Title:
PYRIMIDINE DERIVATIVES
Document Type and Number:
WIPO Patent Application WO/2004/011442
Kind Code:
A1
Abstract:
Pyrimidine derivatives represented by the following general formula (1): (1) Because of having an excellent PA activity promoting effect and a PAI−1 inhibitory effect, these pyrimidine derivatives are usable as antithrombotic agents and thrombolytic agents which can be orally administered.
Inventors:
NAKATOGAWA KIYOSHI (JP)
MURATA MASANAO (JP)
TAKEUCHI AKIRA (JP)
SUZUKI KAORU (JP)
MURATA MASANAO (JP)
TAKEUCHI AKIRA (JP)
SUZUKI KAORU (JP)
Application Number:
PCT/JP2002/007678
Publication Date:
February 05, 2004
Filing Date:
July 29, 2002
Export Citation:
Assignee:
SHIZUOKA COFFEIN CO LTD (JP)
NAKATOGAWA KIYOSHI (JP)
MURATA MASANAO (JP)
TAKEUCHI AKIRA (JP)
SUZUKI KAORU (JP)
NAKATOGAWA KIYOSHI (JP)
MURATA MASANAO (JP)
TAKEUCHI AKIRA (JP)
SUZUKI KAORU (JP)
International Classes:
A61K31/505; A61K31/506; A61K31/5377; A61P7/02; A61P43/00; C07D401/04; C07D401/12; (IPC1-7): C07D239/34; A61K31/505; A61K31/506; A61K31/5377; A61P7/02; A61P43/00; C07D239/36; C07D239/47; C07D239/70; C07D401/04; C07D401/12; C07D403/12; C07D405/04
Domestic Patent References:
WO2001094299A1 | 2001-12-13 |
Foreign References:
JP2000159751A | 2000-06-13 |
Attorney, Agent or Firm:
Asamura, Kiyoshi (New Ohtemachi Bldg. 2-1, Ohtemachi 2-chom, Chiyoda-ku Tokyo, JP)
Download PDF: