Title:
SUBSTITUTED ARYL KETONES
Document Type and Number:
WIPO Patent Application WO2001053275
Kind Code:
A3
Abstract:
The invention relates to novel aryl ketones of general formula (I), wherein n represents the numbers 0, 1 or 2, A represents alkanediyl (alkylene), R<1> represents one of the following groupings, m, R<5>, R<6>, R<7>, R<8>, R<9>, R<10>, R<11>, R<12> and R<13> having one of the meanings given in the description, R<2> represents hydrogen, nitro, cyano, carboxy, carbamoyl, thiocarbamoyl, halogen, or optionally substituted alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, dialkylamino or dialkylaminosulfonyl, R<3> represents nitro, cyano, carboxy, carbamoyl, thiocarbamoyl, halogen or optionally substituted alkyl, alkoxy, alkylthio, alkylsulfinyl, alkylsulfonyl, alkylamino, dialkylamino or dialkylaminosulfonyl and R<4> represents an optionally substituted 4- to 12-membered, saturated or unsaturated, monocyclic or bicyclic, heterocyclic grouping. The invention also relates to methods for producing said substituted arylketones, to intermediate products and to the use of these compounds as herbicides.
Inventors:
SCHALLNER OTTO (DE)
LEHR STEFAN (DE)
SCHWARZ HANS-GEORG (DE)
MUELLER KLAUS-HELMUT (DE)
HOISCHEN DOROTHEE (DE)
DREWES MARK WILHELM (DE)
DAHMEN PETER (DE)
FEUCHT DIETER (DE)
PONTZEN ROLF (DE)
YANAGI AKIHIKO (JP)
NARABU SHINICHI (JP)
GOTO TOSHIO (JP)
LEHR STEFAN (DE)
SCHWARZ HANS-GEORG (DE)
MUELLER KLAUS-HELMUT (DE)
HOISCHEN DOROTHEE (DE)
DREWES MARK WILHELM (DE)
DAHMEN PETER (DE)
FEUCHT DIETER (DE)
PONTZEN ROLF (DE)
YANAGI AKIHIKO (JP)
NARABU SHINICHI (JP)
GOTO TOSHIO (JP)
Application Number:
PCT/EP2001/000092
Publication Date:
April 17, 2003
Filing Date:
January 05, 2001
Export Citation:
Assignee:
BAYER AG (DE)
BAYER AGROCHEM KK (JP)
SCHALLNER OTTO (DE)
LEHR STEFAN (DE)
SCHWARZ HANS-GEORG (DE)
MUELLER KLAUS-HELMUT (DE)
HOISCHEN DOROTHEE (DE)
DREWES MARK WILHELM (DE)
DAHMEN PETER (DE)
FEUCHT DIETER (DE)
PONTZEN ROLF (DE)
YANAGI AKIHIKO (JP)
NARABU SHINICHI (JP)
GOTO TOSHIO (JP)
BAYER AGROCHEM KK (JP)
SCHALLNER OTTO (DE)
LEHR STEFAN (DE)
SCHWARZ HANS-GEORG (DE)
MUELLER KLAUS-HELMUT (DE)
HOISCHEN DOROTHEE (DE)
DREWES MARK WILHELM (DE)
DAHMEN PETER (DE)
FEUCHT DIETER (DE)
PONTZEN ROLF (DE)
YANAGI AKIHIKO (JP)
NARABU SHINICHI (JP)
GOTO TOSHIO (JP)
International Classes:
A01N43/36; A01N43/40; A01N43/56; A01N43/653; A01N43/713; C07D207/26; C07D213/64; C07D249/12; C07D257/04; C07D403/12; (IPC1-7): C07D403/12; C07D249/12; C07D213/64; C07D207/26; C07D257/04; A01N43/653; A01N43/40; A01N43/56; A01N43/36; A01N43/713
Domestic Patent References:
| WO1997045404A1 | 1997-12-04 | |||
| WO1998041089A1 | 1998-09-24 | |||
| WO2000017194A1 | 2000-03-30 | |||
| WO2001014303A1 | 2001-03-01 | |||
| WO1999010328A1 | 1999-03-04 | |||
| WO1999010327A1 | 1999-03-04 | |||
| WO1999003856A1 | 1999-01-28 | |||
| WO1997027187A1 | 1997-07-31 | |||
| WO1999007688A1 | 1999-02-18 | |||
| WO1997046530A1 | 1997-12-11 | |||
| WO2001000206A1 | 2001-01-04 | |||
| WO2000075130A1 | 2000-12-14 | |||
| WO2000066120A1 | 2000-11-09 | |||
| WO2000058295A2 | 2000-10-05 | |||
| WO1999043672A1 | 1999-09-02 | |||
| WO1999041235A1 | 1999-08-19 | |||
| WO1992019603A1 | 1992-11-12 | |||
| WO1996011023A1 | 1996-04-18 | |||
| WO1996006094A1 | 1996-02-29 |
Foreign References:
| EP0352543A1 | 1990-01-31 | |||
| EP0609797A1 | 1994-08-10 | |||
| US5804532A | 1998-09-08 | |||
| EP0741128A2 | 1996-11-06 |
Other References:
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; MORITA, TAKESHI ET AL: "Preparation of 2-[3-(1,3-dioxolan-4-ylmethoxy)benzoyl]-1,3- cyclohexanedione derivatives as herbicides", XP002166959, retrieved from STN Database accession no. 122:155301
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; MORITA, TAKESHI ET AL: "Preparation of dioxane and dioxolane derivatives as herbicides", XP002166960, retrieved from STN Database accession no. 122:160651
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; SOMEYA, SHINZO ET AL: "Pyrazole derivatives as herbicides and process of their preparation", XP002166961, retrieved from STN Database accession no. 110:173224
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; FATTAKHOV, S. G. ET AL: "Synthesis and transformations of 1,3-bis[.omega.-(2- formylphenoxy)alkyl]-6-methyluracils", XP002166962, retrieved from STN Database accession no. 133:335208
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; GRABOWSKA, URSZULA ET AL: "5-(Hydroxymethyl)oxazoles: Versatile Scaffolds for Combinatorial Solid-Phase Synthesis of 5-Substituted Oxazoles", XP002166963, retrieved from STN Database accession no. 133:222636
