Substituted N-(tetrazol-5-yl)- and N-(triazol-5-yl)arylcarboxamide compounds and their use as herbicides

Description

The present invention relates to substituted N-(tetrazol-5-yl)- and N-(triazol-5- yl)arylcarboxamide compounds and the N-oxides and salts thereof and to compositions comprising the same. The invention also relates to the use of the N-(tetrazol-5-yl)- and N- (triazol-5-yl)arylcarboxamide compounds or of the compositions comprising such compounds for controlling unwanted vegetation. Furthermore, the invention relates to methods of applying such compounds.

For the purposes of controlling unwanted vegetation, especially in crops, there is an ongoing need for new herbicides which have high activities and selectivities together with a substantial lack of toxicity for humans and animals.

WO 201 1/035874 describes N-(1 ,2,5-oxadiazol-3-yl)benzamides carrying 3 substituents in the 2-, 3- and 4-positions of the phenyl ring and their use as herbicides.

WO 2012/028579 describes N-(tetrazol-4-yl)- and N-(triazol-3-yl)arylcarboxylic acid amides carrying 3 substituents in the 2-, 3- and 4-positions of the aryl ring and their use as herbicides.

The compounds of the prior art often suffer form insufficient herbicidal activity in particular at low application rates and/or unsatisfactory selectivity resulting in a low compatibility with crop plants.

Accordingly, it is an object of the present invention to provide further N-(tetrazol-5-yl)- and N-(triazol-5-yl)arylcarboxamide compounds having a strong herbicidal activity, in particular even at low application rates, a sufficiently low toxicity for humans and animals and/or a high compatibility with crop plants. The N-(tetrazol-5-yl)- and N-(triazol-5-yl)arylcarboxamide compounds should also show a broad activity spectrum against a large number of different unwanted plants.

These and further objectives are achieved by the compounds of formula I defined below and their N-oxides and also their agriculturally suitable salts.

It has been found that the above objectives can be achieved by substituted N-(tetrazol-5- yl)- and N-(triazol-5-yl)arylcarboxamide compounds of the general formula I, as defined below, including their N-oxides and their salts, in particular their agriculturally suitable salts.

Therefore, in a first aspect the present invention relates to compounds of formula I,

where

B is N or CH; R is selected from the group consisting of hydrogen, Ci-C6-alkyl, C3-C7-cycloalkyl, C3-C7- cycloalkyl-Ci-C4-alkyl, where the C3-C7-cycloalkyl groups in the two aforementioned radicals are unsubstituted or partially or completely halogenated, Ci-C6-haloalkyl, C2-C6- alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, Ci-C4-alkoxy-Ci-C4-alkyl, Ci- C ₄ -haloalkoxy-Ci-C ₄ -alkyl, R ^b -S(0) _n -Ci-C ₃ -alkyl, R ^d O-C(=0)-Ci-C ₃ - alkyl, R ^e R ^f N-C(=0)-Ci-C ₃ -alkyl, R9R ^h N-Ci-C ₃ -alkyl, phenyl-Z and heterocyclyl-Z, where heterocyclyl is a 5- or 6-membered monocyclic or 8-, 9- or 10-membered bicyclic saturated, partially unsaturated or aromatic heterocycle, which contains 1 , 2, 3 or 4 heteroatoms as ring members, which are selected from the group consisting of O, N and S, where phe- nyl and heterocyclyl are unsubstituted or substituted by 1 , 2, 3 or 4 groups R', which are identical or different;

R ¹ is selected from the group consisting of cyano-Z ¹ , halogen, nitro, Ci-Cs-alkyl, C2-C8- alkenyl, C2-Cs-alkynyl, Ci-Cs-haloalkyl, d-Cs-alkoxy, Ci-C ₄ -alkoxy-Ci-C ₄ -alkyl, Ci-C ₄ - alkoxy-Ci-C -alkoxy-Z ¹ , Ci-C -alkylthio-Ci-C -alkyl, Ci-C -alkylthio-Ci-C -alkylthio-Z ¹ , C ₂ - C6-alkenyloxy, C2-C6-alkynyloxy, Ci-C6-haloalkoxy, Ci-C ₄ -haloalkoxy-Ci-C ₄ -alkyl, Ci-C ₄ - haloalkoxy-Ci-C ₄ -alkoxy-Z ¹ , R ^1b -S(0) _k -Z ¹ , phenoxy-Z ¹ , and heterocyclyloxy-Z ¹ , where het- erocyclyloxy is an oxygen bound 5- or 6-membered monocyclic or 8-, 9- or 10-membered bicyclic saturated, partially unsaturated or aromatic heterocycle, which contains 1 , 2, 3 or 4 heteroatoms as ring members, which are selected from the group consisting of O, N and S, where the cyclic groups in phenoxy and heterocyclyloxy are unsubstituted or substituted by 1 , 2, 3 or 4 groups R ¹¹ , which are identical or different;

R ² , R ³ are identical or different and independently selected from the group consisting of hydrogen, halogen, OH-Z ² , NO2-Z ² , cyano-Z ² , Ci-C6-alkyl, C2-Cs-alkenyl, C2-Cs-alkynyl, C ₃ -Cio- cycloalkyl-Z ² , C ₃ -Cio-cycloalkoxy-Z ² , where the C ₃ -Cio-cycloalkyl groups in the two afore- mentioned radicals are unsubstituted or partially or completely halogenated, Ci-Cs- haloalkyl, Ci-Cs-alkoxy-Z ² , Ci-Cs-haloalkoxy-Z ² , Ci-C ₄ -alkoxy-Ci-C ₄ -alkoxy-Z ² , Ci-C ₄ - a I ky 11 h i o-C1 -C ₄ -a I kyl th i0-Z ² , C ₂ -C ₈ -alkenyloxy-Z ² , C ₂ -C ₈ -alkynyloxy-Z ² , C ₂ -C ₈ - haloalkenyloxy-Z ² , C2-C8-haloalkynyloxy-Z ² , Ci-C ₄ -haloalkoxy-Ci-C ₄ -alkoxy-Z ² , (tri-Ci-C ₄ - alkyl)silyl-Z ² , R ^2b -S(0) _k -Z ² , R ^2c -C(=0)-Z ² , R ^2d O-C(=0)-Z ² , R ^2e R ^2f N-C(=0)-Z ² , R¾R ^2h N-Z ² , phenyl-Z ^2a and heterocyclyl-Z ^2a , where heterocyclyl is a 3-, 4-, 5- or 6-membered monocyclic or 8-, 9- or 10-membered bicyclic saturated, partially unsaturated or aromatic heterocycle, which contains 1 , 2, 3 or 4 heteroatoms as ring members, which are selected from the group consisting of O, N and S, where the cyclic groups in phenyl-Z ^2a and heterocyclyl-Z ²³ are unsubstituted or substituted by 1 , 2, 3 or 4 groups R ²¹ , which are identical or different;

R ⁴ , R ⁵ are identical or different and independently selected from the group consisting of hydrogen, cyano- Z ¹ , halogen, nitro, Ci-Cs-alkyl, C ₃ -C7-cycloalkyl, C ₃ -C7-cycloalkyl-Ci-C ₄ -alkyl, where the C ₃ -C7-cycloalkyl groups in the two aforementioned radicals are unsubstituted or partially or completely halogenated, C2-Cs-alkenyl, C2-Cs-alkynyl, Ci-Cs-haloalkyl, Ci-C ₃ - alkylamino, Ci-C ₃ -dialkylamino, Ci-C ₃ -alkylamino-S(0)k, Ci-C ₃ -alkylcarbonyl, Ci-C ₃ - alkoxy, Ci-C ₄ -alkoxy-Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy-Ci-C ₄ -alkoxy-Z ¹ , Ci-C ₄ -alkylthio-Ci-C ₄ - alkyl, Ci-C ₄ -alkylthio-Ci-C ₄ -alkylthio-Z ¹ , C2-C6-alkenyloxy, C2-C6-alkynyloxy, C1-C6- haloalkoxy, Ci-C ₄ -haloalkoxy-Ci-C ₄ -alkyl, Ci-C -haloalkoxy-Ci-C -alkoxy-Z ¹ , R ^1b -S(0) _k -Z ¹ , phenoxy-Z ¹ and heterocyclyloxy-Z ¹ , where heterocyclyloxy is an oxygen bound 5- or 6- membered monocyclic or 8-, 9- or 10-membered bicyclic saturated, partially unsaturated or aromatic heterocycle, which contains 1 , 2, 3 or 4 heteroatoms as ring members, which are selected from the group consisting of O, N and S, where the cyclic groups in phenoxy and heterocyclyloxy are unsubstituted or substituted by 1 , 2, 3 or 4 groups R ¹¹ , which are identical or different;

provided that at least one of the radicals R ⁴ and R ⁵ is different from hydrogen; and further provided that if R ⁴ is hydrogen, halogen, cyano, nitro, Ci-C ₄ -alkyl or Ci-C ₄ -haloalkyl, R ⁵ is not hydrogen, halogen, Ci-C ₄ -alkyl or Ci-C ₄ -haloalkyl;

n is 0, 1 or 2;

k is 0, 1 or 2;

R', R ¹¹ , R ²¹ independently of each other are selected from the group consisting of halogen, NO2, CN, d-Ce-alkyl, C ₃ -C ₇ -cycloalkyl, C ₃ -C ₇ -halocycloalkyl, Ci-C ₆ -haloalkyl, C ₂ -C ₆ -alkenyl, C ₂ - C6-haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, Ci-C6-alkoxy, Ci-C ₄ -alkoxy-Ci-C ₄ -alkyl,

Ci-C ₄ -alkylthio-Ci-C ₄ -alkyl, Ci-C ₄ -haloalkoxy-Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy-Ci-C ₄ -alkoxy, C3- C7-cycloalkoxy and Ci-C6-haloalkyloxy, or two vicinal radicals R', R ¹¹ or R ²¹ together may form a group =0;

Z, Z ¹ , Z ² independently of each other are selected from the group consisting of a covalent bond and Ci-C ₄ -alkanediyl;

Z ^2a is selected from the group consisting of a covalent bond, Ci-C ₄ -alkanediyl, 0-Ci-C ₄ - alkanediyl, Ci-C ₄ -alkanediyl-0 and Ci-C ₄ -alkanediyl-0-Ci-C ₄ -alkanediyl;

R ^b , R ^1b , R ^2b independently of each other are selected from the group consisting of Ci-C6-alkyl, C3-C7-cycloalkyl, Ci-C6-haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C2-C6- haloalkynyl, phenyl and heterocyclyl, where heterocyclyl is a 5- or 6-membered monocyclic saturated, partially unsaturated or aromatic heterocycle, which contains 1 , 2, 3 or 4 heteroatoms as ring members, which are selected from the group consisting of O, N and S, where phenyl and heterocyclyl are unsubstituted or substituted by 1 , 2, 3 or 4 groups, which are identical or different and selected from the group consisting of halogen, Ci-C ₄ -alkyl, Ci-C ₄ -haloalkyl, Ci-C ₄ -alkoxy and Ci-C ₄ -haloalkoxy;

R ^c , R ^2c independently of each other are selected from the group consisting of hydrogen, C1-C6- alkyl, C3-C7-cycloalkyl, C3-C7-cycloalkyl-Ci-C ₄ -alkyl, where the C3-C7-cycloalkyl groups in the two aforementioned radicals are unsubstituted or partially or completely halogenated, Ci-C6-haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, Ci-C ₄ - alkoxy-Ci-C ₄ -alkyl, phenyl, benzyl and heterocyclyl, where heterocyclyl is a 5- or 6- membered monocyclic saturated, partially unsaturated or aromatic heterocycle, which contains 1 , 2, 3 or 4 heteroatoms as ring members, which are selected from the group consisting of O, N and S, where phenyl, benzyl and heterocyclyl are unsubstituted or substituted by 1 , 2, 3 or 4 groups, which are identical or different and selected from the group consisting of halogen, Ci-C ₄ -alkyl, Ci-C ₄ -haloalkyl, Ci-C ₄ -alkoxy and Ci-C ₄ - haloalkoxy;

R ^d , R ^2d independently of each other are selected from the group consisting of Ci-C6-alkyl, C3-C7- cycloalkyl, C3-C7-cycloalkyl-Ci-C4-alkyl, where the C3-C7-cycloalkyl groups in the two aforementioned radicals are unsubstituted or partially or completely halogenated, C1-C6- haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, C1-C4- alkoxy-Ci-C4-alkyl, phenyl and benzyl, where phenyl and benzyl are unsubstituted or substituted by 1 , 2, 3 or 4 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy and C1-C4- haloalkoxy;

R ^e , R ^f independently of each other are selected from the group consisting of hydrogen, C1-C6- alkyl, C3-C7-cycloalkyl, C3-C7-cycloalkyl-Ci-C4-alkyl, where the C3-C7-cycloalkyl groups in the two aforementioned radicals are unsubstituted or partially or completely halogenated,

Ci-C6-haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, C1-C4- alkoxy-Ci-C4-alkyl, phenyl and benzyl, where phenyl and benzyl are unsubstituted or substituted by 1 , 2, 3 or 4 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy and C1-C4- haloalkoxy, or

R ^e , R ^f together with the nitrogen atom, to which they are bound may form a 5-, 6 or 7- membered, saturated or unsaturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is unsubstituted or may carry 1 , 2, 3 or 4 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy and Ci-C4-haloalkoxy;

R ^2e , R ^2f independently of each other have the meanings given for R ^e , R ^f ;

R9 is selected from the group consisting of hydrogen, Ci-C6-alkyl, C3-C7-cycloalkyl, C3-C7- cycloalkyl-Ci-C4-alkyl, where the C3-C7-cycloalkyl groups in the two aforementioned radicals are unsubstituted or partially or completely halogenated, Ci-C6-haloalkyl, C2-C6- alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, Ci-C4-alkoxy-Ci-C4-alkyl, phenyl and benzyl, where phenyl and benzyl are unsubstituted or substituted by 1 , 2, 3 or 4 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy and Ci-C4-haloalkoxy;

R ^h is selected from the group consisting of hydrogen, Ci-C6-alkyl, C3-C7-cycloalkyl, C3-C7- cycloalkyl-Ci-C4-alkyl, where the C3-C7-cycloalkyl groups in the two aforementioned radicals are unsubstituted or partially or completely halogenated, Ci-C6-haloalkyl, C2-C6- alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, Ci-C4-alkoxy-Ci-C4-alkyl, a radical C(=0)-R ^k , phenyl and benzyl, where phenyl and benzyl are unsubstituted or substituted by 1 , 2, 3 or 4 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy and C1-C4- haloalkoxy, or

R9, R ^h together with the nitrogen atom, to which they are bound may form a 5-, 6 or 7- membered, saturated or unsaturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is unsubstituted or may carry 1 , 2, 3 or 4 groups, which are identical or different and selected from the group consisting of =0, halogen, Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy and C1-C4- haloalkoxy; R¾, R ^2h independently of each other have the meanings given for Rs, R ^h ; and

R ^k has the meanings given for R ^c ;

or an N-oxide or an agriculturally suitable salt thereof. The compounds of the present invention, i.e. the compounds of formula I, their N-oxides, or their salts are particularly useful for controlling unwanted vegetation. Therefore, the invention also relates to the use of a compound of the present invention, an N-oxide or a salt thereof or of a composition comprising at least one compound of the invention, an N-oxide or an agriculturally suitable salt thereof for combating or controlling unwanted vegetation.

The invention also relates to a composition comprising at least one compound according to the invention, including an N-oxide or a salt thereof, and at least one auxiliary. In particular, the invention relates to an agricultural composition comprising at least one compound according to the invention including an N-oxide or an agriculturally suitable salt thereof, and at least one auxiliary customary for crop protection formulations.

The present invention also relates to a method for combating or controlling unwanted vegetation, which method comprises allowing a herbicidally effective amount of at least one compound according to the invention, including an N-oxide or a salt thereof, to act on unwanted plants, their seed and/or their habitat.

Depending on the substitution pattern, the compounds of formula I may have one or more centers of chirality, in which case they are present as mixtures of enantiomers or diastereomers. The invention provides both the pure enantiomers or pure diastereomers of the compounds of formula I, and their mixtures and the use according to the invention of the pure enantiomers or pure diastereomers of the compound of formula I or its mixtures. Suitable compounds of formula I also include all possible geometrical stereoisomers (cis/trans isomers) and mixtures thereof. Cis/trans isomers may be present with respect to an alkene, carbon-nitrogen double-bond, nitrogen-sulfur double bond or amide group. The term "stereoisomer(s)" encompasses both optical isomers, such as enantiomers or diastereomers, the latter existing due to more than one center of chirality in the molecule, as well as geometrical isomers (cis/trans isomers).

Depending on the substitution pattern, the compounds of formula I may be present in the form of their tautomers. Hence the invention also relates to the tautomers of the formula I and the stereoisomers, salts and N-oxides of said tautomers.

The term "N-oxide" includes any compound of the present invention which has at least one tertiary nitrogen atom that is oxidized to an N-oxide moiety. N-oxides in compounds of formula I can in particular be prepared by oxidizing the ring nitrogen atom(s) of the N-(tetrazol-5- yl)- and N-(triazol-5-yl)arylcarboxamide ring with a suitable oxidizing agent, such as peroxo car- boxylic acids or other peroxides, or the ring nitrogen atom(s) of a heterocyclic substituent R, R ¹ , R ² or R ³ .

The present invention moreover relates to compounds as defined herein, wherein one or more of the atoms depicted in formula I have been replaced by its stable, preferably non- radioactive isotope (e.g., hydrogen by deuterium, ¹² C by ¹³ C, ¹⁴ N by ¹⁵ N, ¹⁶ 0 by ¹⁸ 0) and in particular wherein at least one hydrogen atom has been replaced by a deuterium atom. Of course, the compounds according to the invention contain more of the respective isotope than this naturally occurs and thus is anyway present in the compounds of formula I.

The compounds of the present invention may be amorphous or may exist in one ore more different crystalline states (polymorphs) which may have different macroscopic properties such as stability or show different biological properties such as activities. The present invention includes both amorphous and crystalline compounds of formula I, their enantiomers or diastere- omers, mixtures of different crystalline states of the respective compound of formula I, its enantiomers or diastereomers, as well as amorphous or crystalline salts thereof.

Salts of the compounds of the present invention are preferably agriculturally suitable salts. They can be formed in a customary method, e.g. by reacting the compound with an acid if the compound of the present invention has a basic functionality or by reacting the compound with a suitable base if the compound of the present invention has an acidic functionality.

Useful agriculturally suitable salts are especially the salts of those cations or the acid addition salts of those acids whose cations and anions, respectively, do not have any adverse effect on the herbicidal action of the compounds according to the present invention. Suitable cations are in particular the ions of the alkali metals, preferably lithium, sodium and potassium, of the alkaline earth metals, preferably calcium, magnesium and barium, and of the transition metals, preferably manganese, copper, zinc and iron, and also ammonium (NhV) and substituted ammonium in which one to four of the hydrogen atoms are replaced by Ci-C4-alkyl, C1-C4- hydroxyalkyl, Ci-C4-alkoxy, Ci-C4-alkoxy-Ci-C4-alkyl, hydroxy-Ci-C4-alkoxy-Ci-C4-alkyl, phenyl or benzyl. Examples of substituted ammonium ions comprise methylammonium, isoprop- ylammonium, dimethylammonium, diisopropylammonium, trimethylammonium, tetrame- thylammonium, tetraethylammonium, tetrabutylammonium, 2-hydroxyethylammonium, 2-(2- hydroxyethoxy)ethylammonium, bis(2-hydroxyethyl)ammonium, benzyltrimethylammonium and benzl-triethylammonium, furthermore phosphonium ions, sulfonium ions, preferably tri(Ci-C4- alkyl)sulfonium, and sulfoxonium ions, preferably tri(Ci-C4-alkyl)sulfoxonium.

Anions of useful acid addition salts are primarily chloride, bromide, fluoride, hydrogensul- fate, sulfate, dihydrogenphosphate, hydrogenphosphate, phosphate, nitrate, bicarbonate, carbonate, hexafluorosilicate, hexafluorophosphate, benzoate, and the anions of Ci-C4-alkanoic acids, preferably formate, acetate, propionate and butyrate. They can be formed by reacting compounds of the present invention with an acid of the corresponding anion, preferably with hydrochloric acid, hydrobromic acid, sulfuric acid, phosphoric acid or nitric acid.

The term "undesired vegetation" ("weeds") is understood to include any vegetation growing in non-crop-areas or at a crop plant site or locus of seeded and otherwise desired crop, where the vegetation is any plant species, including their germinant seeds, emerging seedlings and established vegetation, other than the seeded or desired crop (if any). Weeds, in the broadest sense, are plants considered undesirable in a particular location.

The organic moieties mentioned in the above definitions of the variables are - like the term halogen - collective terms for individual listings of the individual group members. The prefix C _n - Cm indicates in each case the possible number of carbon atoms in the group.

The term "halogen" denotes in each case fluorine, bromine, chlorine or iodine, in particular fluorine, chlorine or bromine. The term "partially or completely halogenated" will be taken to mean that 1 or more, e.g. 1 , 2, 3, 4 or 5 or all of the hydrogen atoms of a given radical have been replaced by a halogen atom, in particular by fluorine or chlorine. A partially or completely halogenated radical is termed below also "halo-radical". For example, partially or completely halogenated alkyl is also termed haloalkyl.

The term "alkyl" as used herein (and in the alkyl moieties of other groups comprising an alkyl group, e.g. alkoxy, alkylamino, alkylcarbonyl, alkoxycarbonyl, alkylthio, alkylsulfonyl and alkoxyalkyi) denotes in each case a straight-chain or branched alkyl group having usually from 1 to 10 carbon atoms, frequently from 1 to 6 carbon atoms, preferably 1 to 4 carbon atoms and in particular from 1 to 3 carbon atoms. Examples of Ci-C4-alkyl are methyl, ethyl, n-propyl, iso- propyl, n-butyl, 2-butyl (sec-butyl), isobutyl and tert-butyl. Examples for Ci-C6-alkyl are, apart those mentioned for Ci-C4-alkyl, n-pentyl, 1 -methylbutyl, 2-methylbutyl, 3-methylbutyl, 2,2- dimethylpropyl, 1 -ethylpropyl, n-hexyl, 1 ,1 -dimethylpropyl, 1 ,2-dimethylpropyl, 1 -methylpentyl, 2- methylpentyl, 3-methylpentyl, 4-methylpentyl, 1 ,1 -dimethylbutyl, 1 ,2-dimethylbutyl, 1 ,3- dimethylbutyl, 2,2-dimethylbutyl, 2,3-dimethylbutyl, 3,3-dimethylbutyl, 1 -ethylbutyl, 2-ethylbutyl,

1 .1 .2- trimethylpropyl, 1 ,2,2-trimethylpropyl, 1 -ethyl-1 -methylpropyl and 1 -ethyl-2-methylpropyl. Examples for Ci-Cio-alkyl are, apart those mentioned for Ci-C6-alkyl, n-heptyl, 1 -methylhexyl, 2- methylhexyl, 3-methylhexyl, 4-methylhexyl, 5-methylhexyl, 1 -ethylpentyl, 2-ethylpentyl, 3- ethylpentyl, n-octyl, 1 -methyloctyl, 2-methylheptyl, 1 -ethylhexyl, 2-ethylhexyl, 1 ,2-dimethylhexyl, 1 -propylpentyl, 2-propylpentyl, nonyl, decyl, 2-propylheptyl and 3-propylheptyl.

The term "alkylene" (or alkanediyl) as used herein in each case denotes an alkyl radical as defined above, wherein one hydrogen atom at any position of the carbon backbone is replaced by one further binding site, thus forming a bivalent moiety.

The term "haloalkyl" as used herein (and in the haloalkyl moieties of other groups com- prising a haloalkyl group, e.g. haloalkoxy, haloalkylthio, haloalkylcarbonyl, haloalkylsulfonyl and haloalkylsulfinyl) denotes in each case a straight-chain or branched alkyl group having usually from 1 to 8 carbon atoms ("Ci-Cs-haloalkyl"), frequently from 1 to 6 carbon atoms ("C1-C6- haloalkyl"), more frequently 1 to 4 carbon atoms ("Ci-C4-haloalkyl"), wherein the hydrogen atoms of this group are partially or totally replaced with halogen atoms. Preferred haloalkyl moie- ties are selected from Ci-C4-haloalkyl, more preferably from Ci-C2-haloalkyl, more preferably from halomethyl, in particular from Ci-C2-fluoroalkyl. Halomethyl is methyl in which 1 , 2 or 3 of the hydrogen atoms are replaced by halogen atoms. Examples are bromomethyl, chloromethyl, dichloromethyl, trichloromethyl, fluoromethyl, difluoromethyl, trifluoromethyl, chlorofluoromethyl, dichlorofluoromethyl, chlorodifluoromethyl and the like. Examples for Ci-C2-fluoroalkyl are fluo- romethyl, difluoromethyl, trifluoromethyl, 1 -fluoroethyl, 2-fluoroethyl, 2,2-difluoroethyl, 2,2,2- trifluoroethyl, pentafluoroethyl, and the like. Examples for Ci-C2-haloalkyl are, apart those mentioned for Ci-C2-fluoroalkyl, chloromethyl, dichloromethyl, trichloromethyl, bromomethyl, chlorofluoromethyl, dichlorofluoromethyl, chlorodifluoromethyl, 1 -chloroethyl, 2-chloroethyl, 2,2,- dichloroethyl, 2,2,2-trichloroethyl, 2-chloro-2-fluoroethyl, 2-chloro-2,2-difluoroethyl, 2,2-dichloro- 2-fluoroethyl, 1 -bromoethyl, and the like. Examples for Ci-C4-haloalkyl are, apart those mentioned for Ci-C2-haloalkyl, 1 -fluoropropyl, 2-fluoropropyl, 3-fluoropropyl, 3,3-difluoropropyl,

3.3.3- trifluoropropyl, heptafluoropropyl, 1 ,1 ,1 -trif I uoroprop-2-yl , 3-chloropropyl, 4-chlorobutyl and the like.

The term "cycloalkyi" as used herein (and in the cycloalkyi moieties of other groups comprising a cycloalkyi group, e.g. cycloalkoxy and cycloalkylalkyi) denotes in each case a mono- or bicyclic cycloaliphatic radical having usually from 3 to 10 carbon atoms ("C3-Cio-cycloalkyl"), preferably 3 to 7 carbon atoms ("C3-C7-cycloalkyl") or in particular 3 to 6 carbon atoms ("C3-C6- cycloalkyl"). Examples of monocyclic radicals having 3 to 6 carbon atoms comprise cyclopropyl, cyclobutyl, cyclopentyl and cyclohexyl. Examples of monocyclic radicals having 3 to 7 carbon atoms comprise cyclopropyl, cyclobutyl, cyclopentyl, cyclohexyl and cycloheptyl. Examples of bicyclic radicals having 7 or 8 carbon atoms comprise bicyclo[2.1.1]hexyl, bicyclo[2.2.1]heptyl, bicyclo[3.1.1]heptyl, bicyclo[2.2.1]heptyl, bicyclo[2.2.2]octyl and bicyclo[3.2.1]octyl.

The term "halocycloalkyl" as used herein (and in the halocycloalkyl moieties of other groups comprising an halocycloalkyl group, e.g. halocycloalkylmethyl) denotes in each case a mono- or bicyclic cycloaliphatic radical having usually from 3 to 10 carbon atoms, preferably 3 to 7 carbon atoms or in particular 3 to 6 carbon atoms, wherein at least one, e.g. 1 , 2, 3, 4 or 5 of the hydrogen atoms are replaced by halogen, in particular by fluorine or chlorine. Examples are

1 - and 2- fluorocyclopropyl, 1 ,2-, 2,2- and 2,3-difluorocyclopropyl, 1 ,2,2-trifluorocyclopropyl, 2,2,3,3-tetrafluorocyclpropyl, 1 - and 2-chlorocyclopropyl, 1 ,2-, 2,2- and 2,3-dichlorocyclopropyl, 1 ,2,2-trichlorocyclopropyl, 2,2,3,3-tetrachlorocyclpropyl, 1 -,2- and 3-fluorocyclopentyl, 1 ,2-, 2,2-, 2,3-, 3,3-, 3,4-, 2,5-difluorocyclopentyl, 1 -,2- and 3-chlorocyclopentyl, 1 ,2-, 2,2-, 2,3-, 3,3-, 3,4-, 2,5-dichlorocyclopentyl and the like.

The term "cycloalkyl-alkyl" used herein denotes a cycloalkyi group, as defined above, which is bound to the remainder of the molecule via an alkylene group. The term "C3-C7- cycloalkyl-Ci-C4-alkyl" refers to a C3-C7-cycloalkyl group as defined above which is bound to the remainder of the molecule via a Ci-C4-alkyl group, as defined above. Examples are cyclo- propylmethyl, cyclopropylethyl, cyclopropylpropyl, cyclobutylmethyl, cyclobutylethyl, cyclobu- tylpropyl, cyclopentylmethyl, cyclopentylethyl, cyclopentylpropyl, cyclohexylmethyl, cyclo- hexylethyl, cyclohexylpropyl, and the like.

The term "alkenyl" as used herein denotes in each case a monounsaturated straight-chain or branched hydrocarbon radical having usually 2 to 8 ("C2-C8-alkenyl"), preferably 2 to 6 carbon atoms ("C2-C6-alkenyl"), in particular 2 to 4 carbon atoms ("C2-C4-alkenyl"), and a double bond in any position, for example C2-C4-alkenyl, such as ethenyl, 1 -propenyl, 2-propenyl, 1 - methylethenyl, 1 -butenyl, 2-butenyl, 3-butenyl, 1 -methyl-1 -propenyl, 2-methyl-1 -propenyl, 1 - methyl-2-propenyl or 2-methyl-2-propenyl; C2-C6-alkenyl, such as ethenyl, 1 -propenyl, 2- propenyl, 1 -methylethenyl, 1 -butenyl, 2-butenyl, 3-butenyl, 1 -methyl-1 -propenyl, 2-methyl-1 - propenyl, 1 -methyl-2-propenyl, 2-methyl-2-propenyl, 1 -pentenyl, 2-pentenyl, 3-pentenyl, 4- pentenyl, 1 -methyl-1 -butenyl, 2-methyl-1 -butenyl, 3-methyl-1 -butenyl, 1 -methyl-2-butenyl,

2- methyl-2-butenyl, 3-methyl-2-butenyl, 1 -methyl-3-butenyl, 2-methyl-3-butenyl, 3-methyl-3- butenyl, 1 ,1 -dimethyl-2-propenyl, 1 ,2-dimethyl-1 -propenyl, 1 ,2-dimethyl-2-propenyl, 1 -ethyl-1 - propenyl, 1 -ethyl-2-propenyl, 1 -hexenyl, 2-hexenyl, 3-hexenyl, 4-hexenyl, 5-hexenyl, 1 -methyl-1 - pentenyl, 2-methyl-1 -pentenyl, 3-methyl-1 -pentenyl, 4-methyl-1 -pentenyl, 1 -methyl-2-pentenyl,

2- methyl-2-pentenyl, 3-methyl-2-pentenyl, 4-methyl-2-pentenyl, 1 -methyl-3-pentenyl, 2-methyl-

3- pentenyl, 3-methyl-3-pentenyl, 4-methyl-3-pentenyl, 1 -methyl-4-pentenyl, 2-methyl-4-pentenyl, 3-methyl-4-pentenyl, 4-methyl-4-pentenyl, 1 ,1 -dimethyl-2-butenyl, 1 ,1 -dimethyl-3-butenyl,

1 .2- dimethyl-1 -butenyl, 1 ,2-dimethyl-2-butenyl, 1 ,2-dimethyl-3-butenyl, 1 ,3-dimethyl-1 -butenyl,

1 .3- dimethyl-2-butenyl, 1 ,3-dimethyl-3-butenyl, 2,2-dimethyl-3-butenyl, 2,3-dimethyl-1 -butenyl, 2,3-dimethyl-2-butenyl, 2,3-dimethyl-3-butenyl, 3,3-dimethyl-1 -butenyl, 3,3-dimethyl-2-butenyl, 1 -ethyl-1 -butenyl, 1 -ethyl-2-butenyl, 1 -ethyl-3-butenyl, 2-ethyl-1 -butenyl, 2-ethyl-2-butenyl, 2- ethyl-3-butenyl, 1 ,1 ,2-trimethyl-2-propenyl, 1 -ethyl-1 -methyl-2-propenyl, 1 -ethyl-2-methyl-1 - propenyl, 1 -ethyl-2-methyl-2-propenyl and the like, or C2-C8-alkenyl, such as the radicals mentioned for C2-C6-alkenyl and additionally 1 -heptenyl, 2-heptenyl, 3-heptenyl, 1 -octenyl, 2-octenyl, 3-octenyl, 4-octenyl and the positional isomers thereof.

The term "haloalkenyl" as used herein, which may also be expressed as "alkenyl which is substituted by halogen", and the haloalkenyl moieties in haloalkenyloxy and the like refers to unsaturated straight-chain or branched hydrocarbon radicals having 2 to 8 ("C2-C8-haloalkenyl") or 2 to 6 ("C2-C6-haloalkenyl") or 2 to 4 ("C2-C4-haloalkenyl") carbon atoms and a double bond in any position, where some or all of the hydrogen atoms in these groups are replaced by halogen atoms as mentioned above, in particular fluorine, chlorine and bromine, for example chlorovinyl, chloroallyl and the like.

The term "alkynyl" as used herein denotes unsaturated straight-chain or branched hydrocarbon radicals having usually 2 to 8 ("C2-C8-alkynyl"), frequently 2 to 6 ("C2-C6-alkynyl"), preferably 2 to 4 carbon atoms ("C2-C4-alkynyl") and a triple bond in any position, for example C2- C4-alkynyl, such as ethynyl, 1 -propynyl, 2-propynyl, 1 -butynyl, 2-butynyl, 3-butynyl, 1 -methyl-2- propynyl and the like, C2-C6-alkynyl, such as ethynyl, 1 -propynyl, 2-propynyl, 1 -butynyl, 2- butynyl, 3-butynyl, 1 -methyl-2-propynyl, 1 -pentynyl, 2-pentynyl, 3-pentynyl, 4-pentynyl, 1 - methyl-2-butynyl, 1 -methyl-3-butynyl, 2-methyl-3-butynyl, 3-methyl-1 -butynyl, 1 ,1 -dimethyl-2- propynyl, 1 -ethyl-2-propynyl, 1 -hexynyl, 2-hexynyl, 3-hexynyl, 4-hexynyl, 5-hexynyl, 1 -methyl-2- pentynyl, 1 -methyl-3-pentynyl, 1 -methyl-4-pentynyl, 2-methyl-3-pentynyl, 2-methyl-4-pentynyl, 3- methyl-1 -pentynyl, 3-methyl-4-pentynyl, 4-methyl-1 -pentynyl, 4-methyl-2-pentynyl, 1 ,1 -dimethyl- 2-butynyl, 1 ,1 -dimethyl-3-butynyl, 1 ,2-dimethyl-3-butynyl, 2,2-dimethyl-3-butynyl, 3,3-dimethyl-1 - butynyl, 1 -ethyl-2-butynyl, 1 -ethyl-3-butynyl, 2-ethyl-3-butynyl, 1 -ethyl-1 -methyl-2-propynyl and the like.

The term "haloalkynyl" as used herein, which is also expressed as "alkynyl which is substituted by halogen", refers to unsaturated straight-chain or branched hydrocarbon radicals having usually 2 to 8 carbon atoms ("C2-C8-haloalkynyl"), frequently 2 to 6 ("C2-C6-haloalkynyl"), preferabyl 2 to 4 carbon atoms ("C2-C4-haloalkynyl"), and a triple bond in any position (as mentioned above), where some or all of the hydrogen atoms in these groups are replaced by halo- gen atoms as mentioned above, in particular fluorine, chlorine and bromine.

The term "alkoxy" as used herein denotes in each case a straight-chain or branched alkyl group usually having from 1 to 8 carbon atoms ("d-Cs-alkoxy"), frequently from 1 to 6 carbon atoms ("Ci-C6-alkoxy"), preferably 1 to 4 carbon atoms ("Ci-C4-alkoxy"), which is bound to the remainder of the molecule via an oxygen atom. Ci-C2-Alkoxy is methoxy or ethoxy. C1-C4- Alkoxy is additionally, for example, n-propoxy, 1 -methylethoxy (isopropoxy), butoxy,

1 -methylpropoxy (sec-butoxy), 2-methylpropoxy (isobutoxy) or 1 ,1 -dimethylethoxy (tert-butoxy). Ci-C6-Alkoxy is additionally, for example, pentoxy, 1 -methylbutoxy, 2-methylbutoxy, 3- methylbutoxy, 1 ,1 -dimethylpropoxy, 1 ,2-dimethylpropoxy, 2,2-dimethylpropoxy, 1 -ethylpropoxy, hexoxy, 1 -methylpentoxy, 2-methylpentoxy, 3-methylpentoxy, 4-methylpentoxy, 1 ,1 - dimethylbutoxy, 1 ,2-dimethylbutoxy, 1 ,3-dimethylbutoxy, 2,2-dimethylbutoxy, 2,3- dimethylbutoxy, 3,3-dimethylbutoxy, 1 -ethylbutoxy, 2-ethylbutoxy, 1 ,1 ,2-trimethylpropoxy, 1 ,2,2- trimethylpropoxy, 1 -ethyl-1 -methylpropoxy or 1 -ethyl-2-methylpropoxy. Ci-Cs-Alkoxy is additionally, for example, heptyloxy, octyloxy, 2-ethylhexyloxy and positional isomers thereof.

The term "haloalkoxy" as used herein denotes in each case a straight-chain or branched alkoxy group, as defined above, having from 1 to 8 carbon atoms ("Ci-Cs-haloalkoxy"), frequently from 1 to 6 carbon atoms ("Ci-C6-haloalkoxy"), preferably 1 to 4 carbon atoms ("C1-C4- haloalkoxy"), more preferably 1 to 3 carbon atoms ("Ci-C3-haloalkoxy"), wherein the hydrogen atoms of this group are partially or totally replaced with halogen atoms, in particular fluorine atoms. Ci-C ₂ -Haloalkoxy is, for example, OCH ₂ F, OCHF ₂ , OCF ₃ , OCH2CI, OCHC , OCCI ₃ , chlorofluoromethoxy, dichlorofluoromethoxy, chlorodifluoromethoxy, 2-fluoroethoxy, 2- chloroethoxy, 2-bromoethoxy, 2-iodoethoxy, 2,2-difluoroethoxy, 2,2,2-trifluoroethoxy, 2-chloro-2- fluoroethoxy, 2-chloro-2,2-difluoroethoxy, 2,2-dichloro-2-fluoroethoxy, 2,2,2-trichloroethoxy or OC2F5. Ci-C4-Haloalkoxy is additionally, for example, 2-fluoropropoxy, 3-fluoropropoxy, 2,2- difluoropropoxy, 2,3-difluoropropoxy, 2-chloropropoxy, 3-chloropropoxy, 2,3-dichloropropoxy, 2- bromopropoxy, 3-bromopropoxy, 3,3,3-trifluoropropoxy, 3,3,3-trichloropropoxy, OCH2-C2F5, OCF2-C2F5, 1 -(CH ₂ F)-2-fluoroethoxy, 1 -(CH ₂ CI)-2-chloroethoxy, 1 -(CH ₂ Br)-2-bromoethoxy, 4-fluorobutoxy, 4-chlorobutoxy, 4-bromobutoxy or nonafluorobutoxy. Ci-C6-Haloalkoxy is additionally, for example, 5-fluoropentoxy, 5-chloropentoxy, 5-brompentoxy, 5-iodopentoxy, unde- cafluoropentoxy, 6-fluorohexoxy, 6-chlorohexoxy, 6-bromohexoxy, 6-iodohexoxy or dodecafluo- rohexoxy.

The term "alkoxyalkyl" as used herein denotes in each case alkyl usually comprising 1 to 6 carbon atoms, preferably 1 to 4 carbon atoms, wherein 1 carbon atom carries an alkoxy radical usually comprising 1 to 8, frequently 1 to 6, in particular 1 to 4, carbon atoms as defined above. "Ci-C6-alkoxy-Ci-C6-alkyl" is a Ci-C6-alkyl group, as defined above, in which one hydrogen atom is replaced by a Ci-C6-alkoxy group, as defined above. Examples are CH2OCH3, CH2-OC2H5, n-propoxymethyl, CH2-OCH(CH3)2, n-butoxymethyl, (l -methylpropoxy)-methyl, (2- methylpropoxy)methyl, CH2-OC(CH3)3, 2-(methoxy)ethyl, 2-(ethoxy)ethyl, 2-(n-propoxy)-ethyl, 2- (1 -methylethoxy)-ethyl, 2-(n-butoxy)ethyl, 2-(1 -methylpropoxy)-ethyl, 2-(2-methylpropoxy)-ethyl, 2-(1 ,1 -dimethylethoxy)-ethyl, 2-(methoxy)-propyl, 2-(ethoxy)-propyl, 2-(n-propoxy)-propyl, 2-(1 - methylethoxy)-propyl, 2-(n-butoxy)-propyl, 2-(1 -methylpropoxy)-propyl, 2-(2-methylpropoxy)- propyl, 2-(1 ,1 -dimethylethoxy)-propyl, 3-(methoxy)-propyl, 3-(ethoxy)-propyl, 3-(n-propoxy)- propyl, 3-(1 -methylethoxy)-propyl, 3-(n-butoxy)-propyl, 3-(1 -methylpropoxy)-propyl, 3-(2- methylpropoxy)-propyl, 3-(1 ,1 -dimethylethoxy)-propyl, 2-(methoxy)-butyl, 2-(ethoxy)-butyl, 2-(n- propoxy)-butyl, 2-(1 -methylethoxy)-butyl, 2-(n-butoxy)-butyl, 2-(1 -methylpropoxy)-butyl, 2-(2- methyl-propoxy)-butyl, 2-(1 ,1 -dimethylethoxy)-butyl, 3-(methoxy)-butyl, 3-(ethoxy)-butyl, 3-(n- propoxy)-butyl, 3-(1 -methylethoxy)-butyl, 3-(n-butoxy)-butyl, 3-(1 -methylpropoxy)-butyl, 3-(2- methylpropoxy)-butyl, 3-(1 ,1 -dimethylethoxy)-butyl, 4-(methoxy)-butyl, 4-(ethoxy)-butyl, 4-(n- propoxy)-butyl, 4-(1 -methylethoxy)-butyl, 4-(n-butoxy)-butyl, 4-(1 -methylpropoxy)-butyl, 4-(2- methylpropoxy)-butyl, 4-(1 ,1 -dimethylethoxy)-butyl and the like. The term "haloalkoxy-alkyl" as used herein denotes in each case alkyl as defined above, usually comprising 1 to 6 carbon atoms, preferably 1 to 4 carbon atoms, wherein 1 carbon atom carries an haloalkoxy radical as defined above, usually comprising 1 to 8, frequently 1 to 6, in particular 1 to 4, carbon atoms as defined above. Examples are fluoromethoxymethyl, difluoro- methoxymethyl, trifluoromethoxymethyl, 1 -fluoroethoxymethyl, 2-fluoroethoxymethyl, 1 ,1 - difluoroethoxymethyl, 1 ,2-difluoroethoxymethyl, 2,2-difluoroethoxymethyl, 1 ,1 ,2- trifluoroethoxymethyl, 1 ,2,2-trifluoroethoxymethyl, 2,2,2-trifluoroethoxymethyl, pentafluoroethox- ymethyl, 1 -fluoroethoxy-1 -ethyl, 2-fluoroethoxy-1 -ethyl, 1 ,1 -difluoroethoxy-1 -ethyl, 1 ,2- difluoroethoxy-1 -ethyl, 2,2-difluoroethoxy-1 -ethyl, 1 ,1 ,2-trifluoroethoxy-1 -ethyl, 1 ,2,2- trifluoroethoxy-1 -ethyl, 2,2,2-trifluoroethoxy-1 -ethyl, pentafluoroethoxy-1 -ethyl, 1 -fluoroethoxy-2- ethyl, 2-fluoroethoxy-2-ethyl, 1 ,1 -difluoroethoxy-2 -ethyl, 1 ,2-difluoroethoxy-2-ethyl, 2,2- difluoroethoxy-2-ethyl, 1 ,1 ,2-trifluoroethoxy-2-ethyl, 1 ,2,2-trifluoroethoxy-2-ethyl, 2,2,2- trifluoroethoxy-2-ethyl, pentafluoroethoxy-2-ethyl, and the like.

The term "alkylthio" (also alkylsulfanyl, "alkyl-S" or "alkyl-S(0) _k " (wherein k is 0)) as used herein denotes in each case a straight-chain or branched saturated alkyl group as defined above, usually comprising 1 to 8 carbon atoms ("Ci-Cs-alkylthio"), frequently comprising 1 to 6 carbon atoms ("Ci-C6-alkylthio"), preferably 1 to 4 carbon atoms ("Ci-C4-alkylthio"), which is attached via a sulfur atom at any position in the alkyl group. Ci-C2-Alkylthio is methylthio or ethylthio. Ci-C4-Alkylthio is additionally, for example, n-propylthio, 1 -methylethylthio (iso- propylthio), butylthio, 1 -methylpropylthio (sec-butylthio), 2-methylpropylthio (isobutylthio) or 1 ,1 - dimethylethylthio (tert-butylthio). Ci-C6-Alkylthio is additionally, for example, pentylthio, 1 - methylbutylthio, 2-methylbutylthio, 3-methylbutylthio, 1 ,1 -dimethylpropylthio, 1 ,2- dimethylpropylthio, 2,2-dimethylpropylthio, 1 -ethylpropylthio, hexylthio, 1 -methylpentylthio, 2- methylpentylthio, 3-methylpentylthio, 4-methylpentylthio, 1 ,1 -dimethylbutylthio, 1 ,2- dimethylbutylthio, 1 ,3-dimethylbutylthio, 2,2-dimethylbutylthio, 2,3-dimethylbutylthio,

3,3-dimethylbutylthio, 1 -ethylbutylthio, 2-ethylbutylthio, 1 ,1 ,2-trimethylpropylthio, 1 ,2,2- trimethylpropylthio, 1 -ethyl-1 -methylpropylthio or 1-ethyl-2-methylpropylthio. Ci-Cs-Alkylthio is additionally, for example, heptylthio, octylthio, 2-ethylhexylthio and positional isomers thereof.

