Title:
SUBSTITUTED PIPERIDINES/PIPERAZINES AS MELANOCORTIN RECEPTOR AGONISTS
Document Type and Number:
WIPO Patent Application WO2002059107
Kind Code:
A8
Abstract:
The present invention relates to melanocortin receptor agonists of formula I, which is useful in the treatment of obesity, diabetes and male and/or female sexual dysfunction.
Inventors:
BACKER RYAN THOMAS (US)
BRINER KARIN (US)
DOECKE CHRISTOPHER WILLIAM (US)
FISHER MATTHEW JOSEPH (US)
KUKLISH STEVEN LEE (US)
MANCUSO VINCENT (BE)
MARTINELLI MICHAEL JOHN (US)
MULLANEY JEFFREY THOMAS (US)
XIE CHAOYU (US)
BRINER KARIN (US)
DOECKE CHRISTOPHER WILLIAM (US)
FISHER MATTHEW JOSEPH (US)
KUKLISH STEVEN LEE (US)
MANCUSO VINCENT (BE)
MARTINELLI MICHAEL JOHN (US)
MULLANEY JEFFREY THOMAS (US)
XIE CHAOYU (US)
Application Number:
PCT/US2002/000516
Publication Date:
November 06, 2003
Filing Date:
January 23, 2002
Export Citation:
Assignee:
LILLY CO ELI (US)
BACKER RYAN THOMAS (US)
BRINER KARIN (US)
DOECKE CHRISTOPHER WILLIAM (US)
FISHER MATTHEW JOSEPH (US)
KUKLISH STEVEN LEE (US)
MANCUSO VINCENT (BE)
MARTINELLI MICHAEL JOHN (US)
MULLANEY JEFFREY THOMAS (US)
XIE CHAOYU (US)
BACKER RYAN THOMAS (US)
BRINER KARIN (US)
DOECKE CHRISTOPHER WILLIAM (US)
FISHER MATTHEW JOSEPH (US)
KUKLISH STEVEN LEE (US)
MANCUSO VINCENT (BE)
MARTINELLI MICHAEL JOHN (US)
MULLANEY JEFFREY THOMAS (US)
XIE CHAOYU (US)
International Classes:
A61K31/4725; A61K31/496; A61K31/5377; A61P3/04; A61P3/10; A61P15/00; A61P15/10; C07B61/00; C07D209/44; C07D217/26; C07D401/12; C07D401/14; (IPC1-7): C07D401/12; A61K31/44; A61K31/495; A61P15/10; C07D401/14
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