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; VAZ, ROY J. ET AL: "Use of CoMFA in validating the conformation used in designing 4-(1H-benzimidazole-2-carbonyl)piperidines with H1/NK1 receptor antagonist activity", XP002166964, retrieved from STN Database accession no. 128:110371
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; MAYNARD, GEORGE D. ET AL: "Synthesis and structure-activity relationship of 4-(1H-benzimidazole-2-carbonyl)piperidines with dual histamine H1/tachykinin NK1 receptor antagonist activity", XP002166965, retrieved from STN Database accession no. 128:75364
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; WALTON, PAUL H. ET AL: "Stereognostic coordination chemistry 4. The design and synthesis of a selective uranyl ion complexant", XP002166966, retrieved from STN Database accession no. 124:248683
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; MORITA, TAKESHI ET AL: "Cyclohexanediones and herbicides containing them", XP002167114, retrieved from STN Database accession no. 123:278720
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; NAOHARA, KAZUO ET AL: "Synergistic herbicides containing phenoxymethylpyrimidine derivatives", XP002166967, retrieved from STN Database accession no. 122:3573
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; OONISHI, AKIRA ET AL: "Silver halide photographic photosensitive material containing diffusion-resistant dyes", XP002166968, retrieved from STN Database accession no. 121:311734
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; DAINES, ROBERT A. ET AL: "Trisubstituted pyridine leukotriene B4 receptor antagonists: synthesis and structure-activity relationships", XP002166969, retrieved from STN Database accession no. 120:77146
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; WADA, NOBUHIDE ET AL: "Preparation of 2-phenoxypyrimidines as herbicides", XP002166970, retrieved from STN Database accession no. 110:192853
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; MORITA, TAKESHI ET AL: "Preparation of dioxane and dioxolane derivatives as herbicides", XP002166960, retrieved from STN Database accession no. 122:160651
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; SOMEYA, SHINZO ET AL: "Pyrazole derivatives as herbicides and process of their preparation", XP002166961, retrieved from STN Database accession no. 110:173224
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; FATTAKHOV, S. G. ET AL: "Synthesis and transformations of 1,3-bis[.omega.-(2- formylphenoxy)alkyl]-6-methyluracils", XP002166962, retrieved from STN Database accession no. 133:335208
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; GRABOWSKA, URSZULA ET AL: "5-(Hydroxymethyl)oxazoles: Versatile Scaffolds for Combinatorial Solid-Phase Synthesis of 5-Substituted Oxazoles", XP002166963, retrieved from STN Database accession no. 133:222636
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; VAZ, ROY J. ET AL: "Use of CoMFA in validating the conformation used in designing 4-(1H-benzimidazole-2-carbonyl)piperidines with H1/NK1 receptor antagonist activity", XP002166964, retrieved from STN Database accession no. 128:110371
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; MAYNARD, GEORGE D. ET AL: "Synthesis and structure-activity relationship of 4-(1H-benzimidazole-2-carbonyl)piperidines with dual histamine H1/tachykinin NK1 receptor antagonist activity", XP002166965, retrieved from STN Database accession no. 128:75364
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; WALTON, PAUL H. ET AL: "Stereognostic coordination chemistry 4. The design and synthesis of a selective uranyl ion complexant", XP002166966, retrieved from STN Database accession no. 124:248683
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; MORITA, TAKESHI ET AL: "Cyclohexanediones and herbicides containing them", XP002167114, retrieved from STN Database accession no. 123:278720
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; NAOHARA, KAZUO ET AL: "Synergistic herbicides containing phenoxymethylpyrimidine derivatives", XP002166967, retrieved from STN Database accession no. 122:3573
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; OONISHI, AKIRA ET AL: "Silver halide photographic photosensitive material containing diffusion-resistant dyes", XP002166968, retrieved from STN Database accession no. 121:311734
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; DAINES, ROBERT A. ET AL: "Trisubstituted pyridine leukotriene B4 receptor antagonists: synthesis and structure-activity relationships", XP002166969, retrieved from STN Database accession no. 120:77146
DATABASE CHEMABS [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; WADA, NOBUHIDE ET AL: "Preparation of 2-phenoxypyrimidines as herbicides", XP002166970, retrieved from STN Database accession no. 110:192853
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