The term "haloalkylthio" as used herein refers to an alkylthio group as defined above wherein the hydrogen atoms are partially or completely substituted by fluorine, chlorine, bromine and/or iodine. Ci-C ₂ -Haloalkylthio is, for example, SCH ₂ F, SCHF ₂ , SCF ₃ , SCH ₂ CI, SCHCI ₂ , SCC , chlorofluoromethylthio, dichlorofluoromethylthio, chlorodifluoromethylthio, 2- fluoroethylthio, 2-chloroethylthio, 2-bromoethylthio, 2-iodoethylthio, 2,2-difluoroethylthio, 2,2,2- trifluoroethylthio, 2-chloro-2-fluoroethylthio, 2-chloro-2,2-difluoroethylthio, 2,2-dichloro-2- fluoroethylthio, 2,2,2-trichloroethylthio or SC ₂ F ₅ . Ci-C4-Haloalkylthio is additionally, for example, 2-fluoropropylthio, 3-fluoropropylthio, 2,2-difluoropropylthio, 2,3-difluoropropylthio,

2- chloropropylthio, 3-chloropropylthio, 2,3-dichloropropylthio, 2-bromopropylthio,

3- bromopropylthio, 3,3,3-trifluoropropylthio, 3,3,3-trichloropropylthio, SCH ₂ -C ₂ F ₅ , SCF ₂ -C ₂ F ₅ , 1 - (CH ₂ F)-2-fluoroethylthio, 1 -(CH ₂ CI)-2-chloroethylthio, 1 -(CH ₂ Br)-2-bromoethylthio,

4-fluorobutylthio, 4-chlorobutylthio, 4-bromobutylthio or nonafluorobutylthio. Ci-C6-Haloalkylthio is additionally, for example, 5-fluoropentylthio, 5-chloropentylthio, 5-brompentylthio, 5- iodopentylthio, undecafluoropentylthio, 6-fluorohexylthio, 6-chlorohexylthio, 6-bromohexylthio,

6- iodohexylthio or dodecafluorohexylthio.

The terms "alkylsulfinyl" and "alkyl-S(0)k" (wherein k is 1 ) are equivalent and, as used herein, denote an alkyl group, as defined above, attached via a sulfinyl [S(O)] group. For exam- pie, the term "Ci-C2-a I kylsu If i nyl " refers to a Ci-C2-alkyl group, as defined above, attached via a sulfinyl [S(O)] group. The term "Ci-C4-alkylsulfinyl" refers to a Ci-C4-alkyl group, as defined above, attached via a sulfinyl [S(O)] group. The term "Ci-C6-alkylsulfinyl" refers to a Ci-C6-alkyl group, as defined above, attached via a sulfinyl [S(O)] group. Ci-C2-alkylsulfinyl is methylsulfinyl or ethylsulfinyl. Ci-C4-alkylsulfinyl is additionally, for example, n-propylsulfinyl,

1 -methylethylsulfinyl (isopropylsulfinyl), butylsulfinyl, 1 -methylpropylsulfinyl (sec-butylsulfinyl), 2- methylpropylsulfinyl (isobutylsulfinyl) or 1 ,1 -dimethylethylsulfinyl (tert-butylsulfinyl). C1-C6- alkylsulfinyl is additionally, for example, pentylsulfinyl, 1 -methylbutylsulfinyl, 2- methylbutylsulfinyl, 3-methylbutylsulfinyl, 1 ,1 -dimethylpropylsulfinyl, 1 ,2-dimethylpropylsulfinyl, 2,2-dimethylpropylsulfinyl, 1 -ethylpropylsulfinyl, hexylsulfinyl, 1 -methylpentylsulfinyl, 2- methylpentylsulfinyl, 3-methylpentylsulfinyl, 4-methylpentylsulfinyl, 1 ,1 -dimethylbutylsulfinyl,

1 .2- dimethylbutylsulfinyl, 1 ,3-dimethylbutylsulfinyl, 2,2-dimethylbutylsulfinyl,

2.3- dimethylbutylsulfinyl, 3,3-dimethylbutylsulfinyl, 1 -ethylbutylsulf inyl , 2-ethylbutylsulfinyl, 1 ,1 ,2- trimethylpropylsulfinyl, 1 ,2,2-trimethylpropylsulfinyl, 1 -ethyl-1 -methylpropylsulfinyl or 1 -ethyl-2- methylpropylsulfinyl.

The terms "alkylsulfonyl" and "alkyl-S(0)k" (wherein k is 2) are equivalent and, as used herein, denote an alkyl group, as defined above, attached via a sulfonyl [S(0)2] group. The term "Ci-C2-alkylsulfonyl" refers to a Ci-C2-alkyl group, as defined above, attached via a sulfonyl [S(0)2] group. The term "Ci-C4-alkylsulfonyl" refers to a Ci-C4-alkyl group, as defined above, attached via a sulfonyl [S(0)2] group. The term "Ci-C6-alkylsulfonyl" refers to a Ci-C6-alkyl group, as defined above, attached via a sulfonyl [S(0)2] group. Ci-C2-alkylsulfonyl is methyl- sulfonyl or ethylsulfonyl. Ci-C4-alkylsulfonyl is additionally, for example, n-propylsulfonyl, 1 -methylethylsulfonyl (isopropylsulfonyl), butylsulfonyl, 1 -methylpropylsulfonyl (sec- butylsulfonyl), 2-methylpropylsulfonyl (isobutylsulfonyl) or 1 ,1 -dimethylethylsulfonyl (tert- butylsulfonyl). Ci-C6-alkylsulfonyl is additionally, for example, pentylsulfonyl,

1 -methylbutylsulfonyl, 2-methylbutylsulfonyl, 3-methylbutylsulfonyl, 1 ,1 -dimethylpropylsulfonyl, 1 ,2-dimethylpropylsulfonyl, 2,2-dimethylpropylsulfonyl, 1 -ethylpropylsulfonyl, hexylsulfonyl, 1 - methylpentylsulfonyl, 2-methylpentylsulfonyl, 3-methylpentylsulfonyl, 4-methylpentylsulfonyl,

1 .1 - dimethylbutylsulfonyl, 1 ,2-dimethylbutylsulfonyl, 1 ,3-dimethylbutylsulfonyl,

2.2- dimethylbutylsulfonyl, 2,3-dimethylbutylsulfonyl, 3,3-dimethylbutylsulfonyl,

1 -ethylbutylsulfonyl, 2-ethylbutylsulfonyl, 1 ,1 ,2-trimethylpropylsulfonyl,

1 ,2,2-trimethylpropylsulfonyl, 1 -ethyl-1 -methylpropylsulfonyl or 1 -ethyl-2-methylpropylsulfonyl.

The term "alkylamino" as used herein denotes in each case a group R ^* HN-, wherein R ^* is a straight-chain or branched alkyl group usually having from 1 to 6 carbon atoms ("Ci-Ce- alkylamino"), preferably 1 to 4 carbon atoms("Ci-C4-alkylamino"). Examples of Ci-C6-alkylamino are methylamino, ethylamino, n-propylamino, isopropylamino, n-butylamino, 2-butylamino, iso- butylamino, tert-butylamino, and the like.

The term "dialkylamino" as used herein denotes in each case a group R ^* R°N-, wherein R ^* and R°, independently of each other, are a straight-chain or branched alkyl group each usually having from 1 to 6 carbon atoms ("di-(Ci-C6-alkyl)-amino"), preferably 1 to 4 carbon atoms ("di- (Ci-C4-alkyl)-amino"). Examples of a di-(Ci-C6-alkyl)-amino group are dimethylamino, diethyla- mino, dipropylamino, dibutylamino, methyl-ethyl-amino, methyl-propyl-amino, methyl- isopropylamino, methyl-butyl-amino, methyl-isobutyl-amino, ethyl-propyl-amino, ethyl- isopropylamino, ethyl-butyl-amino, ethyl-isobutyl-amino, and the like.

The suffix "-carbonyl" in a group denotes in each case that the group is bound to the remainder of the molecule via a carbonyl C=0 group. This is the case e.g. in alkylcarbonyl, haloalkylcarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoxycarbonyl, haloalkoxycarbonyl.

The term "aryl" as used herein refers to a mono-, bi- or tricyclic aromatic hydrocarbon radical such as phenyl or naphthyl, in particular phenyl.

The term "het(ero)aryl" as used herein refers to a mono-, bi- or tricyclic heteroaromatic hydrocarbon radical, preferably to a monocyclic heteroaromatic radical, such as pyridyl, pyrim- idyl and the like.

The term "3-, 4-, 5- or 6-membered monocyclic or 8-, 9- or 10-membered bicyclic saturated, unsaturated or aromatic heterocyde containing 1 , 2, 3 or 4 heteroatoms as ring members selected from the groups consisting of N, O and S" as used herein denotes monocyclic or bicyclic radicals, the monocyclic or bicyclic radicals being saturated, unsaturated or aromatic where N can optionally be oxidized, i.e. in the form of an N-oxide, and S can also optionally be oxidized to various oxidation states, i.e. as SO or SO2. An unsaturated heterocyde contains at least one C-C and/or C-N and/or N-N double bond(s). A fully unsaturated heterocyde contains as many conjugated C-C and/or C-N and/or N-N double bonds as allowed by the size(s) of the ring(s). An aromatic monocyclic heterocyde is a fully unsaturated 5- or 6-membered monocyclic heterocyde. An aromatic bicyclic heterocyde is an 8-, 9- or 10-membered bicyclic heterocyde consisting of a 5- or 6-membered heteroaromatic ring which is fused to a phenyl ring or to another 5- or 6-membered heteroaromatic ring. The heterocyde may be attached to the remainder of the molecule via a carbon ring member or via a nitrogen ring member. As a matter of course, the heterocyclic ring contains at least one carbon ring atom. If the ring contains more than one O ring atom, these are not adjacent.

Examples of a 3-, 4-, 5- or 6-membered monocyclic saturated heterocyde include:

oxirane-2-yl, aziridine-1 -yl, aziridine-2-yl, oxetan-2-yl, azetidine-1 -yl, azetidine-2-yl, azetidine-3- yl, thietane-1 -yl, thietan-2-yl, thietane-3-yl, tetrahydrofuran-2-yl, tetrahydrofuran-3-yl, tetrahy- drothien-2-yl, tetrahydrothien-3-yl, pyrrolidin-1 -yl, pyrrolidin-2-yl, pyrrolidin-3-yl, pyrazolidin-1 -yl, pyrazolidin-3-yl, pyrazolidin-4-yl, pyrazolidin-5-yl, imidazolidin-1 -yl, imidazolidin-2-yl, imidazoli- din-4-yl, oxazolidin-2-yl, oxazolidin-3-yl, oxazolidin-4-yl, oxazolidin-5-yl, isoxazolidin-2-yl, isoxa- zolidin-3-yl, isoxazolidin-4-yl, isoxazolidin-5-yl, thiazolidin-2-yl, thiazolidin-3-yl, thiazolidin-4-yl, thiazolidin-5-yl, isothiazolidin-2-yl, isothiazolidin-3-yl, isothiazolidin-4-yl, isothiazolidin-5-yl, 1 ,2,4- oxadiazolidin-3-yl, 1 ,2,4-oxadiazolidin-5-yl, 1 ,2,4-thiadiazolidin-3-yl, 1 ,2,4-thiadiazolidin-5-yl, 1 ,2,4-triazolidin-3-yl, 1 ,3,4-oxadiazolidin-2-yl, 1 ,3,4-thiadiazolidin-2-yl, 1 ,3,4-triazolidin-1 -yl,

1 ,3,4-triazolidin-2-yl, 2-tetrahydropyranyl, 4-tetrahydropyranyl, 1 ,3-dioxan-5-yl, 1 ,4-dioxan-2-yl, piperidin-1 -yl, piperidin-2-yl, piperidin-3-yl, piperidin-4-yl, hexahydropyridazin-3-yl, hexahydro- pyridazin-4-yl, hexahydropyrimidin-2-yl, hexahydropyrimidin-4-yl, hexahydropyrimidin-5-yl, pi- perazin-1 -yl, piperazin-2-yl, 1 ,3,5-hexahydrotriazin-1 -yl, 1 ,3,5-hexahydrotriazin-2-yl and

1 ,2,4-hexahydrotriazin-3-yl, morpholin-2-yl, morpholin-3-yl, morpholin-4-yl, thiomorpholin-2-yl, thiomorpholin-3-yl, thiomorpholin-4-yl, 1 -oxothiomorpholin-2-yl, 1 -oxothiomorpholin-3-yl, 1 - oxothiomorpholin-4-yl, 1 ,1 -dioxothiomorpholin-2-yl, 1 ,1 -dioxothiomorpholin-3-yl, 1 ,1 - dioxothiomorpholin-4-yl and the like.

Examples of a 5- or 6-membered monocyclic partially unsaturated heterocycle include: 2,3-dihydrofur-2-yl, 2,3-dihydrofur-3-yl, 2,4-dihydrofur-2-yl, 2,4-dihydrofur-3-yl, 2,3-dihydrothien- 2-yl, 2,3-dihydrothien-3-yl, 2,4-dihydrothien-2-yl, 2,4-dihydrothien-3-yl, 2-pyrrolin-2-yl, 2-pyrrolin- 3-yl, 3-pyrrolin-2-yl, 3-pyrrolin-3-yl, 2-isoxazolin-3-yl, 3-isoxazolin-3-yl, 4-isoxazolin-3-yl, 2- isoxazolin-4-yl, 3-isoxazolin-4-yl, 4-isoxazolin-4-yl, 2-isoxazolin-5-yl, 3-isoxazolin-5-yl, 4- isoxazolin-5-yl, 2-isothiazolin-3-yl, 3-isothiazolin-3-yl, 4-isothiazolin-3-yl, 2-isothiazolin-4-yl, 3- isothiazolin-4-yl, 4-isothiazolin-4-yl, 2-isothiazolin-5-yl, 3-isothiazolin-5-yl, 4-isothiazolin-5-yl, 2,3- dihydropyrazol-1 -yl, 2,3-dihydropyrazol-2-yl, 2,3-dihydropyrazol-3-yl, 2,3-dihydropyrazol-4-yl, 2,3-dihydropyrazol-5-yl, 3,4-dihydropyrazol-1 -yl, 3,4-dihydropyrazol-3-yl, 3,4-dihydropyrazol-4- yl, 3,4-dihydropyrazol-5-yl, 4,5-dihydropyrazol-1 -yl, 4,5-dihydropyrazol-3-yl, 4,5-dihydropyrazol- 4-yl, 4,5-dihydropyrazol-5-yl, 2,3-dihydrooxazol-2-yl, 2,3-dihydrooxazol-3-yl, 2,3-dihydrooxazol-

4- yl, 2,3-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4- yl, 3,4-dihydrooxazol-5-yl, 3,4-dihydrooxazol-2-yl, 3,4-dihydrooxazol-3-yl, 3,4-dihydrooxazol-4- yl, 2-, 3-, 4-, 5- or 6-di- or tetrahydropyridinyl, 3-di- or tetrahydropyridazinyl, 4-di- or tetrahydro- pyridazinyl, 2-di- or tetrahydropyrimidinyl, 4-di- or tetrahydropyrimidinyl, 5-di- or tetrahydropyrim- idinyl, di- or tetrahydropyrazinyl, 1 ,3, 5-di- or tetrahydrotriazin-2-yl and 1 ,2, 4-di- or tetrahydrotria- zin-3-yl.

A 5- or 6-membered monocyclic fully unsaturated (including aromatic) heterocyclic ring is e.g. a 5- or 6-membered monocyclic fully unsaturated (including aromatic) heterocyclic ring.

Examples are: 2-furyl, 3-furyl, 2-thienyl, 3-thienyl, 1 -pyrrolyl, 2-pyrrolyl, 3-pyrrolyl, 1-pyrazolyl, 3- pyrazolyl, 4-pyrazolyl, 5-pyrazolyl, 2-oxazolyl, 4-oxazolyl, 5-oxazolyl, 2-thiazolyl, 4-thiazolyl,

5- thiazolyl, 1 -imidazolyl, 2-imidazolyl, 4-imidazolyl, 1 ,3,4-triazol-1 -yl, 1 ,3,4-triazol-2-yl, 2- pyridinyl, 3-pyridinyl, 4-pyridinyl, 1 -oxopyridin-2-yl, 1 -oxopyridin-3-yl, 1 -oxopyridin-4-yl,3- pyridazinyl, 4-pyridazinyl, 2-pyrimidinyl, 4-pyrimidinyl, 5-pyrimidinyl and 2-pyrazinyl.

Examples of a 5- or 6-membered heteroaromatic ring fused to a phenyl ring or to a 5- or

6- membered heteroaromatic radical include benzofuranyl, benzothienyl, indolyl, indazolyl, ben- zimidazolyl, benzoxathiazolyl, benzoxadiazolyl, benzothiadiazolyl, benzoxazinyl, chinolinyl, iso- chinolinyl, purinyl, 1 ,8-naphthyridyl, pteridyl, pyrido[3,2-d]pyrimidyl or pyridoimidazolyl and the like.

If two radicals bound on the same nitrogen atom (for example R ^e and R ^f or R ^2e and R ^2f or R9 and R ^h or R¾ and R ^2h ) together with the nitrogen atom, to which they are bound, form a 5-, 6 or 7-membered, saturated or unsaturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N, this is for example pyrrolidine-1 -yl, pyrazolidin-1 -yl, imidazolidin-1 -yl, oxazolidin-3-yl, thiazolidin-3-yl, isoxazolidin-2-yl, isothiazolin- 2-yl, [1 ,2,3]-triazolidin-1 -yl, [1 ,2,3]-triazolidin-2-yl, [1 ,2,4]-triazolidin-1 -yl, [1 ,2,4]-triazolidin-4-yl, [1 ,2,3]-oxadiazolidin-2-yl, [1 ,2,3]-oxadiazolidin-3-yl, [1 ,2,5]-oxadiazolidin-2-yl, [1 ,2,4]- oxadiazolidin-2-yl, [1 ,2,4]-oxadiazolidin-4-yl, [1 ,3,4]-oxadiazolidin-3-yl, [1 ,2,3]-thiadiazolidin-2-yl, [1 ,2,3]- thiadiazolidin-3-yl, [1 ,2,5]-thiadiazolidin-2-yl, [1 ,2,4]-thiadiazolidin-2-yl, [1 ,2,4]- thiadiazolidin-4-yl, [1 ,3,4]-thiadiazolidin-3-yl, piperdin-1 -yl, piperazine-1 -yl, morpholin-1 -yl, thio- morpholin-1 -yl, 1 -oxothiomorpholin-1 -yl, 1 ,1 -dioxothiomorpholin-1 -yl, azepan-1 -yl, 1 ,4-diazepan- 1 -yl, pyrrolin-1 -yl, pyrazolin-1 -yl, imidazolin-1 -yl, oxazolin-3-yl, isoxazolin-2-yl, thiazolin-3-yl, isothiazolin-1 -yl, 1 ,2-dihydropyridin-1 -yl, 1 ,2,3,4-tetrahydropyridin-1 -yl, 1 ,2,5,6-tetrahydropyridin- 1 -yl, 1 ,2-dihydropyridazin, 1 ,6-dihydropyridazin, 1 ,2,3,4-tetrahydropyridazin-1 -yl, 1 ,2,5,6- tetrahydropyridazin-1 -yl, 1 ,2-dihydropyrimidin, 1 ,6-dihydropyrimidin, 1 ,2,3,4-tetrahydropyrimidin- 1 -yl, 1 ,2,5,6-tetrahydropyrimidin-1 -yl, 1 ,2-dihydropyrazin-1 -yl, 1 ,2,3,4-tetrahydropyrazin-1 -yl, 1 ,2,5,6-tetrahydropyrazin-1 -yl, pyrrol-1 -yl, pyrazol-1 -yl, imidazol-1 -yl, [1 ,2,3]-1 H-triazol-1 -yl, [1 ,2,3]-2H-triazol-2-yl, [1 ,2,4]-1 H-triazol-1 -yl and [1 ,2,4]-4H-triazol-4-yl.

The remarks made below as to preferred embodiments of the variables (substituents) of the compounds of formula I are valid on their own as well as preferably in combination with each other, as well as in combination with the stereoisomers, salts, tautomers or N-oxides thereof.

The remarks made below concerning preferred embodiments of the variables further are valid on their own as well as preferably in combination with each other concerning the compounds of formulae I, where applicable, as well as concerning the uses and methods according to the invention and the composition according to the invention.

Preferred compounds according to the invention are compounds of formula I or a stereoi- somer, salt or N-oxide thereof, wherein the salt is an agriculturally suitable salt. Further preferred compounds according to the invention are compounds of formula I or an N-oxide or salt thereof, especially an agriculturally suitable salt. Particularly preferred compounds according to the invention are compounds of formula I or a salt thereof, especially an agriculturally suitable salt thereof.

According to one embodiment of the invention the variable B in the compounds of formula

I is N.

According to another embodiment of the invention the variable B in the compounds of formula I is CH.

According to a preferred embodiment of the invention the variable R in the compounds of formula I is selected from the group consisting of Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, Ci-C ₄ -alkoxy-Ci-C ₄ -alkyl, C ₃ -C ₇ -cycloalkyl, Ci-C ₆ -haloalkyl, R ^c -C(=0)-Ci-C ₂ -alkyl, R ^d O-C(=0)- Ci-C ₂ -alkyl, and R ^k -C(=0)NH-Ci-C ₂ -alkyl; where R ^c , R ^d , R ^e , R ^f , R ^k , Rs and R ^h are as defined above and which preferably have on their own or in particular in combination the following meanings:

R ^c is hydrogen, Ci-C6-alkyl C3-C7-cycloalkyl, C ₂ -C6-alkenyl, C ₂ -C6-haloalkenyl, Ci-C6-haloalkyl or phenyl, in particular Ci-C ₄ -alkyl or Ci-C ₄ -haloalkyl;

R ^d is Ci-C6-alkyl or Ci-C6-haloalkyl, in particular Ci-C ₄ -alkyl,

R ^e , R ^f are independently of each other selected from hydrogen, Ci-C6-alkyl, Ci-C6-haloalkyl and benzyl, and in particular from the group consisting of hydrogen and Ci-C ₄ -alkyl, or R ^e , R ^f together with the nitrogen atom, to which they are bound form a 5-, 6- or 7-membered, saturated or unsaturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is unsubstituted or may carry 1 , 2, 3 or 4 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl and Ci-C4-haloalkyl, and in particular R ^e , R ^f together with the nitrogen atom, to which they are bound may form a 5-, 6- or 7-membered, saturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is unsubstituted or may carry 1 , 2, 3 or 4 methyl groups;

R9, R ^h are independently of each other selected from hydrogen, Ci-C6-alkyl, Ci-C6-haloalkyl and benzyl and in particular from the group consisting of hydrogen or Ci-C4-alkyl, or

R9, R ^h together with the nitrogen atom, to which they are bound form a 5-, 6 or 7-membered, saturated or unsaturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is unsubstituted or may carry 1 , 2, 3 or 4 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl and Ci-C4-haloalkyl, and in particular Rs, R ^h together with the nitrogen atom, to which they are bound may form a 5-, 6- or 7-membered, saturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is unsubstituted or may carry 1 , 2, 3 or 4 methyl groups; and

R ^k is H, Ci-C4-alkyl, Ci-C4-haloalkyl or phenyl, in particular Ci-C4-alkyl.

According to a more preferred embodiment the variable R of the compounds of the formula I is selected from the group consisting of Ci-C4-alkyl, Ci-C4-alkoxy-Ci-C4-alkyl, C3-C7- cycloalkyl, Ci-C ₄ -haloalkyl, R ^d O-C(=0)-Ci-C ₂ -alkyl,

alkyl and R ^k -C(=0)NH-Ci-C ₂ -alkyl, where R ^c , R ^d , R ^e , R ^f and R ^k are as defined above and which preferably have on their own or in particular in combination the following meanings:

R ^c is Ci-C ₄ -alkyl or Ci-C ₄ -haloalkyl,

R ^d is Ci-C ₄ -alkyl,

R ^e is hydrogen or Ci-C4-alkyl,

R ^f is hydrogen or Ci-C4-alkyl, or

R ^e , R ^f together with the nitrogen atom, to which they are bound may form a 5-, 6 or 7- membered, saturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is unsubstituted or may carry 1 , 2, 3 or 4 methyl groups, and

R ^k is Ci-C ₄ -alkyl.

According to a particular preferred embodiment of the invention the variable R in the compounds of formula I is selected from Ci-C4-alkyl, C3-C7-cycloalkyl, Ci-C4-haloalkyl and C1-C4- alkoxy-Ci-C4-alkyl, in particular from methyl, ethyl, isopropyl, tert-butyl, cyclopropyl, cyclopentyl, cyclohexyl, CF ₃ , CHF ₂ , CCIF ₂ , CH ₂ CF ₃ , CF ₂ CF ₃ , CH ₂ CI, CHCI ₂ , ethoxyethyl, ethoxymethyl, methoxyethyl and methoxymethyl.

According to another particular preferred embodiment of the invention the variable R in the compounds of formula I is selected from Ci-C4-alkyl, C3-C7-cycloalkyl, Ci-C4-haloalkyl, methoxyethyl and methoxymethyl, in particular from methyl, ethyl, isopropyl, tert-butyl, cyclopropyl, cy- clopentyl, cyclohexyl, CF ₃ , CHF ₂ , CCIF ₂ , CH ₂ CF ₃ , CF ₂ CF ₃ , CH ₂ CI, CHCI ₂ , methoxyethyl and methoxymethyl.

According to another preferred embodiment of the invention the variable R in the com- pounds of formula I is phenyl or heterocyclyl, where heterocyclyl is a 5- or 6-membered monocyclic or 8-, 9- or 10-membered bicyclic saturated, partially unsaturated or aromatic heterocycle, which contains 1 , 2, 3 or 4 heteroatoms as ring members, which are selected from the group consisting of O, N and S, where phenyl and heterocyclyl are unsubstituted or substituted by 1 , 2, 3 or 4 groups R' which are as defined above and which are independently from one another are preferably selected from the group consisting of halogen, Ci-C4-alkyl, C3-C6-cycloalkyl, C3- C6-halocycloalkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy, Ci-C4-alkoxy-Ci-C4-alkyl and C1-C6- haloalkyloxy, more preferably from halogen, Ci-C4-alkyl, C3-C6-cycloalkyl, Ci-C4-haloalkyl and Ci-C4-alkoxy, in particular from halogen, methyl, ethyl, methoxy and trifluoromethyl, and specifically from CI, F, Br, methyl, methoxy and trifluoromethyl.

According to a more preferred embodiment of the invention the variable R in the compounds of formula I is phenyl or heterocyclyl, where heterocyclyl is a partially unsaturated or aromatic 5- or 6-membered monocyclic or 9- or 10-membered bicyclic heterocycle containing 1 , 2, 3 or 4 heteroatoms as ring members, which are selected from the group consisting of O, N and S, where the bicyclic heterocycle consists of a 5- or 6-membered heteroaromatic ring which is fused to a phenyl ring, and where phenyl and heterocyclyl are unsubstituted or substituted by 1 , 2, 3 or 4 groups R' which independently from one another have the aforementioned preferred meanings.

According to particular preferred embodiments the variable R in the compounds of the formula I is phenyl or heterocyclyl selected from pyridin-2-yl, pyridin-3-yl, pyridin-4-yl, piperidin- 2-yl, piperidin-3-yl, piperidin-4-yl, benzisoxazole-2-yl, 1 ,2,4-oxadiazol-3-yl, 1 ,2,4-triazol-3-yl, 1 - ethylbenzimidazol-2-yl, 4-methylthiazol-2-yl, thiophen-2-yl, furan-2-yl, furan-3-yl, tetrahydrofu- ran-2-yl, tetrahydrofuran-3-yl, isoxazol-2-yl, isoxazol-3-yl, isoxazol-4-yl, isoxazol-5-yl, oxazol-2- yl, oxazol-3-yl, oxazol-4-yl, oxazol-5-yl, pyrrol-2-yl, pyrrol-3-yl, imidazol-2-yl, imidazol-4-yl, imid- azol-5-yl, pyrazol-3-yl, pyrazol-4-yl, pyrazol-5-yl, isothiazol-3-yl, isothiazol-4-yl, isothiazol-5-yl, thiazol-2-yl, thiazol-4-yl, thiazol-5-yl, 1 ,2,3-triazol-4-yl, 1 ,2,3-triazol-5-yl, 1 ,2,5-triazol-3-yl, 1 ,3,4- triazol-2-yl, 1 ,2,4-triazol-3-yl, 1 ,2,4-triazol-5-yl, 1 ,2,4-oxadiazol-3-yl, 1 ,2,4-oxadiazol-5-yl, 1 ,3,4- oxadiazol-2-yl, 1 ,2,3-oxadiazol-4-yl, 1 ,2,3-oxadiazol-5-yl, 1 ,2,5-oxadiazol-3-yl, 1 ,2,4-thiadiazol- 3-yl, 1 ,2,4-thiadiazol-5-yl, 1 ,3,4-thiadiazol-2-yl, 1 ,2,3-thiadiazol-4-yl, 1 ,2,3-thiadiazol-5-yl, 1 ,2,5- thiadiazol-3-yl, 2H-1 ,2,3,4-tetrazol-5-yl, 1 H-1 ,2,3,4-tetrazol-1 -yl, 1 ,2,3,4-oxatriazol-5-yl, 1 ,2,3,5- oxatriazol-4-yl, 1 ,2,3,4-thiatriazol-5-yl, 1 ,2,3,5-thiatriazol-4-yl, pyrazin-2-yl, pyrazin-3-yl, pyrim- idin-2-yl, pyrimidin-4-yl, pyrimidin-5-yl, pyridazin-3-yl and pyridazin-4-yl, where phenyl and heterocyclyl are unsubstituted or carry 1 , 2, or 3 groups R' which independently from one another have the aforementioned preferred meanings.

According to a preferred embodiment of the invention the variable R in the compounds of formula I is R ^b -S(0) _n -Ci-C3-alkyl, where R ^b is as defined above and in particular selected from the group consisting of Ci-C6-alkyl, C3-C7-cycloalkyl, Ci-C6-haloalkyl, C ₂ -C6-alkenyl, C ₂ -C6- haloalkenyl, C ₂ -C6-alkynyl, C ₂ -C6-haloalkynyl, phenyl and heterocyclyl, where heterocyclyl is a 5- or 6-membered monocyclic saturated, partially unsaturated or aromatic heterocycle, which contains 1 , 2 or 3 heteroatoms as ring members, which are selected from the group consisting of O, N and S, where phenyl and heterocyclyl are unsubstituted or substituted by 1 , 2 or 3 groups, which are identical or different and preferably selected from the group consisting of hal- ogen, Ci-C4-alkyl, Ci-C2-haloalkyl and Ci-C2-alkoxy.

According to a more preferred embodiment of the invention the variable R in the compounds of formula I is R ^b -S(0) _n -Ci-C3-alkyl, where R ^b is selected from the group consisting of Ci-C6-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, Ci-C6-haloalkyl, C2-C6-haloalkenyl, C2-C6-haloalkynyl, C3-C7-cycloalkyl, phenyl and heterocyclyl, where heterocyclyl is a 5- or 6-membered monocyclic saturated, partially unsaturated or aromatic heterocycle, which contains 1 , 2 or 3 heteroatoms as ring members, which are selected from the group consisting of O, N and S.

According to an even more preferred embodiment of the invention the variable R in the compounds of formula I is R ^b -S(0) _n -Ci-C2-alkyl, where R ^b is selected from Ci-C6-alkyl, C1-C6- haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C3-C7-cycloalkyl, phenyl and hetero- cyclyl, where heterocyclyl is a 6-membered aromatic heterocyclic radical having 1 or 2 nitrogen atoms as ring members.

According to a particularly preferred embodiment of the invention the variable R in the compounds of formula I is R ^b -S(0) ₂ -Ci-C ₂ -alkyl, where R ^b is CH ₃ , CH ₂ H ₃ , CH(CH ₃ ) ₂ ,

CH2CH2CH3, CH ₂ CH=CH ₂ , CH ₂ C≡CH or phenyl.

According to specifically preferred embodiments of the invention the variable R in the compounds of formula I is selected from the group consisting of methyl, ethyl, isopropyl, tert- butyl, cyclopropyl, cyclopentyl, cyclohexyl, CF ₃ , CHF ₂ , CCIF ₂ , CH2CF3, CF2CF3, CH ₂ CI, CHC , methoxyethyl, methoxymethyl, and in particular from methyl and ethyl.

Preferred compounds according to the invention are compounds of formula I, wherein R ¹ is selected from the group consisting of CN, halogen, nitro, Ci-C6-alkyl, C2-C6-alkenyl, C2-C6- alkynyl, Ci-C6-haloalkyl, Ci-C6-alkoxy, Ci-C4-alkoxy-Ci-C4-alkyl, Ci-C4-haloalkoxy-Ci-C4-alkyl, Ci-C ₄ -alkoxy-Ci-C ₄ -alkoxy-Z ¹ , Ci-C ₄ -alkylthio-Ci-C ₄ -alkyl, Ci-C4-alkylthio-Ci-C ₄ -alkylthio-Z ¹ , C ₂ - C6-alkenyloxy, C2-C6-alkynyloxy, Ci-C6-haloalkoxy, Ci-C4-haloalkoxy-Ci-C4-alkoxy and R ^1b -

S(0)k, where k and Z ¹ are as defined herein and where R ^1b is as defined above and in particular selected from the group consisting of Ci-C4-alkyl and Ci-C4-haloalkyl. In this context Z ¹ is in particular a covalent bond.

More preferably, R ¹ is selected from halogen, CN, nitro, Ci-C4-alkyl, Ci-C4-haloalkyl, Ci- C4-alkoxy-Ci-C4-alkyl, Ci-C4-haloalkoxy-Ci-C4-alkyl, Ci-C4-alkoxy-Ci-C4-alkoxy-Ci-C4-alkyl, Ci- C ₄ -a I ky 11 h i o-C1 -C ₄ -a I ky I , Ci-C4-alkylthio-Ci-C4-alkylthio-Ci-C ₄ -alkyl, Ci-C ₄ -alkoxy, C1-C4- haloalkoxy, C3-C4-alkenyloxy, C3-C4-alkynyloxy, Ci-C4-alkoxy-Ci-C4-alkoxy, Ci-C4-haloalkoxy- Ci-C ₄ -alkoxy, Ci-C ₄ -alkyl-S(0) _k and Ci-C ₄ -haloalkyl-S(0) _k , where k is 0 or 2.

In particular, R ¹ is selected from the group consisting of halogen, nitro, Ci-C4-alkyl, C1-C4- haloalkyl, Ci-C4-alkoxy-Ci-C4-alkyl, Ci-C4-alkoxy-Ci-C4-alkoxy-Ci-C4-alkyl, Ci-C4-alkoxy, C1-C4- haloalkoxy, Ci-C4-alkylthio, Ci-C4-haloalkylthio and Ci-C4-alkylsulfonyl, specifically R ¹ is F, CI, Br, I, nitro, CH ₃ , CF ₃ , OCH ₃ , OCF ₃ , SCH ₃ , SCF ₃ , S0 ₂ CH ₃ or CH2OCH2CH2OCH3, and more specifically R ¹ is F, CI, Br, I, nitro, CH ₃ , CF ₃ , OCH ₃ , SCH ₃ or S0 ₂ CH ₃ .

In one group of embodiments of the invention, the variable R ² is hydrogen.

In one group of embodiments of the invention the variable R ² of the compounds of formula I has any one of the meanings given above for R ² with the exception of hydrogen.

According to preferred embodiment of the invention the variable R ² in the compounds of formula I is a 5- or 6-membered heterocyclyl, where heterocyclyl is a saturated, partially unsaturated or aromatic heterocyclic radical, which contains as ring member 1 heteroatom selected from the group consisting of O, N and S and 0, 1 , 2 or 3 further nitrogen atom(s), where hetero- cyclyl is unsubstituted or carries 1 , 2 or 3 radicals R ²¹ , as defined herein, which are identical or different.

According to an even more preferred embodiment of the invention the variable R ² in the compounds of formula I is a 5- or 6-membered heterocyclyl selected from the group consisting of isoxazolinyl (4,5-dihydroisoxazolyl), 1 ,2-dihydrotetrazolonyl, 1 ,4-dihydrotetrazolonyl, tetrahy- drofuryl, dioxolanyl, piperidinyl, morpholinyl, piperazinyl, isoxazolyl, pyrazolyl, thiazolyl, oxazolyl, furyl, pyridinyl, pyrimidinyl and pyrazinyl, where heterocyclyl is unsubstituted or carries 1 , 2 or 3 radicals R ²¹ which are identical or different and are selected from the group consisting of C1-C4- alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy, Ci-C4-alkoxy-Ci-C4-alkyl and Ci-C4-alkylthio-Ci-C4-alkyl.

According to a particular embodiment of the invention the variable R ² in the compounds of formula I is a 5- or 6-membered heterocyclyl selected from 4,5-dihydroisoxazol-3-yl, which is unsubstituted or substituted in position 5 with CH ₃ , CH2F or CHF2, 4,5-dihydroisoxazol-5-yl, which is unsubstituted or substituted in position 3 with CH ₃ , OCH ₃ , CH2OCH3, CH2SCH3, 1 - methyl-5-oxo-1 ,5-dihydrotetrazol-2-yl, 4-methyl-5-oxo-4,5-dihydrotetrazol-1 -yl, morpholin-4-yl, isoxazol-3-yl, 5-methyl-isoxazol-3-yl, isoxazol-5-yl, 3-methyl-isoxazol-5-yl, 1 -methyl-1 H-pyrazol- 3-yl, 2-methyl-2H-pyrazol-3-yl and thiazol-2-yl.

According to a preferred embodiment of the invention the variable R ² in the compounds of formula I is phenyl-Z ^2a , where Z ^2a is as defined herein, and where phenyl is unsubstituted or carries 1 , 2 or 3 radicals R ²¹ which are identical or different and as defined above and which are in particular selected from halogen, Ci-C4-alkyl, Ci-C4-alkoxy, Ci-C4-haloalkyl, Ci-C4-alkoxy-Ci- C4-alkyl and Ci-C4-alkoxy-Ci-C4-alkoxy, and preferably from halogen, Ci-C2-alkyl, Ci-C2-alkoxy, Ci-C2-haloalkyl and Ci-C2-alkoxy-Ci-C2-alkoxy.

According to a more preferred embodiment of the invention the variable R ² in the compounds of formula I is a radical of the following formula:

in which # denotes the bond through which the group R ² is attached and:

R ^P1 is hydrogen or halogen, preferably hydrogen, CI, Br or F, and in particular H or F;

R ^P2 is hydrogen, halogen or Ci-C2-alkoxy, preferably hydrogen, CI, Br, F, OCH3 or OCH2CH3, and in particular H, F, CI or OCH3; and R ^P3 is hydrogen, halogen, Ci-C2-alkyl, Ci-C2-haloalkyl, Ci-C2-alkoxy, Ci-C2-alkoxy-Ci-C2- alkoxy, preferably hydrogen, CI, Br, F, CH ₃ , C ₂ H ₅ , CF ₃ , CHF ₂ , CH ₂ F, CCI ₂ F, CF ₂ CI, CH2CF3, CH2CHF2, CF2CF3, OCH3, OCH2CH3, OCH2OCH3, OCH2CH2OCH2CH3,

OCH2OCH2CH3 or OCH2CH2OCH3, and in particular is H, F, CI, CH ₃ , CF ₃ , OCH ₃ ,

OCH2CH3, OCH2OCH3 or OCH2CH2OCH3.

According to a particular embodiment of the invention the variable R ² in the compounds of formula I is phenyl which is unsubstituted or carries one radical R ²¹ , where R ²¹ is preferably attached to position 4 of the phenyl group and is as defined above and in particular selected from Ci-C2-alkyl, Ci-C2-alkoxy, Ci-C2-haloalkyl and Ci-C2-alkoxy-Ci-C2-alkoxy, preferably form CH3, C ₂ H ₅ , OCH3, OC ₂ H ₅ , CHF ₂ , CF ₃ , OCH2OCH3 and OCH ₂ CH ₂ OCH ₃ , and specifically from OCH ₃

According to a preferred embodiment of the invention the variable R ² in the compounds of formula I is selected from the group consisting of hydrogen, halogen, Ci-C6-alkyl, Ci-C4-alkoxy- Ci-C4-alkyl, Ci-C4-haloalkoxy-Ci-C4-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, Ci-C4-alkoxy, C1-C4- haloalkoxy, C3-C6-alkenyloxy, C3-C6-alkynyloxy, C3-C6-haloalkenyloxy, C3-C6-haloalkynyloxy, Ci-C ₄ -alkoxycarbonyl, Ci-C ₄ -alkyl-S(0) _k , k is 0, 1 , 2, and Ci-C ₄ -haloalkyl-S(0) ₂ .

According to another preferred embodiment of the invention the variable R ² in the compounds of formula I is selected from the group consisting of halogen, Ci-C6-alkyl, Ci-C4-alkoxy- Ci-C4-alkyl, Ci-C4-haloalkoxy-Ci-C4-alkyl, C2-C6-alkenyl, C2-C6-alkynyl, Ci-C4-alkoxy, C1-C4- haloalkoxy, C3-C6-alkenyloxy, C3-C6-alkynyloxy, C3-C6-haloalkenyloxy, C3-C6-haloalkynyloxy, Ci-C4-alkoxycarbonyl, Ci-C4-alkylsulfonyl, Ci-C4-alkylsulfinyl, Ci-C4-alkylsulfanyl, and C1-C4- haloalkyl-S(0) ₂ .

According to a more preferred embodiment of the invention the variable R ² in the compounds of formula I is selected from C2-C4-alkenyl, C2-C4-alkynyl, Ci-C4-alkoxy, C1-C2- haloalkoxy-Ci-C2-alkyl, C3-C4-alkenyloxy, C3-C4-alkynyloxy, Ci-C4-alkoxycarbonyl, C1-C4- alkylsulfonyl, Ci-C4-alkylsulfinyl and Ci-C4-alkylsulfanyl, and in particular from CH=CH2, CH=CHCH ₃ , CH2OCH2CF3, OC ₂ H ₅ , OCH ₂ CH=CH ₂ , OCH ₂ C≡CH, C(0)OCH ₃ , C(0)OC ₂ H ₅ , SO2CH3, S0 ₂ C ₂ H ₅ , S0 ₂ CH(CH ₃ ) ₂ , SOCH3, SOC ₂ H ₅ , SOCH(CH ₃ ) ₂ , SCH ₃ , SC ₂ H ₅ and

SCH(CH ₃ ) ₂ .

According to a specifically preferred embodiment of the invention the variable R ² in the compounds of formula I is selected from the group consisting of hydrogen, 4,5-dihydroisoxazol- 3-yl, which is unsubstituted or substituted in position 5 with CH3, CH2F or CHF2, 4,5- dihydroisoxazol-5-yl, which is unsubstituted or substituted in position 3 with CH3, OCH3, CH2OCH3, CH2SCH3, 1 -methyl-5-oxo-1 ,5-dihydrotetrazol-2-yl, 4-methyl-5-oxo-4,5- dihydrotetrazol-1 -yl, morpholin-4-yl, isoxazol-3-yl, 5-methyl-isoxazol-3-yl, isoxazol-5-yl, 3- methyl-isoxazol-5-yl, 1 -methyl-1 H-pyrazol-3-yl, 2-methyl-2H-pyrazol-3-yl, thiazol-2-yl, 4-CH3- phenyl, 4-C ₂ H ₅ -phenyl, 4-OCH ₃ -phenyl, 4-OC ₂ H ₅ -phenyl, 4-CHF ₂ -phenyl, 4-CF ₃ -phenyl, 4- OCH ₂ OCH ₃ -phenyl, 4-OCH ₂ CH ₂ OCH ₃ -phenyl, CH=CH ₂ , CH=CHCH ₃ , CH ₂ OCH ₂ CF ₃ , OC ₂ H ₅ , OCH ₂ CH=CH ₂ , OCH ₂ C≡CH, C(0)OCH ₃ , C(0)OC ₂ H ₅ , SO2CH3, S0 ₂ C ₂ H ₅ , S0 ₂ CH(CH ₃ ) ₂ , SOCH3, SOC2H5, SOCH(CH ₃ ) ₂ , SCH3, SC2H5 and SCH(CH ₃ ) ₂ , in particular selected from hydrogen, halogen, methyl, CH2OCH2CF3, methylsulfonyl, methylsulfinyl, methylsulfanyl, 3- isoxazolinyl, 5-methyl-3-isoxazolinyl, 5-isoxazolinyl, 3-methyl-5-isoxazolinyl, 3-isoxazolyl, 5- methyl-3-isoxazolyl, 5-isoxazolyl and 3-methyl-5-isoxazolyl, and specifically selected from hydrogen, chlorine, methylsulfonyl, methylsulfinyl, methylsulfanyl, CH2OCH2CF3, 3-isoxazolinyl, 5- methyl-3-isoxazolinyl, 3-methyl-5-isoxazolinyl, 3-isoxazolyl, 5-methyl-3-isoxazolyl and 3-methyl- 5-isoxazolyl.

Preferred compounds according to the invention are compounds of formula I, wherein R ³ is selected from the group consisting of hydrogen, cyano, halogen, nitro, Ci-C4-alkyl, C1-C4- haloalkyl, Ci-C4-alkoxy, Ci-C4-haloalkoxy, C2-C4-alkenyl, C2-C4-alkynyl, C2-C4-alkenyloxy, C2- C4-alkynyloxy or R ^2b -S(0)k, where the variables k and R ^2b have one of the herein defined meanings.

More preferably, R ³ is selected from the group consisting of hydrogen, halogen, CN, NO2,

Ci-C4-alkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy, Ci-C4-haloalkoxy, Ci-C4-alkylthio, C1-C4- haloalkylthio, Ci-C ₄ -alkyl-S(0) ₂ and Ci-C ₄ -haloalkyl-S(0) ₂ .

In particular, R ³ is selected from the group consisting of hydrogen, halogen, CN, NO2, Ci- C2-alkyl, Ci-C2-haloalkyl, Ci-C2-alkoxy, Ci-C2-haloalkoxy, Ci-C2-alkylthio, Ci-C2-haloalkylthio, Ci-C ₂ -alkyl-S(0) ₂ and Ci-C ₂ -haloalkyl-S(0) ₂ , specifically from H, CI, F, CN, N0 ₂ , CH ₃ , CF ₃ ,

CHF ₂ , OCH3, OCF3, OCHF2, SCHs, SCFs, SCHF ₂ , S(0) ₂ CH ₃ and S(0) ₂ CH ₂ CH ₃ , and more specifically from H, CI, F, CN, CF ₃ and S(0) ₂ CH ₃ .

