035 122; EP-A 1 201 648; EP-A 1 122 244,

JP 2002316902; DE 19650197; DE 10021412; DE 102005009458; US 3,296,272;

US 3,325,503; WO 98/46608; WO 99/14187; WO 99/24413; WO 99/27783; WO 00/29404; WO 00/46148; WO 00/65913; WO 01/54501 ; WO 01/56358; WO 02/22583; WO 02/40431 ; WO 03/10149; WO 03/1 1853; WO 03/14103; WO 03/16286; WO 03/53145; WO 03/61388; WO 03/66609; WO 03/74491 ; WO 04/49804; WO 04/83193; WO 05/120234; WO 05/123689; WO 05/123690; WO 05/63721 ; WO 05/87772; WO 05/87773; WO 06/15866; WO 06/87325; WO 06/87343; WO 07/82098; WO 07/90624, WO 1 1/028657, WO2012/168188, WO

2007/006670, WO 201 1/77514; WO13/047749, WO 10/069882, WO 13/047441 , WO 03/16303, WO 09/90181 , WO 13/007767, WO 13/010862, WO 13/127704, WO 13/024009,

WO 13/024010 and WO 13/047441 , WO 13/162072, WO 13/092224, WO 1 1/135833). The present invention furthermore relates to agrochemical mixtures comprising at least one compound I (component 1 ) and at least one further active substance useful for plant protection, e. g. selected from the groups A) to O) (component 2), in particular one further fungicide, e. g. one or more fungicide from the groups A) to K), as described above, and if desired one suitable solvent or solid carrier. Those mixtures are of particular interest, since many of them at the same application rate show higher efficiencies against harmful fungi. Furthermore, combating harmful fungi with a mixture of compounds I and at least one fungicide from groups A) to K), as described above, is more efficient than combating those fungi with individual compounds I or individual fungicides from groups A) to K).

By applying compounds I together with at least one active substance from groups A) to O) a synergistic effect can be obtained, i.e. more than simple addition of the individual effects is obtained (synergistic mixtures).

This can be obtained by applying the compounds I and at least one further active substance simultaneously, either jointly (e. g. as tank-mix) or seperately, or in succession, wherein the time interval between the individual applications is selected to ensure that the active substance ap- plied first still occurs at the site of action in a sufficient amount at the time of application of the further active substance(s). The order of application is not essential for working of the present invention.

When applying compound I and a pesticide II sequentially the time between both applications may vary e. g. between 2 hours to 7 days. Also a broader range is possible ranging from 0.25 hour to 30 days, preferably from 0.5 hour to 14 days, particularly from 1 hour to 7 days or from 1 .5 hours to 5 days, even more preferred from 2 hours to 1 day.

In the binary mixtures and compositions according to the invention the weight ratio of the component 1 ) and the component 2) generally depends on the properties of the active components used, usually it is in the range of from 1 :100 to 100:1 , regularly in the range of from 1 :50 to 50:1 , preferably in the range of from 1 :20 to 20:1 , more preferably in the range of from 1 :10 to 10:1 , even more preferably in the range of from 1 :4 to 4:1 and in particular in the range of from 1 :2 to 2:1 . According to a further embodiment of the binary mixtures and compositions thereof, the weight ratio of the component 1) and the component 2) usually is in the range of from 1000:1 to 1:1, often in the range of from 100: 1 to 1:1, regularly in the range of from 50:1 to 1:1, preferably in the range of from 20:1 to 1:1, more preferably in the range of from 10:1 to 1:1, even more pref- erably in the range of from 4:1 to 1 :1 and in particular in the range of from 2:1 to 1:1.

According to a further embodiment of the binary mixtures and compositions thereof, the weight ratio of the component 1) and the component 2) usually is in the range of from 1:1 to 1:1000, often in the range of from 1:1 to 1:100, regularly in the range of from 1:1 to 1:50, preferably in the range of from 1:1 to 1:20, more preferably in the range of from 1:1 to 1:10, even more pref- erably in the range of from 1:1 to 1:4 and in particular in the range of from 1:1 to 1:2.

In the ternary mixtures, i.e. compositions according to the invention comprising the component 1) and component 2) and a compound III (component 3), the weight ratio of component 1) and component 2) depends on the properties of the active substances used, usually it is in the range of from 1:100 to 100:1, regularly in the range of from 1:50 to 50:1, preferably in the range of from 1:20 to 20:1, more preferably in the range of from 1:10 to 10:1 and in particular in the range of from 1 :4 to 4: 1 , and the weight ratio of component 1 ) and component 3) usually it is in the range of from 1:100 to 100:1, regularly in the range of from 1:50 to 50:1, preferably in the range of from 1:20 to 20:1, more preferably in the range of from 1:10 to 10:1 and in particular in the range of from 1 :4 to 4:1.

Any further active components are, if desired, added in a ratio of from 20:1 to 1 :20 to the component 1).

These ratios are also suitable for inventive mixtures applied by seed treatment.

Preference is also given to mixtures comprising as component 2) at least one active sub- stance selected from group A), which is particularly selected from (A.1.1), (A.1.4), (A.1.8),

(A.1.9), (A.1.12), (A.1.13), (A.1.14), (A.1.17), (A.1.19), (A.1.21), (A.2.1), (A.2.2), (A.2.8), (A.3.2), (A.3.3), (A.3.4), (A.3.7), (A.3.8), (A.3.9), (A.3.12), (A.3.14), (A.3.15), (A.3.16), (A.3.19), (A.3.20), (A.3.21), (A.3.22), (A.3.23), (A.3.24), (A.3.25), (A.3.26), (A.3.27); (A.4.5), (A.4.6), (A.4.8), (A.4.9), (A.4.11), (A.1.23), (A.1.24), (A.1.25), (A.1.26), (A.1.27), (A.1.28), (A.1.29), (A.1.30), (A.1.31), (A.1.32), and (A.1.33).

Preference is given to mixtures comprising as component 2) at least one active substance selected from group B), which is particularly selected from (B.1.4), (B.1.5), diniconazole (B.1.6), (B.1.8), (B.1.10), (B.1.11), (B.1.12), (B.1.17), (B.1.18), (B.1.21), (B.1.22), (B.1.23), (B.1.25), (B.1.26), (B.1.27), (B.1.28), (B.1.29), uni (B.1.31), (B.1.32), (B.1.33), (B.1.34), (B.1.35), (B.1.36), (B.1.37), (B.1.38), (B.1.39), (B.1.40), (B.1.41), (B.1.42), (B.1.44), (B.1.46), (B.1.49) and (B.1.50; (B.2.2), (B.2.4), (B.2.5), (B.2.6), piperalin (B.2.7), (B.2.8); and (B.3.1).

Preference is given to mixtures comprising as component 2) at least one active substance selected from group C), which is particularly selected from (C.1.4), C.1.5), (C.1.6), and (C.2.4).

Preference is given to mixtures comprising as component 2) at least one active substance se- lected from group D), which is particularly selected from (D1.1 ), (D1.2), (D1.4), (D1.5); (D2.2), (D2.4), (D2.5), (D2.6) and (D2.7); Preference is also given to mixtures comprising as component 2) at least one active substance selected from group E), which is particularly selected from (E.1.1 ), (E.1.2), and (E.1.3);

Preference is also given to mixtures comprising as component 2) at least one active substance selected from group F), which is particularly selected from (F.1.2), (F.1 .4), (F.1.5), (F.1 .6) and (F.2.1 ).

Preference is also given to mixtures as component 2) at least one active substance selected from group G), which is particularly selected from (G.3.1 ), (G.3.2), (G.3.3), (G.3.4), (G.3.5), (G.3.6), (G.4.1 ) and (G.5.1 ).

Preference is also given to mixtures comprising as component 2) at least one active sub- stance selected from group H), which is and particularly selected from (H.1.2), (H.1 .3), copper oxychloride (H.1 .4), (H.1.5), (H.1 .6); (H.2.2), (H.2.5), (H.2.7), (H.3.2), (H.3.3), (H.3.4), (H.3.5), (H.3.6), (H.3.12); (H.4.2), (H.4.6), dithianon (H.4.9) and (H.4.10).

Preference is also given to mixtures comprising as component 2) at least one active substance selected from group I), which is particularly selected from (1.2.3) and (1.2.5).

Preference is also given to mixtures comprising as component 2) at least one active substance selected from group J), which is particularly selected from (J.1 .1 ), (J.1.2), (J.1.3), (J.1 .4), (J.1.6), (J.1 .7), (J.1.8) and (J.1 .9).

Preference is also given to mixtures comprising as component 2) at least one active substance selected from group K), which is particularly selected from (K.1 .4), (K.1 .5), (K.1 .8), (K.1.12), (K.1 .14), (K.1.15), (K.1 .19) and(K.1.22).

Accordingly, the present invention furthermore relates to mixtures comprising one compound of the formula I (component 1 ) and one pesticide II (component 2), wherein pesticide II is selected from the column "Co. 2" of the lines B-1 to B-580 of Table B.

A further embodiment relates to the mixtures B-1 to B-580 listed in Table B, where a row of Table B corresponds in each case to a fungicidal mixture comprising as active components one of the in the present specification individualized compounds of formula I, i.e. compounds 1-1 to I- 890 as defined in table A (component 1 in column "Co.1 ") and the respective pesticide II from groups A) to O) (component 2) stated in the row in question.

Another embodiment relates to the mixtures B-1 to B-580 listed in Table B, where a row of Ta- ble B corresponds in each case to a fungicidal mixture comprising as active components one of the compounds Ex-1 to Ex-7 of formula I as defined below in table I (component 1 in column "Co.1 ") and the respective pesticide II from groups A) to O) (component 2) stated in the row in question.

Preferably, the compositions described in Table B comprise the active components in syner- gistically effective amounts.

