Title:
QUINAZOLINONE COMPOUND CRYSTAL FORM, PREPARATION METHOD THEREFOR, AND USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2022/016420
Kind Code:
A1
Abstract:
A quinazolinone compound crystal form, a preparation method therefor, and a use thereof. The crystal form 1 of the compound of formula I has good stability and is easy to form into a drug, can inhibit PI3K kinase activity well, and also has higher subtype selectivity for PI3Kβ/γ/δ.
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Inventors:
TANG WEI (CN)
HUANG JITING (CN)
WANG ZHENYU (CN)
YANG WENQIAN (CN)
HUANG JITING (CN)
WANG ZHENYU (CN)
YANG WENQIAN (CN)
Application Number:
PCT/CN2020/103532
Publication Date:
January 27, 2022
Filing Date:
July 22, 2020
Export Citation:
Assignee:
LUOXIN PHARMACEUTICAL SHANGHAI CO LTD (CN)
SHANDONG LUOXIN PHARMACY STOCK (CN)
SHANDONG LUOXIN PHARMACY STOCK (CN)
International Classes:
C07D401/04; A61K31/517; A61P35/00
Domestic Patent References:
WO2019091476A1 | 2019-05-16 |
Foreign References:
CN102149711A | 2011-08-10 |
Attorney, Agent or Firm:
SHANGHAI BESHINING LAW OFFICE (CN)
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