Title:
PYRUVATE KINASE MODULATORS AND USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2019/035865
Kind Code:
A8
Abstract:
Described herein are methods of using compounds of Formula (I) to modulate PKM2 activity in a subject. These compounds are represented by Formula (I): wherein R1, R2, L1, and L2 are as defined herein.
Inventors:
KUNG CHARLES (US)
CIANCHETTA GIOVANNI (US)
LIU TAO (US)
PADYANA ANIL (US)
SUI ZHIHUA (US)
CAI ZHENWEI (CN)
CUI DAWEI (CN)
JI JINGJING (CN)
CIANCHETTA GIOVANNI (US)
LIU TAO (US)
PADYANA ANIL (US)
SUI ZHIHUA (US)
CAI ZHENWEI (CN)
CUI DAWEI (CN)
JI JINGJING (CN)
Application Number:
PCT/US2018/000129
Publication Date:
March 28, 2019
Filing Date:
August 15, 2018
Export Citation:
Assignee:
AGIOS PHARMACEUTICALS INC (US)
KUNG CHARLES (US)
KUNG CHARLES (US)
International Classes:
A61K31/5025; A61P3/10; A61P7/06; A61P7/08; A61P35/00; C07D513/14
Attorney, Agent or Firm:
DAVIS, Steven, G. et al. (US)
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