Preferred compounds according to the invention are compounds of formula I, wherein R ⁴ and R ⁵ are identical or different and independently selected from the group consisting of hydro- gen, CN, halogen, nitro, Ci-C6-alkyl, C ₃ -C7-cycloalkyl, C ₃ -C7-cycloalkyl-Ci-C4-alkyl, where the C ₃ -C7-cycloalkyl groups in the two aforementioned radicals are unsubstituted or partially or completely halogenated, C2-C6-alkenyl, C2-C6-alkynyl, Ci-C6-haloalkyl, Ci-C ₃ -alkylamino, Ci-C ₃ - dialkylamino, Ci-C ₃ -alkylamino-S(0)k, Ci-C ₃ -alkylcarbonyl, Ci-C6-alkoxy, Ci-C4-alkoxy-Ci-C4- alkyl, Ci-C ₄ -alkoxy-Ci-C ₄ -alkoxy-Z ¹ , Ci-C ₄ -alkylthio-Ci-C ₄ -alkyl, Ci-C ₄ -alkylthio-Ci-C ₄ -alkylthio- Z ¹ , C2-C6-alkenyloxy, C2-C6-alkynyloxy, Ci-C6-haloalkoxy, Ci-C4-haloalkoxy-Ci-C4-alkyl, C1-C4- haloalkoxy-Ci-C4-alkoxy, R ^1b -S(0)k and phenoxy where k and Z ¹ are as defined herein and where R ^1b is as defined above and in particular selected from the group consisting of Ci-C4-alkyl and Ci-C4-haloalkyl, provided that at least one of the radicals R ⁴ and R ⁵ is different from hydrogen, and further provided that if R ⁴ is hydrogen, halogen, cyano, nitro, Ci-C4-alkyl or Ci-C4- haloalkyl, R ⁵ is not hydrogen, halogen, Ci-C4-alkyl or Ci-C4-haloalkyl. In this context, Z ¹ is in particular a covalent bond.

More preferably, R ⁴ and R ⁵ are identical or different and independently selected from the group consisting of hydrogen, halogen, CN, nitro, Ci-C4-alkyl, C ₃ -C5-cycloalkyl, C ₃ -C5-cycloalkyl- Ci-C4-alkyl, where the C ₃ -Cs-cycloalkyl groups in the two aforementioned radicals are unsubsti- tuted or partially or completely halogenated, Ci-C4-haloalkyl, Ci-C ₃ -alkylamino, Ci-C ₃ - dialkylamino, Ci-C ₃ -alkylamino-S(0)k, Ci-C ₃ -alkylcarbonyl, Ci-C4-alkoxy, Ci-C4-alkoxy-Ci-C4- alkyl, Ci-C4-alkoxy-Ci-C4-alkoxy-Ci-C4-alkyl, Ci-C4-alkoxy-Ci-C4-alkoxy, Ci-C4-alkylthio-Ci-C4- alkyl, Ci-C4-alkylthio-Ci-C4-alkylthio-Ci-C4-alkyl, C ₃ -C4-alkenyloxy, C ₃ -C4-alkynyloxy, C1-C4- haloalkoxy, Ci-C4-haloalkoxy-Ci-C4-alkyl, Ci-C4-haloalkoxy-Ci-C4-alkoxy, Ci-C4-alkyl-S(0)k, Ci- C4-haloalkyl-S(0)k, where k is 0, 1 or 2, provided that at least one of the radicals R ⁴ and R ⁵ is different from hydrogen, and further provided that if R ⁴ is hydrogen, halogen, cyano, nitro, Ci- C4-alkyl or Ci-C4-haloalkyl, R ⁵ is not hydrogen, halogen, Ci-C4-alkyl or Ci-C4-haloalkyl. In particular, R ⁴ and R ⁵ are identical or different and independently selected from the group consisting of hydrogen, halogen, CN, nitro, Ci-C4-alkyl, C3-C4-cycloalkyl, C3-C4-cycloalkyl- Ci-C2-alkyl, where the C3-C4-cycloalkyl groups in the two aforementioned radicals are unsubsti- tuted or partially or completely halogenated, Ci-C4-haloalkyl, Ci-C3 alkylcarbonyl, Ci-C4-alkoxy, Ci-C4-alkoxy-Ci-C4-alkyl, Ci-C4-alkoxy-Ci-C4-alkoxy-Ci-C4-alkyl, Ci-C4-haloalkoxy, C1-C4- alkylthio, Ci-C4-haloalkylthio, Ci-C4-alkylsulfinyl, Ci-C4-alkylsulfonyl; specifically R ⁴ and R ⁵ are identical or different and independently selected from the group consisting of H, F, CI, Br, I, CN, nitro, CH3, CH2CH3, CH(CH ₃ ) ₂ , cyclopropyl, cyclopropylmethyl, CF ₃ , OCH ₃ , OCH2CH3,

OCH(CH ₃ ) ₂ , CH2OCH3, CH2OCH2CH2OCH3, OCF3, OCHF2, SCH ₃ , SCF ₃ , SCH2CH3, SCH2CF3, SOCH3, SOCH2CH3, SO2CH3, SO2CH2CH3; and more specifically R ⁴ and R ⁵ are identical or different and independently selected from the group consisting of H, F, CI, Br, I, CN, nitro, CH3, CH2CH3, CH(CH ₃ ) ₂ , cyclopropyl, CF ₃ , OCH ₃ , OCF ₃ , SCH ₃ , SOCH ₃ , SO2CH3 or CH ₂ OCH ₃ ; provided that at least one of the radicals R ⁴ and R ⁵ is different from hydrogen; and further provided that if R ⁴ is hydrogen, halogen, cyano, nitro, Ci-C4-alkyl or Ci-C4-haloalkyl, R ⁵ is not hydrogen, halogen, Ci-C4-alkyl or Ci-C4-haloalkyl;

Preferred compounds according to the invention are compounds of formula I, wherein R ⁴ is H and R ⁵ is selected from the group consisting of CN, nitro, cyclopropyl, cyclopropylmethyl, OCH3, OCH2CH3, OCH(CH ₃ ) ₂ , CH2OCH3, CH2OCH2CH2OCH3, OCF3, OCHF2, SCH ₃ , SCF ₃ , SCH2CH3, SCH2CF3, SOCH3, SOCH2CH3, SO2CH3, SO2CH2CH3; more preferably R ⁵ is selected from the group consisting of CN, nitro, cyclopropyl, OCH ₃ , CH2OCH3, OCF ₃ , SCH ₃ , SOCH ₃ ,

Further preferred compounds according to the invention are compounds of formula I, wherein R ⁵ is H and R ⁴ is selected from the group consisting of cyclopropyl, cyclopropylmethyl, OCH3, OCH2CH3, OCH(CH ₃ ) ₂ , CH2OCH3, CH2OCH2CH2OCH3, OCF3, OCHF2, SCH ₃ , SCF ₃ , SCH2CH3, SCH2CF3, SOCH3, SOCH2CH3, SO2CH3, SO2CH2CH3; more preferably R ⁴ is selected from the group consisting of cyclopropyl, OCH ₃ , CH2OCH3, OCF ₃ , SCH ₃ , SOCH ₃ , SO2CH3. In this context, the variables R', R ¹¹ , R ²¹ , Z, Z , Z ² , Z ^2a , R ^b , R ^b , R ^2b , R ^c , R ^2c , R ^d , R ^2d , R ^e ,

R ^2e , R ^f , R ^2f , R9, R¾, R ^h , R ^2h , R ^k , n and k, independently of each other, preferably have one of the following meanings:

R', R ¹¹ , R ²¹ independently of each other are selected from halogen, Ci-C4-alkyl, C3-C6- cycloalkyl, C3-C6-halocycloalkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy, Ci-C4-alkoxy-Ci-C4-alkyl, C1-C4- alkylthio-Ci-C4-alkyl, Ci-C4-alkoxy-Ci-C4-alkoxy and Ci-C6-haloalkyloxy, more preferably from halogen, Ci-C4-alkyl, C3-C6-cycloalkyl, Ci-C4-haloalkyl and Ci-C4-alkoxy.

More preferably R', R ¹¹ , R ²¹ independently of each other are selected from the group consisting of halogen, Ci-C4-alkyl, C3-C6-cycloalkyl, Ci-C4-haloalkyl, Ci-C4-alkoxy, Ci-C4-alkoxy-Ci- C4-alkyl, Ci-C4-alkylthio-Ci-C4-alkyl and Ci-C4-alkoxy-Ci-C4-alkoxy; in particular selected from halogen, Ci-C4-alkyl, Ci-C4-alkoxy, Ci-C4-haloalkyl, Ci-C4-alkoxy-Ci-C4-alkyl and Ci-C4-alkoxy- Ci-C4-alkoxy; and specifically from CI, F, Br, methyl, ethyl, methoxy and trifluoromethyl.

Z, Z ¹ , Z ² independently of each other are selected from a covalent bond, methanediyl and ethanediyl, and in particular are a covalent bond.

Z ^2a is selected from a covalent bond, Ci-C2-alkanediyl, 0-Ci-C2-alkanediyl, C1-C2- alkanediyl-0 and Ci-C2-alkanediyl-0-Ci-C2-alkanediyl; more preferably from a covalent bond, methanediyl, ethanediyl, O-methanediyl, O-ethanediyl, methanediyl-O, and ethanediyl-O; and in particular from a covalent bond, methanediyl and ethanediyl.

R ^b , R ^1b , R ^2b independently of each other are selected from Ci-C6-alkyl, C3-C7-cycloalkyl, Ci-C6-haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, phenyl and heterocyclyl, where heterocyclyl is a 5- or 6-membered monocyclic saturated, partially unsaturated or aromatic heterocycle, which contains 1 , 2 or 3 heteroatoms as ring members, which are selected from the group consisting of O, N and S, where phenyl and heterocyclyl are unsubstituted or substituted by 1 , 2 or 3 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl, Ci-C2-haloalkyl and Ci-C2-alkoxy.

More preferably R ^b ,R ^1b , R ^2b independently of each other are selected from the group consisting of Ci-C4-alkyl, C2-C4-alkenyl, C2-C4-alkynyl, Ci-C4-haloalkyl, C2-C4-haloalkenyl, C2-C4- haloalkynyl, C3-C6-cycloalkyl, phenyl and heterocyclyl, where heterocyclyl is a 5- or 6- membered monocyclic saturated, partially unsaturated or aromatic heterocycle, which contains 1 , 2 or 3 heteroatoms as ring members, which are selected from the group consisting of O, N and S.

In particular, R ^b , R ^1b , R ^2b independently of each other are selected from Ci-C4-alkyl, C1-C4- haloalkyl, C2-C4-alkenyl, C2-C4-haloalkenyl, C2-C4-alkynyl, C3-C6-cycloalkyl, phenyl and heterocyclyl, where heterocyclyl is a 5- or 6-membered aromatic heterocyclic radical having 1 or 2 nitrogen atoms as ring members.

R ^c , R ^2c , R ^k independently of each other are selected from hydrogen, Ci-C6-alkyl, C3-C7- cycloalkyl, which is unsubstituted or partly or completely halogenated, Ci-C6-haloalkyl, C2-C6- alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, Ci-C4-alkoxy-Ci-C4-alkyl, phenyl, benzyl and heterocyclyl, where heterocyclyl is a 5- or 6-membered monocyclic saturated, partially unsaturated or aromatic heterocycle, which contains 1 , 2 or 3 heteroatoms as ring members, which are selected from the group consisting of O, N and S, where phenyl, benzyl and heterocyclyl are unsubstituted or substituted by 1 , 2 or 3 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl, Ci-C4-haloalkyl and Ci- C4-alkoxy.

More preferably R ^c , R ^2c , R ^k independently of each other are selected from hydrogen, Ci- C4-alkyl, Ci-C4-haloalkyl, C2-C-alkenyl, C2-C-haloalkenyl, C2-C-alkynyl, C3-C6-cycloalkyl, phenyl and heterocyclyl, where heterocyclyl is a 5- or 6-membered monocyclic saturated, partially un- saturated or aromatic heterocycle, which contains 1 , 2 or 3 heteroatoms as ring members, which are selected from the group consisting of O, N and S.

In particular, R ^c , R ^2c , R ^k independently of each other are selected from hydrogen, C1-C4- alkyl, Ci-C4-haloalkyl, C2-C4-alkenyl, C2-C4-haloalkenyl, C3-C6-cycloalkyl, phenyl and heterocyclyl, where heterocyclyl is a 5- or 6-membered aromatic heterocyclic radical having 1 or 2 nitro- gen atoms as ring members.

R ^d , R ^2d independently of each other are selected from Ci-C6-alkyl, C3-C7-cycloalkyl, which is unsubstituted or partly or completely halogenated, Ci-C6-haloalkyl, C2-C6-alkenyl, C2-C6- haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, Ci-C4-alkoxy-Ci-C4-alkyl, phenyl and benzyl.

More preferably R ^d , R ^2d independently of each other are selected from Ci-C6-alkyl, C1-C6- haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, Ci-C4-alkoxy-Ci-C4-alkyl and C3-C7- cycloalkyl, which is unsubstituted or partly or completely halogenated, and in particular selected from Ci-C4-alkyl, Ci-C4-haloalkyl, C2-C4-alkenyl, C2-C4-haloalkenyl, C2-C4-alkynyl and C3-C6- cycloalkyl.

R ^e , R ^f , R ^2e , R ^2f independently of each other are selected from the group consisting of hydrogen, Ci-C6-alkyl, C3-C7-cycloalkyl, which is unsubstituted or partially or completely halogenated, Ci-C6-haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, Ci-C4-alkoxy-Ci-C4-alkyl, phenyl and benzyl, where phenyl and benzyl are unsubstituted or substituted by 1 , 2 or 3 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl, C1-C4- haloalkyl and Ci-C4-alkoxy, or R ^e and R ^f or R ^2e and R ^2f together with the nitrogen atom, to which they are bound may form a 5-, 6 or 7-membered, saturated or unsaturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is unsubstituted or may carry 1 , 2, 3 or 4 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl, Ci-C4-haloalkyl and Ci-C4-alkoxy.

More preferably R ^e , R ^f , R ^2e , R ^2f independently of each other are selected from hydrogen, Ci-C6-alkyl, Ci-C6-haloalkyl and benzyl, or R ^e and R ^f or R ^2e and R ^2f together with the nitrogen atom, to which they are bound may form a 5- or 6-membered, saturated or unsaturated N- bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is unsubstituted or may carry 1 , 2 or 3 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl and Ci-C4-haloalkyl.

In particular, R ^e , R ^f , R ^2e , R ^2f independently of each other are selected from hydrogen and Ci-C4-alkyl, or R ^e and R ^f or R ^2e and R ^2f together with the nitrogen atom, to which they are bound may form a 5- or 6-membered, saturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is unsubstituted or may carry 1 , 2 or 3 methyl groups.

R9, R¾ independently of each other are selected from hydrogen, Ci-C6-alkyl, C3-C7- cycloalkyl, which is unsubstituted or partly or completely halogenated, Ci-C6-haloalkyl, C2-C6- alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, Ci-C4-alkoxy-Ci-C4-alkyl, phenyl and benzyl.

More preferably Rs, R¾ independently of each other are selected from hydrogen, C1-C6- alkyl, Ci-C6-haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, benzyl, Ci-C4-alkoxy-Ci-C4-alkyl and C3-C7-cycloalkyl, which is unsubstituted or partly or completely halogenated, and in particular selected from hydrogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C2-C4-alkenyl, C2-C4-haloalkenyl, benzyl and C3-C6-cycloalkyl.

R ^h , R ^2h independently of each other are selected from hydrogen, Ci-C6-alkyl, C3-C7- cycloalkyl, which is unsubstituted or partly or completely halogenated, Ci-C6-haloalkyl, C2-C6- alkenyl, C2-C6-haloalkenyl, C2-C6-alkynyl, C2-C6-haloalkynyl, Ci-C4-alkoxy-Ci-C4-alkyl, phenyl, benzyl and a radical C(=0)-R ^k , where R ^k is H, Ci-C4-alkyl, Ci-C4-haloalkyl or phenyl.

More preferably R ^h , R ^2h independently of each other are selected from hydrogen, C1-C6- alkyl, Ci-C6-haloalkyl, C2-C6-alkenyl, C2-C6-haloalkenyl, benzyl, Ci-C4-alkoxy-Ci-C4-alkyl and C3-C7-cycloalkyl, which is unsubstituted or partly or completely halogenated, and in particular selected from hydrogen, Ci-C4-alkyl, Ci-C4-haloalkyl, C2-C4-alkenyl, C2-C4-haloalkenyl, benzyl and C3-C6-cycloalkyl; or

R9 and R ^h or R¾ and R ^2h together with the nitrogen atom, to which they are bound may form a 5-, 6 or 7-membered, saturated or unsaturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is

unsubstituted or may carry 1 , 2, 3 or 4 groups, which are identical or different and selected from the group consisting of =0, halogen, Ci-C4-alkyl and Ci-C4-haloalkyl and Ci-C4-alkoxy;

more preferably Rs and R ^h or R¾ and R ^2h together with the nitrogen atom, to which they are bound may form a 5- or 6-membered, saturated or unsaturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is unsubstituted or may carry 1 , 2 or 3 groups, which are identical or different and selected from the group consisting of halogen, Ci-C4-alkyl and Ci-C4-haloalkyl;

and in particular, Rs and R ^h or R¾ and R ^2h together with the nitrogen atom, to which they are bound may form a 5- or 6-membered, saturated N-bound heterocyclic radical, which may carry as a ring member a further heteroatom selected from O, S and N and which is unsubstituted or may carry 1 , 2 or 3 methyl groups.

n and k independently of each other are 0 or 2, and in particular 2.

Particularly preferred are compounds of formula I, wherein the variables R ¹ and R ³ have the following meanings:

R ¹ is selected from the group consisting of halogen, nitro, Ci-C4-alkyl, Ci-C4-haloalkyl, Ci- C4-alkoxy-Ci-C4-alkyl, Ci-C4-alkoxy-Ci-C4-alkoxy-Ci-C4-alkyl, Ci-C4-alkoxy, Ci-C4-haloalkoxy, Ci-C4-alkylthio, Ci-C4-haloalkylthio and Ci-C4-alkylsulfonyl, in particular from F, CI, Br, nitro, CH ₃ , CF ₃ , OCHs, SCHs, OCF ₃ , SCF ₃ , SO2CH3, CH2OCH3 and CH2OCH2CH2OCH3; and

R ³ is selected from the group consisting of hydrogen, halogen, CN, NO2, Ci-C4-alkyl, Ci-

C4-haloalkyl, Ci-C4-alkoxy, Ci-C4-haloalkoxy, Ci-C4-haloalkylthio and Ci-C4-alkylsulfonyl, in particular from H, CI, F, CN, N0 ₂ , CH ₃ , CF ₃ , CHF ₂ , OCH ₃ , OCF ₃ , OCHF ₂ , SCH ₃ , SCF ₃ , SCHF ₂ , S(0) ₂ CH ₃ and S(0) ₂ CH ₂ CH ₃ .

Especially preferred are compounds of formula I, wherein B is N and the variables R, R ¹ , R ² , R ³ , R ⁴ and R ⁵ have the following meanings:

R is selected from Ci-C ₄ -alkyl, in particular from CH ₃ , CH ₂ CH ₃ , CH(CH ₃ ) ₂ and C(CH ₃ ) ₃ ; R ¹ is selected from the group consisting of halogen, nitro, Ci-C4-alkyl, Ci-C4-haloalkyl and Ci-C ₄ -alkyl-S(0) ₂ , in particular from CI, Br, F, nitro, CH ₃ , CH ₂ CH ₃ , CH(CH ₃ ) ₂ , CF ₃ , CHF ₂ , S(0) ₂ CH ₃ and S(0) ₂ CH ₂ CH ₃ ;

R ² is selected from the group consisting of hydrogen, halogen, Ci-C2-alkoxy-Ci-C2-alkyl,

Ci-C2-haloalkoxy-Ci-C2-alkyl, Ci-C4-alkylsulfonyl, Ci-C4-alkylsulfinyl, Ci-C4-alkylsulfanyl, isoxa- zolyl and isoxazolinyl, where the last two mentioned radicals may be unsubstituted or carry 1 or 2 radicals selected from halogen and Ci-C4-alkyl. In particular, R ² is selected from CH20CH ₃ , CH ₂ OCH ₂ CH ₃ , CH ₂ CH ₂ OCH ₃ , CH ₂ CH ₂ OCH ₂ CH ₃ , CH ₂ OCF ₃ , CH ₂ OCHF ₂ , CH ₂ OCH ₂ F,

CH2OCH2CHF2, CH ₂ OCH ₂ CF ₃ , CH ₂ OCF ₂ CF ₃ , methylsulfonyl, methylsulfinyl, methylsulfanyl, isoxazolyl and isoxazolinyl; R ³ is selected from the group consisting of hydrogen, halogen, CN, Ci-C4-haloalkyl and Ci-C ₄ -alkyl-S(0) ₂ , in particular from H, CI, F, CN, CF ₃ , CHF ₂ , S(0) ₂ CH ₃ and S(0) ₂ CH ₂ CH ₃ ;

R ⁴ and R ⁵ are identical or different and independently selected from the group consisting of H, F, CI, Br, I, CN, nitro, CH ₃ , CH ₂ CH ₃ , CH(CH ₃ ) ₂ , cyclopropyl, cyclopropylmethyl, CF ₃ , OCH ₃ , OCH ₂ CH ₃ , OCH(CH ₃ ) ₂ , CH ₂ OCH ₃ , CH ₂ OCH ₂ CH ₂ OCH ₃ , OCF ₃ , OCHF ₂ , SCH ₃ , SCF ₃ , SCH ₂ CH ₃ , SCH ₂ CF ₃ , SOCH ₃ , SOCH ₂ CH ₃ , S0 ₂ CH ₃ , S0 ₂ CH ₂ CH ₃ ; and more specifically R ⁴ and R ⁵ are identical or different and independently selected from the group consisting of H, F, CI, Br, I, CN, nitro, CH ₃ , CH ₂ CH ₃ , CH(CH ₃ ) ₂ , cyclopropyl, CF ₃ , OCH ₃ , OCF ₃ , SCH ₃ , SOCH ₃ , S0 ₂ CH ₃ or CH ₂ OCH ₃ ; provided that at least one of the radicals R ⁴ and R ⁵ is different from hydrogen; and further provided that if R ⁴ is hydrogen, halogen, cyano, nitro, Ci-C ₄ -alkyl or Ci-C ₄ -haloalkyl, R ⁵ is not hydrogen, halogen, Ci-C ₄ -alkyl or Ci-C ₄ -haloalkyl;

Specifically preferred are compounds of formula I, wherein B is N and the variables R, R ¹ , R ² , R ³ , R ⁴ and R ⁵ have the following meanings:

R is selected from the group consisting of methyl and ethyl;

R ¹ is selected from the group consisting of chlorine, nitro, methyl, trifluoromethyl and me- thylsulfonyl;

R ² is selected from the group consisting of hydrogen, CI, F, methyl, methylsulfonyl, me- thylsulfinyl, methylsulfanyl, 3-isoxazolinyl, 5-methyl-3-isoxazolinyl, 5-isoxazolinyl, 3-methyl-5- isoxazolinyl, 3-isoxazolyl, 5-methyl-3-isoxazolyl, 5-isoxazolyl and 3-methyl-5-isoxazolyl;

R ³ is selected from the group consisting of hydrogen, fluorine, chlorine, trifluoromethyl, CN and methylsulfonyl;

and either R ⁴ is H and R ⁵ is selected from the group consisting of CN, nitro, cyclopropyl, cyclopropylmethyl, OCH ₃ , OCH ₂ CH ₃ , OCH(CH ₃ ) ₂ , CH ₂ OCH ₃ , CH ₂ OCH ₂ CH ₂ OCH ₃ , OCF ₃ , OCHF ₂ , SCH ₃ , SCF ₃ , SCH ₂ CH ₃ , SCH ₂ CF ₃ , SOCH ₃ , SOCH ₂ CH ₃ , S0 ₂ CH ₃ , S0 ₂ CH ₂ CH ₃ ; more preferably R ⁵ is selected from the group consisting of CN, nitro, cyclopropyl, OCH ₃ , CH ₂ OCH ₃ , OCF ₃ , SCH ₃ , SOCHs, S0 ₂ CH ₃ ; or

R ⁵ is H and R ⁴ is selected from the group consisting of cyclopropyl, cyclopropylmethyl, OCH ₃ , OCH ₂ CH ₃ , OCH(CH ₃ ) ₂ , CH ₂ OCH ₃ , CH ₂ OCH ₂ CH ₂ OCH ₃ , OCF ₃ , OCHF ₂ , SCH ₃ , SCF ₃ , SCH ₂ CH ₃ , SCH ₂ CF ₃ , SOCH ₃ , SOCH ₂ CH ₃ , S0 ₂ CH ₃ , S0 ₂ CH ₂ CH ₃ ; more preferably R ⁴ is selected from the group consisting of cyclopropyl, OCH ₃ , CH ₂ OCH ₃ , OCF ₃ , SCH ₃ , SOCH ₃ , S0 ₂ CH ₃ .

Also specifically preferred are compounds of formula I, wherein B is N and the variables R, R ¹ , R ² , R ³ , R ⁴ and R ⁵ have the following meanings:

R is selected from the group consisting of methoxyethyl and methoxymethyl;

R ¹ is selected from the group consisting of chlorine, nitro, methyl, trifluoromethyl and me- thylsulfonyl;

R ² is selected from the group consisting of hydrogen, CI, F, methyl, methylsulfonyl, me- thylsulfinyl, methylsulfanyl, 3-isoxazolinyl, 5-methyl-3-isoxazolinyl, 5-isoxazolinyl, 3-methyl-5- isoxazolinyl, 3-isoxazolyl, 5-methyl-3-isoxazolyl, 5-isoxazolyl and 3-methyl-5-isoxazolyl;

R ³ is selected from the group consisting of hydrogen, fluorine, chlorine, trifluoromethyl, CN and methylsulfonyl;

and either R ⁴ is H and R ⁵ is selected from the group consisting of CN, nitro, cyclopropyl, cyclopropylmethyl, OCH ₃ , OCH ₂ CH ₃ , OCH(CH ₃ ) ₂ , CH ₂ OCH ₃ , CH ₂ OCH ₂ CH ₂ OCH ₃ , OCF ₃ , OCHF2, SCHs, SCFs, SCH2CH3, SCH2CF3, SOCH3, SOCH2CH3, SO2CH3, SO2CH2CH3; more preferably R ⁵ is selected from the group consisting of CN, nitro, cyclopropyl, OCH3, CH2OCH3, OCF3, SCH3, SOCH3, SO2CH3 ; or

R ⁵ is H and R ⁴ is selected from the group consisting of cyclopropyl, cyclopropylmethyl, OCH3, OCH2CH3, OCH(CH ₃ ) ₂ , CH2OCH3, CH2OCH2CH2OCH3, OCF3, OCHF2, SCH3, SCF ₃ , SCH2CH3, SCH2CF3, SOCH3, SOCH2CH3, SO2CH3, SO2CH2CH3; more preferably R ⁴ is selected from the group consisting of cyclopropyl, OCH ₃ , CH2OCH3, OCF ₃ , SCH ₃ , SOCH ₃ , SO2CH3.

Especially preferred are compounds of formula I, wherein B is CH and the variables R, R ¹ , R ² , R ³ , R ⁴ and R ⁵ have the following meanings:

R is selected from Ci-C ₄ -alkyl, in particular from CH ₃ , CH2CH3, CH(CH ₃ ) ₂ and C(CH ₃ ) ₃ ; R ¹ is selected from the group consisting of halogen, nitro, Ci-C ₄ -alkyl, Ci-C ₄ -haloalkyl and Ci-C ₄ -alkyl-S(0) ₂ , in particular from CI, Br, F, nitro, CH ₃ , CH2CH3, CH(CH ₃ ) ₂ , CF ₃ , CHF ₂ , S(0) ₂ CH ₃ and S(0) ₂ CH ₂ CH ₃ ;

R ² is selected from the group consisting of hydrogen, halogen, Ci-C2-alkoxy-Ci-C2-alkyl,

Ci-C2-haloalkoxy-Ci-C2-alkyl, Ci-C ₄ -alkylsulfonyl, Ci-C ₄ -alkylsulfinyl, Ci-C ₄ -alkylsulfanyl, isoxa- zolyl and isoxazolinyl, where the last two mentioned radicals may be unsubstituted or carry 1 or 2 radicals selected from halogen and Ci-C ₄ -alkyl. In particular, R ² is selected from CH2OCH3, CH2OCH2CH3, CH2CH2OCH3, CH2CH2OCH2CH3, CH2OCF3, CH2OCHF2, CH2OCH2F,

CH2OCH2CHF2, CH2OCH2CF3, CH2OCF2CF3, methylsulfonyl, methylsulfinyl, methylsulfanyl, isoxazolyl and isoxazolinyl;

R ³ is selected from the group consisting of hydrogen, halogen, CN, Ci-C ₄ -haloalkyl and Ci-C ₄ -alkyl-S(0) ₂ , in particular from H, CI, F, CN, CF ₃ , CHF ₂ , S(0) ₂ CH ₃ and S(0) ₂ CH ₂ CH ₃ ;

R ⁴ and R ⁵ are identical or different and independently selected from the group consisting of H, F, CI, Br, I, CN, nitro, CH ₃ , CH2CH3, CH(CH ₃ ) ₂ , cyclopropyl, cyclopropylmethyl, CF ₃ , OCH ₃ , OCH2CH3, OCH(CH ₃ ) ₂ , CH2OCH3, CH2OCH2CH2OCH3, OCF3, OCHF2, SCH3, SCFs, SCH2CH3, SCH2CF3, SOCH3, SOCH2CH3, SO2CH3, SO2CH2CH3; and more specifically R ⁴ and R ⁵ are identical or different and independently selected from the group consisting of H, F, CI, Br, I, CN, nitro, CH ₃ , CH2CH3, CH(CH ₃ ) ₂ , cyclopropyl, CF ₃ , OCH ₃ , OCF ₃ , SCH ₃ , SOCH ₃ , SO2CH3 or CH2OCH3; provided that at least one of the radicals R ⁴ and R ⁵ is different from hydrogen; and further provided that if R ⁴ is hydrogen, halogen, cyano, nitro, Ci-C ₄ -alkyl or Ci-C ₄ -haloalkyl, R ⁵ is not hydrogen, halogen, Ci-C ₄ -alkyl or Ci-C ₄ -haloalkyl;

Specifically preferred are compounds of formula I, wherein B is CH and the variables R, R ¹ , R ² , R ³ , R ⁴ and R ⁵ have the following meanings:

R is selected from the group consisting of methyl and ethyl;

R ¹ is selected from the group consisting of chlorine, nitro, methyl, trifluoromethyl and methylsulfonyl;

R ² is selected from the group consisting of hydrogen, CI, F, methyl, methylsulfonyl, methylsulfinyl, methylsulfanyl, 3-isoxazolinyl, 5-methyl-3-isoxazolinyl, 5-isoxazolinyl, 3-methyl-5- isoxazolinyl, 3-isoxazolyl, 5-methyl-3-isoxazolyl, 5-isoxazolyl and 3-methyl-5-isoxazolyl;

R ³ is selected from the group consisting of hydrogen, fluorine, chlorine, trifluoromethyl, CN and methylsulfonyl; and either R ⁴ is H and R ⁵ is selected from the group consisting of CN, nitro, cyclopropyl, cyclopropyl methyl, OCH ₃ , OCH ₂ CH ₃ , OCH(CH ₃ ) ₂ , CH ₂ OCH ₃ , CH ₂ OCH ₂ CH ₂ OCH ₃ , OCF ₃ , OCHF ₂ , SCH ₃ , SCF ₃ , SCH ₂ CH ₃ , SCH ₂ CF ₃ , SOCH ₃ , SOCH ₂ CH ₃ , S0 ₂ CH ₃ , S0 ₂ CH ₂ CH ₃ ; more preferably R ⁵ is selected from the group consisting of CN, nitro, cyclopropyl, OCH ₃ , CH ₂ OCH ₃ , OCF ₃ , SCH ₃ , SOCHs, S0 ₂ CH ₃ ; or

R ⁵ is H and R ⁴ is selected from the group consisting of cyclopropyl, cyclopropylmethyl, OCH ₃ , OCH ₂ CH ₃ , OCH(CH ₃ ) ₂ , CH ₂ OCH ₃ , CH ₂ OCH ₂ CH ₂ OCH ₃ , OCF ₃ , OCHF ₂ , SCH ₃ , SCF ₃ , SCH ₂ CH ₃ , SCH ₂ CF ₃ , SOCH ₃ , SOCH ₂ CH ₃ , S0 ₂ CH ₃ , S0 ₂ CH ₂ CH ₃ ; more preferably R ⁴ is selected from the group consisting of cyclopropyl, OCH ₃ , CH ₂ OCH ₃ , OCF ₃ , SCH ₃ , SOCH ₃ , S0 ₂ CH ₃ .

Also specifically preferred are compounds of formula I, wherein B is CH and the variables

R, R ¹ , R ² , R ³ , R ⁴ and R ⁵ have the following meanings:

R is selected from the group consisting of methoxyethyl and methoxymethyl;

R ¹ is selected from the group consisting of chlorine, nitro, methyl, trifluoromethyl and me- thylsulfonyl;

R ² is selected from the group consisting of hydrogen, CI, F, methyl, methylsulfonyl, me- thylsulfinyl, methylsulfanyl, 3-isoxazolinyl, 5-methyl-3-isoxazolinyl, 5-isoxazolinyl, 3-methyl-5- isoxazolinyl, 3-isoxazolyl, 5-methyl-3-isoxazolyl, 5-isoxazolyl and 3-methyl-5-isoxazolyl;

R ³ is selected from the group consisting of hydrogen, fluorine, chlorine, trifluoromethyl, CN and methylsulfonyl;

and either R ⁴ is H and R ⁵ is selected from the group consisting of CN, nitro, cyclopropyl, cyclopropylmethyl, OCH ₃ , OCH ₂ CH ₃ , OCH(CH ₃ ) ₂ , CH ₂ OCH ₃ , CH ₂ OCH ₂ CH ₂ OCH ₃ , OCF ₃ , OCHF ₂ , SCH ₃ , SCF ₃ , SCH ₂ CH ₃ , SCH ₂ CF ₃ , SOCH ₃ , SOCH ₂ CH ₃ , S0 ₂ CH ₃ , S0 ₂ CH ₂ CH ₃ ; more preferably R ⁵ is selected from the group consisting of CN, nitro, cyclopropyl, OCH ₃ , CH ₂ OCH ₃ , OCF ₃ , SCH ₃ , SOCHs, S0 ₂ CH ₃ ; or

R ⁵ is H and R ⁴ is selected from the group consisting of cyclopropyl, cyclopropylmethyl,

OCH ₃ , OCH ₂ CH ₃ , OCH(CH ₃ ) ₂ , CH ₂ OCH ₃ , CH ₂ OCH ₂ CH ₂ OCH ₃ , OCF ₃ , OCHF ₂ , SCH ₃ , SCF ₃ , SCH ₂ CH ₃ , SCH ₂ CF ₃ , SOCH ₃ , SOCH ₂ CH ₃ , S0 ₂ CH ₃ , S0 ₂ CH ₂ CH ₃ ; more preferably R ⁴ is selected from the group consisting of cyclopropyl, OCH ₃ , CH ₂ OCH ₃ , OCF ₃ , SCH ₃ , SOCH ₃ , S0 ₂ CH ₃ . Examples of preferred compounds are the individual compounds compiled in Tables 1 to

8 below. Moreover, the meanings mentioned below for the individual variables in the Tables are per se, independently of the combination in which they are mentioned, a particularly preferred embodiment of the substituents in question.

Table 1 Compounds of formula I (I.A-1 - I.A-5280) in which B is CH and R is methyl and the combination of R ¹ , R ² , R ³ , R ⁴ and R ⁵ for a compound corresponds in each case to one row of Table A;

Table 2 Compounds of formula I (I I.A-1 - II.A-5280) in which B is CH and R is ethyl and the combination of R ¹ , R ² , R ³ , R ⁴ and R ⁵ for a compound corresponds in each case to one row of Table A;

Table 3 Compounds of formula I (I I I.A-1 - III.A-5280) in which B is CH and R is methoxymethyl and the combination of R ¹ , R ² , R ³ , R ⁴ and R ⁵ for a compound corresponds in each case to one row of Table A; Table 4 Compounds of formula I (IV.A-1 - IV.A-5280) in which B is CH and R is methoxy- ethyl and the combination of R ¹ , R ² , R ³ , R ⁴ and R ⁵ for a compound corresponds in each case to one row of Table A;

Table 5 Compounds of formula I (V.A-1 - V.A-5280) in which B is N and R is methyl and the combination of R ¹ , R ² , R ³ , R ⁴ and R ⁵ for a compound corresponds in each case to one row of Table A;

Table 6 Compounds of formula I (VI.A-1 - VI.A-5280) in which B is N and R is ethyl and the combination of R ¹ , R ² , R ³ , R ⁴ and R ⁵ for a compound corresponds in each case to one row of Table A;

Table 7 Compounds of formula I (VII.A-1 - VII.A-5280) in which B is N and R is methox- ymethyl and the combination of R ¹ , R ² , R ³ , R ⁴ and R ⁵ for a compound corresponds in each case to one row of Table A;

Table 8 Compounds of formula I (VIII.A-1 - VIII.A-5280) in which B is N and R is methoxy- ethyl and the combination of R ¹ , R ² , R ³ , R ⁴ and R ⁵ for a compound corresponds in each case to one row of Table A;

Table A

A-391 CI CH20CH2CF3 CI H SOCH3

A-392 CI CH20CH2CF3 CI H SO2CH3

A-393 CI CH20CH2CF3 CI H CH2OCH3

A-394 CI CH20CH2CF3 CI cyclopropyl H

A-395 CI CH20CH2CF3 CI OCH3 H

A-396 CI CH20CH2CF3 CI OCF3 H

A-397 CI CH20CH2CF3 CI SCH ₃ H

A-398 CI CH20CH2CF3 CI SOCH3 H

A-399 CI CH20CH2CF3 CI SO2CH3 H

A-400 CI CH20CH2CF3 CI CH2OCH3 H

A-401 CI CH20CH2CF3 F H CN

A-402 CI CH20CH2CF3 F H N0 ₂

A-403 CI CH20CH2CF3 F H cyclopropyl

A-404 CI CH20CH2CF3 F H OCH3

A-405 CI CH20CH2CF3 F H OCF3

A-406 CI CH20CH2CF3 F H SCH ₃

A-407 CI CH20CH2CF3 F H SOCH3

A-408 CI CH20CH2CF3 F H SO2CH3

A-409 CI CH20CH2CF3 F H CH2OCH3

A-410 CI CH20CH2CF3 F cyclopropyl H

A-41 1 CI CH20CH2CF3 F OCH3 H

A-412 CI CH20CH2CF3 F OCF3 H

A-413 CI CH20CH2CF3 F SCH ₃ H

A-414 CI CH20CH2CF3 F SOCH3 H

A-415 CI CH20CH2CF3 F SO2CH3 H

A-416 CI CH20CH2CF3 F CH2OCH3 H

A-417 CI CH20CH2CF3 CF ₃ H CN

A-418 CI CH20CH2CF3 CF ₃ H N0 ₂

A-419 CI CH20CH2CF3 CF ₃ H cyclopropyl

A-420 CI CH20CH2CF3 CF ₃ H OCH3

A-421 CI CH20CH2CF3 CF ₃ H OCF3

A-422 CI CH20CH2CF3 CF ₃ H SCH ₃

A-423 CI CH20CH2CF3 CF ₃ H SOCH3

A-424 CI CH20CH2CF3 CF ₃ H SO2CH3

A-425 CI CH20CH2CF3 CF ₃ H CH2OCH3

A-426 CI CH20CH2CF3 CF ₃ cyclopropyl H

A-427 CI CH20CH2CF3 CF ₃ OCH3 H A-428 CI CH20CH2CF3 CF ₃ OCF3 H

A-429 CI CH20CH2CF3 CF ₃ SCH ₃ H

A-430 CI CH20CH2CF3 CF ₃ SOCH3 H

A-431 CI CH20CH2CF3 CF ₃ SO2CH3 H

A-432 CI CH20CH2CF3 CF ₃ CH2OCH3 H

A-433 CI CH20CH2CF3 S02CH3 H CN

A-434 CI CH20CH2CF3 S02CH3 H N0 ₂

A-435 CI CH20CH2CF3 S02CH3 H cyclopropyl

A-436 CI CH20CH2CF3 S02CH3 H OCH3

A-437 CI CH20CH2CF3 S02CH3 H OCF3

A-438 CI CH20CH2CF3 S02CH3 H SCH ₃

A-439 CI CH20CH2CF3 S02CH3 H SOCH3

A-440 CI CH20CH2CF3 S02CH3 H SO2CH3

A-441 CI CH20CH2CF3 S02CH3 H CH2OCH3

A-442 CI CH20CH2CF3 S02CH3 cyclopropyl H

A-443 CI CH20CH2CF3 S02CH3 OCH3 H

A-444 CI CH20CH2CF3 S02CH3 OCF3 H

A-445 CI CH20CH2CF3 S02CH3 SCH ₃ H

A-446 CI CH20CH2CF3 S02CH3 SOCH3 H

A-447 CI CH20CH2CF3 S02CH3 SO2CH3 H

A-448 CI CH20CH2CF3 S02CH3 CH2OCH3 H

A-449 CI CH20CH2CF3 CN H CN

A-450 CI CH20CH2CF3 CN H N0 ₂

A-451 CI CH20CH2CF3 CN H cyclopropyl

A-452 CI CH20CH2CF3 CN H OCH3

A-453 CI CH20CH2CF3 CN H OCF3

A-454 CI CH20CH2CF3 CN H SCH ₃

A-455 CI CH20CH2CF3 CN H SOCH3

A-456 CI CH20CH2CF3 CN H SO2CH3

A-457 CI CH20CH2CF3 CN H CH2OCH3

A-458 CI CH20CH2CF3 CN cyclopropyl H

A-459 CI CH20CH2CF3 CN OCH3 H

A-460 CI CH20CH2CF3 CN OCF3 H

A-461 CI CH20CH2CF3 CN SCH ₃ H

A-462 CI CH20CH2CF3 CN SOCH3 H

A-463 CI CH20CH2CF3 CN SO2CH3 H

A-464 CI CH20CH2CF3 CN CH2OCH3 H A-465 CI CH20CH2CF3 H H CN

A-466 CI CH20CH2CF3 H H N0 ₂

A-467 CI CH20CH2CF3 H H cyclopropyl

A-468 CI CH20CH2CF3 H H OCH3

A-469 CI CH20CH2CF3 H H OCF3

A-470 CI CH20CH2CF3 H H SCH ₃

A-471 CI CH20CH2CF3 H H SOCH3

A-472 CI CH20CH2CF3 H H SO2CH3

A-473 CI CH20CH2CF3 H H CH2OCH3

A-474 CI CH20CH2CF3 H cyclopropyl H

A-475 CI CH20CH2CF3 H OCH3 H

A-476 CI CH20CH2CF3 H OCF3 H

A-477 CI CH20CH2CF3 H SCH ₃ H

A-478 CI CH20CH2CF3 H SOCH3 H

A-479 CI CH20CH2CF3 H SO2CH3 H

A-480 CI CH20CH2CF3 H CH2OCH3 H

A-481 CI lsoxazolin-3-yl CI H CN

A-482 CI lsoxazolin-3-yl CI H N0 ₂

A-483 CI lsoxazolin-3-yl CI H cyclopropyl

A-484 CI lsoxazolin-3-yl CI H OCH3

A-485 CI lsoxazolin-3-yl CI H OCF3

A-486 CI lsoxazolin-3-yl CI H SCH ₃

A-487 CI lsoxazolin-3-yl CI H SOCH3

A-488 CI lsoxazolin-3-yl CI H SO2CH3

A-489 CI lsoxazolin-3-yl CI H CH2OCH3

A-490 CI lsoxazolin-3-yl CI cyclopropyl H

A-491 CI lsoxazolin-3-yl CI OCH3 H

A-492 CI lsoxazolin-3-yl CI OCF3 H

A-493 CI lsoxazolin-3-yl CI SCH ₃ H

A-494 CI lsoxazolin-3-yl CI SOCH3 H

A-495 CI lsoxazolin-3-yl CI SO2CH3 H

A-496 CI lsoxazolin-3-yl CI CH2OCH3 H

A-497 CI lsoxazolin-3-yl F H CN

A-498 CI lsoxazolin-3-yl F H N0 ₂

A-499 CI lsoxazolin-3-yl F H cyclopropyl

A-500 CI lsoxazolin-3-yl F H OCH3

A-501 CI lsoxazolin-3-yl F H OCF3 A-502 CI lsoxazolin-3-yl F H SCHs

A-503 CI lsoxazolin-3-yl F H SOCH3

A-504 CI lsoxazolin-3-yl F H SO2CH3

A-505 CI lsoxazolin-3-yl F H CH2OCH3

A-506 CI lsoxazolin-3-yl F cyclopropyl H

A-507 CI lsoxazolin-3-yl F OCHs H

A-508 CI lsoxazolin-3-yl F OCF3 H

A-509 CI lsoxazolin-3-yl F SCHs H

A-510 CI lsoxazolin-3-yl F SOCH3 H

A-51 1 CI lsoxazolin-3-yl F SO2CH3 H

A-512 CI lsoxazolin-3-yl F CH2OCH3 H

A-513 CI lsoxazolin-3-yl CFs H CN

A-514 CI lsoxazolin-3-yl CFs H N0 ₂

A-515 CI lsoxazolin-3-yl CFs H cyclopropyl

A-516 CI lsoxazolin-3-yl CFs H OCHs

A-517 CI lsoxazolin-3-yl CFs H OCF3

A-518 CI lsoxazolin-3-yl CFs H SCHs

A-519 CI lsoxazolin-3-yl CFs H SOCH3

A-520 CI lsoxazolin-3-yl CFs H SO2CH3

A-521 CI lsoxazolin-3-yl CFs H CH2OCH3

A-522 CI lsoxazolin-3-yl CFs cyclopropyl H

A-523 CI lsoxazolin-3-yl CFs OCHs H

A-524 CI lsoxazolin-3-yl CFs OCF3 H

A-525 CI lsoxazolin-3-yl CFs SCHs H

A-526 CI lsoxazolin-3-yl CFs SOCH3 H

A-527 CI lsoxazolin-3-yl CFs SO2CH3 H

A-528 CI lsoxazolin-3-yl CFs CH2OCH3 H

A-529 CI lsoxazolin-3-yl SO2CH3 H CN

A-530 CI lsoxazolin-3-yl SO2CH3 H N0 ₂

A-531 CI lsoxazolin-3-yl SO2CH3 H cyclopropyl

A-532 CI lsoxazolin-3-yl SO2CH3 H OCHs

A-533 CI lsoxazolin-3-yl SO2CH3 H OCF3

A-534 CI lsoxazolin-3-yl SO2CH3 H SCHs

A-535 CI lsoxazolin-3-yl SO2CH3 H SOCH3

A-536 CI lsoxazolin-3-yl SO2CH3 H SO2CH3

A-537 CI lsoxazolin-3-yl SO2CH3 H CH2OCH3

A-538 CI lsoxazolin-3-yl SO2CH3 cyclopropyl H A-539 CI lsoxazolin-3-yl SO2CH3 OCH3 H