Table B: Mixtures comprising as active components one indiviualized compound of the fomula I (in column Co. 1 ), in particular compounds 1-1 to I-890 as defined in table A, or more particularly compounds Ex-1 to Ex-7, as defined below in table I, and as component 2) (in column Co. 2) one pesticide from groups A) to O) [which is coded e. g. as (A.1 .1 ) for azoxystrobin as de- fined above].

Mixt. Co. Co.2 Mixt. Co. Co.2 Mixt. Co. Co.2

1 1 1

B-1 (I) (A.1.1) B-30 (I) (A.1.30) B-59 (I) (A.3.18)

B-2 (I) (A.1.2) B-31 (I) (A.1.31) B-60 (I) (A.3.19)

B-3 (I) (A.1.3) B-32 (I) (A.1.32) B-61 (I) (A.3.20)

B-4 (I) (A.1.4) B-33 (I) (A.1.33) B-62 (I) (A.3.21)

B-5 (I) (A.1.5) B-34 (I) (A.2.1) B-63 (I) (A.3.22)

B-6 (I) (A.1.6) B-35 (I) (A.2.2) B-64 (I) (A.3.23)

B-7 (I) (A.1.7) B-36 (I) (A.2.3) B-65 (I) (A.3.24)

B-8 (I) (A.1.8) B-37 (I) (A.2.4) B-66 (I) (A.3.25)

B-9 (I) (A.1.9) B-38 (I) (A.2.5) B-67 (I) (A.3.26)

B-10 (I) (A.1.10) B-39 (I) (A.2.6) B-68 (I) (A.3.27)

B-11 (I) (A.1.11) B-40 (I) (A.2.7) B-69 (I) (A.4.1)

B-12 (I) (A.1.12) B-41 (I) (A.2.8) B-70 (I) (A.4.2)

B-13 (I) (A.1.13) B-42 (I) (A.3.1) B-71 (I) (A.4.3)

B-14 (I) (A.1.14) B-43 (I) (A.3.2) B-72 (I) (A.4.4)

B-15 (I) (A.1.15) B-44 (I) (A.3.3) B-73 (I) (A.4.5)

B-16 (I) (A.1.16) B-45 (I) (A.3.4) B-74 (I) (A.4.6)

B-17 (I) (A.1.17) B-46 (I) (A.3.5) B-75 (I) (A.4.7)

B-18 (I) (A.1.18) B-47 (I) (A.3.6) B-76 (I) (A.4.8)

B-19 (I) (A.1.19) B-48 (I) (A.3.7) B-77 (I) (A.4.9)

B-20 (I) (A.1.20) B-49 (I) (A.3.8) B-78 (I) (A.4.10)

B-21 (I) (A.1.21) B-50 (I) (A.3.9) B-79 (I) (A.4.11)

B-22 (I) (A.1.22) B-51 (I) (A.3.10) B-80 (I) (A.4.12)

B-23 (I) (A.1.23) B-52 (I) (A.3.11) B-81 (I) (B.1.1)

B-24 (I) (A.1.24) B-53 (I) (A.3.12) B-82 (I) (B.1.2)

B-25 (I) (A.1.25) B-54 (I) (A.3.13) B-83 (I) (B.1.3)

B-26 (I) (A.1.26) B-55 (I) (A.3.14) B-84 (I) (B.1.4)

B-27 (I) (A.1.27) B-56 (I) (A.3.15) B-85 (I) (B.1.5)

B-28 (I) (A.1.28) B-57 (I) (A.3.16) B-86 (I) (B.1.6)

B-29 (I) (A.1.29) B-58 (I) (A.3.17) B-87 (I) (B.1.7) Mixt. Co. Co.2 Mixt. Co. Co.2 Mixt. Co. Co.2 1 1 1

B-88 (I) (B.1.8) B-118 (I) (B.1.38) B-148 (I) (C.2.1)

B-89 (I) (B.1.9) B-119 (I) (B.1.39) B-149 (I) (C.2.2)

B-90 (I) (B.1.10) B-120 (I) (B.1.40) B-150 (I) (C.2.3)

B-91 (I) (B.1.11) B-121 (I) (B.1.41) B-151 (I) (C.2.4)

B-92 (I) (B.1.12) B-122 (I) (B.1.42) B-152 (I) (C.2.5)

B-93 (I) (B.1.13) B-123 (I) (B.1.43) B-153 (I) (C.2.6)

B-94 (I) (B.1.14) B-124 (I) (B.1.44) B-154 (I) (C.2.7)

B-95 (I) (B.1.15) B-125 (I) (B.1.45) B-155 (I) (D.1.1)

B-96 (I) (B.1.16) B-126 (I) (B.1.46) B-156 (I) (D.1.2)

B-97 (I) (B.1.17) B-127 (I) (B.1.47) B-157 (I) (D.1.3)

B-98 (I) (B.1.18) B-128 (I) (B.1.48) B-158 (I) (D.1.4)

