Title:
SUBSTITUTED CAPROLACTAMS AND DERIVATIVES THEREOF USEFUL FOR TREATMENT OF AIDS
Document Type and Number:
WIPO Patent Application WO/1994/008977
Kind Code:
A1
Abstract:
This invention relates to novel substituted caprolactams of formula (I), including 4-azacaprolactams, and derivatives thereof which inhibit HIV protease and are useful for treatment of HIV disease. Also included in this invention are pharmaceutical compositions containing such substituted caprolactams and to methods of using such caprolactams for the treatment of HIV disease.
Inventors:
HODGE CARL NICHOLAS
FERNANDEZ CHRISTINA HOWARD
FERNANDEZ CHRISTINA HOWARD
Application Number:
PCT/US1993/009807
Publication Date:
April 28, 1994
Filing Date:
October 20, 1993
Export Citation:
Assignee:
DU PONT MERCK PHARMA (US)
International Classes:
C07D243/08; C07D245/02; C07D255/02; C07D257/02; C07D267/10; C07D281/06; (IPC1-7): C07D243/08; A61K31/55
Domestic Patent References:
| WO1992009297A1 | 1992-06-11 |
Download PDF:
Previous Patent: FUNGICIDAL AND MITICIDAL AMINOPYRIMIDINES
Next Patent: FUNGICIDAL SUBSTITUTED AZOLE DERIVATIVES
Next Patent: FUNGICIDAL SUBSTITUTED AZOLE DERIVATIVES