A-540 CI lsoxazolin-3-yl SO2CH3 OCF3 H

A-541 CI lsoxazolin-3-yl SO2CH3 SCH ₃ H

A-542 CI lsoxazolin-3-yl SO2CH3 SOCH3 H

A-543 CI lsoxazolin-3-yl SO2CH3 SO2CH3 H

A-544 CI lsoxazolin-3-yl SO2CH3 CH2OCH3 H

A-545 CI lsoxazolin-3-yl CN H CN

A-546 CI lsoxazolin-3-yl CN H N0 ₂

A-547 CI lsoxazolin-3-yl CN H cyclopropyl

A-548 CI lsoxazolin-3-yl CN H OCH3

A-549 CI lsoxazolin-3-yl CN H OCF3

A-550 CI lsoxazolin-3-yl CN H SCH ₃

A-551 CI lsoxazolin-3-yl CN H SOCH3

A-552 CI lsoxazolin-3-yl CN H SO2CH3

A-553 CI lsoxazolin-3-yl CN H CH2OCH3

A-554 CI lsoxazolin-3-yl CN cyclopropyl H

A-555 CI lsoxazolin-3-yl CN OCH3 H

A-556 CI lsoxazolin-3-yl CN OCF3 H

A-557 CI lsoxazolin-3-yl CN SCH ₃ H

A-558 CI lsoxazolin-3-yl CN SOCH3 H

A-559 CI lsoxazolin-3-yl CN SO2CH3 H

A-560 CI lsoxazolin-3-yl CN CH2OCH3 H

A-561 CI lsoxazolin-3-yl H H CN

A-562 CI lsoxazolin-3-yl H H N0 ₂

A-563 CI lsoxazolin-3-yl H H cyclopropyl

A-564 CI lsoxazolin-3-yl H H OCH3

A-565 CI lsoxazolin-3-yl H H OCF3

A-566 CI lsoxazolin-3-yl H H SCH ₃

A-567 CI lsoxazolin-3-yl H H SOCH3

A-568 CI lsoxazolin-3-yl H H SO2CH3

A-569 CI lsoxazolin-3-yl H H CH2OCH3

A-570 CI lsoxazolin-3-yl H cyclopropyl H

A-571 CI lsoxazolin-3-yl H OCH3 H

A-572 CI lsoxazolin-3-yl H OCF3 H

A-573 CI lsoxazolin-3-yl H SCH ₃ H

A-574 CI lsoxazolin-3-yl H SOCH3 H

A-575 CI lsoxazolin-3-yl H SO2CH3 H A-576 CI lsoxazolin-3-yl H CH2OCH3 H

A-577 CI 5-Me-lsoxazolin-3-yl CI H CN

A-578 CI 5-Me-lsoxazolin-3-yl CI H N0 ₂

A-579 CI 5-Me-lsoxazolin-3-yl CI H cyclopropyl

A-580 CI 5-Me-lsoxazolin-3-yl CI H OCHs

A-581 CI 5-Me-lsoxazolin-3-yl CI H OCFs

A-582 CI 5-Me-lsoxazolin-3-yl CI H SCHs

A-583 CI 5-Me-lsoxazolin-3-yl CI H SOCHs

A-584 CI 5-Me-lsoxazolin-3-yl CI H SO2CH3

A-585 CI 5-Me-lsoxazolin-3-yl CI H CH2OCH3

A-586 CI 5-Me-lsoxazolin-3-yl CI cyclopropyl H

A-587 CI 5-Me-lsoxazolin-3-yl CI OCHs H

A-588 CI 5-Me-lsoxazolin-3-yl CI OCFs H

A-589 CI 5-Me-lsoxazolin-3-yl CI SCHs H

A-590 CI 5-Me-lsoxazolin-3-yl CI SOCHs H

A-591 CI 5-Me-lsoxazolin-3-yl CI SO2CH3 H

A-592 CI 5-Me-lsoxazolin-3-yl CI CH2OCH3 H

A-593 CI 5-Me-lsoxazolin-3-yl F H CN

A-594 CI 5-Me-lsoxazolin-3-yl F H N0 ₂

A-595 CI 5-Me-lsoxazolin-3-yl F H cyclopropyl

A-596 CI 5-Me-lsoxazolin-3-yl F H OCHs

A-597 CI 5-Me-lsoxazolin-3-yl F H OCFs

A-598 CI 5-Me-lsoxazolin-3-yl F H SCHs

A-599 CI 5-Me-lsoxazolin-3-yl F H SOCHs

A-600 CI 5-Me-lsoxazolin-3-yl F H SO2CH3

A-601 CI 5-Me-lsoxazolin-3-yl F H CH2OCH3

A-602 CI 5-Me-lsoxazolin-3-yl F cyclopropyl H

A-603 CI 5-Me-lsoxazolin-3-yl F OCHs H

A-604 CI 5-Me-lsoxazolin-3-yl F OCFs H

A-605 CI 5-Me-lsoxazolin-3-yl F SCHs H

A-606 CI 5-Me-lsoxazolin-3-yl F SOCHs H

A-607 CI 5-Me-lsoxazolin-3-yl F SO2CH3 H

A-608 CI 5-Me-lsoxazolin-3-yl F CH2OCH3 H

A-609 CI 5-Me-lsoxazolin-3-yl CFs H CN

A-610 CI 5-Me-lsoxazolin-3-yl CFs H N0 ₂

A-61 1 CI 5-Me-lsoxazolin-3-yl CFs H cyclopropyl

A-612 CI 5-Me-lsoxazolin-3-yl CFs H OCHs A-613 CI 5-Me-lsoxazolin-3-yl CFs H OCFs

A-614 CI 5-Me-lsoxazolin-3-yl CFs H SCHs

A-615 CI 5-Me-lsoxazolin-3-yl CFs H SOCHs

A-616 CI 5-Me-lsoxazolin-3-yl CFs H SO2CH3

A-617 CI 5-Me-lsoxazolin-3-yl CFs H CH2OCH3

A-618 CI 5-Me-lsoxazolin-3-yl CFs cyclopropyl H

A-619 CI 5-Me-lsoxazolin-3-yl CFs OCHs H

A-620 CI 5-Me-lsoxazolin-3-yl CFs OCF3 H

A-621 CI 5-Me-lsoxazolin-3-yl CFs SCHs H

A-622 CI 5-Me-lsoxazolin-3-yl CFs SOCH3 H

A-623 CI 5-Me-lsoxazolin-3-yl CFs SO2CH3 H

A-624 CI 5-Me-lsoxazolin-3-yl CFs CH2OCH3 H

A-625 CI 5-Me-lsoxazolin-3-yl SO2CH3 H CN

A-626 CI 5-Me-lsoxazolin-3-yl SO2CH3 H N0 ₂

A-627 CI 5-Me-lsoxazolin-3-yl SO2CH3 H cyclopropyl

A-628 CI 5-Me-lsoxazolin-3-yl SO2CH3 H OCHs

A-629 CI 5-Me-lsoxazolin-3-yl SO2CH3 H OCFs

A-630 CI 5-Me-lsoxazolin-3-yl SO2CH3 H SCHs

A-631 CI 5-Me-lsoxazolin-3-yl SO2CH3 H SOCHs

A-632 CI 5-Me-lsoxazolin-3-yl SO2CH3 H SO2CH3

A-633 CI 5-Me-lsoxazolin-3-yl SO2CH3 H CH2OCH3

A-634 CI 5-Me-lsoxazolin-3-yl SO2CH3 cyclopropyl H

A-635 CI 5-Me-lsoxazolin-3-yl SO2CH3 OCHs H

A-636 CI 5-Me-lsoxazolin-3-yl SO2CH3 OCF3 H

A-637 CI 5-Me-lsoxazolin-3-yl SO2CH3 SCHs H

A-638 CI 5-Me-lsoxazolin-3-yl SO2CH3 SOCH3 H

A-639 CI 5-Me-lsoxazolin-3-yl SO2CH3 SO2CH3 H

A-640 CI 5-Me-lsoxazolin-3-yl SO2CH3 CH2OCH3 H

A-641 CI 5-Me-lsoxazolin-3-yl CN H CN

A-642 CI 5-Me-lsoxazolin-3-yl CN H N0 ₂

A-643 CI 5-Me-lsoxazolin-3-yl CN H cyclopropyl

A-644 CI 5-Me-lsoxazolin-3-yl CN H OCHs

A-645 CI 5-Me-lsoxazolin-3-yl CN H OCFs

A-646 CI 5-Me-lsoxazolin-3-yl CN H SCHs

A-647 CI 5-Me-lsoxazolin-3-yl CN H SOCHs

A-648 CI 5-Me-lsoxazolin-3-yl CN H SO2CH3

A-649 CI 5-Me-lsoxazolin-3-yl CN H CH2OCH3 A-650 CI 5-Me-lsoxazolin-3-yl CN cyclopropyl H

A-651 CI 5-Me-lsoxazolin-3-yl CN OCHs H

A-652 CI 5-Me-lsoxazolin-3-yl CN OCF3 H

A-653 CI 5-Me-lsoxazolin-3-yl CN SCHs H

A-654 CI 5-Me-lsoxazolin-3-yl CN SOCH3 H

A-655 CI 5-Me-lsoxazolin-3-yl CN SO2CH3 H

A-656 CI 5-Me-lsoxazolin-3-yl CN CH2OCH3 H

A-657 CI 5-Me-lsoxazolin-3-yl H H CN

A-658 CI 5-Me-lsoxazolin-3-yl H H N0 ₂

A-659 CI 5-Me-lsoxazolin-3-yl H H cyclopropyl

A-660 CI 5-Me-lsoxazolin-3-yl H H OCH3

A-661 CI 5-Me-lsoxazolin-3-yl H H OCF3

A-662 CI 5-Me-lsoxazolin-3-yl H H SCH ₃

A-663 CI 5-Me-lsoxazolin-3-yl H H SOCH3

A-664 CI 5-Me-lsoxazolin-3-yl H H SO2CH3

A-665 CI 5-Me-lsoxazolin-3-yl H H CH2OCH3

A-666 CI 5-Me-lsoxazolin-3-yl H cyclopropyl H

A-667 CI 5-Me-lsoxazolin-3-yl H OCH3 H

A-668 CI 5-Me-lsoxazolin-3-yl H OCF3 H

A-669 CI 5-Me-lsoxazolin-3-yl H SCH ₃ H

A-670 CI 5-Me-lsoxazolin-3-yl H SOCH3 H

A-671 CI 5-Me-lsoxazolin-3-yl H SO2CH3 H

A-672 CI 5-Me-lsoxazolin-3-yl H CH2OCH3 H

A-673 CI lsoxazol-3-yl CI H CN

A-674 CI lsoxazol-3-yl CI H N0 ₂

A-675 CI lsoxazol-3-yl CI H cyclopropyl

A-676 CI lsoxazol-3-yl CI H OCH3

A-677 CI lsoxazol-3-yl CI H OCF3

A-678 CI lsoxazol-3-yl CI H SCH ₃

A-679 CI lsoxazol-3-yl CI H SOCH3

A-680 CI lsoxazol-3-yl CI H SO2CH3

A-681 CI lsoxazol-3-yl CI H CH2OCH3

A-682 CI lsoxazol-3-yl CI cyclopropyl H

A-683 CI lsoxazol-3-yl CI OCH3 H

A-684 CI lsoxazol-3-yl CI OCF3 H

A-685 CI lsoxazol-3-yl CI SCH ₃ H

A-686 CI lsoxazol-3-yl CI SOCH3 H A-687 CI lsoxazol-3-yl CI SO2CH3 H

A-688 CI lsoxazol-3-yl CI CH2OCH3 H

A-689 CI lsoxazol-3-yl F H CN

A-690 CI lsoxazol-3-yl F H N0 ₂

A-691 CI lsoxazol-3-yl F H cyclopropyl

A-692 CI lsoxazol-3-yl F H OCH3

A-693 CI lsoxazol-3-yl F H OCFs

A-694 CI lsoxazol-3-yl F H SCHs

A-695 CI lsoxazol-3-yl F H SOCHs

A-696 CI lsoxazol-3-yl F H SO2CH3

A-697 CI lsoxazol-3-yl F H CH2OCH3

A-698 CI lsoxazol-3-yl F cyclopropyl H

A-699 CI lsoxazol-3-yl F OCH3 H

A-700 CI lsoxazol-3-yl F OCFs H

A-701 CI lsoxazol-3-yl F SCHs H

A-702 CI lsoxazol-3-yl F SOCHs H

A-703 CI lsoxazol-3-yl F SO2CH3 H

A-704 CI lsoxazol-3-yl F CH2OCH3 H

A-705 CI lsoxazol-3-yl CFs H CN

A-706 CI lsoxazol-3-yl CFs H N0 ₂

A-707 CI lsoxazol-3-yl CFs H cyclopropyl

A-708 CI lsoxazol-3-yl CFs H OCH3

A-709 CI lsoxazol-3-yl CFs H OCFs

A-710 CI lsoxazol-3-yl CFs H SCHs

A-71 1 CI lsoxazol-3-yl CFs H SOCHs

A-712 CI lsoxazol-3-yl CFs H SO2CH3

A-713 CI lsoxazol-3-yl CFs H CH2OCH3

A-714 CI lsoxazol-3-yl CFs cyclopropyl H

A-715 CI lsoxazol-3-yl CFs OCH3 H

A-716 CI lsoxazol-3-yl CFs OCFs H

A-717 CI lsoxazol-3-yl CFs SCHs H

A-718 CI lsoxazol-3-yl CFs SOCHs H

A-719 CI lsoxazol-3-yl CFs SO2CH3 H

A-720 CI lsoxazol-3-yl CFs CH2OCH3 H

A-721 CI lsoxazol-3-yl SO2CH3 H CN

A-722 CI lsoxazol-3-yl SO2CH3 H N0 ₂

A-723 CI lsoxazol-3-yl SO2CH3 H cyclopropyl A-724 CI lsoxazol-3-yl SO2CH3 H OCH3

A-725 CI lsoxazol-3-yl SO2CH3 H OCF3

A-726 CI lsoxazol-3-yl SO2CH3 H SCH ₃

A-727 CI lsoxazol-3-yl SO2CH3 H SOCH3

A-728 CI lsoxazol-3-yl SO2CH3 H SO2CH3

A-729 CI lsoxazol-3-yl SO2CH3 H CH2OCH3

A-730 CI lsoxazol-3-yl SO2CH3 cyclopropyl H

A-731 CI lsoxazol-3-yl SO2CH3 OCH3 H

A-732 CI lsoxazol-3-yl SO2CH3 OCF3 H

A-733 CI lsoxazol-3-yl SO2CH3 SCH ₃ H

A-734 CI lsoxazol-3-yl SO2CH3 SOCH3 H

A-735 CI lsoxazol-3-yl SO2CH3 SO2CH3 H

A-736 CI lsoxazol-3-yl SO2CH3 CH2OCH3 H

A-737 CI lsoxazol-3-yl CN H CN

A-738 CI lsoxazol-3-yl CN H N0 ₂

A-739 CI lsoxazol-3-yl CN H cyclopropyl

A-740 CI lsoxazol-3-yl CN H OCH3

A-741 CI lsoxazol-3-yl CN H OCF3

A-742 CI lsoxazol-3-yl CN H SCH ₃

A-743 CI lsoxazol-3-yl CN H SOCH3

A-744 CI lsoxazol-3-yl CN H SO2CH3

A-745 CI lsoxazol-3-yl CN H CH2OCH3

A-746 CI lsoxazol-3-yl CN cyclopropyl H

A-747 CI lsoxazol-3-yl CN OCH3 H

A-748 CI lsoxazol-3-yl CN OCF3 H

A-749 CI lsoxazol-3-yl CN SCH ₃ H

A-750 CI lsoxazol-3-yl CN SOCH3 H

A-751 CI lsoxazol-3-yl CN SO2CH3 H

A-752 CI lsoxazol-3-yl CN CH2OCH3 H

A-753 CI lsoxazol-3-yl H H CN

A-754 CI lsoxazol-3-yl H H N0 ₂

A-755 CI lsoxazol-3-yl H H cyclopropyl

A-756 CI lsoxazol-3-yl H H OCH3

A-757 CI lsoxazol-3-yl H H OCF3

A-758 CI lsoxazol-3-yl H H SCH ₃

A-759 CI lsoxazol-3-yl H H SOCH3

A-760 CI lsoxazol-3-yl H H SO2CH3 A-761 CI lsoxazol-3-yl H H CH2OCH3

A-762 CI lsoxazol-3-yl H cyclopropyl H

A-763 CI lsoxazol-3-yl H OCHs H

A-764 CI lsoxazol-3-yl H OCF3 H

A-765 CI lsoxazol-3-yl H SCHs H

A-766 CI lsoxazol-3-yl H SOCH3 H

A-767 CI lsoxazol-3-yl H SO2CH3 H

A-768 CI lsoxazol-3-yl H CH2OCH3 H

A-769 CI 5-Me-lsoxazol-3-yl CI H CN

A-770 CI 5-Me-lsoxazol-3-yl CI H N0 ₂

A-771 CI 5-Me-lsoxazol-3-yl CI H cyclopropyl

A-772 CI 5-Me-lsoxazol-3-yl CI H OCH3

A-773 CI 5-Me-lsoxazol-3-yl CI H OCF3

A-774 CI 5-Me-lsoxazol-3-yl CI H SCH ₃

A-775 CI 5-Me-lsoxazol-3-yl CI H SOCH3

A-776 CI 5-Me-lsoxazol-3-yl CI H SO2CH3

A-777 CI 5-Me-lsoxazol-3-yl CI H CH2OCH3

A-778 CI 5-Me-lsoxazol-3-yl CI cyclopropyl H

A-779 CI 5-Me-lsoxazol-3-yl CI OCH3 H

A-780 CI 5-Me-lsoxazol-3-yl CI OCF3 H

A-781 CI 5-Me-lsoxazol-3-yl CI SCH ₃ H

A-782 CI 5-Me-lsoxazol-3-yl CI SOCH3 H

A-783 CI 5-Me-lsoxazol-3-yl CI SO2CH3 H

A-784 CI 5-Me-lsoxazol-3-yl CI CH2OCH3 H

A-785 CI 5-Me-lsoxazol-3-yl F H CN

A-786 CI 5-Me-lsoxazol-3-yl F H N0 ₂

A-787 CI 5-Me-lsoxazol-3-yl F H cyclopropyl

A-788 CI 5-Me-lsoxazol-3-yl F H OCH3

A-789 CI 5-Me-lsoxazol-3-yl F H OCF3

A-790 CI 5-Me-lsoxazol-3-yl F H SCH ₃

A-791 CI 5-Me-lsoxazol-3-yl F H SOCH3

A-792 CI 5-Me-lsoxazol-3-yl F H SO2CH3

A-793 CI 5-Me-lsoxazol-3-yl F H CH2OCH3

A-794 CI 5-Me-lsoxazol-3-yl F cyclopropyl H

A-795 CI 5-Me-lsoxazol-3-yl F OCH3 H

A-796 CI 5-Me-lsoxazol-3-yl F OCF3 H

A-797 CI 5-Me-lsoxazol-3-yl F SCH ₃ H A-798 CI 5-Me-lsoxazol-3-yl F SOCHs H

A-799 CI 5-Me-lsoxazol-3-yl F SO2CH3 H

A-800 CI 5-Me-lsoxazol-3-yl F CH2OCH3 H

A-801 CI 5-Me-lsoxazol-3-yl CFs H CN

A-802 CI 5-Me-lsoxazol-3-yl CFs H N0 ₂

A-803 CI 5-Me-lsoxazol-3-yl CFs H cyclopropyl

A-804 CI 5-Me-lsoxazol-3-yl CFs H OCH3

A-805 CI 5-Me-lsoxazol-3-yl CFs H OCFs

A-806 CI 5-Me-lsoxazol-3-yl CFs H SCHs

A-807 CI 5-Me-lsoxazol-3-yl CFs H SOCHs

A-808 CI 5-Me-lsoxazol-3-yl CFs H SO2CH3

A-809 CI 5-Me-lsoxazol-3-yl CFs H CH2OCH3

A-810 CI 5-Me-lsoxazol-3-yl CFs cyclopropyl H

A-81 1 CI 5-Me-lsoxazol-3-yl CFs OCH3 H

A-812 CI 5-Me-lsoxazol-3-yl CFs OCFs H

A-813 CI 5-Me-lsoxazol-3-yl CFs SCHs H

A-814 CI 5-Me-lsoxazol-3-yl CFs SOCHs H

A-815 CI 5-Me-lsoxazol-3-yl CFs SO2CH3 H

A-816 CI 5-Me-lsoxazol-3-yl CFs CH2OCH3 H

A-817 CI 5-Me-lsoxazol-3-yl SO2CH3 H CN

A-818 CI 5-Me-lsoxazol-3-yl SO2CH3 H N0 ₂

A-819 CI 5-Me-lsoxazol-3-yl SO2CH3 H cyclopropyl

A-820 CI 5-Me-lsoxazol-3-yl SO2CH3 H OCH3

A-821 CI 5-Me-lsoxazol-3-yl SO2CH3 H OCFs

A-822 CI 5-Me-lsoxazol-3-yl SO2CH3 H SCHs

A-823 CI 5-Me-lsoxazol-3-yl SO2CH3 H SOCHs

A-824 CI 5-Me-lsoxazol-3-yl SO2CH3 H SO2CH3

A-825 CI 5-Me-lsoxazol-3-yl SO2CH3 H CH2OCH3

A-826 CI 5-Me-lsoxazol-3-yl SO2CH3 cyclopropyl H

A-827 CI 5-Me-lsoxazol-3-yl SO2CH3 OCH3 H

A-828 CI 5-Me-lsoxazol-3-yl SO2CH3 OCFs H

A-829 CI 5-Me-lsoxazol-3-yl SO2CH3 SCHs H

A-830 CI 5-Me-lsoxazol-3-yl SO2CH3 SOCHs H

A-831 CI 5-Me-lsoxazol-3-yl SO2CH3 SO2CH3 H

A-832 CI 5-Me-lsoxazol-3-yl SO2CH3 CH2OCH3 H

A-833 CI 5-Me-lsoxazol-3-yl CN H CN

A-834 CI 5-Me-lsoxazol-3-yl CN H N0 ₂ A-835 CI 5-Me-lsoxazol-3-yl CN H cyclopropyl

A-836 CI 5-Me-lsoxazol-3-yl CN H OCH3

A-837 CI 5-Me-lsoxazol-3-yl CN H OCF3

A-838 CI 5-Me-lsoxazol-3-yl CN H SCH ₃

A-839 CI 5-Me-lsoxazol-3-yl CN H SOCH3

A-840 CI 5-Me-lsoxazol-3-yl CN H SO2CH3

A-841 CI 5-Me-lsoxazol-3-yl CN H CH2OCH3

A-842 CI 5-Me-lsoxazol-3-yl CN cyclopropyl H

A-843 CI 5-Me-lsoxazol-3-yl CN OCHs H

A-844 CI 5-Me-lsoxazol-3-yl CN OCF3 H

A-845 CI 5-Me-lsoxazol-3-yl CN SCHs H

A-846 CI 5-Me-lsoxazol-3-yl CN SOCH3 H

A-847 CI 5-Me-lsoxazol-3-yl CN SO2CH3 H

A-848 CI 5-Me-lsoxazol-3-yl CN CH2OCH3 H

A-849 CI 5-Me-lsoxazol-3-yl H H CN

A-850 CI 5-Me-lsoxazol-3-yl H H N0 ₂

A-851 CI 5-Me-lsoxazol-3-yl H H cyclopropyl

A-852 CI 5-Me-lsoxazol-3-yl H H OCH3

A-853 CI 5-Me-lsoxazol-3-yl H H OCF3

A-854 CI 5-Me-lsoxazol-3-yl H H SCH ₃

A-855 CI 5-Me-lsoxazol-3-yl H H SOCH3

A-856 CI 5-Me-lsoxazol-3-yl H H SO2CH3

A-857 CI 5-Me-lsoxazol-3-yl H H CH2OCH3

A-858 CI 5-Me-lsoxazol-3-yl H cyclopropyl H

A-859 CI 5-Me-lsoxazol-3-yl H OCH3 H

A-860 CI 5-Me-lsoxazol-3-yl H OCF3 H

A-861 CI 5-Me-lsoxazol-3-yl H SCH ₃ H

A-862 CI 5-Me-lsoxazol-3-yl H SOCH3 H

A-863 CI 5-Me-lsoxazol-3-yl H SO2CH3 H

A-864 CI 5-Me-lsoxazol-3-yl H CH2OCH3 H

A-865 CI 3-Me-lsoxazolin-5-yl CI H CN

A-866 CI 3-Me-lsoxazolin-5-yl CI H N0 ₂

A-867 CI 3-Me-lsoxazolin-5-yl CI H cyclopropyl

A-868 CI 3-Me-lsoxazolin-5-yl CI H OCH3

A-869 CI 3-Me-lsoxazolin-5-yl CI H OCF3

A-870 CI 3-Me-lsoxazolin-5-yl CI H SCH ₃

A-871 CI 3-Me-lsoxazolin-5-yl CI H SOCH3 A-872 CI 3-Me-lsoxazolin-5-yl CI H SO2CH3

A-873 CI 3-Me-lsoxazolin-5-yl CI H CH2OCH3

A-874 CI 3-Me-lsoxazolin-5-yl CI cyclopropyl H

A-875 CI 3-Me-lsoxazolin-5-yl CI OCHs H

A-876 CI 3-Me-lsoxazolin-5-yl CI OCFs H

A-877 CI 3-Me-lsoxazolin-5-yl CI SCHs H

A-878 CI 3-Me-lsoxazolin-5-yl CI SOCHs H

A-879 CI 3-Me-lsoxazolin-5-yl CI SO2CH3 H

A-880 CI 3-Me-lsoxazolin-5-yl CI CH2OCH3 H

A-881 CI 3-Me-lsoxazolin-5-yl F H CN

A-882 CI 3-Me-lsoxazolin-5-yl F H N0 ₂

A-883 CI 3-Me-lsoxazolin-5-yl F H cyclopropyl

A-884 CI 3-Me-lsoxazolin-5-yl F H OCHs

A-885 CI 3-Me-lsoxazolin-5-yl F H OCFs

A-886 CI 3-Me-lsoxazolin-5-yl F H SCHs

A-887 CI 3-Me-lsoxazolin-5-yl F H SOCHs

A-888 CI 3-Me-lsoxazolin-5-yl F H SO2CH3

A-889 CI 3-Me-lsoxazolin-5-yl F H CH2OCH3

A-890 CI 3-Me-lsoxazolin-5-yl F cyclopropyl H

A-891 CI 3-Me-lsoxazolin-5-yl F OCHs H

A-892 CI 3-Me-lsoxazolin-5-yl F OCFs H

A-893 CI 3-Me-lsoxazolin-5-yl F SCHs H

A-894 CI 3-Me-lsoxazolin-5-yl F SOCHs H

A-895 CI 3-Me-lsoxazolin-5-yl F SO2CH3 H

A-896 CI 3-Me-lsoxazolin-5-yl F CH2OCH3 H

A-897 CI 3-Me-lsoxazolin-5-yl CFs H CN

A-898 CI 3-Me-lsoxazolin-5-yl CFs H N0 ₂

A-899 CI 3-Me-lsoxazolin-5-yl CFs H cyclopropyl

A-900 CI 3-Me-lsoxazolin-5-yl CFs H OCHs

A-901 CI 3-Me-lsoxazolin-5-yl CFs H OCFs

A-902 CI 3-Me-lsoxazolin-5-yl CFs H SCHs

A-903 CI 3-Me-lsoxazolin-5-yl CFs H SOCHs

A-904 CI 3-Me-lsoxazolin-5-yl CFs H SO2CH3

A-905 CI 3-Me-lsoxazolin-5-yl CFs H CH2OCH3

A-906 CI 3-Me-lsoxazolin-5-yl CFs cyclopropyl H

A-907 CI 3-Me-lsoxazolin-5-yl CFs OCHs H

A-908 CI 3-Me-lsoxazolin-5-yl CFs OCFs H A-909 CI 3-Me-lsoxazolin-5-yl CFs SCH ₃ H

A-910 CI 3-Me-lsoxazolin-5-yl CFs SOCH3 H

A-91 1 CI 3-Me-lsoxazolin-5-yl CFs SO2CH3 H

A-912 CI 3-Me-lsoxazolin-5-yl CFs CH2OCH3 H

A-913 CI 3-Me-lsoxazolin-5-yl SO2CH3 H CN

A-914 CI 3-Me-lsoxazolin-5-yl SO2CH3 H N0 ₂

A-915 CI 3-Me-lsoxazolin-5-yl SO2CH3 H cyclopropyl

A-916 CI 3-Me-lsoxazolin-5-yl SO2CH3 H OCH3

A-917 CI 3-Me-lsoxazolin-5-yl SO2CH3 H OCF3

A-918 CI 3-Me-lsoxazolin-5-yl SO2CH3 H SCH ₃

A-919 CI 3-Me-lsoxazolin-5-yl SO2CH3 H SOCH3

A-920 CI 3-Me-lsoxazolin-5-yl SO2CH3 H SO2CH3

A-921 CI 3-Me-lsoxazolin-5-yl SO2CH3 H CH2OCH3

A-922 CI 3-Me-lsoxazolin-5-yl SO2CH3 cyclopropyl H

A-923 CI 3-Me-lsoxazolin-5-yl SO2CH3 OCH3 H

A-924 CI 3-Me-lsoxazolin-5-yl SO2CH3 OCF3 H

A-925 CI 3-Me-lsoxazolin-5-yl SO2CH3 SCH ₃ H

A-926 CI 3-Me-lsoxazolin-5-yl SO2CH3 SOCH3 H

A-927 CI 3-Me-lsoxazolin-5-yl SO2CH3 SO2CH3 H

A-928 CI 3-Me-lsoxazolin-5-yl SO2CH3 CH2OCH3 H

A-929 CI 3-Me-lsoxazolin-5-yl CN H CN

A-930 CI 3-Me-lsoxazolin-5-yl CN H N0 ₂

A-931 CI 3-Me-lsoxazolin-5-yl CN H cyclopropyl

A-932 CI 3-Me-lsoxazolin-5-yl CN H OCH3

A-933 CI 3-Me-lsoxazolin-5-yl CN H OCF3

A-934 CI 3-Me-lsoxazolin-5-yl CN H SCH ₃

A-935 CI 3-Me-lsoxazolin-5-yl CN H SOCH3

A-936 CI 3-Me-lsoxazolin-5-yl CN H SO2CH3

A-937 CI 3-Me-lsoxazolin-5-yl CN H CH2OCH3

A-938 CI 3-Me-lsoxazolin-5-yl CN cyclopropyl H

A-939 CI 3-Me-lsoxazolin-5-yl CN OCH3 H

A-940 CI 3-Me-lsoxazolin-5-yl CN OCF3 H

A-941 CI 3-Me-lsoxazolin-5-yl CN SCH ₃ H

A-942 CI 3-Me-lsoxazolin-5-yl CN SOCH3 H

A-943 CI 3-Me-lsoxazolin-5-yl CN SO2CH3 H

A-944 CI 3-Me-lsoxazolin-5-yl CN CH2OCH3 H

A-945 CI 3-Me-lsoxazolin-5-yl H H CN A-946 CI 3-Me-lsoxazolin-5-yl H H N0 ₂

A-947 CI 3-Me-lsoxazolin-5-yl H H cyclopropyl

A-948 CI 3-Me-lsoxazolin-5-yl H H OCH3

A-949 CI 3-Me-lsoxazolin-5-yl H H OCF3

A-950 CI 3-Me-lsoxazolin-5-yl H H SCH ₃

A-951 CI 3-Me-lsoxazolin-5-yl H H SOCH3

A-952 CI 3-Me-lsoxazolin-5-yl H H SO2CH3

A-953 CI 3-Me-lsoxazolin-5-yl H H CH2OCH3

A-954 CI 3-Me-lsoxazolin-5-yl H cyclopropyl H

A-955 CI 3-Me-lsoxazolin-5-yl H OCHs H

A-956 CI 3-Me-lsoxazolin-5-yl H OCF3 H

A-957 CI 3-Me-lsoxazolin-5-yl H SCHs H

A-958 CI 3-Me-lsoxazolin-5-yl H SOCH3 H

A-959 CI 3-Me-lsoxazolin-5-yl H SO2CH3 H

A-960 CI 3-Me-lsoxazolin-5-yl H CH2OCH3 H

A-961 CI 3-Me-lsoxazol-5-yl CI H CN

A-962 CI 3-Me-lsoxazol-5-yl CI H N0 ₂

A-963 CI 3-Me-lsoxazol-5-yl CI H cyclopropyl

A-964 CI 3-Me-lsoxazol-5-yl CI H OCH3

A-965 CI 3-Me-lsoxazol-5-yl CI H OCF3

A-966 CI 3-Me-lsoxazol-5-yl CI H SCH ₃

A-967 CI 3-Me-lsoxazol-5-yl CI H SOCH3

A-968 CI 3-Me-lsoxazol-5-yl CI H SO2CH3

A-969 CI 3-Me-lsoxazol-5-yl CI H CH2OCH3

A-970 CI 3-Me-lsoxazol-5-yl CI cyclopropyl H

A-971 CI 3-Me-lsoxazol-5-yl CI OCH3 H

A-972 CI 3-Me-lsoxazol-5-yl CI OCF3 H

A-973 CI 3-Me-lsoxazol-5-yl CI SCH ₃ H

A-974 CI 3-Me-lsoxazol-5-yl CI SOCH3 H

A-975 CI 3-Me-lsoxazol-5-yl CI SO2CH3 H

A-976 CI 3-Me-lsoxazol-5-yl CI CH2OCH3 H

A-977 CI 3-Me-lsoxazol-5-yl F H CN

A-978 CI 3-Me-lsoxazol-5-yl F H N0 ₂

A-979 CI 3-Me-lsoxazol-5-yl F H cyclopropyl

A-980 CI 3-Me-lsoxazol-5-yl F H OCH3

A-981 CI 3-Me-lsoxazol-5-yl F H OCF3

A-982 CI 3-Me-lsoxazol-5-yl F H SCH ₃ A-983 CI 3-Me-lsoxazol-5-yl F H SOCHs

A-984 CI 3-Me-lsoxazol-5-yl F H SO2CH3

A-985 CI 3-Me-lsoxazol-5-yl F H CH2OCH3

A-986 CI 3-Me-lsoxazol-5-yl F cyclopropyl H

A-987 CI 3-Me-lsoxazol-5-yl F OCH3 H

A-988 CI 3-Me-lsoxazol-5-yl F OCFs H

A-989 CI 3-Me-lsoxazol-5-yl F SCHs H

A-990 CI 3-Me-lsoxazol-5-yl F SOCHs H

A-991 CI 3-Me-lsoxazol-5-yl F SO2CH3 H

A-992 CI 3-Me-lsoxazol-5-yl F CH2OCH3 H

A-993 CI 3-Me-lsoxazol-5-yl CFs H CN

A-994 CI 3-Me-lsoxazol-5-yl CFs H N0 ₂

A-995 CI 3-Me-lsoxazol-5-yl CFs H cyclopropyl

A-996 CI 3-Me-lsoxazol-5-yl CFs H OCHs

A-997 CI 3-Me-lsoxazol-5-yl CFs H OCFs

A-998 CI 3-Me-lsoxazol-5-yl CFs H SCHs

A-999 CI 3-Me-lsoxazol-5-yl CFs H SOCHs

A-1000 CI 3-Me-lsoxazol-5-yl CFs H SO2CH3

A-1001 CI 3-Me-lsoxazol-5-yl CFs H CH2OCH3

A-1002 CI 3-Me-lsoxazol-5-yl CFs cyclopropyl H

A-1003 CI 3-Me-lsoxazol-5-yl CFs OCH3 H

A-1004 CI 3-Me-lsoxazol-5-yl CFs OCFs H

A-1005 CI 3-Me-lsoxazol-5-yl CFs SCHs H

A-1006 CI 3-Me-lsoxazol-5-yl CFs SOCHs H

A-1007 CI 3-Me-lsoxazol-5-yl CFs SO2CH3 H

A-1008 CI 3-Me-lsoxazol-5-yl CFs CH2OCH3 H

A-1009 CI 3-Me-lsoxazol-5-yl SO2CH3 H CN

A-1010 CI 3-Me-lsoxazol-5-yl SO2CH3 H N0 ₂

A-101 1 CI 3-Me-lsoxazol-5-yl SO2CH3 H cyclopropyl

A-1012 CI 3-Me-lsoxazol-5-yl SO2CH3 H OCHs

A-1013 CI 3-Me-lsoxazol-5-yl SO2CH3 H OCFs

A-1014 CI 3-Me-lsoxazol-5-yl SO2CH3 H SCHs

A-1015 CI 3-Me-lsoxazol-5-yl SO2CH3 H SOCHs

A-1016 CI 3-Me-lsoxazol-5-yl SO2CH3 H SO2CH3

A-1017 CI 3-Me-lsoxazol-5-yl SO2CH3 H CH2OCH3

A-1018 CI 3-Me-lsoxazol-5-yl SO2CH3 cyclopropyl H

A-1019 CI 3-Me-lsoxazol-5-yl SO2CH3 OCH3 H A-1020 CI 3-Me-lsoxazol-5-yl SO2CH3 OCF3 H

A-1021 CI 3-Me-lsoxazol-5-yl SO2CH3 SCH ₃ H

A-1022 CI 3-Me-lsoxazol-5-yl SO2CH3 SOCH3 H

A-1023 CI 3-Me-lsoxazol-5-yl SO2CH3 SO2CH3 H

A-1024 CI 3-Me-lsoxazol-5-yl SO2CH3 CH2OCH3 H

A-1025 CI 3-Me-lsoxazol-5-yl CN H CN

A-1026 CI 3-Me-lsoxazol-5-yl CN H N0 ₂

A-1027 CI 3-Me-lsoxazol-5-yl CN H cyclopropyl

A-1028 CI 3-Me-lsoxazol-5-yl CN H OCH3

A-1029 CI 3-Me-lsoxazol-5-yl CN H OCF3

A-1030 CI 3-Me-lsoxazol-5-yl CN H SCH ₃

A-1031 CI 3-Me-lsoxazol-5-yl CN H SOCH3

A-1032 CI 3-Me-lsoxazol-5-yl CN H SO2CH3

A-1033 CI 3-Me-lsoxazol-5-yl CN H CH2OCH3

A-1034 CI 3-Me-lsoxazol-5-yl CN cyclopropyl H

A-1035 CI 3-Me-lsoxazol-5-yl CN OCH3 H

A-1036 CI 3-Me-lsoxazol-5-yl CN OCF3 H

A-1037 CI 3-Me-lsoxazol-5-yl CN SCH ₃ H

A-1038 CI 3-Me-lsoxazol-5-yl CN SOCH3 H

A-1039 CI 3-Me-lsoxazol-5-yl CN SO2CH3 H

A-1040 CI 3-Me-lsoxazol-5-yl CN CH2OCH3 H

A-1041 CI 3-Me-lsoxazol-5-yl H H CN

A-1042 CI 3-Me-lsoxazol-5-yl H H N0 ₂

A-1043 CI 3-Me-lsoxazol-5-yl H H cyclopropyl

A-1044 CI 3-Me-lsoxazol-5-yl H H OCH3

A-1045 CI 3-Me-lsoxazol-5-yl H H OCF3

A-1046 CI 3-Me-lsoxazol-5-yl H H SCH ₃

A-1047 CI 3-Me-lsoxazol-5-yl H H SOCH3

A-1048 CI 3-Me-lsoxazol-5-yl H H SO2CH3

A-1049 CI 3-Me-lsoxazol-5-yl H H CH2OCH3

A-1050 CI 3-Me-lsoxazol-5-yl H cyclopropyl H

A-1051 CI 3-Me-lsoxazol-5-yl H OCH3 H

A-1052 CI 3-Me-lsoxazol-5-yl H OCF3 H

A-1053 CI 3-Me-lsoxazol-5-yl H SCH ₃ H

A-1054 CI 3-Me-lsoxazol-5-yl H SOCH3 H

A-1055 CI 3-Me-lsoxazol-5-yl H SO2CH3 H

A-1056 CI 3-Me-lsoxazol-5-yl H CH2OCH3 H A-1242 CHs SOCHs H cyclopropyl H

A-1243 CHs SOCHs H OCHs H

A-1244 CHs SOCHs H OCFs H

A-1245 CHs SOCHs H SCHs H

A-1246 CHs SOCHs H SOCHs H

A-1247 CHs SOCHs H SO2CH3 H

A-1248 CHs SOCHs H CH2OCH3 H

A-1249 CHs SOCHs CI H CN

A-1250 CHs SOCHs CI H N0 ₂

A-1251 CHs SOCHs CI H cyclopropyl

A-1252 CHs SOCHs CI H OCHs

A-1253 CHs SOCHs CI H OCFs

A-1254 CHs SOCHs CI H SCHs

A-1255 CHs SOCHs CI H SOCHs

A-1256 CHs SOCHs CI H SO2CH3

A-1257 CHs SOCHs CI H CH2OCH3

A-1258 CHs SOCHs CI cyclopropyl H

A-1259 CHs SOCHs CI OCHs H

A-1260 CHs SOCHs CI OCFs H

A-1261 CHs SOCHs CI SCHs H

A-1262 CHs SOCHs CI SOCHs H

A-1263 CHs SOCHs CI SO2CH3 H

A-1264 CHs SOCHs CI CH2OCH3 H

A-1265 CHs SOCHs F H CN

A-1266 CHs SOCHs F H N0 ₂

A-1267 CHs SOCHs F H cyclopropyl

A-1268 CHs SOCHs F H OCHs

A-1269 CHs SOCHs F H OCFs

A-1270 CHs SOCHs F H SCHs

A-1271 CHs SOCHs F H SOCHs

A-1272 CHs SOCHs F H SO2CH3

A-1273 CHs SOCHs F H CH2OCH3

A-1274 CHs SOCHs F cyclopropyl H

A-1275 CHs SOCHs F OCHs H

A-1276 CHs SOCHs F OCFs H

A-1277 CHs SOCHs F SCHs H

A-1278 CHs SOCHs F SOCHs H A-1279 CHs SOCHs F SO2CH3 H

A-1280 CHs SOCHs F CH2OCH3 H

A-1281 CHs SOCHs CFs H CN

A-1282 CHs SOCHs CFs H N0 ₂

A-1283 CHs SOCHs CFs H cyclopropyl

A-1284 CHs SOCHs CFs H OCH3

A-1285 CHs SOCHs CFs H OCFs

A-1286 CHs SOCHs CFs H SCHs

A-1287 CHs SOCHs CFs H SOCHs

A-1288 CHs SOCHs CFs H SO2CH3

A-1289 CHs SOCHs CFs H CH2OCH3

A-1290 CHs SOCHs CFs cyclopropyl H

A-1291 CHs SOCHs CFs OCH3 H

A-1292 CHs SOCHs CFs OCFs H

A-1293 CHs SOCHs CFs SCHs H

A-1294 CHs SOCHs CFs SOCHs H

A-1295 CHs SOCHs CFs SO2CH3 H

A-1296 CHs SOCHs CFs CH2OCH3 H

A-1297 CHs SOCHs SO2CH3 H CN

A-1298 CHs SOCHs SO2CH3 H N0 ₂

A-1299 CHs SOCHs SO2CH3 H cyclopropyl

A-1300 CHs SOCHs SO2CH3 H OCH3

A-1301 CHs SOCHs SO2CH3 H OCFs

A-1302 CHs SOCHs SO2CH3 H SCHs

A-1303 CHs SOCHs SO2CH3 H SOCHs

A-1304 CHs SOCHs SO2CH3 H SO2CH3

A-1305 CHs SOCHs SO2CH3 H CH2OCH3

A-1306 CHs SOCHs SO2CH3 cyclopropyl H

A-1307 CHs SOCHs SO2CH3 OCH3 H

A-1308 CHs SOCHs SO2CH3 OCFs H

A-1309 CHs SOCHs SO2CH3 SCHs H

A-1310 CHs SOCHs SO2CH3 SOCHs H

A-131 1 CHs SOCHs SO2CH3 SO2CH3 H

A-1312 CHs SOCHs SO2CH3 CH2OCH3 H

A-1313 CHs SOCHs CN H CN

A-1314 CHs SOCHs CN H N0 ₂

A-1315 CHs SOCHs CN H cyclopropyl A-1427 CHs SO2CH3 H H cyclopropyl

A-1428 CHs SO2CH3 H H OCHs

A-1429 CHs SO2CH3 H H OCF3

A-1430 CHs SO2CH3 H H SCHs

A-1431 CHs SO2CH3 H H SOCH3

A-1432 CHs SO2CH3 H H SO2CH3

A-1433 CHs SO2CH3 H H CH2OCH3

A-1434 CHs SO2CH3 H cyclopropyl H

A-1435 CHs SO2CH3 H OCHs H

A-1436 CHs SO2CH3 H OCF3 H

A-1437 CHs SO2CH3 H SCHs H

A-1438 CHs SO2CH3 H SOCH3 H

A-1439 CHs SO2CH3 H SO2CH3 H

A-1440 CHs SO2CH3 H CH2OCH3 H

A-1441 CHs CH2OCH2CF3 CI H CN

A-1442 CHs CH2OCH2CF3 CI H N0 ₂

A-1443 CHs CH2OCH2CF3 CI H cyclopropyl

A-1444 CHs CH2OCH2CF3 CI H OCHs

A-1445 CHs CH2OCH2CF3 CI H OCF3

A-1446 CHs CH2OCH2CF3 CI H SCHs

A-1447 CHs CH2OCH2CF3 CI H SOCH3

A-1448 CHs CH2OCH2CF3 CI H SO2CH3

A-1449 CHs CH2OCH2CF3 CI H CH2OCH3

A-1450 CHs CH2OCH2CF3 CI cyclopropyl H

A-1451 CHs CH2OCH2CF3 CI OCHs H

A-1452 CHs CH2OCH2CF3 CI OCF3 H

A-1453 CHs CH2OCH2CF3 CI SCHs H

A-1454 CHs CH2OCH2CF3 CI SOCH3 H

A- 1455 CHs CH2OCH2CF3 CI SO2CH3 H

A-1456 CHs CH2OCH2CF3 CI CH2OCH3 H

A-1457 CHs CH2OCH2CF3 F H CN

A-1458 CHs CH2OCH2CF3 F H N0 ₂

A-1459 CHs CH2OCH2CF3 F H cyclopropyl

A-1460 CHs CH2OCH2CF3 F H OCHs

A-1461 CHs CH2OCH2CF3 F H OCF3

A-1462 CHs CH2OCH2CF3 F H SCHs

A-1463 CHs CH2OCH2CF3 F H SOCH3 A-1464 CHs CH2OCH2CF3 F H SO2CH3

A-1465 CHs CH2OCH2CF3 F H CH2OCH3

A-1466 CHs CH2OCH2CF3 F cyclopropyl H

A-1467 CHs CH2OCH2CF3 F OCHs H

A-1468 CHs CH2OCH2CF3 F OCF3 H

A-1469 CHs CH2OCH2CF3 F SCHs H

A-1470 CHs CH2OCH2CF3 F SOCH3 H

A-1471 CHs CH2OCH2CF3 F SO2CH3 H

A-1472 CHs CH2OCH2CF3 F CH2OCH3 H

A-1473 CHs CH2OCH2CF3 CFs H CN

A-1474 CHs CH2OCH2CF3 CFs H N0 ₂

A-1475 CHs CH2OCH2CF3 CFs H cyclopropyl

A-1476 CHs CH2OCH2CF3 CFs H OCHs

A-1477 CHs CH2OCH2CF3 CFs H OCFs

A-1478 CHs CH2OCH2CF3 CFs H SCHs

A-1479 CHs CH2OCH2CF3 CFs H SOCHs

A-1480 CHs CH2OCH2CF3 CFs H SO2CH3

A-1481 CHs CH2OCH2CF3 CFs H CH2OCH3

A-1482 CHs CH2OCH2CF3 CFs cyclopropyl H

A-1483 CHs CH2OCH2CF3 CFs OCHs H

A-1484 CHs CH2OCH2CF3 CFs OCF3 H

A-1485 CHs CH2OCH2CF3 CFs SCHs H

A-1486 CHs CH2OCH2CF3 CFs SOCH3 H

A-1487 CHs CH2OCH2CF3 CFs SO2CH3 H

A-1488 CHs CH2OCH2CF3 CFs CH2OCH3 H

A-1489 CHs CH2OCH2CF3 SO2CH3 H CN

A-1490 CHs CH2OCH2CF3 SO2CH3 H N0 ₂

A-1491 CHs CH2OCH2CF3 SO2CH3 H cyclopropyl

A-1492 CHs CH2OCH2CF3 SO2CH3 H OCHs

A-1493 CHs CH2OCH2CF3 SO2CH3 H OCFs

A-1494 CHs CH2OCH2CF3 SO2CH3 H SCHs

A-1495 CHs CH2OCH2CF3 SO2CH3 H SOCHs

A-1496 CHs CH2OCH2CF3 SO2CH3 H SO2CH3

A-1497 CHs CH2OCH2CF3 SO2CH3 H CH2OCH3

A-1498 CHs CH2OCH2CF3 SO2CH3 cyclopropyl H

A-1499 CHs CH2OCH2CF3 SO2CH3 OCHs H

A-1500 CHs CH2OCH2CF3 SO2CH3 OCF3 H A-1501 CHs CH2OCH2CF3 SO2CH3 SCHs H

A-1502 CHs CH2OCH2CF3 SO2CH3 SOCHs H

A-1503 CHs CH2OCH2CF3 SO2CH3 SO2CH3 H

A-1504 CHs CH2OCH2CF3 SO2CH3 CH2OCH3 H

A-1505 CHs CH2OCH2CF3 CN H CN

A-1506 CHs CH2OCH2CF3 CN H N0 ₂

A-1507 CHs CH2OCH2CF3 CN H cyclopropyl

A-1508 CHs CH2OCH2CF3 CN H OCH3

A-1509 CHs CH2OCH2CF3 CN H OCFs

A-1510 CHs CH2OCH2CF3 CN H SCHs

A-151 1 CHs CH2OCH2CF3 CN H SOCHs

A-1512 CHs CH2OCH2CF3 CN H SO2CH3

A-1513 CHs CH2OCH2CF3 CN H CH2OCH3

A-1514 CHs CH2OCH2CF3 CN cyclopropyl H

A-1515 CHs CH2OCH2CF3 CN OCH3 H

A-1516 CHs CH2OCH2CF3 CN OCFs H

A-1517 CHs CH2OCH2CF3 CN SCHs H

A-1518 CHs CH2OCH2CF3 CN SOCHs H

A-1519 CHs CH2OCH2CF3 CN SO2CH3 H

A-1520 CHs CH2OCH2CF3 CN CH2OCH3 H

A-1521 CHs CH2OCH2CF3 H H CN

A-1522 CHs CH2OCH2CF3 H H N0 ₂

A-1523 CHs CH2OCH2CF3 H H cyclopropyl

A-1524 CHs CH2OCH2CF3 H H OCH3

A-1525 CHs CH2OCH2CF3 H H OCFs

A-1526 CHs CH2OCH2CF3 H H SCHs

A-1527 CHs CH2OCH2CF3 H H SOCHs

A-1528 CHs CH2OCH2CF3 H H SO2CH3

A-1529 CHs CH2OCH2CF3 H H CH2OCH3

A-1530 CHs CH2OCH2CF3 H cyclopropyl H

A-1531 CHs CH2OCH2CF3 H OCH3 H

A-1532 CHs CH2OCH2CF3 H OCFs H

A-1533 CHs CH2OCH2CF3 H SCHs H

A-1534 CHs CH2OCH2CF3 H SOCHs H

A-1535 CHs CH2OCH2CF3 H SO2CH3 H

A-1536 CHs CH2OCH2CF3 H CH2OCH3 H

A-1537 CHs lsoxazolin-3-yl CI H CN A-1538 CHs lsoxazolin-3-yl CI H N0 ₂

A-1539 CHs lsoxazolin-3-yl CI H cyclopropyl

A-1540 CHs lsoxazolin-3-yl CI H OCHs

A-1541 CHs lsoxazolin-3-yl CI H OCFs

A-1542 CHs lsoxazolin-3-yl CI H SCHs

A-1543 CHs lsoxazolin-3-yl CI H SOCHs

A-1544 CHs lsoxazolin-3-yl CI H SO2CH3

A-1545 CHs lsoxazolin-3-yl CI H CH2OCH3

A-1546 CHs lsoxazolin-3-yl CI cyclopropyl H

A-1547 CHs lsoxazolin-3-yl CI OCHs H

A-1548 CHs lsoxazolin-3-yl CI OCFs H

A-1549 CHs lsoxazolin-3-yl CI SCHs H

A-1550 CHs lsoxazolin-3-yl CI SOCHs H

A-1551 CHs lsoxazolin-3-yl CI SO2CH3 H

A-1552 CHs lsoxazolin-3-yl CI CH2OCH3 H

A-1553 CHs lsoxazolin-3-yl F H CN

A- 1554 CHs lsoxazolin-3-yl F H N0 ₂

A-1555 CHs lsoxazolin-3-yl F H cyclopropyl

A-1556 CHs lsoxazolin-3-yl F H OCHs

A- 1557 CHs lsoxazolin-3-yl F H OCFs

A-1558 CHs lsoxazolin-3-yl F H SCHs

A-1559 CHs lsoxazolin-3-yl F H SOCHs

A-1560 CHs lsoxazolin-3-yl F H SO2CH3

A-1561 CHs lsoxazolin-3-yl F H CH2OCH3

A-1562 CHs lsoxazolin-3-yl F cyclopropyl H

A-1563 CHs lsoxazolin-3-yl F OCHs H

A-1564 CHs lsoxazolin-3-yl F OCFs H

A-1565 CHs lsoxazolin-3-yl F SCHs H

A-1566 CHs lsoxazolin-3-yl F SOCHs H

A-1567 CHs lsoxazolin-3-yl F SO2CH3 H

A-1568 CHs lsoxazolin-3-yl F CH2OCH3 H

A-1569 CHs lsoxazolin-3-yl CFs H CN

A-1570 CHs lsoxazolin-3-yl CFs H N0 ₂

A-1571 CHs lsoxazolin-3-yl CFs H cyclopropyl

A-1572 CHs lsoxazolin-3-yl CFs H OCHs

A-1573 CHs lsoxazolin-3-yl CFs H OCFs

A-1574 CHs lsoxazolin-3-yl CFs H SCHs A- 1575 CHs lsoxazolin-3-yl CFs H SOCH3

A-1576 CHs lsoxazolin-3-yl CFs H SO2CH3

A- 1577 CHs lsoxazolin-3-yl CFs H CH2OCH3

A-1578 CHs lsoxazolin-3-yl CFs cyclopropyl H

A-1579 CHs lsoxazolin-3-yl CFs OCHs H

A-1580 CHs lsoxazolin-3-yl CFs OCF3 H

A-1581 CHs lsoxazolin-3-yl CFs SCHs H

A-1582 CHs lsoxazolin-3-yl CFs SOCH3 H

A-1583 CHs lsoxazolin-3-yl CFs SO2CH3 H

A-1584 CHs lsoxazolin-3-yl CFs CH2OCH3 H

A-1585 CHs lsoxazolin-3-yl SO2CH3 H CN

A-1586 CHs lsoxazolin-3-yl SO2CH3 H N0 ₂

A-1587 CHs lsoxazolin-3-yl SO2CH3 H cyclopropyl

A-1588 CHs lsoxazolin-3-yl SO2CH3 H OCHs

A-1589 CHs lsoxazolin-3-yl SO2CH3 H OCF3

A-1590 CHs lsoxazolin-3-yl SO2CH3 H SCHs

A-1591 CHs lsoxazolin-3-yl SO2CH3 H SOCH3

A-1592 CHs lsoxazolin-3-yl SO2CH3 H SO2CH3

A-1593 CHs lsoxazolin-3-yl SO2CH3 H CH2OCH3

A-1594 CHs lsoxazolin-3-yl SO2CH3 cyclopropyl H

A-1595 CHs lsoxazolin-3-yl SO2CH3 OCHs H

A-1596 CHs lsoxazolin-3-yl SO2CH3 OCF3 H

A-1597 CHs lsoxazolin-3-yl SO2CH3 SCHs H

A-1598 CHs lsoxazolin-3-yl SO2CH3 SOCH3 H

A-1599 CHs lsoxazolin-3-yl SO2CH3 SO2CH3 H

A-1600 CHs lsoxazolin-3-yl SO2CH3 CH2OCH3 H

A-1601 CHs lsoxazolin-3-yl CN H CN

A-1602 CHs lsoxazolin-3-yl CN H N0 ₂

A-1603 CHs lsoxazolin-3-yl CN H cyclopropyl

A-1604 CHs lsoxazolin-3-yl CN H OCHs

A-1605 CHs lsoxazolin-3-yl CN H OCF3

A-1606 CHs lsoxazolin-3-yl CN H SCHs

A-1607 CHs lsoxazolin-3-yl CN H SOCH3

A-1608 CHs lsoxazolin-3-yl CN H SO2CH3

A-1609 CHs lsoxazolin-3-yl CN H CH2OCH3

A-1610 CHs lsoxazolin-3-yl CN cyclopropyl H

A-161 1 CHs lsoxazolin-3-yl CN OCHs H A-1612 CHs lsoxazolin-3-yl CN OCFs H

A-1613 CHs lsoxazolin-3-yl CN SCHs H

A-1614 CHs lsoxazolin-3-yl CN SOCHs H

A-1615 CHs lsoxazolin-3-yl CN SO2CH3 H

A-1616 CHs lsoxazolin-3-yl CN CH2OCH3 H

A-1617 CHs lsoxazolin-3-yl H H CN

A-1618 CHs lsoxazolin-3-yl H H N0 ₂

A-1619 CHs lsoxazolin-3-yl H H cyclopropyl

A-1620 CHs lsoxazolin-3-yl H H OCHs

A-1621 CHs lsoxazolin-3-yl H H OCFs

A-1622 CHs lsoxazolin-3-yl H H SCHs

A-1623 CHs lsoxazolin-3-yl H H SOCHs

A-1624 CHs lsoxazolin-3-yl H H SO2CH3

A-1625 CHs lsoxazolin-3-yl H H CH2OCH3

A-1626 CHs lsoxazolin-3-yl H cyclopropyl H

A-1627 CHs lsoxazolin-3-yl H OCHs H

A-1628 CHs lsoxazolin-3-yl H OCFs H

A-1629 CHs lsoxazolin-3-yl H SCHs H

A-1630 CHs lsoxazolin-3-yl H SOCHs H

A-1631 CHs lsoxazolin-3-yl H SO2CH3 H

A-1632 CHs lsoxazolin-3-yl H CH2OCH3 H

A-1633 CHs 5-Me-lsoxazolin-3-yl CI H CN

A-1634 CHs 5-Me-lsoxazolin-3-yl CI H N0 ₂

A-1635 CHs 5-Me-lsoxazolin-3-yl CI H cyclopropyl

A-1636 CHs 5-Me-lsoxazolin-3-yl CI H OCHs

A-1637 CHs 5-Me-lsoxazolin-3-yl CI H OCFs

A-1638 CHs 5-Me-lsoxazolin-3-yl CI H SCHs

A-1639 CHs 5-Me-lsoxazolin-3-yl CI H SOCHs

A-1640 CHs 5-Me-lsoxazolin-3-yl CI H SO2CH3

A-1641 CHs 5-Me-lsoxazolin-3-yl CI H CH2OCH3

A-1642 CHs 5-Me-lsoxazolin-3-yl CI cyclopropyl H

A-1643 CHs 5-Me-lsoxazolin-3-yl CI OCHs H

A-1644 CHs 5-Me-lsoxazolin-3-yl CI OCFs H

A-1645 CHs 5-Me-lsoxazolin-3-yl CI SCHs H

A-1646 CHs 5-Me-lsoxazolin-3-yl CI SOCHs H

A-1647 CHs 5-Me-lsoxazolin-3-yl CI SO2CH3 H

A-1648 CHs 5-Me-lsoxazolin-3-yl CI CH2OCH3 H A-1649 CHs 5-Me-lsoxazolin-3-yl F H CN

A-1650 CHs 5-Me-lsoxazolin-3-yl F H N0 ₂

A-1651 CHs 5-Me-lsoxazolin-3-yl F H cyclopropyl

A-1652 CHs 5-Me-lsoxazolin-3-yl F H OCH3

A-1653 CHs 5-Me-lsoxazolin-3-yl F H OCFs

A-1654 CHs 5-Me-lsoxazolin-3-yl F H SCHs

A-1655 CHs 5-Me-lsoxazolin-3-yl F H SOCHs

A-1656 CHs 5-Me-lsoxazolin-3-yl F H SO2CH3

A-1657 CHs 5-Me-lsoxazolin-3-yl F H CH2OCH3

A-1658 CHs 5-Me-lsoxazolin-3-yl F cyclopropyl H

A-1659 CHs 5-Me-lsoxazolin-3-yl F OCH3 H

A-1660 CHs 5-Me-lsoxazolin-3-yl F OCFs H

A-1661 CHs 5-Me-lsoxazolin-3-yl F SCHs H

A-1662 CHs 5-Me-lsoxazolin-3-yl F SOCHs H

A-1663 CHs 5-Me-lsoxazolin-3-yl F SO2CH3 H

A-1664 CHs 5-Me-lsoxazolin-3-yl F CH2OCH3 H

A-1665 CHs 5-Me-lsoxazolin-3-yl CFs H CN

A-1666 CHs 5-Me-lsoxazolin-3-yl CFs H N0 ₂

A-1667 CHs 5-Me-lsoxazolin-3-yl CFs H cyclopropyl

A-1668 CHs 5-Me-lsoxazolin-3-yl CFs H OCH3

A-1669 CHs 5-Me-lsoxazolin-3-yl CFs H OCFs

A-1670 CHs 5-Me-lsoxazolin-3-yl CFs H SCHs

A-1671 CHs 5-Me-lsoxazolin-3-yl CFs H SOCHs

A-1672 CHs 5-Me-lsoxazolin-3-yl CFs H SO2CH3

A-1673 CHs 5-Me-lsoxazolin-3-yl CFs H CH2OCH3

A-1674 CHs 5-Me-lsoxazolin-3-yl CFs cyclopropyl H

A-1675 CHs 5-Me-lsoxazolin-3-yl CFs OCH3 H

A-1676 CHs 5-Me-lsoxazolin-3-yl CFs OCFs H

A-1677 CHs 5-Me-lsoxazolin-3-yl CFs SCHs H

A-1678 CHs 5-Me-lsoxazolin-3-yl CFs SOCHs H

A-1679 CHs 5-Me-lsoxazolin-3-yl CFs SO2CH3 H

A-1680 CHs 5-Me-lsoxazolin-3-yl CFs CH2OCH3 H

A-1681 CHs 5-Me-lsoxazolin-3-yl SO2CH3 H CN

A-1682 CHs 5-Me-lsoxazolin-3-yl SO2CH3 H N0 ₂

A-1683 CHs 5-Me-lsoxazolin-3-yl SO2CH3 H cyclopropyl

A-1684 CHs 5-Me-lsoxazolin-3-yl SO2CH3 H OCH3

A-1685 CHs 5-Me-lsoxazolin-3-yl SO2CH3 H OCFs A-1686 CHs 5-Me-lsoxazolin-3-yl SO2CH3 H SCHs

A-1687 CHs 5-Me-lsoxazolin-3-yl SO2CH3 H SOCHs

A-1688 CHs 5-Me-lsoxazolin-3-yl SO2CH3 H SO2CH3

A-1689 CHs 5-Me-lsoxazolin-3-yl SO2CH3 H CH2OCH3

A-1690 CHs 5-Me-lsoxazolin-3-yl SO2CH3 cyclopropyl H

A-1691 CHs 5-Me-lsoxazolin-3-yl SO2CH3 OCH3 H

A-1692 CHs 5-Me-lsoxazolin-3-yl SO2CH3 OCFs H

A-1693 CHs 5-Me-lsoxazolin-3-yl SO2CH3 SCHs H

A-1694 CHs 5-Me-lsoxazolin-3-yl SO2CH3 SOCHs H

A-1695 CHs 5-Me-lsoxazolin-3-yl SO2CH3 SO2CH3 H

A-1696 CHs 5-Me-lsoxazolin-3-yl SO2CH3 CH2OCH3 H

A-1697 CHs 5-Me-lsoxazolin-3-yl CN H CN

A-1698 CHs 5-Me-lsoxazolin-3-yl CN H N0 ₂

A-1699 CHs 5-Me-lsoxazolin-3-yl CN H cyclopropyl

A-1700 CHs 5-Me-lsoxazolin-3-yl CN H OCH3

A-1701 CHs 5-Me-lsoxazolin-3-yl CN H OCFs

A-1702 CHs 5-Me-lsoxazolin-3-yl CN H SCHs

A-1703 CHs 5-Me-lsoxazolin-3-yl CN H SOCHs

A-1704 CHs 5-Me-lsoxazolin-3-yl CN H SO2CH3

A-1705 CHs 5-Me-lsoxazolin-3-yl CN H CH2OCH3

A-1706 CHs 5-Me-lsoxazolin-3-yl CN cyclopropyl H

A-1707 CHs 5-Me-lsoxazolin-3-yl CN OCH3 H

A-1708 CHs 5-Me-lsoxazolin-3-yl CN OCFs H

A-1709 CHs 5-Me-lsoxazolin-3-yl CN SCHs H

A-1710 CHs 5-Me-lsoxazolin-3-yl CN SOCHs H

A-171 1 CHs 5-Me-lsoxazolin-3-yl CN SO2CH3 H

A-1712 CHs 5-Me-lsoxazolin-3-yl CN CH2OCH3 H

A-1713 CHs 5-Me-lsoxazolin-3-yl H H CN

A-1714 CHs 5-Me-lsoxazolin-3-yl H H N0 ₂

A-1715 CHs 5-Me-lsoxazolin-3-yl H H cyclopropyl

A-1716 CHs 5-Me-lsoxazolin-3-yl H H OCH3

A-1717 CHs 5-Me-lsoxazolin-3-yl H H OCFs

A-1718 CHs 5-Me-lsoxazolin-3-yl H H SCHs

A-1719 CHs 5-Me-lsoxazolin-3-yl H H SOCHs

A-1720 CHs 5-Me-lsoxazolin-3-yl H H SO2CH3

A-1721 CHs 5-Me-lsoxazolin-3-yl H H CH2OCH3

A-1722 CHs 5-Me-lsoxazolin-3-yl H cyclopropyl H A-1723 CHs 5-Me-lsoxazolin-3-yl H OCHs H

A-1724 CHs 5-Me-lsoxazolin-3-yl H OCFs H

A-1725 CHs 5-Me-lsoxazolin-3-yl H SCHs H

A-1726 CHs 5-Me-lsoxazolin-3-yl H SOCHs H

A-1727 CHs 5-Me-lsoxazolin-3-yl H SO2CH3 H

A-1728 CHs 5-Me-lsoxazolin-3-yl H CH2OCH3 H

A-1729 CHs lsoxazol-3-yl CI H CN

A-1730 CHs lsoxazol-3-yl CI H N0 ₂

A-1731 CHs lsoxazol-3-yl CI H cyclopropyl

A-1732 CHs lsoxazol-3-yl CI H OCHs

A-1733 CHs lsoxazol-3-yl CI H OCFs

A-1734 CHs lsoxazol-3-yl CI H SCHs

A-1735 CHs lsoxazol-3-yl CI H SOCHs

A-1736 CHs lsoxazol-3-yl CI H SO2CH3

A-1737 CHs lsoxazol-3-yl CI H CH2OCH3

A-1738 CHs lsoxazol-3-yl CI cyclopropyl H

A-1739 CHs lsoxazol-3-yl CI OCHs H

A-1740 CHs lsoxazol-3-yl CI OCFs H

A-1741 CHs lsoxazol-3-yl CI SCHs H

A-1742 CHs lsoxazol-3-yl CI SOCHs H

A-1743 CHs lsoxazol-3-yl CI SO2CH3 H

A-1744 CHs lsoxazol-3-yl CI CH2OCH3 H

A-1745 CHs lsoxazol-3-yl F H CN

A-1746 CHs lsoxazol-3-yl F H N0 ₂

A-1747 CHs lsoxazol-3-yl F H cyclopropyl

A-1748 CHs lsoxazol-3-yl F H OCHs

A-1749 CHs lsoxazol-3-yl F H OCFs

A-1750 CHs lsoxazol-3-yl F H SCHs

A-1751 CHs lsoxazol-3-yl F H SOCHs

A-1752 CHs lsoxazol-3-yl F H SO2CH3

A-1753 CHs lsoxazol-3-yl F H CH2OCH3

A-1754 CHs lsoxazol-3-yl F cyclopropyl H

A- 1755 CHs lsoxazol-3-yl F OCHs H

A-1756 CHs lsoxazol-3-yl F OCFs H

A- 1757 CHs lsoxazol-3-yl F SCHs H

A-1758 CHs lsoxazol-3-yl F SOCHs H

A-1759 CHs lsoxazol-3-yl F SO2CH3 H A-1760 CHs lsoxazol-3-yl F CH2OCH3 H

A-1761 CHs lsoxazol-3-yl CFs H CN

A-1762 CHs lsoxazol-3-yl CFs H N0 ₂

A-1763 CHs lsoxazol-3-yl CFs H cyclopropyl

A-1764 CHs lsoxazol-3-yl CFs H OCHs

A-1765 CHs lsoxazol-3-yl CFs H OCF3

A-1766 CHs lsoxazol-3-yl CFs H SCHs

A-1767 CHs lsoxazol-3-yl CFs H SOCH3

A-1768 CHs lsoxazol-3-yl CFs H SO2CH3

A-1769 CHs lsoxazol-3-yl CFs H CH2OCH3

A-1770 CHs lsoxazol-3-yl CFs cyclopropyl H

A-1771 CHs lsoxazol-3-yl CFs OCHs H

A-1772 CHs lsoxazol-3-yl CFs OCF3 H

A-1773 CHs lsoxazol-3-yl CFs SCHs H

A-1774 CHs lsoxazol-3-yl CFs SOCH3 H

A- 1775 CHs lsoxazol-3-yl CFs SO2CH3 H

A-1776 CHs lsoxazol-3-yl CFs CH2OCH3 H

A- 1777 CHs lsoxazol-3-yl SO2CH3 H CN

A-1778 CHs lsoxazol-3-yl SO2CH3 H N0 ₂

A-1779 CHs lsoxazol-3-yl SO2CH3 H cyclopropyl

A-1780 CHs lsoxazol-3-yl SO2CH3 H OCHs

A-1781 CHs lsoxazol-3-yl SO2CH3 H OCF3

A-1782 CHs lsoxazol-3-yl SO2CH3 H SCHs

A-1783 CHs lsoxazol-3-yl SO2CH3 H SOCH3

A-1784 CHs lsoxazol-3-yl SO2CH3 H SO2CH3

A-1785 CHs lsoxazol-3-yl SO2CH3 H CH2OCH3

A-1786 CHs lsoxazol-3-yl SO2CH3 cyclopropyl H

A-1787 CHs lsoxazol-3-yl SO2CH3 OCHs H

A-1788 CHs lsoxazol-3-yl SO2CH3 OCF3 H

A-1789 CHs lsoxazol-3-yl SO2CH3 SCHs H

A-1790 CHs lsoxazol-3-yl SO2CH3 SOCH3 H

A-1791 CHs lsoxazol-3-yl SO2CH3 SO2CH3 H

A-1792 CHs lsoxazol-3-yl SO2CH3 CH2OCH3 H

A-1793 CHs lsoxazol-3-yl CN H CN

A-1794 CHs lsoxazol-3-yl CN H N0 ₂

A-1795 CHs lsoxazol-3-yl CN H cyclopropyl

A-1796 CHs lsoxazol-3-yl CN H OCHs A-1797 CHs lsoxazol-3-yl CN H OCFs

A-1798 CHs lsoxazol-3-yl CN H SCHs

A-1799 CHs lsoxazol-3-yl CN H SOCHs

A-1800 CHs lsoxazol-3-yl CN H SO2CH3

A-1801 CHs lsoxazol-3-yl CN H CH2OCH3

A-1802 CHs lsoxazol-3-yl CN cyclopropyl H

A-1803 CHs lsoxazol-3-yl CN OCHs H

A-1804 CHs lsoxazol-3-yl CN OCFs H

A-1805 CHs lsoxazol-3-yl CN SCHs H

A-1806 CHs lsoxazol-3-yl CN SOCHs H

A-1807 CHs lsoxazol-3-yl CN SO2CH3 H

A-1808 CHs lsoxazol-3-yl CN CH2OCH3 H

A-1809 CHs lsoxazol-3-yl H H CN

A-1810 CHs lsoxazol-3-yl H H N0 ₂

A-181 1 CHs lsoxazol-3-yl H H cyclopropyl

A-1812 CHs lsoxazol-3-yl H H OCHs

A-1813 CHs lsoxazol-3-yl H H OCFs

A-1814 CHs lsoxazol-3-yl H H SCHs

A-1815 CHs lsoxazol-3-yl H H SOCHs

A-1816 CHs lsoxazol-3-yl H H SO2CH3

A-1817 CHs lsoxazol-3-yl H H CH2OCH3

A-1818 CHs lsoxazol-3-yl H cyclopropyl H

A-1819 CHs lsoxazol-3-yl H OCHs H

A-1820 CHs lsoxazol-3-yl H OCFs H

A-1821 CHs lsoxazol-3-yl H SCHs H

A-1822 CHs lsoxazol-3-yl H SOCHs H

A-1823 CHs lsoxazol-3-yl H SO2CH3 H

A-1824 CHs lsoxazol-3-yl H CH2OCH3 H

A-1825 CHs 5-Me-lsoxazol-3-yl CI H CN

A-1826 CHs 5-Me-lsoxazol-3-yl CI H N0 ₂

A-1827 CHs 5-Me-lsoxazol-3-yl CI H cyclopropyl

A-1828 CHs 5-Me-lsoxazol-3-yl CI H OCHs

A-1829 CHs 5-Me-lsoxazol-3-yl CI H OCFs

A-1830 CHs 5-Me-lsoxazol-3-yl CI H SCHs

A-1831 CHs 5-Me-lsoxazol-3-yl CI H SOCHs

A-1832 CHs 5-Me-lsoxazol-3-yl CI H SO2CH3

A-1833 CHs 5-Me-lsoxazol-3-yl CI H CH2OCH3 A-1834 CHs 5-Me-lsoxazol-3-yl CI cyclopropyl H

A-1835 CHs 5-Me-lsoxazol-3-yl CI OCHs H

A-1836 CHs 5-Me-lsoxazol-3-yl CI OCFs H

A-1837 CHs 5-Me-lsoxazol-3-yl CI SCHs H

A-1838 CHs 5-Me-lsoxazol-3-yl CI SOCHs H

A-1839 CHs 5-Me-lsoxazol-3-yl CI SO2CH3 H

A-1840 CHs 5-Me-lsoxazol-3-yl CI CH2OCH3 H

A-1841 CHs 5-Me-lsoxazol-3-yl F H CN

A-1842 CHs 5-Me-lsoxazol-3-yl F H N0 ₂

A-1843 CHs 5-Me-lsoxazol-3-yl F H cyclopropyl

A-1844 CHs 5-Me-lsoxazol-3-yl F H OCHs

A-1845 CHs 5-Me-lsoxazol-3-yl F H OCFs

A-1846 CHs 5-Me-lsoxazol-3-yl F H SCHs

A-1847 CHs 5-Me-lsoxazol-3-yl F H SOCHs

A-1848 CHs 5-Me-lsoxazol-3-yl F H SO2CH3

A-1849 CHs 5-Me-lsoxazol-3-yl F H CH2OCH3

A-1850 CHs 5-Me-lsoxazol-3-yl F cyclopropyl H

A-1851 CHs 5-Me-lsoxazol-3-yl F OCHs H

A-1852 CHs 5-Me-lsoxazol-3-yl F OCFs H

A-1853 CHs 5-Me-lsoxazol-3-yl F SCHs H

A-1854 CHs 5-Me-lsoxazol-3-yl F SOCHs H

A-1855 CHs 5-Me-lsoxazol-3-yl F SO2CH3 H

A-1856 CHs 5-Me-lsoxazol-3-yl F CH2OCH3 H

A-1857 CHs 5-Me-lsoxazol-3-yl CFs H CN

A-1858 CHs 5-Me-lsoxazol-3-yl CFs H N0 ₂

A-1859 CHs 5-Me-lsoxazol-3-yl CFs H cyclopropyl

A-1860 CHs 5-Me-lsoxazol-3-yl CFs H OCHs

A-1861 CHs 5-Me-lsoxazol-3-yl CFs H OCFs

A-1862 CHs 5-Me-lsoxazol-3-yl CFs H SCHs

A-1863 CHs 5-Me-lsoxazol-3-yl CFs H SOCHs

A-1864 CHs 5-Me-lsoxazol-3-yl CFs H SO2CH3

A-1865 CHs 5-Me-lsoxazol-3-yl CFs H CH2OCH3

A-1866 CHs 5-Me-lsoxazol-3-yl CFs cyclopropyl H

A-1867 CHs 5-Me-lsoxazol-3-yl CFs OCHs H

A-1868 CHs 5-Me-lsoxazol-3-yl CFs OCFs H

A-1869 CHs 5-Me-lsoxazol-3-yl CFs SCHs H

A-1870 CHs 5-Me-lsoxazol-3-yl CFs SOCHs H A-1871 CHs 5-Me-lsoxazol-3-yl CFs SO2CH3 H

A-1872 CHs 5-Me-lsoxazol-3-yl CFs CH2OCH3 H

A-1873 CHs 5-Me-lsoxazol-3-yl SO2CH3 H CN

A-1874 CHs 5-Me-lsoxazol-3-yl SO2CH3 H N0 ₂

A-1875 CHs 5-Me-lsoxazol-3-yl SO2CH3 H cyclopropyl

A-1876 CHs 5-Me-lsoxazol-3-yl SO2CH3 H OCH3

A-1877 CHs 5-Me-lsoxazol-3-yl SO2CH3 H OCFs

A-1878 CHs 5-Me-lsoxazol-3-yl SO2CH3 H SCHs

A-1879 CHs 5-Me-lsoxazol-3-yl SO2CH3 H SOCHs

A-1880 CHs 5-Me-lsoxazol-3-yl SO2CH3 H SO2CH3

A-1881 CHs 5-Me-lsoxazol-3-yl SO2CH3 H CH2OCH3

A-1882 CHs 5-Me-lsoxazol-3-yl SO2CH3 cyclopropyl H

A-1883 CHs 5-Me-lsoxazol-3-yl SO2CH3 OCH3 H

A-1884 CHs 5-Me-lsoxazol-3-yl SO2CH3 OCFs H

A-1885 CHs 5-Me-lsoxazol-3-yl SO2CH3 SCHs H

A-1886 CHs 5-Me-lsoxazol-3-yl SO2CH3 SOCHs H

A-1887 CHs 5-Me-lsoxazol-3-yl SO2CH3 SO2CH3 H

A-1888 CHs 5-Me-lsoxazol-3-yl SO2CH3 CH2OCH3 H

A-1889 CHs 5-Me-lsoxazol-3-yl CN H CN

A-1890 CHs 5-Me-lsoxazol-3-yl CN H N0 ₂

A-1891 CHs 5-Me-lsoxazol-3-yl CN H cyclopropyl

A-1892 CHs 5-Me-lsoxazol-3-yl CN H OCH3

A-1893 CHs 5-Me-lsoxazol-3-yl CN H OCFs

A-1894 CHs 5-Me-lsoxazol-3-yl CN H SCHs

A-1895 CHs 5-Me-lsoxazol-3-yl CN H SOCHs

A-1896 CHs 5-Me-lsoxazol-3-yl CN H SO2CH3

A-1897 CHs 5-Me-lsoxazol-3-yl CN H CH2OCH3

A-1898 CHs 5-Me-lsoxazol-3-yl CN cyclopropyl H

A-1899 CHs 5-Me-lsoxazol-3-yl CN OCH3 H

A-1900 CHs 5-Me-lsoxazol-3-yl CN OCFs H

A-1901 CHs 5-Me-lsoxazol-3-yl CN SCHs H

A-1902 CHs 5-Me-lsoxazol-3-yl CN SOCHs H

A-1903 CHs 5-Me-lsoxazol-3-yl CN SO2CH3 H

A-1904 CHs 5-Me-lsoxazol-3-yl CN CH2OCH3 H

A-1905 CHs 5-Me-lsoxazol-3-yl H H CN

A-1906 CHs 5-Me-lsoxazol-3-yl H H N0 ₂

A-1907 CHs 5-Me-lsoxazol-3-yl H H cyclopropyl A-1908 CHs 5-Me-lsoxazol-3-yl H H OCHs

A-1909 CHs 5-Me-lsoxazol-3-yl H H OCFs

A-1910 CHs 5-Me-lsoxazol-3-yl H H SCHs

A-191 1 CHs 5-Me-lsoxazol-3-yl H H SOCHs

A-1912 CHs 5-Me-lsoxazol-3-yl H H SO2CH3

A-1913 CHs 5-Me-lsoxazol-3-yl H H CH2OCH3

A-1914 CHs 5-Me-lsoxazol-3-yl H cyclopropyl H

A-1915 CHs 5-Me-lsoxazol-3-yl H OCHs H

A-1916 CHs 5-Me-lsoxazol-3-yl H OCFs H

A-1917 CHs 5-Me-lsoxazol-3-yl H SCHs H

A-1918 CHs 5-Me-lsoxazol-3-yl H SOCHs H

A-1919 CHs 5-Me-lsoxazol-3-yl H SO2CH3 H

A-1920 CHs 5-Me-lsoxazol-3-yl H CH2OCH3 H

A-1921 CHs 3-Me-lsoxazolin-5-yl CI H CN

A-1922 CHs 3-Me-lsoxazolin-5-yl CI H N0 ₂

A-1923 CHs 3-Me-lsoxazolin-5-yl CI H cyclopropyl

A-1924 CHs 3-Me-lsoxazolin-5-yl CI H OCHs

A-1925 CHs 3-Me-lsoxazolin-5-yl CI H OCFs

A-1926 CHs 3-Me-lsoxazolin-5-yl CI H SCHs

A-1927 CHs 3-Me-lsoxazolin-5-yl CI H SOCHs

A-1928 CHs 3-Me-lsoxazolin-5-yl CI H SO2CH3

A-1929 CHs 3-Me-lsoxazolin-5-yl CI H CH2OCH3

A-1930 CHs 3-Me-lsoxazolin-5-yl CI cyclopropyl H

A-1931 CHs 3-Me-lsoxazolin-5-yl CI OCHs H

A-1932 CHs 3-Me-lsoxazolin-5-yl CI OCFs H

A-1933 CHs 3-Me-lsoxazolin-5-yl CI SCHs H

A-1934 CHs 3-Me-lsoxazolin-5-yl CI SOCHs H

A-1935 CHs 3-Me-lsoxazolin-5-yl CI SO2CH3 H

A-1936 CHs 3-Me-lsoxazolin-5-yl CI CH2OCH3 H

A-1937 CHs 3-Me-lsoxazolin-5-yl F H CN

A-1938 CHs 3-Me-lsoxazolin-5-yl F H N0 ₂

A-1939 CHs 3-Me-lsoxazolin-5-yl F H cyclopropyl

A-1940 CHs 3-Me-lsoxazolin-5-yl F H OCHs

A-1941 CHs 3-Me-lsoxazolin-5-yl F H OCFs

A-1942 CHs 3-Me-lsoxazolin-5-yl F H SCHs

A-1943 CHs 3-Me-lsoxazolin-5-yl F H SOCHs

A-1944 CHs 3-Me-lsoxazolin-5-yl F H SO2CH3 A-1945 CHs 3-Me-lsoxazolin-5-yl F H CH2OCH3

A-1946 CHs 3-Me-lsoxazolin-5-yl F cyclopropyl H

A-1947 CHs 3-Me-lsoxazolin-5-yl F OCH3 H

A-1948 CHs 3-Me-lsoxazolin-5-yl F OCFs H

A-1949 CHs 3-Me-lsoxazolin-5-yl F SCHs H

A-1950 CHs 3-Me-lsoxazolin-5-yl F SOCHs H

A-1951 CHs 3-Me-lsoxazolin-5-yl F SO2CH3 H

A-1952 CHs 3-Me-lsoxazolin-5-yl F CH2OCH3 H

A-1953 CHs 3-Me-lsoxazolin-5-yl CFs H CN

A-1954 CHs 3-Me-lsoxazolin-5-yl CFs H N0 ₂

A-1955 CHs 3-Me-lsoxazolin-5-yl CFs H cyclopropyl

A-1956 CHs 3-Me-lsoxazolin-5-yl CFs H OCHs

A-1957 CHs 3-Me-lsoxazolin-5-yl CFs H OCFs

A-1958 CHs 3-Me-lsoxazolin-5-yl CFs H SCHs

A-1959 CHs 3-Me-lsoxazolin-5-yl CFs H SOCHs

A-1960 CHs 3-Me-lsoxazolin-5-yl CFs H SO2CH3

A-1961 CHs 3-Me-lsoxazolin-5-yl CFs H CH2OCH3

A-1962 CHs 3-Me-lsoxazolin-5-yl CFs cyclopropyl H

A-1963 CHs 3-Me-lsoxazolin-5-yl CFs OCH3 H

A-1964 CHs 3-Me-lsoxazolin-5-yl CFs OCFs H

A-1965 CHs 3-Me-lsoxazolin-5-yl CFs SCHs H

A-1966 CHs 3-Me-lsoxazolin-5-yl CFs SOCHs H

A-1967 CHs 3-Me-lsoxazolin-5-yl CFs SO2CH3 H

A-1968 CHs 3-Me-lsoxazolin-5-yl CFs CH2OCH3 H

A-1969 CHs 3-Me-lsoxazolin-5-yl SO2CH3 H CN

A-1970 CHs 3-Me-lsoxazolin-5-yl SO2CH3 H N0 ₂

A-1971 CHs 3-Me-lsoxazolin-5-yl SO2CH3 H cyclopropyl

A-1972 CHs 3-Me-lsoxazolin-5-yl SO2CH3 H OCHs

A-1973 CHs 3-Me-lsoxazolin-5-yl SO2CH3 H OCFs

A-1974 CHs 3-Me-lsoxazolin-5-yl SO2CH3 H SCHs

A-1975 CHs 3-Me-lsoxazolin-5-yl SO2CH3 H SOCHs

A-1976 CHs 3-Me-lsoxazolin-5-yl SO2CH3 H SO2CH3

A-1977 CHs 3-Me-lsoxazolin-5-yl SO2CH3 H CH2OCH3

A-1978 CHs 3-Me-lsoxazolin-5-yl SO2CH3 cyclopropyl H

A-1979 CHs 3-Me-lsoxazolin-5-yl SO2CH3 OCH3 H

A-1980 CHs 3-Me-lsoxazolin-5-yl SO2CH3 OCFs H

A-1981 CHs 3-Me-lsoxazolin-5-yl SO2CH3 SCHs H A-1982 CHs 3-Me-lsoxazolin-5-yl SO2CH3 SOCHs H

A-1983 CHs 3-Me-lsoxazolin-5-yl SO2CH3 SO2CH3 H

A-1984 CHs 3-Me-lsoxazolin-5-yl SO2CH3 CH2OCH3 H

A-1985 CHs 3-Me-lsoxazolin-5-yl CN H CN

A-1986 CHs 3-Me-lsoxazolin-5-yl CN H N0 ₂

A-1987 CHs 3-Me-lsoxazolin-5-yl CN H cyclopropyl

A-1988 CHs 3-Me-lsoxazolin-5-yl CN H OCH3

A-1989 CHs 3-Me-lsoxazolin-5-yl CN H OCFs

A-1990 CHs 3-Me-lsoxazolin-5-yl CN H SCHs

A-1991 CHs 3-Me-lsoxazolin-5-yl CN H SOCHs

A-1992 CHs 3-Me-lsoxazolin-5-yl CN H SO2CH3

A-1993 CHs 3-Me-lsoxazolin-5-yl CN H CH2OCH3

A-1994 CHs 3-Me-lsoxazolin-5-yl CN cyclopropyl H

A-1995 CHs 3-Me-lsoxazolin-5-yl CN OCH3 H

A-1996 CHs 3-Me-lsoxazolin-5-yl CN OCFs H

A-1997 CHs 3-Me-lsoxazolin-5-yl CN SCHs H

A-1998 CHs 3-Me-lsoxazolin-5-yl CN SOCHs H

A-1999 CHs 3-Me-lsoxazolin-5-yl CN SO2CH3 H

A-2000 CHs 3-Me-lsoxazolin-5-yl CN CH2OCH3 H

A-2001 CHs 3-Me-lsoxazolin-5-yl H H CN

A-2002 CHs 3-Me-lsoxazolin-5-yl H H N0 ₂

A-2003 CHs 3-Me-lsoxazolin-5-yl H H cyclopropyl

A-2004 CHs 3-Me-lsoxazolin-5-yl H H OCH3

A-2005 CHs 3-Me-lsoxazolin-5-yl H H OCFs

A-2006 CHs 3-Me-lsoxazolin-5-yl H H SCHs

A-2007 CHs 3-Me-lsoxazolin-5-yl H H SOCHs

A-2008 CHs 3-Me-lsoxazolin-5-yl H H SO2CH3

A-2009 CHs 3-Me-lsoxazolin-5-yl H H CH2OCH3

A-2010 CHs 3-Me-lsoxazolin-5-yl H cyclopropyl H

A-201 1 CHs 3-Me-lsoxazolin-5-yl H OCH3 H

A-2012 CHs 3-Me-lsoxazolin-5-yl H OCFs H

A-2013 CHs 3-Me-lsoxazolin-5-yl H SCHs H

A-2014 CHs 3-Me-lsoxazolin-5-yl H SOCHs H

A-2015 CHs 3-Me-lsoxazolin-5-yl H SO2CH3 H

A-2016 CHs 3-Me-lsoxazolin-5-yl H CH2OCH3 H

A-2017 CHs 3-Me-lsoxazol-5-yl CI H CN

A-2018 CHs 3-Me-lsoxazol-5-yl CI H N0 ₂ A-2019 CHs 3-Me-lsoxazol-5-yl CI H cyclopropyl

A-2020 CHs 3-Me-lsoxazol-5-yl CI H OCHs

A-2021 CHs 3-Me-lsoxazol-5-yl CI H OCFs

A-2022 CHs 3-Me-lsoxazol-5-yl CI H SCHs

A-2023 CHs 3-Me-lsoxazol-5-yl CI H SOCHs

A-2024 CHs 3-Me-lsoxazol-5-yl CI H SO2CH3

A-2025 CHs 3-Me-lsoxazol-5-yl CI H CH2OCH3

A-2026 CHs 3-Me-lsoxazol-5-yl CI cyclopropyl H

A-2027 CHs 3-Me-lsoxazol-5-yl CI OCHs H

A-2028 CHs 3-Me-lsoxazol-5-yl CI OCFs H

A-2029 CHs 3-Me-lsoxazol-5-yl CI SCHs H

A-2030 CHs 3-Me-lsoxazol-5-yl CI SOCHs H

A-2031 CHs 3-Me-lsoxazol-5-yl CI SO2CH3 H

A-2032 CHs 3-Me-lsoxazol-5-yl CI CH2OCH3 H

A-2033 CHs 3-Me-lsoxazol-5-yl F H CN

A-2034 CHs 3-Me-lsoxazol-5-yl F H N0 ₂

A-2035 CHs 3-Me-lsoxazol-5-yl F H cyclopropyl

A-2036 CHs 3-Me-lsoxazol-5-yl F H OCHs

A-2037 CHs 3-Me-lsoxazol-5-yl F H OCFs

A-2038 CHs 3-Me-lsoxazol-5-yl F H SCHs

A-2039 CHs 3-Me-lsoxazol-5-yl F H SOCHs

A-2040 CHs 3-Me-lsoxazol-5-yl F H SO2CH3

A-2041 CHs 3-Me-lsoxazol-5-yl F H CH2OCH3

A-2042 CHs 3-Me-lsoxazol-5-yl F cyclopropyl H

A-2043 CHs 3-Me-lsoxazol-5-yl F OCHs H

A-2044 CHs 3-Me-lsoxazol-5-yl F OCFs H

A-2045 CHs 3-Me-lsoxazol-5-yl F SCHs H

A-2046 CHs 3-Me-lsoxazol-5-yl F SOCHs H

A-2047 CHs 3-Me-lsoxazol-5-yl F SO2CH3 H

A-2048 CHs 3-Me-lsoxazol-5-yl F CH2OCH3 H

A-2049 CHs 3-Me-lsoxazol-5-yl CFs H CN

A-2050 CHs 3-Me-lsoxazol-5-yl CFs H N0 ₂

A-2051 CHs 3-Me-lsoxazol-5-yl CFs H cyclopropyl

A-2052 CHs 3-Me-lsoxazol-5-yl CFs H OCHs

A-2053 CHs 3-Me-lsoxazol-5-yl CFs H OCFs

A-2054 CHs 3-Me-lsoxazol-5-yl CFs H SCHs

A-2055 CHs 3-Me-lsoxazol-5-yl CFs H SOCHs A-2056 CHs 3-Me-lsoxazol-5-yl CFs H SO2CH3