B-99 (I) (B.1.19) B-129 (I) (B.1.49) B-159 (I) (D.1.5)

B-100 (I) (B.1.20) B-130 (I) (B.1.50) B-160 (I) (D.1.6)

B-101 (I) (B.1.21) B-131 (I) (B.1.51) B-161 (I) (D.2.1)

B-102 (I) (B.1.22) B-132 (I) (B.2.1) B-162 (I) (D.2.2)

B-103 (I) (B.1.23) B-133 (I) (B.2.2) B-163 (I) (D.2.3)

B-104 (I) (B.1.24) B-134 (I) (B.2.3) B-164 (I) (D.2.4)

B-105 (I) (B.1.25) B-135 (I) (B.2.4) B-165 (I) (D.2.5)

B-106 (I) (B.1.26) B-136 (I) (B.2.5) B-166 (I) (D.2.6)

B-107 (I) (B.1.27) B-137 (I) (B.2.6) B-167 (I) (D.2.7)

B-108 (I) (B.1.28) B-138 (I) (B.2.7) B-168 (I) (E.1.1)

B-109 (I) (B.1.29) B-139 (I) (B.2.8) B-169 (I) (E.1.2)

B-110 (I) (B.1.30) B-140 (I) (B.3.1) B-170 (I) (E.1.3)

B-111 (I) (B.1.31) B-141 (I) (C.1.1) B-171 (I) (E.2.1)

B-112 (I) (B.1.32) B-142 (I) (C.1.2) B-172 (I) (E.2.2)

B-113 (I) (B.1.33) B-143 (I) (C.1.3) B-173 (I) (E.2.3)

B-114 (I) (B.1.34) B-144 (I) (C.1.4) B-174 (I) (E.2.4)

B-115 (I) (B.1.35) B-145 (I) (C.1.5) B-175 (I) (E.2.5)

B-116 (I) (B.1.36) B-146 (I) (C.1.6) B-176 (I) (E.2.6)

B-117 (I) (B.1.37) B-147 (I) (C.1.7) B-177 (I) (E.2.7) Mixt. Co. Co. 2 Mixt. Co. Co. 2 Mixt. Co. Co. 2 1 1 1

B-178 (I) (E.2.8) B-208 (I) (G.5.3) B-238 (I) (H.4.4)

B-179 (I) (F.1.1 ) B-209 (I) (H.1.1 ) B-239 (I) (H.4.5)

B-180 (I) (F.1.2) B-210 (I) (H.1.2) B-240 (I) (H.4.6)

B-181 (I) (F.1.3) B-21 1 (I) (H.1.3) B-241 (I) (H.4.7)

B-182 (I) (F.1.4) B-212 (I) (H.1.4) B-242 (I) (H.4.8)

B-183 (I) (F.1.5) B-213 (I) (H.1.5) B-243 (I) (H.4.9)

B-184 (I) (F.1.6) B-214 (I) (H.1.6) B-244 (I) (H.4.10)

B-185 (I) (F.2.1 ) B-215 (I) (H.2.1 ) B-245 (I) (1.1 .1 )

B-186 (I) (G.1 .1 ) B-216 (I) (H.2.2) B-246 (I) (1.1 .2)

B-187 (I) (G.1 .2) B-217 (I) (H.2.3) B-247 (I) (1.2.1 )

B-188 (I) (G.1 .3) B-218 (I) (H.2.4) B-248 (I) (I.2.2)

B-189 (I) (G.1 .4) B-219 (I) (H.2.5) B-249 (I) (I.2.3)

B-190 (I) (G.2.1 ) B-220 (I) (H.2.6) B-250 (I) (I.2.4)

B-191 (I) (G.2.2) B-221 (I) (H.2.7) B-251 (I) (I.2.5)

B-192 (I) (G.2.3) B-222 (I) (H.2.8) B-252 (I) (J.1.1 )

B-193 (I) (G.2.4) B-223 (I) (H.2.9) B-253 (I) (J.1.2)

B-194 (I) (G.2.5) B-224 (I) (H.3.1 ) B-254 (I) (J.1.3)

B-195 (I) (G.2.6) B-225 (I) (H.3.2) B-255 (I) (J.1.4)

B-196 (I) (G.2.7) B-226 (I) (H.3.3) B-256 (I) (J.1.5)

B-197 (I) (G.3.1 ) B-227 (I) (H.3.4) B-257 (I) (J.1.6)

B-198 (I) (G.3.2) B-228 (I) (H.3.5) B-258 (I) (J.1.7)

B-199 (I) (G.3.3) B-229 (I) (H.3.6) B-259 (I) (J.1.8)

B-200 (I) (G.3.4) B-230 (I) (H.3.7) B-260 (I) (J.1.9)

B-201 (I) (G.3.5) B-231 (I) (H.3.8) B-261 (I) (K.1 .1 )

B-202 (I) (G.3.6) B-232 (I) (H.3.9) B-262 (I) (K.1 .2)

B-203 (I) (G.3.7) B-233 (I) (H.3.10) B-263 (I) (K.1 .3)

B-204 (I) (G.3.8) B-234 (I) (H.3.1 1 ) B-264 (I) (K.1 .4)

B-205 (I) (G.4.1 ) B-235 (I) (H.4.1 ) B-265 (I) (K.1 .5)

B-206 (I) (G.5.1 ) B-236 (I) (H.4.2) B-266 (I) (K.1 .6)

B-207 (I) (G.5.2) B-237 (I) (H.4.3) B-267 (I) (K.1 .7) Mixt. Co. Co.2 Mixt. Co. Co.2 Mixt. Co. Co.2 1 1 1

B-268 (I) (K.1.8) B-298 (I) (K.1.38) B-328 (I) (M.1.20)

B-269 (I) (K.1.9) B-299 (I) (K.1.39) B-329 (I) (M.1.21)

B-270 (I) (K.1.10) B-300 (I) (K.1.40) B-330 (I) (M.1.22)

B-271 (I) (K.1.11) B-301 (I) (K.1.41) B-331 (I) (M.1.23)

B-272 (I) (K.1.12) B-302 (I) (K.1.42) B-332 (I) (M.1.24)

B-273 (I) (K.1.13) B-303 (I) (K.1.43) B-333 (I) (M.1.25)

B-274 (I) (K.1.14) B-304 (I) (K.1.44) B-334 (I) (M.1.26)

B-275 (I) (K.1.15) B-305 (I) (K.1.45) B-335 (I) (M.1.27)

B-276 (I) (K.1.16) B-306 (I) (K.1.46) B-336 (I) (M.1.28)

B-277 (I) (K.1.17) B-307 (I) (K.1.47) B-337 (I) (M.1.29)

B-278 (I) (K.1.18) B-308 (I) (K.1.48) B-338 (I) (M.1.30)

B-279 (I) (K.1.19) B-309 (I) (M.1.1) B-339 (I) (M.1.31)

B-280 (I) (K.1.20) B-310 (I) (M.1.2) B-340 (I) (M.1.32)

B-281 (I) (K.1.21) B-311 (I) (M.1.3) B-341 (I) (M.1.33)

B-282 (I) (K.1.22) B-312 (I) (M.1.4) B-342 (I) (M.1.34)

B-283 (I) (K.1.23) B-313 (I) (M.1.5) B-343 (I) (M.1.35)

B-284 (I) (K.1.24) B-314 (I) (M.1.6) B-344 (I) (M.1.36)

B-285 (I) (K.1.25) B-315 (I) (M.1.7) B-345 (I) (M.1.37)

B-286 (I) (K.1.26) B-316 (I) (M.1.8) B-346 (I) (M.1.38)

B-287 (I) (K.1.27) B-317 (I) (M.1.9) B-347 (I) (M.1.39)

B-288 (I) (K.1.28) B-318 (I) (M.1.10) B-348 (I) (M.1.40)

B-289 (I) (K.1.29) B-319 (I) (M.1.11) B-349 (I) (M.1.41)

B-290 (I) (K.1.30) B-320 (I) (M.1.12) B-350 (I) (M.1.42)

B-291 (I) (K.1.31) B-321 (I) (M.1.13) B-351 (I) (M.1.43)

B-292 (I) (K.1.32) B-322 (I) (M.1.14) B-352 (I) (M.1.44)

B-293 (I) (K.1.33) B-323 (I) (M.1.15) B-353 (I) (M.1.45)

B-294 (I) (K.1.34) B-324 (I) (M.1.16) B-354 (I) (M.1.46)

B-295 (I) (K.1.35) B-325 (I) (M.1.17) B-355 (I) (M.1.47)

B-296 (I) (K.1.36) B-326 (I) (M.1.18) B-356 (I) (M.1.48)

B-297 (I) (K.1.37) B-327 (I) (M.1.19) B-357 (I) (M.1.49) Mixt. Co. Co.2 Mixt. Co. Co.2 Mixt. Co. Co.2 1 1 1

B-358 (I) (M.1.50) B-388 (I) (N.11.1) B-418 (I) (N.17.11)

B-359 (I) (N.1.1) B-389 (I) (N.12.1) B-419 (I) (N.17.12)

B-360 (I) (N.1.2) B-390 (I) (N.12.2) B-420 (I) (0.1.1)

B-361 (I) (N.1.3) B-391 (I) (N.12.3) B-421 (I) (0.1.2)

B-362 (I) (N.1.4) B-392 (I) (N.12.4) B-422 (I) (0.1.3)

B-363 (I) (N.1.5) B-393 (I) (N.13.1) B-423 (I) (0.1.4)

B-364 (I) (N.2.1) B-394 (I) (N.13.2) B-424 (I) (0.1.5)

B-365 (I) (N.2.2) B-395 (I) (N.13.3) B-425 (I) (0.1.6)