A-2057 CHs 3-Me-lsoxazol-5-yl CFs H CH2OCH3

A-2058 CHs 3-Me-lsoxazol-5-yl CFs cyclopropyl H

A-2059 CHs 3-Me-lsoxazol-5-yl CFs OCHs H

A-2060 CHs 3-Me-lsoxazol-5-yl CFs OCF3 H

A-2061 CHs 3-Me-lsoxazol-5-yl CFs SCHs H

A-2062 CHs 3-Me-lsoxazol-5-yl CFs SOCH3 H

A-2063 CHs 3-Me-lsoxazol-5-yl CFs SO2CH3 H

A-2064 CHs 3-Me-lsoxazol-5-yl CFs CH2OCH3 H

A-2065 CHs 3-Me-lsoxazol-5-yl SO2CH3 H CN

A-2066 CHs 3-Me-lsoxazol-5-yl SO2CH3 H N0 ₂

A-2067 CHs 3-Me-lsoxazol-5-yl SO2CH3 H cyclopropyl

A-2068 CHs 3-Me-lsoxazol-5-yl SO2CH3 H OCHs

A-2069 CHs 3-Me-lsoxazol-5-yl SO2CH3 H OCFs

A-2070 CHs 3-Me-lsoxazol-5-yl SO2CH3 H SCHs

A-2071 CHs 3-Me-lsoxazol-5-yl SO2CH3 H SOCHs

A-2072 CHs 3-Me-lsoxazol-5-yl SO2CH3 H SO2CH3

A-2073 CHs 3-Me-lsoxazol-5-yl SO2CH3 H CH2OCH3

A-2074 CHs 3-Me-lsoxazol-5-yl SO2CH3 cyclopropyl H

A-2075 CHs 3-Me-lsoxazol-5-yl SO2CH3 OCHs H

A-2076 CHs 3-Me-lsoxazol-5-yl SO2CH3 OCF3 H

A-2077 CHs 3-Me-lsoxazol-5-yl SO2CH3 SCHs H

A-2078 CHs 3-Me-lsoxazol-5-yl SO2CH3 SOCH3 H

A-2079 CHs 3-Me-lsoxazol-5-yl SO2CH3 SO2CH3 H

A-2080 CHs 3-Me-lsoxazol-5-yl SO2CH3 CH2OCH3 H

A-2081 CHs 3-Me-lsoxazol-5-yl CN H CN

A-2082 CHs 3-Me-lsoxazol-5-yl CN H N0 ₂

A-2083 CHs 3-Me-lsoxazol-5-yl CN H cyclopropyl

A-2084 CHs 3-Me-lsoxazol-5-yl CN H OCHs

A-2085 CHs 3-Me-lsoxazol-5-yl CN H OCFs

A-2086 CHs 3-Me-lsoxazol-5-yl CN H SCHs

A-2087 CHs 3-Me-lsoxazol-5-yl CN H SOCHs

A-2088 CHs 3-Me-lsoxazol-5-yl CN H SO2CH3

A-2089 CHs 3-Me-lsoxazol-5-yl CN H CH2OCH3

A-2090 CHs 3-Me-lsoxazol-5-yl CN cyclopropyl H

A-2091 CHs 3-Me-lsoxazol-5-yl CN OCHs H

A-2092 CHs 3-Me-lsoxazol-5-yl CN OCF3 H A-2241 CFs SCHs CFs H CN

A-2242 CFs SCHs CFs H N0 ₂

A-2243 CFs SCHs CFs H cyclopropyl

A-2244 CFs SCHs CFs H OCHs

A-2245 CFs SCHs CFs H OCF3

A-2246 CFs SCHs CFs H SCHs

A-2247 CFs SCHs CFs H SOCH3

A-2248 CFs SCHs CFs H SO2CH3

A-2249 CFs SCHs CFs H CH2OCH3

A-2250 CFs SCHs CFs cyclopropyl H

A-2251 CFs SCHs CFs OCHs H

A-2252 CFs SCHs CFs OCF3 H

A-2253 CFs SCHs CFs SCHs H

A-2254 CFs SCHs CFs SOCH3 H

A-2255 CFs SCHs CFs SO2CH3 H

A-2256 CFs SCHs CFs CH2OCH3 H

A-2257 CFs SCHs SO2CH3 H CN

A-2258 CFs SCHs SO2CH3 H N0 ₂

A-2259 CFs SCHs SO2CH3 H cyclopropyl

A-2260 CFs SCHs SO2CH3 H OCHs

A-2261 CFs SCHs SO2CH3 H OCF3

A-2262 CFs SCHs SO2CH3 H SCHs

A-2263 CFs SCHs SO2CH3 H SOCH3

A-2264 CFs SCHs SO2CH3 H SO2CH3

A-2265 CFs SCHs SO2CH3 H CH2OCH3

A-2266 CFs SCHs SO2CH3 cyclopropyl H

A-2267 CFs SCHs SO2CH3 OCHs H

A-2268 CFs SCHs SO2CH3 OCF3 H

A-2269 CFs SCHs SO2CH3 SCHs H

A-2270 CFs SCHs SO2CH3 SOCH3 H

A-2271 CFs SCHs SO2CH3 SO2CH3 H

A-2272 CFs SCHs SO2CH3 CH2OCH3 H

A-2273 CFs SCHs CN H CN

A-2274 CFs SCHs CN H N0 ₂

A-2275 CFs SCHs CN H cyclopropyl

A-2276 CFs SCHs CN H OCHs

A-2277 CFs SCHs CN H OCF3 A-2278 CFs SCHs CN H SCHs

A-2279 CFs SCHs CN H SOCHs

A-2280 CFs SCHs CN H SO2CH3

A-2281 CFs SCHs CN H CH2OCH3

A-2282 CFs SCHs CN cyclopropyl H

A-2283 CFs SCHs CN OCHs H

A-2284 CFs SCHs CN OCFs H

A-2285 CFs SCHs CN SCHs H

A-2286 CFs SCHs CN SOCHs H

A-2287 CFs SCHs CN SO2CH3 H

A-2288 CFs SCHs CN CH2OCH3 H

A-2289 CFs SOCHs H H CN

A-2290 CFs SOCHs H H N0 ₂

A-2291 CFs SOCHs H H cyclopropyl

A-2292 CFs SOCHs H H OCHs

A-2293 CFs SOCHs H H OCFs

A-2294 CFs SOCHs H H SCHs

A-2295 CFs SOCHs H H SOCHs

A-2296 CFs SOCHs H H SO2CH3

A-2297 CFs SOCHs H H CH2OCH3

A-2298 CFs SOCHs H cyclopropyl H

A-2299 CFs SOCHs H OCHs H

A-2300 CFs SOCHs H OCFs H

A-2301 CFs SOCHs H SCHs H

A-2302 CFs SOCHs H SOCHs H

A-2303 CFs SOCHs H SO2CH3 H

A-2304 CFs SOCHs H CH2OCH3 H

A-2305 CFs SOCHs CI H CN

A-2306 CFs SOCHs CI H N0 ₂

A-2307 CFs SOCHs CI H cyclopropyl

A-2308 CFs SOCHs CI H OCHs

A-2309 CFs SOCHs CI H OCFs

A-2310 CFs SOCHs CI H SCHs

A-231 1 CFs SOCHs CI H SOCHs

A-2312 CFs SOCHs CI H SO2CH3

A-2313 CFs SOCHs CI H CH2OCH3

A-2314 CFs SOCHs CI cyclopropyl H A-2315 CFs SOCHs CI OCHs H

A-2316 CFs SOCHs CI OCFs H

A-2317 CFs SOCHs CI SCHs H

A-2318 CFs SOCHs CI SOCHs H

A-2319 CFs SOCHs CI SO2CH3 H

A-2320 CFs SOCHs CI CH2OCH3 H

A-2321 CFs SOCHs F H CN

A-2322 CFs SOCHs F H N0 ₂

A-2323 CFs SOCHs F H cyclopropyl

A-2324 CFs SOCHs F H OCHs

A-2325 CFs SOCHs F H OCFs

A-2326 CFs SOCHs F H SCHs

A-2327 CFs SOCHs F H SOCHs

A-2328 CFs SOCHs F H SO2CH3

A-2329 CFs SOCHs F H CH2OCH3

A-2330 CFs SOCHs F cyclopropyl H

A-2331 CFs SOCHs F OCHs H

A-2332 CFs SOCHs F OCFs H

A-2333 CFs SOCHs F SCHs H

A-2334 CFs SOCHs F SOCHs H

A-2335 CFs SOCHs F SO2CH3 H

A-2336 CFs SOCHs F CH2OCH3 H

A-2337 CFs SOCHs CFs H CN

A-2338 CFs SOCHs CFs H N0 ₂

A-2339 CFs SOCHs CFs H cyclopropyl

A-2340 CFs SOCHs CFs H OCHs

A-2341 CFs SOCHs CFs H OCFs

A-2342 CFs SOCHs CFs H SCHs

A-2343 CFs SOCHs CFs H SOCHs

A-2344 CFs SOCHs CFs H SO2CH3

A-2345 CFs SOCHs CFs H CH2OCH3

A-2346 CFs SOCHs CFs cyclopropyl H

A-2347 CFs SOCHs CFs OCHs H

A-2348 CFs SOCHs CFs OCFs H

A-2349 CFs SOCHs CFs SCHs H

A-2350 CFs SOCHs CFs SOCHs H

A-2351 CFs SOCHs CFs SO2CH3 H A-2352 CFs SOCHs CFs CH2OCH3 H

A-2353 CFs SOCHs SO2CH3 H CN

A-2354 CFs SOCHs SO2CH3 H N0 ₂

A-2355 CFs SOCHs SO2CH3 H cyclopropyl

A-2356 CFs SOCHs SO2CH3 H OCHs

A-2357 CFs SOCHs SO2CH3 H OCF3

A-2358 CFs SOCHs SO2CH3 H SCHs

A-2359 CFs SOCHs SO2CH3 H SOCHs

A-2360 CFs SOCHs SO2CH3 H SO2CH3

A-2361 CFs SOCHs SO2CH3 H CH2OCH3

A-2362 CFs SOCHs SO2CH3 cyclopropyl H

A-2363 CFs SOCHs SO2CH3 OCHs H

A-2364 CFs SOCHs SO2CH3 OCF3 H

A-2365 CFs SOCHs SO2CH3 SCHs H

A-2366 CFs SOCHs SO2CH3 SOCHs H

A-2367 CFs SOCHs SO2CH3 SO2CH3 H

A-2368 CFs SOCHs SO2CH3 CH2OCH3 H

A-2369 CFs SOCHs CN H CN

A-2370 CFs SOCHs CN H N0 ₂

A-2371 CFs SOCHs CN H cyclopropyl

A-2372 CFs SOCHs CN H OCHs

A-2373 CFs SOCHs CN H OCF3

A-2374 CFs SOCHs CN H SCHs

A-2375 CFs SOCHs CN H SOCHs

A-2376 CFs SOCHs CN H SO2CH3

A-2377 CFs SOCHs CN H CH2OCH3

A-2378 CFs SOCHs CN cyclopropyl H

A-2379 CFs SOCHs CN OCHs H

A-2380 CFs SOCHs CN OCF3 H

A-2381 CFs SOCHs CN SCHs H

A-2382 CFs SOCHs CN SOCHs H

A-2383 CFs SOCHs CN SO2CH3 H

A-2384 CFs SOCHs CN CH2OCH3 H

A-2385 CFs SOCHs H H CN

A-2386 CFs SOCHs H H N0 ₂

A-2387 CFs SOCHs H H cyclopropyl

A-2388 CFs SOCHs H H OCHs A-2426 CFs SO2CH3 F cyclopropyl H

A-2427 CFs SO2CH3 F OCHs H

A-2428 CFs SO2CH3 F OCF3 H

A-2429 CFs SO2CH3 F SCHs H

A-2430 CFs SO2CH3 F SOCH3 H

A-2431 CFs SO2CH3 F SO2CH3 H

A-2432 CFs SO2CH3 F CH2OCH3 H

A-2433 CFs SO2CH3 CFs H CN

A-2434 CFs SO2CH3 CFs H N0 ₂

A-2435 CFs SO2CH3 CFs H cyclopropyl

A-2436 CFs SO2CH3 CFs H OCHs

A-2437 CFs SO2CH3 CFs H OCFs

A-2438 CFs SO2CH3 CFs H SCHs

A-2439 CFs SO2CH3 CFs H SOCHs

A-2440 CFs SO2CH3 CFs H SO2CH3

A-2441 CFs SO2CH3 CFs H CH2OCH3

A-2442 CFs SO2CH3 CFs cyclopropyl H

A-2443 CFs SO2CH3 CFs OCHs H

A-2444 CFs SO2CH3 CFs OCF3 H

A-2445 CFs SO2CH3 CFs SCHs H

A-2446 CFs SO2CH3 CFs SOCH3 H

A-2447 CFs SO2CH3 CFs SO2CH3 H

A-2448 CFs SO2CH3 CFs CH2OCH3 H

A-2449 CFs SO2CH3 SO2CH3 H CN

A-2450 CFs SO2CH3 SO2CH3 H N0 ₂

A-2451 CFs SO2CH3 SO2CH3 H cyclopropyl

A-2452 CFs SO2CH3 SO2CH3 H OCHs

A-2453 CFs SO2CH3 SO2CH3 H OCFs

A-2454 CFs SO2CH3 SO2CH3 H SCHs

A-2455 CFs SO2CH3 SO2CH3 H SOCHs

A-2456 CFs SO2CH3 SO2CH3 H SO2CH3

A-2457 CFs SO2CH3 SO2CH3 H CH2OCH3

A-2458 CFs SO2CH3 SO2CH3 cyclopropyl H

A-2459 CFs SO2CH3 SO2CH3 OCHs H

A-2460 CFs SO2CH3 SO2CH3 OCF3 H

A-2461 CFs SO2CH3 SO2CH3 SCHs H

A-2462 CFs SO2CH3 SO2CH3 SOCH3 H A-2500 CFs CH2OCH2CF3 CI H OCHs

A-2501 CFs CH2OCH2CF3 CI H OCFs

A-2502 CFs CH2OCH2CF3 CI H SCHs

A-2503 CFs CH2OCH2CF3 CI H SOCH3

A-2504 CFs CH2OCH2CF3 CI H SO2CH3

A-2505 CFs CH2OCH2CF3 CI H CH2OCH3

A-2506 CFs CH2OCH2CF3 CI cyclopropyl H

A-2507 CFs CH2OCH2CF3 CI OCHs H

A-2508 CFs CH2OCH2CF3 CI OCFs H

A-2509 CFs CH2OCH2CF3 CI SCHs H

A-2510 CFs CH2OCH2CF3 CI SOCH3 H

A-251 1 CFs CH2OCH2CF3 CI SO2CH3 H

A-2512 CFs CH2OCH2CF3 CI CH2OCH3 H

A-2513 CFs CH2OCH2CF3 F H CN

A-2514 CFs CH2OCH2CF3 F H N0 ₂

A-2515 CFs CH2OCH2CF3 F H cyclopropyl

A-2516 CFs CH2OCH2CF3 F H OCHs

A-2517 CFs CH2OCH2CF3 F H OCFs

A-2518 CFs CH2OCH2CF3 F H SCHs

A-2519 CFs CH2OCH2CF3 F H SOCH3

A-2520 CFs CH2OCH2CF3 F H SO2CH3

A-2521 CFs CH2OCH2CF3 F H CH2OCH3

A-2522 CFs CH2OCH2CF3 F cyclopropyl H

A-2523 CFs CH2OCH2CF3 F OCHs H

A-2524 CFs CH2OCH2CF3 F OCFs H

A-2525 CFs CH2OCH2CF3 F SCHs H

A-2526 CFs CH2OCH2CF3 F SOCH3 H

A-2527 CFs CH2OCH2CF3 F SO2CH3 H

A-2528 CFs CH2OCH2CF3 F CH2OCH3 H

A-2529 CFs CH2OCH2CF3 CFs H CN

A-2530 CFs CH2OCH2CF3 CFs H N0 ₂

A-2531 CFs CH2OCH2CF3 CFs H cyclopropyl

A-2532 CFs CH2OCH2CF3 CFs H OCHs

A-2533 CFs CH2OCH2CF3 CFs H OCFs

A-2534 CFs CH2OCH2CF3 CFs H SCHs

A-2535 CFs CH2OCH2CF3 CFs H SOCH3

A-2536 CFs CH2OCH2CF3 CFs H SO2CH3 A-2537 CFs CH2OCH2CF3 CFs H CH2OCH3

A-2538 CFs CH2OCH2CF3 CFs cyclopropyl H

A-2539 CFs CH2OCH2CF3 CFs OCHs H

A-2540 CFs CH2OCH2CF3 CFs OCF3 H

A-2541 CFs CH2OCH2CF3 CFs SCHs H

A-2542 CFs CH2OCH2CF3 CFs SOCH3 H

A-2543 CFs CH2OCH2CF3 CFs SO2CH3 H

A-2544 CFs CH2OCH2CF3 CFs CH2OCH3 H

A-2545 CFs CH2OCH2CF3 SO2CH3 H CN

A-2546 CFs CH2OCH2CF3 SO2CH3 H N0 ₂

A-2547 CFs CH2OCH2CF3 SO2CH3 H cyclopropyl

A-2548 CFs CH2OCH2CF3 SO2CH3 H OCHs

A-2549 CFs CH2OCH2CF3 SO2CH3 H OCFs

A-2550 CFs CH2OCH2CF3 SO2CH3 H SCHs

A-2551 CFs CH2OCH2CF3 SO2CH3 H SOCHs

A-2552 CFs CH2OCH2CF3 SO2CH3 H SO2CH3

A-2553 CFs CH2OCH2CF3 SO2CH3 H CH2OCH3

A-2554 CFs CH2OCH2CF3 SO2CH3 cyclopropyl H

A-2555 CFs CH2OCH2CF3 SO2CH3 OCHs H

A-2556 CFs CH2OCH2CF3 SO2CH3 OCF3 H

A-2557 CFs CH2OCH2CF3 SO2CH3 SCHs H

A-2558 CFs CH2OCH2CF3 SO2CH3 SOCH3 H

A-2559 CFs CH2OCH2CF3 SO2CH3 SO2CH3 H

A-2560 CFs CH2OCH2CF3 SO2CH3 CH2OCH3 H

A-2561 CFs CH2OCH2CF3 CN H CN

A-2562 CFs CH2OCH2CF3 CN H N0 ₂

A-2563 CFs CH2OCH2CF3 CN H cyclopropyl

A-2564 CFs CH2OCH2CF3 CN H OCHs

A-2565 CFs CH2OCH2CF3 CN H OCFs

A-2566 CFs CH2OCH2CF3 CN H SCHs

A-2567 CFs CH2OCH2CF3 CN H SOCHs

A-2568 CFs CH2OCH2CF3 CN H SO2CH3

A-2569 CFs CH2OCH2CF3 CN H CH2OCH3

A-2570 CFs CH2OCH2CF3 CN cyclopropyl H

A-2571 CFs CH2OCH2CF3 CN OCHs H

A-2572 CFs CH2OCH2CF3 CN OCF3 H

A-2573 CFs CH2OCH2CF3 CN SCHs H A-2574 CFs CH2OCH2CF3 CN SOCH3 H

A-2575 CFs CH2OCH2CF3 CN SO2CH3 H

A-2576 CFs CH2OCH2CF3 CN CH2OCH3 H

A-2577 CFs CH2OCH2CF3 H H CN

A-2578 CFs CH2OCH2CF3 H H N0 ₂

A-2579 CFs CH2OCH2CF3 H H cyclopropyl

A-2580 CFs CH2OCH2CF3 H H OCHs

A-2581 CFs CH2OCH2CF3 H H OCF3

A-2582 CFs CH2OCH2CF3 H H SCHs

A-2583 CFs CH2OCH2CF3 H H SOCH3

A-2584 CFs CH2OCH2CF3 H H SO2CH3

A-2585 CFs CH2OCH2CF3 H H CH2OCH3

A-2586 CFs CH2OCH2CF3 H cyclopropyl H

A-2587 CFs CH2OCH2CF3 H OCHs H

A-2588 CFs CH2OCH2CF3 H OCF3 H

A-2589 CFs CH2OCH2CF3 H SCHs H

A-2590 CFs CH2OCH2CF3 H SOCH3 H

A-2591 CFs CH2OCH2CF3 H SO2CH3 H

A-2592 CFs CH2OCH2CF3 H CH2OCH3 H

A-2593 CFs lsoxazolin-3-yl CI H CN

A-2594 CFs lsoxazolin-3-yl CI H N0 ₂

A-2595 CFs lsoxazolin-3-yl CI H cyclopropyl

A-2596 CFs lsoxazolin-3-yl CI H OCHs

A-2597 CFs lsoxazolin-3-yl CI H OCF3

A-2598 CFs lsoxazolin-3-yl CI H SCHs

A-2599 CFs lsoxazolin-3-yl CI H SOCH3

A-2600 CFs lsoxazolin-3-yl CI H SO2CH3

A-2601 CFs lsoxazolin-3-yl CI H CH2OCH3

A-2602 CFs lsoxazolin-3-yl CI cyclopropyl H

A-2603 CFs lsoxazolin-3-yl CI OCHs H

A-2604 CFs lsoxazolin-3-yl CI OCF3 H

A-2605 CFs lsoxazolin-3-yl CI SCHs H

A-2606 CFs lsoxazolin-3-yl CI SOCH3 H

A-2607 CFs lsoxazolin-3-yl CI SO2CH3 H

A-2608 CFs lsoxazolin-3-yl CI CH2OCH3 H

A-2609 CFs lsoxazolin-3-yl F H CN

A-2610 CFs lsoxazolin-3-yl F H N0 ₂ A-261 1 CFs lsoxazolin-3-yl F H cyclopropyl

A-2612 CFs lsoxazolin-3-yl F H OCH3

A-2613 CFs lsoxazolin-3-yl F H OCFs

A-2614 CFs lsoxazolin-3-yl F H SCHs

A-2615 CFs lsoxazolin-3-yl F H SOCHs

A-2616 CFs lsoxazolin-3-yl F H SO2CH3

A-2617 CFs lsoxazolin-3-yl F H CH2OCH3

A-2618 CFs lsoxazolin-3-yl F cyclopropyl H

A-2619 CFs lsoxazolin-3-yl F OCH3 H

A-2620 CFs lsoxazolin-3-yl F OCFs H

A-2621 CFs lsoxazolin-3-yl F SCHs H

A-2622 CFs lsoxazolin-3-yl F SOCHs H

A-2623 CFs lsoxazolin-3-yl F SO2CH3 H

A-2624 CFs lsoxazolin-3-yl F CH2OCH3 H

A-2625 CFs lsoxazolin-3-yl CFs H CN

A-2626 CFs lsoxazolin-3-yl CFs H N0 ₂

A-2627 CFs lsoxazolin-3-yl CFs H cyclopropyl

A-2628 CFs lsoxazolin-3-yl CFs H OCH3

A-2629 CFs lsoxazolin-3-yl CFs H OCFs

A-2630 CFs lsoxazolin-3-yl CFs H SCHs

A-2631 CFs lsoxazolin-3-yl CFs H SOCHs

A-2632 CFs lsoxazolin-3-yl CFs H SO2CH3

A-2633 CFs lsoxazolin-3-yl CFs H CH2OCH3

A-2634 CFs lsoxazolin-3-yl CFs cyclopropyl H

A-2635 CFs lsoxazolin-3-yl CFs OCH3 H

A-2636 CFs lsoxazolin-3-yl CFs OCFs H

A-2637 CFs lsoxazolin-3-yl CFs SCHs H

A-2638 CFs lsoxazolin-3-yl CFs SOCHs H

A-2639 CFs lsoxazolin-3-yl CFs SO2CH3 H

A-2640 CFs lsoxazolin-3-yl CFs CH2OCH3 H

A-2641 CFs lsoxazolin-3-yl SO2CH3 H CN

A-2642 CFs lsoxazolin-3-yl SO2CH3 H N0 ₂

A-2643 CFs lsoxazolin-3-yl SO2CH3 H cyclopropyl

A-2644 CFs lsoxazolin-3-yl SO2CH3 H OCH3

A-2645 CFs lsoxazolin-3-yl SO2CH3 H OCFs

A-2646 CFs lsoxazolin-3-yl SO2CH3 H SCHs

A-2647 CFs lsoxazolin-3-yl SO2CH3 H SOCHs A-2648 CFs lsoxazolin-3-yl SO2CH3 H SO2CH3

A-2649 CFs lsoxazolin-3-yl SO2CH3 H CH2OCH3

A-2650 CFs lsoxazolin-3-yl SO2CH3 cyclopropyl H

A-2651 CFs lsoxazolin-3-yl SO2CH3 OCH3 H

A-2652 CFs lsoxazolin-3-yl SO2CH3 OCFs H

A-2653 CFs lsoxazolin-3-yl SO2CH3 SCHs H

A-2654 CFs lsoxazolin-3-yl SO2CH3 SOCHs H

A-2655 CFs lsoxazolin-3-yl SO2CH3 SO2CH3 H

A-2656 CFs lsoxazolin-3-yl SO2CH3 CH2OCH3 H

A-2657 CFs lsoxazolin-3-yl CN H CN

A-2658 CFs lsoxazolin-3-yl CN H N0 ₂

A-2659 CFs lsoxazolin-3-yl CN H cyclopropyl

A-2660 CFs lsoxazolin-3-yl CN H OCHs

A-2661 CFs lsoxazolin-3-yl CN H OCFs

A-2662 CFs lsoxazolin-3-yl CN H SCHs

A-2663 CFs lsoxazolin-3-yl CN H SOCHs

A-2664 CFs lsoxazolin-3-yl CN H SO2CH3

A-2665 CFs lsoxazolin-3-yl CN H CH2OCH3

A-2666 CFs lsoxazolin-3-yl CN cyclopropyl H

A-2667 CFs lsoxazolin-3-yl CN OCH3 H

A-2668 CFs lsoxazolin-3-yl CN OCFs H

A-2669 CFs lsoxazolin-3-yl CN SCHs H

A-2670 CFs lsoxazolin-3-yl CN SOCHs H

A-2671 CFs lsoxazolin-3-yl CN SO2CH3 H

A-2672 CFs lsoxazolin-3-yl CN CH2OCH3 H

A-2673 CFs lsoxazolin-3-yl H H CN

A-2674 CFs lsoxazolin-3-yl H H N0 ₂

A-2675 CFs lsoxazolin-3-yl H H cyclopropyl

A-2676 CFs lsoxazolin-3-yl H H OCHs

A-2677 CFs lsoxazolin-3-yl H H OCFs

A-2678 CFs lsoxazolin-3-yl H H SCHs

A-2679 CFs lsoxazolin-3-yl H H SOCHs

A-2680 CFs lsoxazolin-3-yl H H SO2CH3

A-2681 CFs lsoxazolin-3-yl H H CH2OCH3

A-2682 CFs lsoxazolin-3-yl H cyclopropyl H

A-2683 CFs lsoxazolin-3-yl H OCH3 H

A-2684 CFs lsoxazolin-3-yl H OCFs H A-2685 CFs lsoxazolin-3-yl H SCHs H

A-2686 CFs lsoxazolin-3-yl H SOCHs H

A-2687 CFs lsoxazolin-3-yl H SO2CH3 H

A-2688 CFs lsoxazolin-3-yl H CH2OCH3 H

A-2689 CFs 5-Me-lsoxazolin-3-yl CI H CN

A-2690 CFs 5-Me-lsoxazolin-3-yl CI H N0 ₂

A-2691 CFs 5-Me-lsoxazolin-3-yl CI H cyclopropyl

A-2692 CFs 5-Me-lsoxazolin-3-yl CI H OCHs

A-2693 CFs 5-Me-lsoxazolin-3-yl CI H OCFs

A-2694 CFs 5-Me-lsoxazolin-3-yl CI H SCHs

A-2695 CFs 5-Me-lsoxazolin-3-yl CI H SOCHs

A-2696 CFs 5-Me-lsoxazolin-3-yl CI H SO2CH3

A-2697 CFs 5-Me-lsoxazolin-3-yl CI H CH2OCH3

A-2698 CFs 5-Me-lsoxazolin-3-yl CI cyclopropyl H

A-2699 CFs 5-Me-lsoxazolin-3-yl CI OCHs H

A-2700 CFs 5-Me-lsoxazolin-3-yl CI OCFs H

A-2701 CFs 5-Me-lsoxazolin-3-yl CI SCHs H

A-2702 CFs 5-Me-lsoxazolin-3-yl CI SOCHs H

A-2703 CFs 5-Me-lsoxazolin-3-yl CI SO2CH3 H

A-2704 CFs 5-Me-lsoxazolin-3-yl CI CH2OCH3 H

A-2705 CFs 5-Me-lsoxazolin-3-yl F H CN

A-2706 CFs 5-Me-lsoxazolin-3-yl F H N0 ₂

A-2707 CFs 5-Me-lsoxazolin-3-yl F H cyclopropyl

A-2708 CFs 5-Me-lsoxazolin-3-yl F H OCHs

A-2709 CFs 5-Me-lsoxazolin-3-yl F H OCFs

A-2710 CFs 5-Me-lsoxazolin-3-yl F H SCHs

A-271 1 CFs 5-Me-lsoxazolin-3-yl F H SOCHs

A-2712 CFs 5-Me-lsoxazolin-3-yl F H SO2CH3

A-2713 CFs 5-Me-lsoxazolin-3-yl F H CH2OCH3

A-2714 CFs 5-Me-lsoxazolin-3-yl F cyclopropyl H

A-2715 CFs 5-Me-lsoxazolin-3-yl F OCHs H

A-2716 CFs 5-Me-lsoxazolin-3-yl F OCFs H

A-2717 CFs 5-Me-lsoxazolin-3-yl F SCHs H

A-2718 CFs 5-Me-lsoxazolin-3-yl F SOCHs H

A-2719 CFs 5-Me-lsoxazolin-3-yl F SO2CH3 H

A-2720 CFs 5-Me-lsoxazolin-3-yl F CH2OCH3 H

A-2721 CFs 5-Me-lsoxazolin-3-yl CFs H CN A-2722 CFs 5-Me-lsoxazolin-3-yl CFs H N0 ₂

A-2723 CFs 5-Me-lsoxazolin-3-yl CFs H cyclopropyl

A-2724 CFs 5-Me-lsoxazolin-3-yl CFs H OCHs

A-2725 CFs 5-Me-lsoxazolin-3-yl CFs H OCF3

A-2726 CFs 5-Me-lsoxazolin-3-yl CFs H SCHs

A-2727 CFs 5-Me-lsoxazolin-3-yl CFs H SOCH3

A-2728 CFs 5-Me-lsoxazolin-3-yl CFs H SO2CH3

A-2729 CFs 5-Me-lsoxazolin-3-yl CFs H CH2OCH3

A-2730 CFs 5-Me-lsoxazolin-3-yl CFs cyclopropyl H

A-2731 CFs 5-Me-lsoxazolin-3-yl CFs OCHs H

A-2732 CFs 5-Me-lsoxazolin-3-yl CFs OCF3 H

A-2733 CFs 5-Me-lsoxazolin-3-yl CFs SCHs H

A-2734 CFs 5-Me-lsoxazolin-3-yl CFs SOCH3 H

A-2735 CFs 5-Me-lsoxazolin-3-yl CFs SO2CH3 H

A-2736 CFs 5-Me-lsoxazolin-3-yl CFs CH2OCH3 H

A-2737 CFs 5-Me-lsoxazolin-3-yl SO2CH3 H CN

A-2738 CFs 5-Me-lsoxazolin-3-yl SO2CH3 H N0 ₂

A-2739 CFs 5-Me-lsoxazolin-3-yl SO2CH3 H cyclopropyl

A-2740 CFs 5-Me-lsoxazolin-3-yl SO2CH3 H OCHs

A-2741 CFs 5-Me-lsoxazolin-3-yl SO2CH3 H OCF3

A-2742 CFs 5-Me-lsoxazolin-3-yl SO2CH3 H SCHs

A-2743 CFs 5-Me-lsoxazolin-3-yl SO2CH3 H SOCH3

A-2744 CFs 5-Me-lsoxazolin-3-yl SO2CH3 H SO2CH3

A-2745 CFs 5-Me-lsoxazolin-3-yl SO2CH3 H CH2OCH3

A-2746 CFs 5-Me-lsoxazolin-3-yl SO2CH3 cyclopropyl H

A-2747 CFs 5-Me-lsoxazolin-3-yl SO2CH3 OCHs H

A-2748 CFs 5-Me-lsoxazolin-3-yl SO2CH3 OCF3 H

A-2749 CFs 5-Me-lsoxazolin-3-yl SO2CH3 SCHs H

A-2750 CFs 5-Me-lsoxazolin-3-yl SO2CH3 SOCH3 H

A-2751 CFs 5-Me-lsoxazolin-3-yl SO2CH3 SO2CH3 H

A-2752 CFs 5-Me-lsoxazolin-3-yl SO2CH3 CH2OCH3 H

A-2753 CFs 5-Me-lsoxazolin-3-yl CN H CN

A-2754 CFs 5-Me-lsoxazolin-3-yl CN H N0 ₂

A-2755 CFs 5-Me-lsoxazolin-3-yl CN H cyclopropyl

A-2756 CFs 5-Me-lsoxazolin-3-yl CN H OCHs

A-2757 CFs 5-Me-lsoxazolin-3-yl CN H OCF3

A-2758 CFs 5-Me-lsoxazolin-3-yl CN H SCHs A-2759 CFs 5-Me-lsoxazolin-3-yl CN H SOCHs

A-2760 CFs 5-Me-lsoxazolin-3-yl CN H SO2CH3

A-2761 CFs 5-Me-lsoxazolin-3-yl CN H CH2OCH3

A-2762 CFs 5-Me-lsoxazolin-3-yl CN cyclopropyl H

A-2763 CFs 5-Me-lsoxazolin-3-yl CN OCHs H

A-2764 CFs 5-Me-lsoxazolin-3-yl CN OCFs H

A-2765 CFs 5-Me-lsoxazolin-3-yl CN SCHs H

A-2766 CFs 5-Me-lsoxazolin-3-yl CN SOCHs H

A-2767 CFs 5-Me-lsoxazolin-3-yl CN SO2CH3 H

A-2768 CFs 5-Me-lsoxazolin-3-yl CN CH2OCH3 H

A-2769 CFs 5-Me-lsoxazolin-3-yl H H CN

A-2770 CFs 5-Me-lsoxazolin-3-yl H H N0 ₂

A-2771 CFs 5-Me-lsoxazolin-3-yl H H cyclopropyl

A-2772 CFs 5-Me-lsoxazolin-3-yl H H OCHs

A-2773 CFs 5-Me-lsoxazolin-3-yl H H OCFs

A-2774 CFs 5-Me-lsoxazolin-3-yl H H SCHs

A-2775 CFs 5-Me-lsoxazolin-3-yl H H SOCHs

A-2776 CFs 5-Me-lsoxazolin-3-yl H H SO2CH3

A-2777 CFs 5-Me-lsoxazolin-3-yl H H CH2OCH3

A-2778 CFs 5-Me-lsoxazolin-3-yl H cyclopropyl H

A-2779 CFs 5-Me-lsoxazolin-3-yl H OCHs H

A-2780 CFs 5-Me-lsoxazolin-3-yl H OCFs H

A-2781 CFs 5-Me-lsoxazolin-3-yl H SCHs H

A-2782 CFs 5-Me-lsoxazolin-3-yl H SOCHs H

A-2783 CFs 5-Me-lsoxazolin-3-yl H SO2CH3 H

A-2784 CFs 5-Me-lsoxazolin-3-yl H CH2OCH3 H

A-2785 CFs lsoxazol-3-yl CI H CN

A-2786 CFs lsoxazol-3-yl CI H N0 ₂

A-2787 CFs lsoxazol-3-yl CI H cyclopropyl

A-2788 CFs lsoxazol-3-yl CI H OCHs

A-2789 CFs lsoxazol-3-yl CI H OCFs

A-2790 CFs lsoxazol-3-yl CI H SCHs

A-2791 CFs lsoxazol-3-yl CI H SOCHs

A-2792 CFs lsoxazol-3-yl CI H SO2CH3

A-2793 CFs lsoxazol-3-yl CI H CH2OCH3

A-2794 CFs lsoxazol-3-yl CI cyclopropyl H

A-2795 CFs lsoxazol-3-yl CI OCHs H A-2796 CFs lsoxazol-3-yl CI OCFs H

A-2797 CFs lsoxazol-3-yl CI SCHs H

A-2798 CFs lsoxazol-3-yl CI SOCHs H

A-2799 CFs lsoxazol-3-yl CI SO2CH3 H

A-2800 CFs lsoxazol-3-yl CI CH2OCH3 H

A-2801 CFs lsoxazol-3-yl F H CN

A-2802 CFs lsoxazol-3-yl F H N0 ₂

A-2803 CFs lsoxazol-3-yl F H cyclopropyl

A-2804 CFs lsoxazol-3-yl F H OCHs

A-2805 CFs lsoxazol-3-yl F H OCFs

A-2806 CFs lsoxazol-3-yl F H SCHs

A-2807 CFs lsoxazol-3-yl F H SOCHs

A-2808 CFs lsoxazol-3-yl F H SO2CH3

A-2809 CFs lsoxazol-3-yl F H CH2OCH3

A-2810 CFs lsoxazol-3-yl F cyclopropyl H

A-281 1 CFs lsoxazol-3-yl F OCHs H

A-2812 CFs lsoxazol-3-yl F OCFs H

A-2813 CFs lsoxazol-3-yl F SCHs H

A-2814 CFs lsoxazol-3-yl F SOCHs H

A-2815 CFs lsoxazol-3-yl F SO2CH3 H

A-2816 CFs lsoxazol-3-yl F CH2OCH3 H

A-2817 CFs lsoxazol-3-yl CFs H CN

A-2818 CFs lsoxazol-3-yl CFs H N0 ₂

A-2819 CFs lsoxazol-3-yl CFs H cyclopropyl

A-2820 CFs lsoxazol-3-yl CFs H OCHs

A-2821 CFs lsoxazol-3-yl CFs H OCFs

A-2822 CFs lsoxazol-3-yl CFs H SCHs

A-2823 CFs lsoxazol-3-yl CFs H SOCHs

A-2824 CFs lsoxazol-3-yl CFs H SO2CH3

A-2825 CFs lsoxazol-3-yl CFs H CH2OCH3

A-2826 CFs lsoxazol-3-yl CFs cyclopropyl H

A-2827 CFs lsoxazol-3-yl CFs OCHs H

A-2828 CFs lsoxazol-3-yl CFs OCFs H

A-2829 CFs lsoxazol-3-yl CFs SCHs H

A-2830 CFs lsoxazol-3-yl CFs SOCHs H

A-2831 CFs lsoxazol-3-yl CFs SO2CH3 H

A-2832 CFs lsoxazol-3-yl CFs CH2OCH3 H A-2833 CFs lsoxazol-3-yl SO2CH3 H CN

A-2834 CFs lsoxazol-3-yl SO2CH3 H N0 ₂

A-2835 CFs lsoxazol-3-yl SO2CH3 H cyclopropyl

A-2836 CFs lsoxazol-3-yl SO2CH3 H OCHs

A-2837 CFs lsoxazol-3-yl SO2CH3 H OCF3

A-2838 CFs lsoxazol-3-yl SO2CH3 H SCHs

A-2839 CFs lsoxazol-3-yl SO2CH3 H SOCH3

A-2840 CFs lsoxazol-3-yl SO2CH3 H SO2CH3

A-2841 CFs lsoxazol-3-yl SO2CH3 H CH2OCH3

A-2842 CFs lsoxazol-3-yl SO2CH3 cyclopropyl H

A-2843 CFs lsoxazol-3-yl SO2CH3 OCHs H

A-2844 CFs lsoxazol-3-yl SO2CH3 OCF3 H

A-2845 CFs lsoxazol-3-yl SO2CH3 SCHs H

A-2846 CFs lsoxazol-3-yl SO2CH3 SOCH3 H

A-2847 CFs lsoxazol-3-yl SO2CH3 SO2CH3 H

A-2848 CFs lsoxazol-3-yl SO2CH3 CH2OCH3 H

A-2849 CFs lsoxazol-3-yl CN H CN

A-2850 CFs lsoxazol-3-yl CN H N0 ₂

A-2851 CFs lsoxazol-3-yl CN H cyclopropyl

A-2852 CFs lsoxazol-3-yl CN H OCHs

A-2853 CFs lsoxazol-3-yl CN H OCF3

A-2854 CFs lsoxazol-3-yl CN H SCHs

A-2855 CFs lsoxazol-3-yl CN H SOCH3

A-2856 CFs lsoxazol-3-yl CN H SO2CH3

A-2857 CFs lsoxazol-3-yl CN H CH2OCH3

A-2858 CFs lsoxazol-3-yl CN cyclopropyl H

A-2859 CFs lsoxazol-3-yl CN OCHs H

A-2860 CFs lsoxazol-3-yl CN OCF3 H

A-2861 CFs lsoxazol-3-yl CN SCHs H

A-2862 CFs lsoxazol-3-yl CN SOCH3 H

A-2863 CFs lsoxazol-3-yl CN SO2CH3 H

A-2864 CFs lsoxazol-3-yl CN CH2OCH3 H

A-2865 CFs lsoxazol-3-yl H H CN

A-2866 CFs lsoxazol-3-yl H H N0 ₂

A-2867 CFs lsoxazol-3-yl H H cyclopropyl

A-2868 CFs lsoxazol-3-yl H H OCHs

A-2869 CFs lsoxazol-3-yl H H OCF3 A-2870 CFs lsoxazol-3-yl H H SCHs

A-2871 CFs lsoxazol-3-yl H H SOCHs

A-2872 CFs lsoxazol-3-yl H H SO2CH3

A-2873 CFs lsoxazol-3-yl H H CH2OCH3

A-2874 CFs lsoxazol-3-yl H cyclopropyl H

A-2875 CFs lsoxazol-3-yl H OCHs H

A-2876 CFs lsoxazol-3-yl H OCFs H

A-2877 CFs lsoxazol-3-yl H SCHs H

A-2878 CFs lsoxazol-3-yl H SOCHs H

A-2879 CFs lsoxazol-3-yl H SO2CH3 H

A-2880 CFs lsoxazol-3-yl H CH2OCH3 H

A-2881 CFs 5-Me-lsoxazol-3-yl CI H CN

A-2882 CFs 5-Me-lsoxazol-3-yl CI H N0 ₂

A-2883 CFs 5-Me-lsoxazol-3-yl CI H cyclopropyl

A-2884 CFs 5-Me-lsoxazol-3-yl CI H OCHs

A-2885 CFs 5-Me-lsoxazol-3-yl CI H OCFs

A-2886 CFs 5-Me-lsoxazol-3-yl CI H SCHs

A-2887 CFs 5-Me-lsoxazol-3-yl CI H SOCHs

A-2888 CFs 5-Me-lsoxazol-3-yl CI H SO2CH3

A-2889 CFs 5-Me-lsoxazol-3-yl CI H CH2OCH3

A-2890 CFs 5-Me-lsoxazol-3-yl CI cyclopropyl H

A-2891 CFs 5-Me-lsoxazol-3-yl CI OCHs H

A-2892 CFs 5-Me-lsoxazol-3-yl CI OCFs H

A-2893 CFs 5-Me-lsoxazol-3-yl CI SCHs H

A-2894 CFs 5-Me-lsoxazol-3-yl CI SOCHs H

A-2895 CFs 5-Me-lsoxazol-3-yl CI SO2CH3 H

A-2896 CFs 5-Me-lsoxazol-3-yl CI CH2OCH3 H

A-2897 CFs 5-Me-lsoxazol-3-yl F H CN

A-2898 CFs 5-Me-lsoxazol-3-yl F H N0 ₂

A-2899 CFs 5-Me-lsoxazol-3-yl F H cyclopropyl

A-2900 CFs 5-Me-lsoxazol-3-yl F H OCHs

A-2901 CFs 5-Me-lsoxazol-3-yl F H OCFs

A-2902 CFs 5-Me-lsoxazol-3-yl F H SCHs

A-2903 CFs 5-Me-lsoxazol-3-yl F H SOCHs

A-2904 CFs 5-Me-lsoxazol-3-yl F H SO2CH3

A-2905 CFs 5-Me-lsoxazol-3-yl F H CH2OCH3

A-2906 CFs 5-Me-lsoxazol-3-yl F cyclopropyl H A-2907 CFs 5-Me-lsoxazol-3-yl F OCH3 H

A-2908 CFs 5-Me-lsoxazol-3-yl F OCFs H

A-2909 CFs 5-Me-lsoxazol-3-yl F SCHs H

A-2910 CFs 5-Me-lsoxazol-3-yl F SOCHs H

A-291 1 CFs 5-Me-lsoxazol-3-yl F SO2CH3 H

A-2912 CFs 5-Me-lsoxazol-3-yl F CH2OCH3 H

A-2913 CFs 5-Me-lsoxazol-3-yl CFs H CN

A-2914 CFs 5-Me-lsoxazol-3-yl CFs H N0 ₂

A-2915 CFs 5-Me-lsoxazol-3-yl CFs H cyclopropyl

A-2916 CFs 5-Me-lsoxazol-3-yl CFs H OCHs

A-2917 CFs 5-Me-lsoxazol-3-yl CFs H OCFs

A-2918 CFs 5-Me-lsoxazol-3-yl CFs H SCHs

A-2919 CFs 5-Me-lsoxazol-3-yl CFs H SOCHs

A-2920 CFs 5-Me-lsoxazol-3-yl CFs H SO2CH3

A-2921 CFs 5-Me-lsoxazol-3-yl CFs H CH2OCH3

A-2922 CFs 5-Me-lsoxazol-3-yl CFs cyclopropyl H

A-2923 CFs 5-Me-lsoxazol-3-yl CFs OCH3 H

A-2924 CFs 5-Me-lsoxazol-3-yl CFs OCFs H

A-2925 CFs 5-Me-lsoxazol-3-yl CFs SCHs H

A-2926 CFs 5-Me-lsoxazol-3-yl CFs SOCHs H

A-2927 CFs 5-Me-lsoxazol-3-yl CFs SO2CH3 H

A-2928 CFs 5-Me-lsoxazol-3-yl CFs CH2OCH3 H

A-2929 CFs 5-Me-lsoxazol-3-yl SO2CH3 H CN

A-2930 CFs 5-Me-lsoxazol-3-yl SO2CH3 H N0 ₂

A-2931 CFs 5-Me-lsoxazol-3-yl SO2CH3 H cyclopropyl

A-2932 CFs 5-Me-lsoxazol-3-yl SO2CH3 H OCHs

A-2933 CFs 5-Me-lsoxazol-3-yl SO2CH3 H OCFs

A-2934 CFs 5-Me-lsoxazol-3-yl SO2CH3 H SCHs

A-2935 CFs 5-Me-lsoxazol-3-yl SO2CH3 H SOCHs

A-2936 CFs 5-Me-lsoxazol-3-yl SO2CH3 H SO2CH3

A-2937 CFs 5-Me-lsoxazol-3-yl SO2CH3 H CH2OCH3

A-2938 CFs 5-Me-lsoxazol-3-yl SO2CH3 cyclopropyl H

A-2939 CFs 5-Me-lsoxazol-3-yl SO2CH3 OCH3 H

A-2940 CFs 5-Me-lsoxazol-3-yl SO2CH3 OCFs H

A-2941 CFs 5-Me-lsoxazol-3-yl SO2CH3 SCHs H

A-2942 CFs 5-Me-lsoxazol-3-yl SO2CH3 SOCHs H

A-2943 CFs 5-Me-lsoxazol-3-yl SO2CH3 SO2CH3 H A-2944 CFs 5-Me-lsoxazol-3-yl SO2CH3 CH2OCH3 H

A-2945 CFs 5-Me-lsoxazol-3-yl CN H CN

A-2946 CFs 5-Me-lsoxazol-3-yl CN H N0 ₂

A-2947 CFs 5-Me-lsoxazol-3-yl CN H cyclopropyl

A-2948 CFs 5-Me-lsoxazol-3-yl CN H OCHs

A-2949 CFs 5-Me-lsoxazol-3-yl CN H OCFs

A-2950 CFs 5-Me-lsoxazol-3-yl CN H SCHs

A-2951 CFs 5-Me-lsoxazol-3-yl CN H SOCH3

A-2952 CFs 5-Me-lsoxazol-3-yl CN H SO2CH3

A-2953 CFs 5-Me-lsoxazol-3-yl CN H CH2OCH3

A-2954 CFs 5-Me-lsoxazol-3-yl CN cyclopropyl H

A-2955 CFs 5-Me-lsoxazol-3-yl CN OCHs H

A-2956 CFs 5-Me-lsoxazol-3-yl CN OCFs H

A-2957 CFs 5-Me-lsoxazol-3-yl CN SCHs H

A-2958 CFs 5-Me-lsoxazol-3-yl CN SOCH3 H

A-2959 CFs 5-Me-lsoxazol-3-yl CN SO2CH3 H

A-2960 CFs 5-Me-lsoxazol-3-yl CN CH2OCH3 H

A-2961 CFs 5-Me-lsoxazol-3-yl H H CN

A-2962 CFs 5-Me-lsoxazol-3-yl H H N0 ₂

A-2963 CFs 5-Me-lsoxazol-3-yl H H cyclopropyl

A-2964 CFs 5-Me-lsoxazol-3-yl H H OCHs

A-2965 CFs 5-Me-lsoxazol-3-yl H H OCFs

A-2966 CFs 5-Me-lsoxazol-3-yl H H SCHs

A-2967 CFs 5-Me-lsoxazol-3-yl H H SOCH3

A-2968 CFs 5-Me-lsoxazol-3-yl H H SO2CH3

A-2969 CFs 5-Me-lsoxazol-3-yl H H CH2OCH3

A-2970 CFs 5-Me-lsoxazol-3-yl H cyclopropyl H

A-2971 CFs 5-Me-lsoxazol-3-yl H OCHs H

A-2972 CFs 5-Me-lsoxazol-3-yl H OCFs H

A-2973 CFs 5-Me-lsoxazol-3-yl H SCHs H

A-2974 CFs 5-Me-lsoxazol-3-yl H SOCH3 H

A-2975 CFs 5-Me-lsoxazol-3-yl H SO2CH3 H

A-2976 CFs 5-Me-lsoxazol-3-yl H CH2OCH3 H

A-2977 CFs 3-Me-lsoxazolin-5-yl CI H CN

A-2978 CFs 3-Me-lsoxazolin-5-yl CI H N0 ₂

A-2979 CFs 3-Me-lsoxazolin-5-yl CI H cyclopropyl

A-2980 CFs 3-Me-lsoxazolin-5-yl CI H OCHs A-2981 CFs 3-Me-lsoxazolin-5-yl CI H OCFs

A-2982 CFs 3-Me-lsoxazolin-5-yl CI H SCHs

A-2983 CFs 3-Me-lsoxazolin-5-yl CI H SOCHs

A-2984 CFs 3-Me-lsoxazolin-5-yl CI H SO2CH3

A-2985 CFs 3-Me-lsoxazolin-5-yl CI H CH2OCH3

A-2986 CFs 3-Me-lsoxazolin-5-yl CI cyclopropyl H

A-2987 CFs 3-Me-lsoxazolin-5-yl CI OCHs H

A-2988 CFs 3-Me-lsoxazolin-5-yl CI OCFs H

A-2989 CFs 3-Me-lsoxazolin-5-yl CI SCHs H

A-2990 CFs 3-Me-lsoxazolin-5-yl CI SOCHs H

A-2991 CFs 3-Me-lsoxazolin-5-yl CI SO2CH3 H

A-2992 CFs 3-Me-lsoxazolin-5-yl CI CH2OCH3 H

A-2993 CFs 3-Me-lsoxazolin-5-yl F H CN

A-2994 CFs 3-Me-lsoxazolin-5-yl F H N0 ₂

A-2995 CFs 3-Me-lsoxazolin-5-yl F H cyclopropyl

A-2996 CFs 3-Me-lsoxazolin-5-yl F H OCHs

A-2997 CFs 3-Me-lsoxazolin-5-yl F H OCFs

A-2998 CFs 3-Me-lsoxazolin-5-yl F H SCHs

A-2999 CFs 3-Me-lsoxazolin-5-yl F H SOCHs

A-3000 CFs 3-Me-lsoxazolin-5-yl F H SO2CH3

A-3001 CFs 3-Me-lsoxazolin-5-yl F H CH2OCH3

A-3002 CFs 3-Me-lsoxazolin-5-yl F cyclopropyl H

A-3003 CFs 3-Me-lsoxazolin-5-yl F OCHs H

A-3004 CFs 3-Me-lsoxazolin-5-yl F OCFs H

A-3005 CFs 3-Me-lsoxazolin-5-yl F SCHs H

A-3006 CFs 3-Me-lsoxazolin-5-yl F SOCHs H

A-3007 CFs 3-Me-lsoxazolin-5-yl F SO2CH3 H

A-3008 CFs 3-Me-lsoxazolin-5-yl F CH2OCH3 H

A-3009 CFs 3-Me-lsoxazolin-5-yl CFs H CN

A-3010 CFs 3-Me-lsoxazolin-5-yl CFs H N0 ₂

A-301 1 CFs 3-Me-lsoxazolin-5-yl CFs H cyclopropyl

A-3012 CFs 3-Me-lsoxazolin-5-yl CFs H OCHs

A-3013 CFs 3-Me-lsoxazolin-5-yl CFs H OCFs

A-3014 CFs 3-Me-lsoxazolin-5-yl CFs H SCHs

A-3015 CFs 3-Me-lsoxazolin-5-yl CFs H SOCHs

A-3016 CFs 3-Me-lsoxazolin-5-yl CFs H SO2CH3

A-3017 CFs 3-Me-lsoxazolin-5-yl CFs H CH2OCH3 A-3018 CFs 3-Me-lsoxazolin-5-yl CFs cyclopropyl H

A-3019 CFs 3-Me-lsoxazolin-5-yl CFs OCHs H

A-3020 CFs 3-Me-lsoxazolin-5-yl CFs OCF3 H

A-3021 CFs 3-Me-lsoxazolin-5-yl CFs SCHs H

A-3022 CFs 3-Me-lsoxazolin-5-yl CFs SOCH3 H

A-3023 CFs 3-Me-lsoxazolin-5-yl CFs SO2CH3 H

A-3024 CFs 3-Me-lsoxazolin-5-yl CFs CH2OCH3 H

A-3025 CFs 3-Me-lsoxazolin-5-yl SO2CH3 H CN

A-3026 CFs 3-Me-lsoxazolin-5-yl SO2CH3 H N0 ₂

A-3027 CFs 3-Me-lsoxazolin-5-yl SO2CH3 H cyclopropyl

A-3028 CFs 3-Me-lsoxazolin-5-yl SO2CH3 H OCHs

A-3029 CFs 3-Me-lsoxazolin-5-yl SO2CH3 H OCFs

A-3030 CFs 3-Me-lsoxazolin-5-yl SO2CH3 H SCHs

A-3031 CFs 3-Me-lsoxazolin-5-yl SO2CH3 H SOCHs

A-3032 CFs 3-Me-lsoxazolin-5-yl SO2CH3 H SO2CH3

A-3033 CFs 3-Me-lsoxazolin-5-yl SO2CH3 H CH2OCH3

A-3034 CFs 3-Me-lsoxazolin-5-yl SO2CH3 cyclopropyl H

A-3035 CFs 3-Me-lsoxazolin-5-yl SO2CH3 OCHs H

A-3036 CFs 3-Me-lsoxazolin-5-yl SO2CH3 OCF3 H

A-3037 CFs 3-Me-lsoxazolin-5-yl SO2CH3 SCHs H

A-3038 CFs 3-Me-lsoxazolin-5-yl SO2CH3 SOCH3 H

A-3039 CFs 3-Me-lsoxazolin-5-yl SO2CH3 SO2CH3 H

A-3040 CFs 3-Me-lsoxazolin-5-yl SO2CH3 CH2OCH3 H

A-3041 CFs 3-Me-lsoxazolin-5-yl CN H CN

A-3042 CFs 3-Me-lsoxazolin-5-yl CN H N0 ₂

A-3043 CFs 3-Me-lsoxazolin-5-yl CN H cyclopropyl

A-3044 CFs 3-Me-lsoxazolin-5-yl CN H OCHs

A-3045 CFs 3-Me-lsoxazolin-5-yl CN H OCFs

A-3046 CFs 3-Me-lsoxazolin-5-yl CN H SCHs

A-3047 CFs 3-Me-lsoxazolin-5-yl CN H SOCHs

A-3048 CFs 3-Me-lsoxazolin-5-yl CN H SO2CH3

A-3049 CFs 3-Me-lsoxazolin-5-yl CN H CH2OCH3

A-3050 CFs 3-Me-lsoxazolin-5-yl CN cyclopropyl H

A-3051 CFs 3-Me-lsoxazolin-5-yl CN OCHs H

A-3052 CFs 3-Me-lsoxazolin-5-yl CN OCF3 H

A-3053 CFs 3-Me-lsoxazolin-5-yl CN SCHs H

A-3054 CFs 3-Me-lsoxazolin-5-yl CN SOCH3 H A-3055 CFs 3-Me-lsoxazolin-5-yl CN SO2CH3 H

A-3056 CFs 3-Me-lsoxazolin-5-yl CN CH2OCH3 H

A-3057 CFs 3-Me-lsoxazolin-5-yl H H CN

A-3058 CFs 3-Me-lsoxazolin-5-yl H H N0 ₂

A-3059 CFs 3-Me-lsoxazolin-5-yl H H cyclopropyl

A-3060 CFs 3-Me-lsoxazolin-5-yl H H OCHs

A-3061 CFs 3-Me-lsoxazolin-5-yl H H OCFs

A-3062 CFs 3-Me-lsoxazolin-5-yl H H SCHs

A-3063 CFs 3-Me-lsoxazolin-5-yl H H SOCH3

A-3064 CFs 3-Me-lsoxazolin-5-yl H H SO2CH3

A-3065 CFs 3-Me-lsoxazolin-5-yl H H CH2OCH3

A-3066 CFs 3-Me-lsoxazolin-5-yl H cyclopropyl H

A-3067 CFs 3-Me-lsoxazolin-5-yl H OCHs H

A-3068 CFs 3-Me-lsoxazolin-5-yl H OCFs H

A-3069 CFs 3-Me-lsoxazolin-5-yl H SCHs H

A-3070 CFs 3-Me-lsoxazolin-5-yl H SOCH3 H

A-3071 CFs 3-Me-lsoxazolin-5-yl H SO2CH3 H

A-3072 CFs 3-Me-lsoxazolin-5-yl H CH2OCH3 H

A-3073 CFs 3-Me-lsoxazol-5-yl CI H CN

A-3074 CFs 3-Me-lsoxazol-5-yl CI H N0 ₂

A-3075 CFs 3-Me-lsoxazol-5-yl CI H cyclopropyl

A-3076 CFs 3-Me-lsoxazol-5-yl CI H OCHs

A-3077 CFs 3-Me-lsoxazol-5-yl CI H OCFs

A-3078 CFs 3-Me-lsoxazol-5-yl CI H SCHs

A-3079 CFs 3-Me-lsoxazol-5-yl CI H SOCH3

A-3080 CFs 3-Me-lsoxazol-5-yl CI H SO2CH3

A-3081 CFs 3-Me-lsoxazol-5-yl CI H CH2OCH3

A-3082 CFs 3-Me-lsoxazol-5-yl CI cyclopropyl H

A-3083 CFs 3-Me-lsoxazol-5-yl CI OCHs H

A-3084 CFs 3-Me-lsoxazol-5-yl CI OCFs H

A-3085 CFs 3-Me-lsoxazol-5-yl CI SCHs H

A-3086 CFs 3-Me-lsoxazol-5-yl CI SOCH3 H

A-3087 CFs 3-Me-lsoxazol-5-yl CI SO2CH3 H

A-3088 CFs 3-Me-lsoxazol-5-yl CI CH2OCH3 H

A-3089 CFs 3-Me-lsoxazol-5-yl F H CN

A-3090 CFs 3-Me-lsoxazol-5-yl F H N0 ₂

A-3091 CFs 3-Me-lsoxazol-5-yl F H cyclopropyl A-3092 CFs 3-Me-lsoxazol-5-yl F H OCHs

A-3093 CFs 3-Me-lsoxazol-5-yl F H OCF3

A-3094 CFs 3-Me-lsoxazol-5-yl F H SCHs

A-3095 CFs 3-Me-lsoxazol-5-yl F H SOCH3

A-3096 CFs 3-Me-lsoxazol-5-yl F H SO2CH3

A-3097 CFs 3-Me-lsoxazol-5-yl F H CH2OCH3

A-3098 CFs 3-Me-lsoxazol-5-yl F cyclopropyl H

A-3099 CFs 3-Me-lsoxazol-5-yl F OCHs H

A-3100 CFs 3-Me-lsoxazol-5-yl F OCF3 H

A-3101 CFs 3-Me-lsoxazol-5-yl F SCHs H

A-3102 CFs 3-Me-lsoxazol-5-yl F SOCH3 H

A-3103 CFs 3-Me-lsoxazol-5-yl F SO2CH3 H

A-3104 CFs 3-Me-lsoxazol-5-yl F CH2OCH3 H

A-3105 CFs 3-Me-lsoxazol-5-yl CFs H CN

A-3106 CFs 3-Me-lsoxazol-5-yl CFs H N0 ₂

A-3107 CFs 3-Me-lsoxazol-5-yl CFs H cyclopropyl

A-3108 CFs 3-Me-lsoxazol-5-yl CFs H OCHs

A-3109 CFs 3-Me-lsoxazol-5-yl CFs H OCF3

A-31 10 CFs 3-Me-lsoxazol-5-yl CFs H SCHs

A-31 1 1 CFs 3-Me-lsoxazol-5-yl CFs H SOCH3

A-31 12 CFs 3-Me-lsoxazol-5-yl CFs H SO2CH3

A-31 13 CFs 3-Me-lsoxazol-5-yl CFs H CH2OCH3

A-31 14 CFs 3-Me-lsoxazol-5-yl CFs cyclopropyl H

A-31 15 CFs 3-Me-lsoxazol-5-yl CFs OCHs H

A-31 16 CFs 3-Me-lsoxazol-5-yl CFs OCF3 H

A-31 17 CFs 3-Me-lsoxazol-5-yl CFs SCHs H

A-31 18 CFs 3-Me-lsoxazol-5-yl CFs SOCH3 H

A-31 19 CFs 3-Me-lsoxazol-5-yl CFs SO2CH3 H

A-3120 CFs 3-Me-lsoxazol-5-yl CFs CH2OCH3 H

A-3121 CFs 3-Me-lsoxazol-5-yl SO2CH3 H CN

A-3122 CFs 3-Me-lsoxazol-5-yl SO2CH3 H N0 ₂

A-3123 CFs 3-Me-lsoxazol-5-yl SO2CH3 H cyclopropyl

A-3124 CFs 3-Me-lsoxazol-5-yl SO2CH3 H OCHs

A-3125 CFs 3-Me-lsoxazol-5-yl SO2CH3 H OCF3

A-3126 CFs 3-Me-lsoxazol-5-yl SO2CH3 H SCHs

A-3127 CFs 3-Me-lsoxazol-5-yl SO2CH3 H SOCH3

A-3128 CFs 3-Me-lsoxazol-5-yl SO2CH3 H SO2CH3 A-3129 CFs 3-Me-lsoxazol-5-yl SO2CH3 H CH2OCH3

A-3130 CFs 3-Me-lsoxazol-5-yl SO2CH3 cyclopropyl H

A-3131 CFs 3-Me-lsoxazol-5-yl SO2CH3 OCHs H

A-3132 CFs 3-Me-lsoxazol-5-yl SO2CH3 OCF3 H

A-3133 CFs 3-Me-lsoxazol-5-yl SO2CH3 SCHs H

A-3134 CFs 3-Me-lsoxazol-5-yl SO2CH3 SOCH3 H

A-3135 CFs 3-Me-lsoxazol-5-yl SO2CH3 SO2CH3 H

A-3136 CFs 3-Me-lsoxazol-5-yl SO2CH3 CH2OCH3 H

A-3137 CFs 3-Me-lsoxazol-5-yl CN H CN

A-3138 CFs 3-Me-lsoxazol-5-yl CN H N0 ₂

A-3139 CFs 3-Me-lsoxazol-5-yl CN H cyclopropyl

A-3140 CFs 3-Me-lsoxazol-5-yl CN H OCHs

A-3141 CFs 3-Me-lsoxazol-5-yl CN H OCFs

A-3142 CFs 3-Me-lsoxazol-5-yl CN H SCHs

A-3143 CFs 3-Me-lsoxazol-5-yl CN H SOCHs

A-3144 CFs 3-Me-lsoxazol-5-yl CN H SO2CH3

A-3145 CFs 3-Me-lsoxazol-5-yl CN H CH2OCH3

A-3146 CFs 3-Me-lsoxazol-5-yl CN cyclopropyl H

A-3147 CFs 3-Me-lsoxazol-5-yl CN OCHs H

A-3148 CFs 3-Me-lsoxazol-5-yl CN OCF3 H

A-3149 CFs 3-Me-lsoxazol-5-yl CN SCHs H

A-3150 CFs 3-Me-lsoxazol-5-yl CN SOCH3 H

A-3151 CFs 3-Me-lsoxazol-5-yl CN SO2CH3 H

A-3152 CFs 3-Me-lsoxazol-5-yl CN CH2OCH3 H

A-3153 CFs 3-Me-lsoxazol-5-yl H H CN

A-3154 CFs 3-Me-lsoxazol-5-yl H H N0 ₂

A-3155 CFs 3-Me-lsoxazol-5-yl H H cyclopropyl

A-3156 CFs 3-Me-lsoxazol-5-yl H H OCHs

A-3157 CFs 3-Me-lsoxazol-5-yl H H OCFs

A-3158 CFs 3-Me-lsoxazol-5-yl H H SCHs

A-3159 CFs 3-Me-lsoxazol-5-yl H H SOCHs

A-3160 CFs 3-Me-lsoxazol-5-yl H H SO2CH3

A-3161 CFs 3-Me-lsoxazol-5-yl H H CH2OCH3

A-3162 CFs 3-Me-lsoxazol-5-yl H cyclopropyl H

A-3163 CFs 3-Me-lsoxazol-5-yl H OCHs H

A-3164 CFs 3-Me-lsoxazol-5-yl H OCF3 H

A-3165 CFs 3-Me-lsoxazol-5-yl H SCHs H A-3314 SO2CH3 SCH ₃ SO2CH3 H N0 ₂

A-3315 SO2CH3 SCH ₃ SO2CH3 H cyclopropyl

A-3316 SO2CH3 SCH ₃ SO2CH3 H OCH3

A-3317 SO2CH3 SCH ₃ SO2CH3 H OCF3

A-3318 SO2CH3 SCH ₃ SO2CH3 H SCH ₃

A-3319 SO2CH3 SCH ₃ SO2CH3 H SOCH3

A-3320 SO2CH3 SCH ₃ SO2CH3 H SO2CH3

A-3321 SO2CH3 SCH ₃ SO2CH3 H CH2OCH3

A-3322 SO2CH3 SCH ₃ SO2CH3 cyclopropyl H

A-3323 SO2CH3 SCH ₃ SO2CH3 OCH3 H

A-3324 SO2CH3 SCH ₃ SO2CH3 OCF3 H

A-3325 SO2CH3 SCH ₃ SO2CH3 SCH ₃ H

A-3326 SO2CH3 SCH ₃ SO2CH3 SOCH3 H

A-3327 SO2CH3 SCH ₃ SO2CH3 SO2CH3 H

A-3328 SO2CH3 SCH ₃ SO2CH3 CH2OCH3 H

A-3329 SO2CH3 SCH ₃ CN H CN

A-3330 SO2CH3 SCH ₃ CN H N0 ₂

A-3331 SO2CH3 SCH ₃ CN H cyclopropyl

A-3332 SO2CH3 SCH ₃ CN H OCH3

A-3333 SO2CH3 SCH ₃ CN H OCF3

A-3334 SO2CH3 SCH ₃ CN H SCH ₃

A-3335 SO2CH3 SCH ₃ CN H SOCH3

A-3336 SO2CH3 SCH ₃ CN H SO2CH3

A-3337 SO2CH3 SCH ₃ CN H CH2OCH3

A-3338 SO2CH3 SCH ₃ CN cyclopropyl H

A-3339 SO2CH3 SCH ₃ CN OCH3 H

A-3340 SO2CH3 SCH ₃ CN OCF3 H

A-3341 SO2CH3 SCH ₃ CN SCH ₃ H

A-3342 SO2CH3 SCH ₃ CN SOCH3 H

A-3343 SO2CH3 SCH ₃ CN SO2CH3 H

A-3344 SO2CH3 SCH ₃ CN CH2OCH3 H

A-3345 SO2CH3 SOCH3 H H CN

A-3346 SO2CH3 SOCH3 H H N0 ₂

A-3347 SO2CH3 SOCH3 H H cyclopropyl

A-3348 SO2CH3 SOCH3 H H OCH3

A-3349 SO2CH3 SOCH3 H H OCF3

A-3350 SO2CH3 SOCH3 H H SCH ₃ A-3351 SO2CH3 SOCH3 H H SOCH3

A-3352 SO2CH3 SOCH3 H H SO2CH3

A-3353 SO2CH3 SOCH3 H H CH2OCH3

A-3354 SO2CH3 SOCH3 H cyclopropyl H

A-3355 SO2CH3 SOCH3 H OCH3 H

A-3356 SO2CH3 SOCH3 H OCF3 H

A-3357 SO2CH3 SOCH3 H SCH ₃ H

A-3358 SO2CH3 SOCH3 H SOCH3 H

A-3359 SO2CH3 SOCH3 H SO2CH3 H

A-3360 SO2CH3 SOCH3 H CH2OCH3 H

A-3361 SO2CH3 SOCH3 CI H CN

A-3362 SO2CH3 SOCH3 CI H N0 ₂

A-3363 SO2CH3 SOCH3 CI H cyclopropyl

A-3364 SO2CH3 SOCH3 CI H OCH3

A-3365 SO2CH3 SOCH3 CI H OCF3

A-3366 SO2CH3 SOCH3 CI H SCH ₃

A-3367 SO2CH3 SOCH3 CI H SOCH3

A-3368 SO2CH3 SOCH3 CI H SO2CH3

A-3369 SO2CH3 SOCH3 CI H CH2OCH3

A-3370 SO2CH3 SOCH3 CI cyclopropyl H

A-3371 SO2CH3 SOCH3 CI OCH3 H

A-3372 SO2CH3 SOCH3 CI OCF3 H

A-3373 SO2CH3 SOCH3 CI SCH ₃ H

A-3374 SO2CH3 SOCH3 CI SOCH3 H

A-3375 SO2CH3 SOCH3 CI SO2CH3 H

A-3376 SO2CH3 SOCH3 CI CH2OCH3 H

A-3377 SO2CH3 SOCH3 F H CN

A-3378 SO2CH3 SOCH3 F H N0 ₂

A-3379 SO2CH3 SOCH3 F H cyclopropyl

A-3380 SO2CH3 SOCH3 F H OCH3

A-3381 SO2CH3 SOCH3 F H OCF3

A-3382 SO2CH3 SOCH3 F H SCH ₃

A-3383 SO2CH3 SOCH3 F H SOCH3

A-3384 SO2CH3 SOCH3 F H SO2CH3

A-3385 SO2CH3 SOCH3 F H CH2OCH3

A-3386 SO2CH3 SOCH3 F cyclopropyl H

A-3387 SO2CH3 SOCH3 F OCH3 H A-3388 SO2CH3 SOCH3 F OCF3 H

A-3389 SO2CH3 SOCH3 F SCH ₃ H

A-3390 SO2CH3 SOCH3 F SOCH3 H

A-3391 SO2CH3 SOCH3 F SO2CH3 H

A-3392 SO2CH3 SOCH3 F CH2OCH3 H

A-3393 SO2CH3 SOCH3 CF ₃ H CN

A-3394 SO2CH3 SOCH3 CF ₃ H N0 ₂

A-3395 SO2CH3 SOCH3 CF ₃ H cyclopropyl

A-3396 SO2CH3 SOCH3 CF ₃ H OCH3

A-3397 SO2CH3 SOCH3 CF ₃ H OCF3

A-3398 SO2CH3 SOCH3 CF ₃ H SCH ₃

A-3399 SO2CH3 SOCH3 CF ₃ H SOCH3

A-3400 SO2CH3 SOCH3 CF ₃ H SO2CH3

A-3401 SO2CH3 SOCH3 CF ₃ H CH2OCH3

A-3402 SO2CH3 SOCH3 CF ₃ cyclopropyl H

A-3403 SO2CH3 SOCH3 CF ₃ OCH3 H

A-3404 SO2CH3 SOCH3 CF ₃ OCF3 H

A-3405 SO2CH3 SOCH3 CF ₃ SCH ₃ H

A-3406 SO2CH3 SOCH3 CF ₃ SOCH3 H

A-3407 SO2CH3 SOCH3 CF ₃ SO2CH3 H

A-3408 SO2CH3 SOCH3 CF ₃ CH2OCH3 H

A-3409 SO2CH3 SOCH3 SO2CH3 H CN

A-3410 SO2CH3 SOCH3 SO2CH3 H N0 ₂

A-341 1 SO2CH3 SOCH3 SO2CH3 H cyclopropyl

A-3412 SO2CH3 SOCH3 SO2CH3 H OCH3

A-3413 SO2CH3 SOCH3 SO2CH3 H OCF3

A-3414 SO2CH3 SOCH3 SO2CH3 H SCH ₃

A-3415 SO2CH3 SOCH3 SO2CH3 H SOCH3

A-3416 SO2CH3 SOCH3 SO2CH3 H SO2CH3

A-3417 SO2CH3 SOCH3 SO2CH3 H CH2OCH3

A-3418 SO2CH3 SOCH3 SO2CH3 cyclopropyl H

A-3419 SO2CH3 SOCH3 SO2CH3 OCH3 H

A-3420 SO2CH3 SOCH3 SO2CH3 OCF3 H

A-3421 SO2CH3 SOCH3 SO2CH3 SCH ₃ H

A-3422 SO2CH3 SOCH3 SO2CH3 SOCH3 H

A-3423 SO2CH3 SOCH3 SO2CH3 SO2CH3 H

A-3424 SO2CH3 SOCH3 SO2CH3 CH2OCH3 H A-3425 SO2CH3 SOCH3 CN H CN

A-3426 SO2CH3 SOCH3 CN H N0 ₂

A-3427 SO2CH3 SOCH3 CN H cyclopropyl

A-3428 SO2CH3 SOCH3 CN H OCH3

A-3429 SO2CH3 SOCH3 CN H OCF3

A-3430 SO2CH3 SOCH3 CN H SCH ₃

A-3431 SO2CH3 SOCH3 CN H SOCH3

A-3432 SO2CH3 SOCH3 CN H SO2CH3

A-3433 SO2CH3 SOCH3 CN H CH2OCH3

A-3434 SO2CH3 SOCH3 CN cyclopropyl H

A-3435 SO2CH3 SOCH3 CN OCH3 H

A-3436 SO2CH3 SOCH3 CN OCF3 H

A-3437 SO2CH3 SOCH3 CN SCH ₃ H

A-3438 SO2CH3 SOCH3 CN SOCH3 H

A-3439 SO2CH3 SOCH3 CN SO2CH3 H

A-3440 SO2CH3 SOCH3 CN CH2OCH3 H

A-3441 SO2CH3 SOCH3 H H CN

A-3442 SO2CH3 SOCH3 H H N0 ₂

A-3443 SO2CH3 SOCH3 H H cyclopropyl

A-3444 SO2CH3 SOCH3 H H OCH3

A-3445 SO2CH3 SOCH3 H H OCF3

A-3446 SO2CH3 SOCH3 H H SCH ₃

A-3447 SO2CH3 SOCH3 H H SOCH3

A-3448 SO2CH3 SOCH3 H H SO2CH3

A-3449 SO2CH3 SOCH3 H H CH2OCH3

A-3450 SO2CH3 SOCH3 H cyclopropyl H

A-3451 SO2CH3 SOCH3 H OCH3 H

A-3452 SO2CH3 SOCH3 H OCF3 H

A-3453 SO2CH3 SOCH3 H SCH ₃ H

A-3454 SO2CH3 SOCH3 H SOCH3 H

A-3455 SO2CH3 SOCH3 H SO2CH3 H

A-3456 SO2CH3 SOCH3 H CH2OCH3 H

A-3457 SO2CH3 SO2CH3 CI H CN

A-3458 SO2CH3 SO2CH3 CI H N0 ₂

A-3459 SO2CH3 SO2CH3 CI H cyclopropyl

A-3460 SO2CH3 SO2CH3 CI H OCH3

A-3461 SO2CH3 SO2CH3 CI H OCF3 A-3462 SO2CH3 SO2CH3 CI H SCH ₃

A-3463 SO2CH3 SO2CH3 CI H SOCH3

A-3464 SO2CH3 SO2CH3 CI H SO2CH3

A-3465 SO2CH3 SO2CH3 CI H CH2OCH3

A-3466 SO2CH3 SO2CH3 CI cyclopropyl H

A-3467 SO2CH3 SO2CH3 CI OCH3 H

A-3468 SO2CH3 SO2CH3 CI OCF3 H

A-3469 SO2CH3 SO2CH3 CI SCH ₃ H

A-3470 SO2CH3 SO2CH3 CI SOCH3 H

A-3471 SO2CH3 SO2CH3 CI SO2CH3 H

A-3472 SO2CH3 SO2CH3 CI CH2OCH3 H

A-3473 SO2CH3 SO2CH3 F H CN

A-3474 SO2CH3 SO2CH3 F H N0 ₂

A-3475 SO2CH3 SO2CH3 F H cyclopropyl

A-3476 SO2CH3 SO2CH3 F H OCH3

A-3477 SO2CH3 SO2CH3 F H OCF3

A-3478 SO2CH3 SO2CH3 F H SCH ₃

A-3479 SO2CH3 SO2CH3 F H SOCH3

A-3480 SO2CH3 SO2CH3 F H SO2CH3

A-3481 SO2CH3 SO2CH3 F H CH2OCH3

A-3482 SO2CH3 SO2CH3 F cyclopropyl H

A-3483 SO2CH3 SO2CH3 F OCH3 H

A-3484 SO2CH3 SO2CH3 F OCF3 H

A-3485 SO2CH3 SO2CH3 F SCH ₃ H

A-3486 SO2CH3 SO2CH3 F SOCH3 H

A-3487 SO2CH3 SO2CH3 F SO2CH3 H

A-3488 SO2CH3 SO2CH3 F CH2OCH3 H

A-3489 SO2CH3 SO2CH3 CF ₃ H CN

A-3490 SO2CH3 SO2CH3 CF ₃ H N0 ₂

A-3491 SO2CH3 SO2CH3 CF ₃ H cyclopropyl

A-3492 SO2CH3 SO2CH3 CF ₃ H OCH3

A-3493 SO2CH3 SO2CH3 CF ₃ H OCF3

A-3494 SO2CH3 SO2CH3 CF ₃ H SCH ₃

A-3495 SO2CH3 SO2CH3 CF ₃ H SOCH3

A-3496 SO2CH3 SO2CH3 CF ₃ H SO2CH3

A-3497 SO2CH3 SO2CH3 CF ₃ H CH2OCH3

A-3498 SO2CH3 SO2CH3 CF ₃ cyclopropyl H A-3499 SO2CH3 SO2CH3 CF ₃ OCH3 H

A-3500 SO2CH3 SO2CH3 CF ₃ OCF3 H

A-3501 SO2CH3 SO2CH3 CF ₃ SCH ₃ H

A-3502 SO2CH3 SO2CH3 CF ₃ SOCH3 H

A-3503 SO2CH3 SO2CH3 CF ₃ SO2CH3 H

A-3504 SO2CH3 SO2CH3 CF ₃ CH2OCH3 H

A-3505 SO2CH3 SO2CH3 SO2CH3 H CN

A-3506 SO2CH3 SO2CH3 SO2CH3 H N0 ₂

A-3507 SO2CH3 SO2CH3 SO2CH3 H cyclopropyl

A-3508 SO2CH3 SO2CH3 SO2CH3 H OCH3

A-3509 SO2CH3 SO2CH3 SO2CH3 H OCF3

A-3510 SO2CH3 SO2CH3 SO2CH3 H SCH ₃

A-351 1 SO2CH3 SO2CH3 SO2CH3 H SOCH3

A-3512 SO2CH3 SO2CH3 SO2CH3 H SO2CH3

A-3513 SO2CH3 SO2CH3 SO2CH3 H CH2OCH3

A-3514 SO2CH3 SO2CH3 SO2CH3 cyclopropyl H

A-3515 SO2CH3 SO2CH3 SO2CH3 OCH3 H

A-3516 SO2CH3 SO2CH3 SO2CH3 OCF3 H

A-3517 SO2CH3 SO2CH3 SO2CH3 SCH ₃ H

A-3518 SO2CH3 SO2CH3 SO2CH3 SOCH3 H

A-3519 SO2CH3 SO2CH3 SO2CH3 SO2CH3 H

A-3520 SO2CH3 SO2CH3 SO2CH3 CH2OCH3 H

A-3521 SO2CH3 SO2CH3 CN H CN

A-3522 SO2CH3 SO2CH3 CN H N0 ₂

A-3523 SO2CH3 SO2CH3 CN H cyclopropyl

A-3524 SO2CH3 SO2CH3 CN H OCH3

A-3525 SO2CH3 SO2CH3 CN H OCF3

A-3526 SO2CH3 SO2CH3 CN H SCH ₃

A-3527 SO2CH3 SO2CH3 CN H SOCH3

A-3528 SO2CH3 SO2CH3 CN H SO2CH3

A-3529 SO2CH3 SO2CH3 CN H CH2OCH3

A-3530 SO2CH3 SO2CH3 CN cyclopropyl H

A-3531 SO2CH3 SO2CH3 CN OCH3 H

A-3532 SO2CH3 SO2CH3 CN OCF3 H

A-3533 SO2CH3 SO2CH3 CN SCH ₃ H

A-3534 SO2CH3 SO2CH3 CN SOCH3 H

A-3535 SO2CH3 SO2CH3 CN SO2CH3 H A-3536 SO2CH3 SO2CH3 CN CH2OCH3 H

A-3537 SO2CH3 SO2CH3 H H CN

A-3538 SO2CH3 SO2CH3 H H N0 ₂

A-3539 SO2CH3 SO2CH3 H H cyclopropyl

A-3540 SO2CH3 SO2CH3 H H OCH3

A-3541 SO2CH3 SO2CH3 H H OCF3

A-3542 SO2CH3 SO2CH3 H H SCH ₃

A-3543 SO2CH3 SO2CH3 H H SOCH3

A-3544 SO2CH3 SO2CH3 H H SO2CH3

A-3545 SO2CH3 SO2CH3 H H CH2OCH3

A-3546 SO2CH3 SO2CH3 H cyclopropyl H

A-3547 SO2CH3 SO2CH3 H OCH3 H

A-3548 SO2CH3 SO2CH3 H OCF3 H

A-3549 SO2CH3 SO2CH3 H SCH ₃ H

A-3550 SO2CH3 SO2CH3 H SOCH3 H

A-3551 SO2CH3 SO2CH3 H SO2CH3 H

A-3552 SO2CH3 SO2CH3 H CH2OCH3 H

A-3553 SO2CH3 CH2OCH2CF3 CI H CN

A-3554 SO2CH3 CH2OCH2CF3 CI H N0 ₂

A-3555 SO2CH3 CH2OCH2CF3 CI H cyclopropyl

A-3556 SO2CH3 CH2OCH2CF3 CI H OCH3

A-3557 SO2CH3 CH2OCH2CF3 CI H OCF3

A-3558 SO2CH3 CH2OCH2CF3 CI H SCH ₃

A-3559 SO2CH3 CH2OCH2CF3 CI H SOCH3

A-3560 SO2CH3 CH2OCH2CF3 CI H SO2CH3

A-3561 SO2CH3 CH2OCH2CF3 CI H CH2OCH3

A-3562 SO2CH3 CH2OCH2CF3 CI cyclopropyl H

A-3563 SO2CH3 CH2OCH2CF3 CI OCH3 H

A-3564 SO2CH3 CH2OCH2CF3 CI OCF3 H

A-3565 SO2CH3 CH2OCH2CF3 CI SCH ₃ H

A-3566 SO2CH3 CH2OCH2CF3 CI SOCH3 H

A-3567 SO2CH3 CH2OCH2CF3 CI SO2CH3 H

A-3568 SO2CH3 CH2OCH2CF3 CI CH2OCH3 H

A-3569 SO2CH3 CH2OCH2CF3 F H CN

A-3570 SO2CH3 CH2OCH2CF3 F H N0 ₂

A-3571 SO2CH3 CH2OCH2CF3 F H cyclopropyl

A-3572 SO2CH3 CH2OCH2CF3 F H OCH3 A-3573 SO2CH3 CH2OCH2CF3 F H OCF3

A-3574 SO2CH3 CH2OCH2CF3 F H SCH ₃

A-3575 SO2CH3 CH2OCH2CF3 F H SOCH3

A-3576 SO2CH3 CH2OCH2CF3 F H SO2CH3

A-3577 SO2CH3 CH2OCH2CF3 F H CH2OCH3

A-3578 SO2CH3 CH2OCH2CF3 F cyclopropyl H

A-3579 SO2CH3 CH2OCH2CF3 F OCH3 H

A-3580 SO2CH3 CH2OCH2CF3 F OCF3 H

A-3581 SO2CH3 CH2OCH2CF3 F SCH ₃ H

A-3582 SO2CH3 CH2OCH2CF3 F SOCH3 H

A-3583 SO2CH3 CH2OCH2CF3 F SO2CH3 H

A-3584 SO2CH3 CH2OCH2CF3 F CH2OCH3 H

A-3585 SO2CH3 CH2OCH2CF3 CF ₃ H CN

A-3586 SO2CH3 CH2OCH2CF3 CF ₃ H N0 ₂

A-3587 SO2CH3 CH2OCH2CF3 CF ₃ H cyclopropyl

A-3588 SO2CH3 CH2OCH2CF3 CF ₃ H OCH3

A-3589 SO2CH3 CH2OCH2CF3 CF ₃ H OCF3

A-3590 SO2CH3 CH2OCH2CF3 CF ₃ H SCH ₃

A-3591 SO2CH3 CH2OCH2CF3 CF ₃ H SOCH3

A-3592 SO2CH3 CH2OCH2CF3 CF ₃ H SO2CH3

A-3593 SO2CH3 CH2OCH2CF3 CF ₃ H CH2OCH3

A-3594 SO2CH3 CH2OCH2CF3 CF ₃ cyclopropyl H

A-3595 SO2CH3 CH2OCH2CF3 CF ₃ OCH3 H

A-3596 SO2CH3 CH2OCH2CF3 CF ₃ OCF3 H

A-3597 SO2CH3 CH2OCH2CF3 CF ₃ SCH ₃ H

A-3598 SO2CH3 CH2OCH2CF3 CF ₃ SOCH3 H

A-3599 SO2CH3 CH2OCH2CF3 CF ₃ SO2CH3 H

A-3600 SO2CH3 CH2OCH2CF3 CF ₃ CH2OCH3 H

A-3601 SO2CH3 CH2OCH2CF3 SO2CH3 H CN

A-3602 SO2CH3 CH2OCH2CF3 SO2CH3 H N0 ₂

A-3603 SO2CH3 CH2OCH2CF3 SO2CH3 H cyclopropyl

A-3604 SO2CH3 CH2OCH2CF3 SO2CH3 H OCH3

A-3605 SO2CH3 CH2OCH2CF3 SO2CH3 H OCF3

A-3606 SO2CH3 CH2OCH2CF3 SO2CH3 H SCH ₃

A-3607 SO2CH3 CH2OCH2CF3 SO2CH3 H SOCH3

A-3608 SO2CH3 CH2OCH2CF3 SO2CH3 H SO2CH3

A-3609 SO2CH3 CH2OCH2CF3 SO2CH3 H CH2OCH3 A-3610 SO2CH3 CH2OCH2CF3 SO2CH3 cyclopropyl H

A-361 1 SO2CH3 CH2OCH2CF3 SO2CH3 OCH3 H

A-3612 SO2CH3 CH2OCH2CF3 SO2CH3 OCF3 H

A-3613 SO2CH3 CH2OCH2CF3 SO2CH3 SCH ₃ H

A-3614 SO2CH3 CH2OCH2CF3 SO2CH3 SOCH3 H

A-3615 SO2CH3 CH2OCH2CF3 SO2CH3 SO2CH3 H

A-3616 SO2CH3 CH2OCH2CF3 SO2CH3 CH2OCH3 H

A-3617 SO2CH3 CH2OCH2CF3 CN H CN

A-3618 SO2CH3 CH2OCH2CF3 CN H N0 ₂

A-3619 SO2CH3 CH2OCH2CF3 CN H cyclopropyl

A-3620 SO2CH3 CH2OCH2CF3 CN H OCH3

A-3621 SO2CH3 CH2OCH2CF3 CN H OCF3

A-3622 SO2CH3 CH2OCH2CF3 CN H SCH ₃

A-3623 SO2CH3 CH2OCH2CF3 CN H SOCH3

A-3624 SO2CH3 CH2OCH2CF3 CN H SO2CH3

A-3625 SO2CH3 CH2OCH2CF3 CN H CH2OCH3

A-3626 SO2CH3 CH2OCH2CF3 CN cyclopropyl H

A-3627 SO2CH3 CH2OCH2CF3 CN OCH3 H

A-3628 SO2CH3 CH2OCH2CF3 CN OCF3 H

A-3629 SO2CH3 CH2OCH2CF3 CN SCH ₃ H

A-3630 SO2CH3 CH2OCH2CF3 CN SOCH3 H

A-3631 SO2CH3 CH2OCH2CF3 CN SO2CH3 H

A-3632 SO2CH3 CH2OCH2CF3 CN CH2OCH3 H

A-3633 SO2CH3 CH2OCH2CF3 H H CN

A-3634 SO2CH3 CH2OCH2CF3 H H N0 ₂

A-3635 SO2CH3 CH2OCH2CF3 H H cyclopropyl

A-3636 SO2CH3 CH2OCH2CF3 H H OCH3

A-3637 SO2CH3 CH2OCH2CF3 H H OCF3

A-3638 SO2CH3 CH2OCH2CF3 H H SCH ₃

A-3639 SO2CH3 CH2OCH2CF3 H H SOCH3

A-3640 SO2CH3 CH2OCH2CF3 H H SO2CH3

A-3641 SO2CH3 CH2OCH2CF3 H H CH2OCH3

A-3642 SO2CH3 CH2OCH2CF3 H cyclopropyl H

A-3643 SO2CH3 CH2OCH2CF3 H OCH3 H

A-3644 SO2CH3 CH2OCH2CF3 H OCF3 H

A-3645 SO2CH3 CH2OCH2CF3 H SCH ₃ H

A-3646 SO2CH3 CH2OCH2CF3 H SOCH3 H A-3647 SO2CH3 CH2OCH2CF3 H SO2CH3 H

A-3648 SO2CH3 CH2OCH2CF3 H CH2OCH3 H

A-3649 SO2CH3 lsoxazolin-3-yl CI H CN

A-3650 SO2CH3 lsoxazolin-3-yl CI H N0 ₂

A-3651 SO2CH3 lsoxazolin-3-yl CI H cyclopropyl

A-3652 SO2CH3 lsoxazolin-3-yl CI H OCH3

A-3653 SO2CH3 lsoxazolin-3-yl CI H OCF3

A-3654 SO2CH3 lsoxazolin-3-yl CI H SCH ₃

A-3655 SO2CH3 lsoxazolin-3-yl CI H SOCH3

A-3656 SO2CH3 lsoxazolin-3-yl CI H SO2CH3

A-3657 SO2CH3 lsoxazolin-3-yl CI H CH2OCH3

A-3658 SO2CH3 lsoxazolin-3-yl CI cyclopropyl H

A-3659 SO2CH3 lsoxazolin-3-yl CI OCH3 H

A-3660 SO2CH3 lsoxazolin-3-yl CI OCF3 H

A-3661 SO2CH3 lsoxazolin-3-yl CI SCH ₃ H

A-3662 SO2CH3 lsoxazolin-3-yl CI SOCH3 H

A-3663 SO2CH3 lsoxazolin-3-yl CI SO2CH3 H

A-3664 SO2CH3 lsoxazolin-3-yl CI CH2OCH3 H

A-3665 SO2CH3 lsoxazolin-3-yl F H CN

A-3666 SO2CH3 lsoxazolin-3-yl F H N0 ₂

A-3667 SO2CH3 lsoxazolin-3-yl F H cyclopropyl

A-3668 SO2CH3 lsoxazolin-3-yl F H OCH3

A-3669 SO2CH3 lsoxazolin-3-yl F H OCF3

A-3670 SO2CH3 lsoxazolin-3-yl F H SCH ₃

A-3671 SO2CH3 lsoxazolin-3-yl F H SOCH3

A-3672 SO2CH3 lsoxazolin-3-yl F H SO2CH3

A-3673 SO2CH3 lsoxazolin-3-yl F H CH2OCH3

A-3674 SO2CH3 lsoxazolin-3-yl F cyclopropyl H

A-3675 SO2CH3 lsoxazolin-3-yl F OCH3 H

A-3676 SO2CH3 lsoxazolin-3-yl F OCF3 H

A-3677 SO2CH3 lsoxazolin-3-yl F SCH ₃ H

A-3678 SO2CH3 lsoxazolin-3-yl F SOCH3 H

A-3679 SO2CH3 lsoxazolin-3-yl F SO2CH3 H

A-3680 SO2CH3 lsoxazolin-3-yl F CH2OCH3 H

A-3681 SO2CH3 lsoxazolin-3-yl CF ₃ H CN

A-3682 SO2CH3 lsoxazolin-3-yl CF ₃ H N0 ₂

A-3683 SO2CH3 lsoxazolin-3-yl CF ₃ H cyclopropyl A-3684 SO2CH3 lsoxazolin-3-yl CF ₃ H OCH3