B-366 (I) (N.2.3) B-396 (I) (N.13.4) B-426 (I) (0.1.7)

B-367 (I) (N.3.1) B-397 (I) (N.13.5) B-427 (I) (0.1.8)

B-368 (I) (N.3.2) B-398 (I) (N.13.6) B-428 (I) (0.1.9)

B-369 (I) (N.3.3) B-399 (I) (N.13.7) B-429 (I) (0.1.10)

B-370 (I) (N.3.4) B-400 (I) (N.13.8) B-430 (I) (0.1.11)

B-371 (I) (N.4.1) B-401 (I) (N.13.9) B-431 (I) (0.1.12)

B-372 (I) (N.5.1) B-402 (I) (N.14.1) B-432 (I) (0.1.13)

B-373 (I) (N.6.1) B-403 (I) (N.14.2) B-433 (I) (0.1.14)

B-374 (I) (N.6.2) B-404 (I) (N.14.3) B-434 (I) (0.1.15)

B-375 (I) (N.6.3) B-405 (I) (N.15.1) B-435 (I) (0.1.16)

B-376 (I) (N.6.4) B-406 (I) (N.16.1) B-436 (I) (0.1.17)

B-377 (I) (N.6.5) B-407 (I) (N.16.2) B-437 (I) (0.1.18)

B-378 (I) (N.7.1) B-408 (I) (N.17.1) B-438 (I) (0.1.19)

B-379 (I) (N.7.2) B-409 (I) (N.17.2) B-439 (I) (0.1.20)

B-380 (I) (N.7.3) B-410 (I) (N.17.3) B-440 (I) (0.1.21)

B-381 (I) (N.8.1) B-411 (I) (N.17.4) B-441 (I) (0.1.22)

B-382 (I) (N.9.1) B-412 (I) (N.17.5) B-442 (I) (0.1.23)

B-383 (I) (N.10.1) B-413 (I) (N.17.6) B-443 (I) (0.1.24)

B-384 (I) (N.10.2) B-414 (I) (N.17.7) B-444 (I) (0.1.25)

B-385 (I) (N.10.3) B-415 (I) (N.17.8) B-445 (I) (0.1.26)

B-386 (I) (N.10.4) B-416 (I) (N.17.9) B-446 (I) (0.1.27)

B-387 (I) (N.10.5) B-417 (I) (N.17.10) B-447 (I) (0.1.28) Mixt. Co. Co. 2 Mixt. Co. Co. 2 Mixt. Co. Co. 2 1 1 1

B-448 (I) (0.1 .29) B-478 (I) (0.3.5) B-508 (I) (0.4.8)

B-449 (I) (0.1 .30) B-479 (I) (0.3.6) B-509 (I) (0.4.9)

B-450 (I) (0.1 .31 ) B-480 (I) (0.3.7) B-510 (I) (0.4.10)

B-451 (I) (0.1 .32) B-481 (I) (0.3.8) B-51 1 (I) (0.4.1 1 )

B-452 (I) (0.1 .33) B-482 (I) (0.3.9) B-512 (I) (0.4.12)

B-453 (I) (0.1 .34) B-483 (I) (0.3.10) B-513 (I) (0.4.13)

B-454 (I) (0.1 .35) B-484 (I) (0.3.1 1 ) B-514 (I) (0.4.14)

B-455 (I) (0.1 .36) B-485 (I) (0.3.12) B-515 (I) (0.4.15)

B-456 (I) (0.1 .37) B-486 (I) (0.3.13) B-516 (I) (0.4.16)

B-457 (I) (0.1 .38) B-487 (I) (0.3.14) B-517 (I) (0.4.17)

B-458 (I) (0.2.1 ) B-488 (I) (0.3.15) B-518 (I) (0.4.18)

B-459 (I) (0.2.2) B-489 (I) (0.3.16) B-519 (I) (0.4.19)

B-460 (I) (0.2.3) B-490 (I) (0.3.17) B-520 (I) (O.4.20)

B-461 (I) (0.2.4) B-491 (I) (0.3.18) B-521 (I) (0.4.21 )

B-462 (I) (0.2.5) B-492 (I) (0.3.19) B-522 (I) (0.4.22)

B-463 (I) (0.2.6) B-493 (I) (O.3.20) B-523 (I) (0.4.23)

B-464 (I) (0.2.7) B-494 (I) (0.3.21 ) B-524 (I) (0.4.24)

B-465 (I) (0.2.8) B-495 (I) (0.3.22) B-525 (I) (0.5.1 )

B-466 (I) (0.2.9) B-496 (I) (0.3.23) B-526 (I) (0.5.2)

B-467 (I) (0.2.10) B-497 (I) (0.3.24) B-527 (I) (0.5.3)

B-468 (I) (0.2.1 1 ) B-498 (I) (0.3.25) B-528 (I) (0.5.4)

B-469 (I) (0.2.12) B-499 (I) (0.3.26) B-529 (I) (0.5.5)

B-470 (I) (0.2.13) B-500 (I) (0.3.27) B-530 (I) (0.5.6)

B-471 (I) (0.2.14) B-501 (I) (0.4.1 ) B-531 (I) (0.5.7)

B-472 (I) (0.2.15) B-502 (I) (0.4.2) B-532 (I) (0.5.8)

B-473 (I) (0.2.16) B-503 (I) (0.4.3) B-533 (I) (0.5.9)

B-474 (I) (0.3.1 ) B-504 (I) (0.4.4) B-534 (I) (0.6.1 )

B-475 (I) (0.3.2) B-505 (I) (0.4.5) B-535 (I) (0.6.2)

B-476 (I) (0.3.3) B-506 (I) (0.4.6) B-536 (I) (0.6.3)

B-477 (I) (0.3.4) B-507 (I) (0.4.7) B-537 (I) (0.6.4) Mixt. Co. Co. 2 Mixt. Co. Co. 2 Mixt. Co. Co. 2 1 1 1

B-538 (I) (0.6.5) B-553 (I) (0.9.2) B-568 (I) (0.15.5)

B-539 (I) (0.6.6) B-554 (I) (0.9.3) B-569 (I) (0.15.6)

B-540 (I) (0.6.7) B-555 (I) (O.10.1 ) B-570 (I) (0.15.7)

B-541 (I) (0.7.1 ) B-556 (I) (0.1 1.1 ) B-571 (I) (0.15.8)

B-542 (I) (0.7.2) B-557 (I) (0.1 1.2) B-572 (I) (0.15.9)

B-543 (I) (0.7.3) B-558 (I) (0.1 1.3) B-573 (I) (O.15.10)

B-544 (I) (0.7.4) B-559 (I) (0.1 1.4) B-574 (I) (0.15.1 1 )

B-545 (I) (0.7.5) B-560 (I) (0.12.1 ) B-575 (I) (0.16.1 )

B-546 (I) (0.7.6) B-561 (I) (0.13.1 ) B-576 (I) (0.16.2)

B-547 (I) (0.8.1 ) B-562 (I) (0.14.1 ) B-577 (I) (0.16.3)

B-548 (I) (0.8.2) B-563 (I) (0.14.2) B-578 (I) (0.16.4)

B-549 (I) (0.8.3) B-564 (I) (0.15.1 ) B-579 (I) (0.16.5)

B-550 (I) (0.8.4) B-565 (I) (0.15.2) B-580 (I) (0.16.6)

B-551 (I) (0.8.5) B-566 (I) (0.15.3)

B-552 (I) (0.9.1 ) B-567 (I) (0.15.4)

The mixtures of active substances can be prepared as compositions comprising besides the active ingredients at least one inert ingredient (auxiliary) by usual means, e. g. by the means given for the compositions of compounds I.

Concerning usual ingredients of such compositions reference is made to the explanations given for the compositions containing compounds I.

I. Synthesis examples:

2,3-Dibromo-5-[3-fluoro-2-(1 -methoxyethyl)phenoxy]pyridine

1.1 1 -[2-[(5,6-dibromo-3-pyridyl)ox -6-fluoro-phenyl]ethanone

10 g (40 mmol) 5,6,dibromopyridin-3-ol and 7,1 g (51 mmol) potassium carbonat in 200 ml 1 ,2- dimethoxyethane were stirred for 30 min at room temperature. Then 8,03 g (51 mmol) 1 -(2,6- difluorophenyl)ethanon were added and the reaction mixture was stirred 3 days at reflux temperature (85°C). Afterwards the reaction mixture was cooled to room temperature and diluted with water. The aqueous layer was extracted three times with methyl-t-butylether and the combined organic layers were extracted with water and brine, dried over sodium sulfate and concentrated. The residue was purified via chromatography over silica using n-heptane/methyl-t- butylether-mixtures as eluent. One obtained 6,95 g (18 mmol (45 %)) of the title compound as colourless oil.

H-NMR (CDCIs, in ppm):

8,1 (s, 1 H); 7,5 (s, 1 H); 7,4 (m, 1 H); 7,0 (t, 1 H); 6,8 (d, 1 H); 2,6 (s, 3H)

1 -[2-[(5,6-dibromo-3-pyridyl)ox -6-fluoro-phenyl]ethanol

At 0°C 0,039 g (1 mmol) sodium bobohydride was added to 0,2 g (1 mmol) 1 -[2-[(5,6-dibromo-3- pyridyl)oxy]-6-fluoro-phenyl]ethanone in 3 ml methanol. The reaction mixture was allowed to warm up to room temperature and was stirred 2 hours in total. Afterwards the reaction mixture was diluted with water and the aqueous layer was extracted three times with methyl-t- butylether. The combined organic layers were extracted with water and brine to yield 0,188 g (93 %) of the title compound as colourless oil.

H-NMR (CDCIs, in ppm):

8,15 (s, 1 H); 7,5 (s, 1 H); 7,25 (m, 1 H); 6,95 (m, 1 H); 6,7 (d, 1 H); 5,3 (m, 1 H); 2,35 (d, 1 H); 1 ,6 (d, 3H) 1 .3 2,3-Dibromo-5-[3-fluoro-2-(1 -methoxyethyl)phenoxy]pyridine

0,31 1 g (2,4 mmol) Di-isopropyl ethylamine and subsequently 0,109 g (0,63 mmol) methane sulfonic anhydride in 1 ml dichloromethane were added to 0,188 g (0,48 mmol) 1 -[2-[(5,6- dibromo-3-pyridyl)oxy]-6-fluoro-phenyl]ethanol (example 1 .2.) in 5 ml dichloromethane at -10°C. Then several portions of methane sulfonic anhydride were added until total conversion of the starting material. Then 10 ml of methanol were added and the reaction mixture was stirred at room temperature over night. Then silica was added and the mixture was concentrated in vac- uo. The residue was collected and added to the top of a silica column and the product was purified by chromatography using n-heptane/methyl-t-butylether-mixtures as eluent. One obtained 0,104 g (53 %) of the title compound as colourless oil.

H-NMR (CDCIs, in ppm):

8,05 (s, 1 H); 7,5 (s, 1 H); 7,3 (m, 1 H); 7,0 (t, 1 H); 6,7 (d, 1 H); 4,8 (q, 1 H); 3,2 (s, 3H); 1 ,6 (d, 3H)

With due modification of the starting compounds, the procedures shown in the synthesis examples below were used to obtain further compounds I. The resulting compounds, together with physical data, are listed in Table I below.

Table I:

# means conntection to O atom.

No. R ¹ R ² R ³ R ⁴ Q ¹ Q ² Q ³ H-NMR(5 in ppm);

HPLC-MS* (El (M ⁺ +H)

Mp (°C)

1-18 Br Br H H CHs H # M ⁺ + H 465,8

c I

1-19 Br Br H H CHs H M ⁺ + H 464

CH ₃

I-20 Br Br H H CHs H

1-21 Br Br H H CHs H M ⁺ + H 533

R _t = 1,123 min

I-22 Br Br H H CHs H M ⁺ + H 429,9

R _t = 1,322 min

c- 1

HPLC-MS: HPLC-column Kinetex XB C18 1 ,7μ (50 x 2,1 mm); eluent: acetonitrile / water + 0.1 % TFA (5 gradient from 5:95 to 100 : 0 in 1.5 min at 60°C, flow gradient from 0.8 to 1 .0 ml/min in 1 .5 min). MS: Quadrupol Electrospray lonisation, 80 V (positive mode). II. Biological trials

Microtest

The active compounds were formulated separately as a stock solution having a concentration of 10000 ppm in dimethyl sulfoxide. Example 1 - Activity against rice blast Pyricularia oryzae in the microtiterplate test The stock solutions were mixed according to the ratio, pipetted onto a micro titer plate (MTP) and diluted with water to the stated concentrations. A spore suspension of Pyricularia oryzae in an aqueous biomalt or yeast-bactopeptone-glycerine solution was then added. The plates were placed in a water vapor-saturated chamber at a temperature of 18°C. Using an absorption pho- tometer, the MTPs were measured at 405 nm 7 days after the inoculation.

In this test, the samples which had been treated with 31 ppm of the active substance from examples I-2, I-3, I-4, I-5, I-6, I-7, I-8, I-9, 1-10, 1-1 1 , 1-12, 1-13 and 1-14 respectively, showed up to at most 0 % growth of the pathogen.

[Example 2 - Activity against early blight caused by Alternaria solani

The stock solutions were mixed according to the ratio, pipetted onto a micro titer plate (MTP) and diluted with water to the stated concentrations. A spore suspension of Alternaria solani in a DOB medium solution was then added. The plates were placed in a water vapor-saturated chamber at a temperature of 18°C. Using an absorption photometer, the MTPs were measured at 405 nm 9 days after the inoculation.

In this test, the samples which had been treated with 31 ppm of the active substance from ex- amples I-4, I-5, I-7, I-8, I-9, 1-1 1 , 1-12 and 1-13 respectively, showed up to at most 14 % growth of the pathogen.

[Example 53 - Activity against wheat leaf spots caused by Leptosphaeria nodorum The stock solutions were mixed according to the ratio, pipetted onto a micro titer plate (MTP) and diluted with water to the stated concentrations. A spore suspension of Leptosphaeria nodorum in a DOB medium solution was then added. The plates were placed in a water vapor- saturated chamber at a temperature of 18°C. Using an absorption photometer, the MTPs were measured at 405 nm 9 days after the inoculation.

In this test, the sample which had been treated with 31 ppm of the active substance from example 1-12, showed up to at most 19 % growth of the pathogen.

The measured parameters were compared to the growth of the active compound-free control variant (100%) and the fungus-free and active compound-free blank value to determine the relative growth in % of the pathogens in the respective active compounds.