A-3685 SO2CH3 lsoxazolin-3-yl CF ₃ H OCF3

A-3686 SO2CH3 lsoxazolin-3-yl CF ₃ H SCH ₃

A-3687 SO2CH3 lsoxazolin-3-yl CF ₃ H SOCH3

A-3688 SO2CH3 lsoxazolin-3-yl CF ₃ H SO2CH3

A-3689 SO2CH3 lsoxazolin-3-yl CF ₃ H CH2OCH3

A-3690 SO2CH3 lsoxazolin-3-yl CF ₃ cyclopropyl H

A-3691 SO2CH3 lsoxazolin-3-yl CF ₃ OCH3 H

A-3692 SO2CH3 lsoxazolin-3-yl CF ₃ OCF3 H

A-3693 SO2CH3 lsoxazolin-3-yl CF ₃ SCH ₃ H

A-3694 SO2CH3 lsoxazolin-3-yl CF ₃ SOCH3 H

A-3695 SO2CH3 lsoxazolin-3-yl CF ₃ SO2CH3 H

A-3696 SO2CH3 lsoxazolin-3-yl CF ₃ CH2OCH3 H

A-3697 SO2CH3 lsoxazolin-3-yl SO2CH3 H CN

A-3698 SO2CH3 lsoxazolin-3-yl SO2CH3 H N0 ₂

A-3699 SO2CH3 lsoxazolin-3-yl SO2CH3 H cyclopropyl

A-3700 SO2CH3 lsoxazolin-3-yl SO2CH3 H OCH3

A-3701 SO2CH3 lsoxazolin-3-yl SO2CH3 H OCF3

A-3702 SO2CH3 lsoxazolin-3-yl SO2CH3 H SCH ₃

A-3703 SO2CH3 lsoxazolin-3-yl SO2CH3 H SOCH3

A-3704 SO2CH3 lsoxazolin-3-yl SO2CH3 H SO2CH3

A-3705 SO2CH3 lsoxazolin-3-yl SO2CH3 H CH2OCH3

A-3706 SO2CH3 lsoxazolin-3-yl SO2CH3 cyclopropyl H

A-3707 SO2CH3 lsoxazolin-3-yl SO2CH3 OCH3 H

A-3708 SO2CH3 lsoxazolin-3-yl SO2CH3 OCF3 H

A-3709 SO2CH3 lsoxazolin-3-yl SO2CH3 SCH ₃ H

A-3710 SO2CH3 lsoxazolin-3-yl SO2CH3 SOCH3 H

A-371 1 SO2CH3 lsoxazolin-3-yl SO2CH3 SO2CH3 H

A-3712 SO2CH3 lsoxazolin-3-yl SO2CH3 CH2OCH3 H

A-3713 SO2CH3 lsoxazolin-3-yl CN H CN

A-3714 SO2CH3 lsoxazolin-3-yl CN H N0 ₂

A-3715 SO2CH3 lsoxazolin-3-yl CN H cyclopropyl

A-3716 SO2CH3 lsoxazolin-3-yl CN H OCH3

A-3717 SO2CH3 lsoxazolin-3-yl CN H OCF3

A-3718 SO2CH3 lsoxazolin-3-yl CN H SCH ₃

A-3719 SO2CH3 lsoxazolin-3-yl CN H SOCH3

A-3720 SO2CH3 lsoxazolin-3-yl CN H SO2CH3 A-3721 SO2CH3 lsoxazolin-3-yl CN H CH2OCH3

A-3722 SO2CH3 lsoxazolin-3-yl CN cyclopropyl H

A-3723 SO2CH3 lsoxazolin-3-yl CN OCH3 H

A-3724 SO2CH3 lsoxazolin-3-yl CN OCF3 H

A-3725 SO2CH3 lsoxazolin-3-yl CN SCH ₃ H

A-3726 SO2CH3 lsoxazolin-3-yl CN SOCH3 H

A-3727 SO2CH3 lsoxazolin-3-yl CN SO2CH3 H

A-3728 SO2CH3 lsoxazolin-3-yl CN CH2OCH3 H

A-3729 SO2CH3 lsoxazolin-3-yl H H CN

A-3730 SO2CH3 lsoxazolin-3-yl H H N0 ₂

A-3731 SO2CH3 lsoxazolin-3-yl H H cyclopropyl

A-3732 SO2CH3 lsoxazolin-3-yl H H OCH3

A-3733 SO2CH3 lsoxazolin-3-yl H H OCF3

A-3734 SO2CH3 lsoxazolin-3-yl H H SCH ₃

A-3735 SO2CH3 lsoxazolin-3-yl H H SOCH3

A-3736 SO2CH3 lsoxazolin-3-yl H H SO2CH3

A-3737 SO2CH3 lsoxazolin-3-yl H H CH2OCH3

A-3738 SO2CH3 lsoxazolin-3-yl H cyclopropyl H

A-3739 SO2CH3 lsoxazolin-3-yl H OCH3 H

A-3740 SO2CH3 lsoxazolin-3-yl H OCF3 H

A-3741 SO2CH3 lsoxazolin-3-yl H SCH ₃ H

A-3742 SO2CH3 lsoxazolin-3-yl H SOCH3 H

A-3743 SO2CH3 lsoxazolin-3-yl H SO2CH3 H

A-3744 SO2CH3 lsoxazolin-3-yl H CH2OCH3 H

A-3745 SO2CH3 5-Me-lsoxazolin-3-yl CI H CN

A-3746 SO2CH3 5-Me-lsoxazolin-3-yl CI H N0 ₂

A-3747 SO2CH3 5-Me-lsoxazolin-3-yl CI H cyclopropyl

A-3748 SO2CH3 5-Me-lsoxazolin-3-yl CI H OCH3

A-3749 SO2CH3 5-Me-lsoxazolin-3-yl CI H OCF3

A-3750 SO2CH3 5-Me-lsoxazolin-3-yl CI H SCH ₃

A-3751 SO2CH3 5-Me-lsoxazolin-3-yl CI H SOCH3

A-3752 SO2CH3 5-Me-lsoxazolin-3-yl CI H SO2CH3

A-3753 SO2CH3 5-Me-lsoxazolin-3-yl CI H CH2OCH3

A-3754 SO2CH3 5-Me-lsoxazolin-3-yl CI cyclopropyl H

A-3755 SO2CH3 5-Me-lsoxazolin-3-yl CI OCH3 H

A-3756 SO2CH3 5-Me-lsoxazolin-3-yl CI OCF3 H

A-3757 SO2CH3 5-Me-lsoxazolin-3-yl CI SCH ₃ H A-3758 SO2CH3 5-Me-lsoxazolin-3-yl CI SOCH3 H

A-3759 SO2CH3 5-Me-lsoxazolin-3-yl CI SO2CH3 H

A-3760 SO2CH3 5-Me-lsoxazolin-3-yl CI CH2OCH3 H

A-3761 SO2CH3 5-Me-lsoxazolin-3-yl F H CN

A-3762 SO2CH3 5-Me-lsoxazolin-3-yl F H N0 ₂

A-3763 SO2CH3 5-Me-lsoxazolin-3-yl F H cyclopropyl

A-3764 SO2CH3 5-Me-lsoxazolin-3-yl F H OCH3

A-3765 SO2CH3 5-Me-lsoxazolin-3-yl F H OCF3

A-3766 SO2CH3 5-Me-lsoxazolin-3-yl F H SCH ₃

A-3767 SO2CH3 5-Me-lsoxazolin-3-yl F H SOCH3

A-3768 SO2CH3 5-Me-lsoxazolin-3-yl F H SO2CH3

A-3769 SO2CH3 5-Me-lsoxazolin-3-yl F H CH2OCH3

A-3770 SO2CH3 5-Me-lsoxazolin-3-yl F cyclopropyl H

A-3771 SO2CH3 5-Me-lsoxazolin-3-yl F OCH3 H

A-3772 SO2CH3 5-Me-lsoxazolin-3-yl F OCF3 H

A-3773 SO2CH3 5-Me-lsoxazolin-3-yl F SCH ₃ H

A-3774 SO2CH3 5-Me-lsoxazolin-3-yl F SOCH3 H

A-3775 SO2CH3 5-Me-lsoxazolin-3-yl F SO2CH3 H

A-3776 SO2CH3 5-Me-lsoxazolin-3-yl F CH2OCH3 H

A-3777 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ H CN

A-3778 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ H N0 ₂

A-3779 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ H cyclopropyl

A-3780 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ H OCH3

A-3781 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ H OCF3

A-3782 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ H SCH ₃

A-3783 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ H SOCH3

A-3784 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ H SO2CH3

A-3785 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ H CH2OCH3

A-3786 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ cyclopropyl H

A-3787 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ OCH3 H

A-3788 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ OCF3 H

A-3789 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ SCH ₃ H

A-3790 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ SOCH3 H

A-3791 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ SO2CH3 H

A-3792 SO2CH3 5-Me-lsoxazolin-3-yl CF ₃ CH2OCH3 H

A-3793 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 H CN

A-3794 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 H N0 ₂ A-3795 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 H cyclopropyl

A-3796 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 H OCH3

A-3797 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 H OCF3

A-3798 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 H SCH ₃

A-3799 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 H SOCH3

A-3800 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 H SO2CH3

A-3801 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 H CH2OCH3

A-3802 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 cyclopropyl H

A-3803 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 OCH3 H

A-3804 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 OCF3 H

A-3805 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 SCH ₃ H

A-3806 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 SOCH3 H

A-3807 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 SO2CH3 H

A-3808 SO2CH3 5-Me-lsoxazolin-3-yl SO2CH3 CH2OCH3 H

A-3809 SO2CH3 5-Me-lsoxazolin-3-yl CN H CN

A-3810 SO2CH3 5-Me-lsoxazolin-3-yl CN H N0 ₂

A-381 1 SO2CH3 5-Me-lsoxazolin-3-yl CN H cyclopropyl

A-3812 SO2CH3 5-Me-lsoxazolin-3-yl CN H OCH3

A-3813 SO2CH3 5-Me-lsoxazolin-3-yl CN H OCF3

A-3814 SO2CH3 5-Me-lsoxazolin-3-yl CN H SCH ₃

A-3815 SO2CH3 5-Me-lsoxazolin-3-yl CN H SOCH3

A-3816 SO2CH3 5-Me-lsoxazolin-3-yl CN H SO2CH3

A-3817 SO2CH3 5-Me-lsoxazolin-3-yl CN H CH2OCH3

A-3818 SO2CH3 5-Me-lsoxazolin-3-yl CN cyclopropyl H

A-3819 SO2CH3 5-Me-lsoxazolin-3-yl CN OCH3 H

A-3820 SO2CH3 5-Me-lsoxazolin-3-yl CN OCF3 H

A-3821 SO2CH3 5-Me-lsoxazolin-3-yl CN SCH ₃ H

A-3822 SO2CH3 5-Me-lsoxazolin-3-yl CN SOCH3 H

A-3823 SO2CH3 5-Me-lsoxazolin-3-yl CN SO2CH3 H

A-3824 SO2CH3 5-Me-lsoxazolin-3-yl CN CH2OCH3 H

A-3825 SO2CH3 5-Me-lsoxazolin-3-yl H H CN

A-3826 SO2CH3 5-Me-lsoxazolin-3-yl H H N0 ₂

A-3827 SO2CH3 5-Me-lsoxazolin-3-yl H H cyclopropyl

A-3828 SO2CH3 5-Me-lsoxazolin-3-yl H H OCH3

A-3829 SO2CH3 5-Me-lsoxazolin-3-yl H H OCF3

A-3830 SO2CH3 5-Me-lsoxazolin-3-yl H H SCH ₃

A-3831 SO2CH3 5-Me-lsoxazolin-3-yl H H SOCH3 A-3832 SO2CH3 5-Me-lsoxazolin-3-yl H H SO2CH3

A-3833 SO2CH3 5-Me-lsoxazolin-3-yl H H CH2OCH3

A-3834 SO2CH3 5-Me-lsoxazolin-3-yl H cyclopropyl H

A-3835 SO2CH3 5-Me-lsoxazolin-3-yl H OCH3 H

A-3836 SO2CH3 5-Me-lsoxazolin-3-yl H OCF3 H

A-3837 SO2CH3 5-Me-lsoxazolin-3-yl H SCH ₃ H

A-3838 SO2CH3 5-Me-lsoxazolin-3-yl H SOCH3 H

A-3839 SO2CH3 5-Me-lsoxazolin-3-yl H SO2CH3 H

A-3840 SO2CH3 5-Me-lsoxazolin-3-yl H CH2OCH3 H

A-3841 SO2CH3 lsoxazol-3-yl CI H CN

A-3842 SO2CH3 lsoxazol-3-yl CI H N0 ₂

A-3843 SO2CH3 lsoxazol-3-yl CI H cyclopropyl

A-3844 SO2CH3 lsoxazol-3-yl CI H OCH3

A-3845 SO2CH3 lsoxazol-3-yl CI H OCF3

A-3846 SO2CH3 lsoxazol-3-yl CI H SCH ₃

A-3847 SO2CH3 lsoxazol-3-yl CI H SOCH3

A-3848 SO2CH3 lsoxazol-3-yl CI H SO2CH3

A-3849 SO2CH3 lsoxazol-3-yl CI H CH2OCH3

A-3850 SO2CH3 lsoxazol-3-yl CI cyclopropyl H

A-3851 SO2CH3 lsoxazol-3-yl CI OCH3 H

A-3852 SO2CH3 lsoxazol-3-yl CI OCF3 H

A-3853 SO2CH3 lsoxazol-3-yl CI SCH ₃ H

A-3854 SO2CH3 lsoxazol-3-yl CI SOCH3 H

A-3855 SO2CH3 lsoxazol-3-yl CI SO2CH3 H

A-3856 SO2CH3 lsoxazol-3-yl CI CH2OCH3 H

A-3857 SO2CH3 lsoxazol-3-yl F H CN

A-3858 SO2CH3 lsoxazol-3-yl F H N0 ₂

A-3859 SO2CH3 lsoxazol-3-yl F H cyclopropyl

A-3860 SO2CH3 lsoxazol-3-yl F H OCH3

A-3861 SO2CH3 lsoxazol-3-yl F H OCF3

A-3862 SO2CH3 lsoxazol-3-yl F H SCH ₃

A-3863 SO2CH3 lsoxazol-3-yl F H SOCH3

A-3864 SO2CH3 lsoxazol-3-yl F H SO2CH3

A-3865 SO2CH3 lsoxazol-3-yl F H CH2OCH3

A-3866 SO2CH3 lsoxazol-3-yl F cyclopropyl H

A-3867 SO2CH3 lsoxazol-3-yl F OCH3 H

A-3868 SO2CH3 lsoxazol-3-yl F OCF3 H A-3869 SO2CH3 lsoxazol-3-yl F SCH ₃ H

A-3870 SO2CH3 lsoxazol-3-yl F SOCH3 H

A-3871 SO2CH3 lsoxazol-3-yl F SO2CH3 H

A-3872 SO2CH3 lsoxazol-3-yl F CH2OCH3 H

A-3873 SO2CH3 lsoxazol-3-yl CF ₃ H CN

A-3874 SO2CH3 lsoxazol-3-yl CF ₃ H N0 ₂

A-3875 SO2CH3 lsoxazol-3-yl CF ₃ H cyclopropyl

A-3876 SO2CH3 lsoxazol-3-yl CF ₃ H OCH3

A-3877 SO2CH3 lsoxazol-3-yl CF ₃ H OCF3

A-3878 SO2CH3 lsoxazol-3-yl CF ₃ H SCH ₃

A-3879 SO2CH3 lsoxazol-3-yl CF ₃ H SOCH3

A-3880 SO2CH3 lsoxazol-3-yl CF ₃ H SO2CH3

A-3881 SO2CH3 lsoxazol-3-yl CF ₃ H CH2OCH3

A-3882 SO2CH3 lsoxazol-3-yl CF ₃ cyclopropyl H

A-3883 SO2CH3 lsoxazol-3-yl CF ₃ OCH3 H

A-3884 SO2CH3 lsoxazol-3-yl CF ₃ OCF3 H

A-3885 SO2CH3 lsoxazol-3-yl CF ₃ SCH ₃ H

A-3886 SO2CH3 lsoxazol-3-yl CF ₃ SOCH3 H

A-3887 SO2CH3 lsoxazol-3-yl CF ₃ SO2CH3 H

A-3888 SO2CH3 lsoxazol-3-yl CF ₃ CH2OCH3 H

A-3889 SO2CH3 lsoxazol-3-yl SO2CH3 H CN

A-3890 SO2CH3 lsoxazol-3-yl SO2CH3 H N0 ₂

A-3891 SO2CH3 lsoxazol-3-yl SO2CH3 H cyclopropyl

A-3892 SO2CH3 lsoxazol-3-yl SO2CH3 H OCH3

A-3893 SO2CH3 lsoxazol-3-yl SO2CH3 H OCF3

A-3894 SO2CH3 lsoxazol-3-yl SO2CH3 H SCH ₃

A-3895 SO2CH3 lsoxazol-3-yl SO2CH3 H SOCH3

A-3896 SO2CH3 lsoxazol-3-yl SO2CH3 H SO2CH3

A-3897 SO2CH3 lsoxazol-3-yl SO2CH3 H CH2OCH3

A-3898 SO2CH3 lsoxazol-3-yl SO2CH3 cyclopropyl H

A-3899 SO2CH3 lsoxazol-3-yl SO2CH3 OCH3 H

A-3900 SO2CH3 lsoxazol-3-yl SO2CH3 OCF3 H

A-3901 SO2CH3 lsoxazol-3-yl SO2CH3 SCH ₃ H

A-3902 SO2CH3 lsoxazol-3-yl SO2CH3 SOCH3 H

A-3903 SO2CH3 lsoxazol-3-yl SO2CH3 SO2CH3 H

A-3904 SO2CH3 lsoxazol-3-yl SO2CH3 CH2OCH3 H

A-3905 SO2CH3 lsoxazol-3-yl CN H CN A-3906 SO2CH3 lsoxazol-3-yl CN H N0 ₂

A-3907 SO2CH3 lsoxazol-3-yl CN H cyclopropyl

A-3908 SO2CH3 lsoxazol-3-yl CN H OCH3

A-3909 SO2CH3 lsoxazol-3-yl CN H OCF3

A-3910 SO2CH3 lsoxazol-3-yl CN H SCH ₃

A-391 1 SO2CH3 lsoxazol-3-yl CN H SOCH3

A-3912 SO2CH3 lsoxazol-3-yl CN H SO2CH3

A-3913 SO2CH3 lsoxazol-3-yl CN H CH2OCH3

A-3914 SO2CH3 lsoxazol-3-yl CN cyclopropyl H

A-3915 SO2CH3 lsoxazol-3-yl CN OCH3 H

A-3916 SO2CH3 lsoxazol-3-yl CN OCF3 H

A-3917 SO2CH3 lsoxazol-3-yl CN SCH ₃ H

A-3918 SO2CH3 lsoxazol-3-yl CN SOCH3 H

A-3919 SO2CH3 lsoxazol-3-yl CN SO2CH3 H

A-3920 SO2CH3 lsoxazol-3-yl CN CH2OCH3 H

A-3921 SO2CH3 lsoxazol-3-yl H H CN

A-3922 SO2CH3 lsoxazol-3-yl H H N0 ₂

A-3923 SO2CH3 lsoxazol-3-yl H H cyclopropyl

A-3924 SO2CH3 lsoxazol-3-yl H H OCH3

A-3925 SO2CH3 lsoxazol-3-yl H H OCF3

A-3926 SO2CH3 lsoxazol-3-yl H H SCH ₃

A-3927 SO2CH3 lsoxazol-3-yl H H SOCH3

A-3928 SO2CH3 lsoxazol-3-yl H H SO2CH3

A-3929 SO2CH3 lsoxazol-3-yl H H CH2OCH3

A-3930 SO2CH3 lsoxazol-3-yl H cyclopropyl H

A-3931 SO2CH3 lsoxazol-3-yl H OCH3 H

A-3932 SO2CH3 lsoxazol-3-yl H OCF3 H

A-3933 SO2CH3 lsoxazol-3-yl H SCH ₃ H

A-3934 SO2CH3 lsoxazol-3-yl H SOCH3 H

A-3935 SO2CH3 lsoxazol-3-yl H SO2CH3 H

A-3936 SO2CH3 lsoxazol-3-yl H CH2OCH3 H

A-3937 SO2CH3 5-Me-lsoxazol-3-yl CI H CN

A-3938 SO2CH3 5-Me-lsoxazol-3-yl CI H N0 ₂

A-3939 SO2CH3 5-Me-lsoxazol-3-yl CI H cyclopropyl

A-3940 SO2CH3 5-Me-lsoxazol-3-yl CI H OCH3

A-3941 SO2CH3 5-Me-lsoxazol-3-yl CI H OCF3

A-3942 SO2CH3 5-Me-lsoxazol-3-yl CI H SCH ₃ A-3943 SO2CH3 5-Me-lsoxazol-3-yl CI H SOCH3

A-3944 SO2CH3 5-Me-lsoxazol-3-yl CI H SO2CH3

A-3945 SO2CH3 5-Me-lsoxazol-3-yl CI H CH2OCH3

A-3946 SO2CH3 5-Me-lsoxazol-3-yl CI cyclopropyl H

A-3947 SO2CH3 5-Me-lsoxazol-3-yl CI OCH3 H

A-3948 SO2CH3 5-Me-lsoxazol-3-yl CI OCF3 H

A-3949 SO2CH3 5-Me-lsoxazol-3-yl CI SCH ₃ H

A-3950 SO2CH3 5-Me-lsoxazol-3-yl CI SOCH3 H

A-3951 SO2CH3 5-Me-lsoxazol-3-yl CI SO2CH3 H

A-3952 SO2CH3 5-Me-lsoxazol-3-yl CI CH2OCH3 H

A-3953 SO2CH3 5-Me-lsoxazol-3-yl F H CN

A-3954 SO2CH3 5-Me-lsoxazol-3-yl F H N0 ₂

A-3955 SO2CH3 5-Me-lsoxazol-3-yl F H cyclopropyl

A-3956 SO2CH3 5-Me-lsoxazol-3-yl F H OCH3

A-3957 SO2CH3 5-Me-lsoxazol-3-yl F H OCF3

A-3958 SO2CH3 5-Me-lsoxazol-3-yl F H SCH ₃

A-3959 SO2CH3 5-Me-lsoxazol-3-yl F H SOCH3

A-3960 SO2CH3 5-Me-lsoxazol-3-yl F H SO2CH3

A-3961 SO2CH3 5-Me-lsoxazol-3-yl F H CH2OCH3

A-3962 SO2CH3 5-Me-lsoxazol-3-yl F cyclopropyl H

A-3963 SO2CH3 5-Me-lsoxazol-3-yl F OCH3 H

A-3964 SO2CH3 5-Me-lsoxazol-3-yl F OCF3 H

A-3965 SO2CH3 5-Me-lsoxazol-3-yl F SCH ₃ H

A-3966 SO2CH3 5-Me-lsoxazol-3-yl F SOCH3 H

A-3967 SO2CH3 5-Me-lsoxazol-3-yl F SO2CH3 H

A-3968 SO2CH3 5-Me-lsoxazol-3-yl F CH2OCH3 H

A-3969 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ H CN

A-3970 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ H N0 ₂

A-3971 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ H cyclopropyl

A-3972 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ H OCH3

A-3973 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ H OCF3

A-3974 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ H SCH ₃

A-3975 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ H SOCH3

A-3976 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ H SO2CH3

A-3977 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ H CH2OCH3

A-3978 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ cyclopropyl H

A-3979 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ OCH3 H A-3980 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ OCF3 H

A-3981 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ SCH ₃ H

A-3982 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ SOCH3 H

A-3983 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ SO2CH3 H

A-3984 SO2CH3 5-Me-lsoxazol-3-yl CF ₃ CH2OCH3 H

A-3985 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 H CN

A-3986 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 H N0 ₂

A-3987 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 H cyclopropyl

A-3988 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 H OCH3

A-3989 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 H OCF3

A-3990 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 H SCH ₃

A-3991 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 H SOCH3

A-3992 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 H SO2CH3

A-3993 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 H CH2OCH3

A-3994 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 cyclopropyl H

A-3995 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 OCH3 H

A-3996 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 OCF3 H

A-3997 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 SCH ₃ H

A-3998 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 SOCH3 H

A-3999 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 SO2CH3 H

A-4000 SO2CH3 5-Me-lsoxazol-3-yl SO2CH3 CH2OCH3 H

A-4001 SO2CH3 5-Me-lsoxazol-3-yl CN H CN

A-4002 SO2CH3 5-Me-lsoxazol-3-yl CN H N0 ₂

A-4003 SO2CH3 5-Me-lsoxazol-3-yl CN H cyclopropyl

A-4004 SO2CH3 5-Me-lsoxazol-3-yl CN H OCH3

A-4005 SO2CH3 5-Me-lsoxazol-3-yl CN H OCF3

A-4006 SO2CH3 5-Me-lsoxazol-3-yl CN H SCH ₃

A-4007 SO2CH3 5-Me-lsoxazol-3-yl CN H SOCH3

A-4008 SO2CH3 5-Me-lsoxazol-3-yl CN H SO2CH3

A-4009 SO2CH3 5-Me-lsoxazol-3-yl CN H CH2OCH3

A-4010 SO2CH3 5-Me-lsoxazol-3-yl CN cyclopropyl H

A-401 1 SO2CH3 5-Me-lsoxazol-3-yl CN OCH3 H

A-4012 SO2CH3 5-Me-lsoxazol-3-yl CN OCF3 H

A-4013 SO2CH3 5-Me-lsoxazol-3-yl CN SCH ₃ H

A-4014 SO2CH3 5-Me-lsoxazol-3-yl CN SOCH3 H

A-4015 SO2CH3 5-Me-lsoxazol-3-yl CN SO2CH3 H

A-4016 SO2CH3 5-Me-lsoxazol-3-yl CN CH2OCH3 H A-4017 SO2CH3 5-Me-lsoxazol-3-yl H H CN

A-4018 SO2CH3 5-Me-lsoxazol-3-yl H H N0 ₂

A-4019 SO2CH3 5-Me-lsoxazol-3-yl H H cyclopropyl

A-4020 SO2CH3 5-Me-lsoxazol-3-yl H H OCH3

A-4021 SO2CH3 5-Me-lsoxazol-3-yl H H OCF3

A-4022 SO2CH3 5-Me-lsoxazol-3-yl H H SCH ₃

A-4023 SO2CH3 5-Me-lsoxazol-3-yl H H SOCH3

A-4024 SO2CH3 5-Me-lsoxazol-3-yl H H SO2CH3

A-4025 SO2CH3 5-Me-lsoxazol-3-yl H H CH2OCH3

A-4026 SO2CH3 5-Me-lsoxazol-3-yl H cyclopropyl H

A-4027 SO2CH3 5-Me-lsoxazol-3-yl H OCH3 H

A-4028 SO2CH3 5-Me-lsoxazol-3-yl H OCF3 H

A-4029 SO2CH3 5-Me-lsoxazol-3-yl H SCH ₃ H

A-4030 SO2CH3 5-Me-lsoxazol-3-yl H SOCH3 H

A-4031 SO2CH3 5-Me-lsoxazol-3-yl H SO2CH3 H

A-4032 SO2CH3 5-Me-lsoxazol-3-yl H CH2OCH3 H

A-4033 SO2CH3 3-Me-lsoxazolin-5-yl CI H CN

A-4034 SO2CH3 3-Me-lsoxazolin-5-yl CI H N0 ₂

A-4035 SO2CH3 3-Me-lsoxazolin-5-yl CI H cyclopropyl

A-4036 SO2CH3 3-Me-lsoxazolin-5-yl CI H OCH3

A-4037 SO2CH3 3-Me-lsoxazolin-5-yl CI H OCF3

A-4038 SO2CH3 3-Me-lsoxazolin-5-yl CI H SCH ₃

A-4039 SO2CH3 3-Me-lsoxazolin-5-yl CI H SOCH3

A-4040 SO2CH3 3-Me-lsoxazolin-5-yl CI H SO2CH3

A-4041 SO2CH3 3-Me-lsoxazolin-5-yl CI H CH2OCH3

A-4042 SO2CH3 3-Me-lsoxazolin-5-yl CI cyclopropyl H

A-4043 SO2CH3 3-Me-lsoxazolin-5-yl CI OCH3 H

A-4044 SO2CH3 3-Me-lsoxazolin-5-yl CI OCF3 H

A-4045 SO2CH3 3-Me-lsoxazolin-5-yl CI SCH ₃ H

A-4046 SO2CH3 3-Me-lsoxazolin-5-yl CI SOCH3 H

A-4047 SO2CH3 3-Me-lsoxazolin-5-yl CI SO2CH3 H

A-4048 SO2CH3 3-Me-lsoxazolin-5-yl CI CH2OCH3 H

A-4049 SO2CH3 3-Me-lsoxazolin-5-yl F H CN

A-4050 SO2CH3 3-Me-lsoxazolin-5-yl F H N0 ₂

A-4051 SO2CH3 3-Me-lsoxazolin-5-yl F H cyclopropyl

A-4052 SO2CH3 3-Me-lsoxazolin-5-yl F H OCH3

A-4053 SO2CH3 3-Me-lsoxazolin-5-yl F H OCF3 A-4054 SO2CH3 3-Me-lsoxazolin-5-yl F H SCH ₃

A-4055 SO2CH3 3-Me-lsoxazolin-5-yl F H SOCH3

A-4056 SO2CH3 3-Me-lsoxazolin-5-yl F H SO2CH3

A-4057 SO2CH3 3-Me-lsoxazolin-5-yl F H CH2OCH3

A-4058 SO2CH3 3-Me-lsoxazolin-5-yl F cyclopropyl H

A-4059 SO2CH3 3-Me-lsoxazolin-5-yl F OCH3 H

A-4060 SO2CH3 3-Me-lsoxazolin-5-yl F OCF3 H

A-4061 SO2CH3 3-Me-lsoxazolin-5-yl F SCH ₃ H

A-4062 SO2CH3 3-Me-lsoxazolin-5-yl F SOCH3 H

A-4063 SO2CH3 3-Me-lsoxazolin-5-yl F SO2CH3 H

A-4064 SO2CH3 3-Me-lsoxazolin-5-yl F CH2OCH3 H

A-4065 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ H CN

A-4066 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ H N0 ₂

A-4067 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ H cyclopropyl

A-4068 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ H OCH3

A-4069 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ H OCF3

A-4070 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ H SCH ₃

A-4071 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ H SOCH3

A-4072 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ H SO2CH3

A-4073 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ H CH2OCH3

A-4074 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ cyclopropyl H

A-4075 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ OCH3 H

A-4076 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ OCF3 H

A-4077 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ SCH ₃ H

A-4078 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ SOCH3 H

A-4079 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ SO2CH3 H

A-4080 SO2CH3 3-Me-lsoxazolin-5-yl CF ₃ CH2OCH3 H

A-4081 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 H CN

A-4082 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 H N0 ₂

A-4083 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 H cyclopropyl

A-4084 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 H OCH3

A-4085 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 H OCF3

A-4086 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 H SCH ₃

A-4087 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 H SOCH3

A-4088 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 H SO2CH3

A-4089 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 H CH2OCH3

A-4090 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 cyclopropyl H A-4091 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 OCH3 H

A-4092 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 OCF3 H

A-4093 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 SCH ₃ H

A-4094 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 SOCH3 H

A-4095 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 SO2CH3 H

A-4096 SO2CH3 3-Me-lsoxazolin-5-yl SO2CH3 CH2OCH3 H

A-4097 SO2CH3 3-Me-lsoxazolin-5-yl CN H CN

A-4098 SO2CH3 3-Me-lsoxazolin-5-yl CN H N0 ₂

A-4099 SO2CH3 3-Me-lsoxazolin-5-yl CN H cyclopropyl

A-4100 SO2CH3 3-Me-lsoxazolin-5-yl CN H OCH3

A-4101 SO2CH3 3-Me-lsoxazolin-5-yl CN H OCF3

A-4102 SO2CH3 3-Me-lsoxazolin-5-yl CN H SCH ₃

A-4103 SO2CH3 3-Me-lsoxazolin-5-yl CN H SOCH3

A-4104 SO2CH3 3-Me-lsoxazolin-5-yl CN H SO2CH3

A-4105 SO2CH3 3-Me-lsoxazolin-5-yl CN H CH2OCH3

A-4106 SO2CH3 3-Me-lsoxazolin-5-yl CN cyclopropyl H

A-4107 SO2CH3 3-Me-lsoxazolin-5-yl CN OCH3 H

A-4108 SO2CH3 3-Me-lsoxazolin-5-yl CN OCF3 H

A-4109 SO2CH3 3-Me-lsoxazolin-5-yl CN SCH ₃ H

A-41 10 SO2CH3 3-Me-lsoxazolin-5-yl CN SOCH3 H

A-41 1 1 SO2CH3 3-Me-lsoxazolin-5-yl CN SO2CH3 H

A-41 12 SO2CH3 3-Me-lsoxazolin-5-yl CN CH2OCH3 H

A-41 13 SO2CH3 3-Me-lsoxazolin-5-yl H H CN

A-41 14 SO2CH3 3-Me-lsoxazolin-5-yl H H N0 ₂

A-41 15 SO2CH3 3-Me-lsoxazolin-5-yl H H cyclopropyl

A-41 16 SO2CH3 3-Me-lsoxazolin-5-yl H H OCH3

A-41 17 SO2CH3 3-Me-lsoxazolin-5-yl H H OCF3

A-41 18 SO2CH3 3-Me-lsoxazolin-5-yl H H SCH ₃

A-41 19 SO2CH3 3-Me-lsoxazolin-5-yl H H SOCH3

A-4120 SO2CH3 3-Me-lsoxazolin-5-yl H H SO2CH3

A-4121 SO2CH3 3-Me-lsoxazolin-5-yl H H CH2OCH3

A-4122 SO2CH3 3-Me-lsoxazolin-5-yl H cyclopropyl H

A-4123 SO2CH3 3-Me-lsoxazolin-5-yl H OCH3 H

A-4124 SO2CH3 3-Me-lsoxazolin-5-yl H OCF3 H

A-4125 SO2CH3 3-Me-lsoxazolin-5-yl H SCH ₃ H

A-4126 SO2CH3 3-Me-lsoxazolin-5-yl H SOCH3 H

A-4127 SO2CH3 3-Me-lsoxazolin-5-yl H SO2CH3 H A-4128 SO2CH3 3-Me-lsoxazolin-5-yl H CH2OCH3 H

A-4129 SO2CH3 3-Me-lsoxazol-5-yl CI H CN

A-4130 SO2CH3 3-Me-lsoxazol-5-yl CI H N0 ₂

A-4131 SO2CH3 3-Me-lsoxazol-5-yl CI H cyclopropyl

A-4132 SO2CH3 3-Me-lsoxazol-5-yl CI H OCH3

A-4133 SO2CH3 3-Me-lsoxazol-5-yl CI H OCF3

A-4134 SO2CH3 3-Me-lsoxazol-5-yl CI H SCH ₃

A-4135 SO2CH3 3-Me-lsoxazol-5-yl CI H SOCH3

A-4136 SO2CH3 3-Me-lsoxazol-5-yl CI H SO2CH3

A-4137 SO2CH3 3-Me-lsoxazol-5-yl CI H CH2OCH3

A-4138 SO2CH3 3-Me-lsoxazol-5-yl CI cyclopropyl H

A-4139 SO2CH3 3-Me-lsoxazol-5-yl CI OCH3 H

A-4140 SO2CH3 3-Me-lsoxazol-5-yl CI OCF3 H

A-4141 SO2CH3 3-Me-lsoxazol-5-yl CI SCH ₃ H

A-4142 SO2CH3 3-Me-lsoxazol-5-yl CI SOCH3 H

A-4143 SO2CH3 3-Me-lsoxazol-5-yl CI SO2CH3 H

A-4144 SO2CH3 3-Me-lsoxazol-5-yl CI CH2OCH3 H

A-4145 SO2CH3 3-Me-lsoxazol-5-yl F H CN

A-4146 SO2CH3 3-Me-lsoxazol-5-yl F H N0 ₂

A-4147 SO2CH3 3-Me-lsoxazol-5-yl F H cyclopropyl

A-4148 SO2CH3 3-Me-lsoxazol-5-yl F H OCH3

A-4149 SO2CH3 3-Me-lsoxazol-5-yl F H OCF3

A-4150 SO2CH3 3-Me-lsoxazol-5-yl F H SCH ₃

A-4151 SO2CH3 3-Me-lsoxazol-5-yl F H SOCH3

A-4152 SO2CH3 3-Me-lsoxazol-5-yl F H SO2CH3

A-4153 SO2CH3 3-Me-lsoxazol-5-yl F H CH2OCH3

A-4154 SO2CH3 3-Me-lsoxazol-5-yl F cyclopropyl H

A-4155 SO2CH3 3-Me-lsoxazol-5-yl F OCH3 H

A-4156 SO2CH3 3-Me-lsoxazol-5-yl F OCF3 H

A-4157 SO2CH3 3-Me-lsoxazol-5-yl F SCH ₃ H

A-4158 SO2CH3 3-Me-lsoxazol-5-yl F SOCH3 H

A-4159 SO2CH3 3-Me-lsoxazol-5-yl F SO2CH3 H

A-4160 SO2CH3 3-Me-lsoxazol-5-yl F CH2OCH3 H

A-4161 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ H CN

A-4162 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ H N0 ₂

A-4163 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ H cyclopropyl

A-4164 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ H OCH3 A-4165 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ H OCF3

A-4166 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ H SCH ₃

A-4167 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ H SOCH3

A-4168 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ H SO2CH3

A-4169 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ H CH2OCH3

A-4170 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ cyclopropyl H

A-4171 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ OCH3 H

A-4172 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ OCF3 H

A-4173 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ SCH ₃ H

A-4174 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ SOCH3 H

A-4175 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ SO2CH3 H

A-4176 SO2CH3 3-Me-lsoxazol-5-yl CF ₃ CH2OCH3 H

A-4177 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 H CN

A-4178 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 H N0 ₂

A-4179 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 H cyclopropyl

A-4180 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 H OCH3

A-4181 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 H OCF3

A-4182 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 H SCH ₃

A-4183 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 H SOCH3

A-4184 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 H SO2CH3

A-4185 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 H CH2OCH3

A-4186 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 cyclopropyl H

A-4187 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 OCH3 H

A-4188 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 OCF3 H

A-4189 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 SCH ₃ H

A-4190 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 SOCH3 H

A-4191 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 SO2CH3 H

A-4192 SO2CH3 3-Me-lsoxazol-5-yl SO2CH3 CH2OCH3 H

A-4193 SO2CH3 3-Me-lsoxazol-5-yl CN H CN

A-4194 SO2CH3 3-Me-lsoxazol-5-yl CN H N0 ₂

A-4195 SO2CH3 3-Me-lsoxazol-5-yl CN H cyclopropyl

A-4196 SO2CH3 3-Me-lsoxazol-5-yl CN H OCH3

A-4197 SO2CH3 3-Me-lsoxazol-5-yl CN H OCF3

A-4198 SO2CH3 3-Me-lsoxazol-5-yl CN H SCH ₃

A-4199 SO2CH3 3-Me-lsoxazol-5-yl CN H SOCH3

A-4200 SO2CH3 3-Me-lsoxazol-5-yl CN H SO2CH3

A-4201 SO2CH3 3-Me-lsoxazol-5-yl CN H CH2OCH3 A-4350 N0 ₂ SCHs F SOCHs H

A-4351 N0 ₂ SCHs F SO2CH3 H

A-4352 N0 ₂ SCHs F CH2OCH3 H

A-4353 N0 ₂ SCHs CFs H CN

A-4354 N0 ₂ SCHs CFs H N0 ₂

A-4355 N0 ₂ SCHs CFs H cyclopropyl

A-4356 N0 ₂ SCHs CFs H OCH3

A-4357 N0 ₂ SCHs CFs H OCFs

A-4358 N0 ₂ SCHs CFs H SCHs

A-4359 N0 ₂ SCHs CFs H SOCHs

A-4360 N0 ₂ SCHs CFs H SO2CH3

A-4361 N0 ₂ SCHs CFs H CH2OCH3

A-4362 N0 ₂ SCHs CFs cyclopropyl H

A-4363 N0 ₂ SCHs CFs OCH3 H

A-4364 N0 ₂ SCHs CFs OCFs H

A-4365 N0 ₂ SCHs CFs SCHs H

A-4366 N0 ₂ SCHs CFs SOCHs H

A-4367 N0 ₂ SCHs CFs SO2CH3 H

A-4368 N0 ₂ SCHs CFs CH2OCH3 H

A-4369 N0 ₂ SCHs SO2CH3 H CN

A-4370 N0 ₂ SCHs SO2CH3 H N0 ₂

A-4371 N0 ₂ SCHs SO2CH3 H cyclopropyl

A-4372 N0 ₂ SCHs SO2CH3 H OCH3

A-4373 N0 ₂ SCHs SO2CH3 H OCFs

A-4374 N0 ₂ SCHs SO2CH3 H SCHs

A-4375 N0 ₂ SCHs SO2CH3 H SOCHs

A-4376 N0 ₂ SCHs SO2CH3 H SO2CH3

A-4377 N0 ₂ SCHs SO2CH3 H CH2OCH3

A-4378 N0 ₂ SCHs SO2CH3 cyclopropyl H

A-4379 N0 ₂ SCHs SO2CH3 OCH3 H

A-4380 N0 ₂ SCHs SO2CH3 OCFs H

A-4381 N0 ₂ SCHs SO2CH3 SCHs H

A-4382 N0 ₂ SCHs SO2CH3 SOCHs H

A-4383 N0 ₂ SCHs SO2CH3 SO2CH3 H

A-4384 N0 ₂ SCHs SO2CH3 CH2OCH3 H

A-4385 N0 ₂ SCHs CN H CN

A-4386 N0 ₂ SCHs CN H N0 ₂ A-4387 N0 ₂ SCHs CN H cyclopropyl

A-4388 N0 ₂ SCHs CN H OCHs

A-4389 N0 ₂ SCHs CN H OCFs

A-4390 N0 ₂ SCHs CN H SCHs

A-4391 N0 ₂ SCHs CN H SOCHs

A-4392 N0 ₂ SCHs CN H SO2CH3

A-4393 N0 ₂ SCHs CN H CH2OCH3

A-4394 N0 ₂ SCHs CN cyclopropyl H

A-4395 N0 ₂ SCHs CN OCHs H

A-4396 N0 ₂ SCHs CN OCFs H

A-4397 N0 ₂ SCHs CN SCHs H

A-4398 N0 ₂ SCHs CN SOCHs H

A-4399 N0 ₂ SCHs CN SO2CH3 H

A-4400 N0 ₂ SCHs CN CH2OCH3 H

A-4401 N0 ₂ SOCHs H H CN

A-4402 N0 ₂ SOCHs H H N0 ₂

A-4403 N0 ₂ SOCHs H H cyclopropyl

A-4404 N0 ₂ SOCHs H H OCHs

A-4405 N0 ₂ SOCHs H H OCFs

A-4406 N0 ₂ SOCHs H H SCHs

A-4407 N0 ₂ SOCHs H H SOCHs

A-4408 N0 ₂ SOCHs H H SO2CH3

A-4409 N0 ₂ SOCHs H H CH2OCH3

A-4410 N0 ₂ SOCHs H cyclopropyl H

A-441 1 N0 ₂ SOCHs H OCHs H

A-4412 N0 ₂ SOCHs H OCFs H

A-4413 N0 ₂ SOCHs H SCHs H

A-4414 N0 ₂ SOCHs H SOCHs H

A-4415 N0 ₂ SOCHs H SO2CH3 H

A-4416 N0 ₂ SOCHs H CH2OCH3 H

A-4417 N0 ₂ SOCHs CI H CN

A-4418 N0 ₂ SOCHs CI H N0 ₂

A-4419 N0 ₂ SOCHs CI H cyclopropyl

A-4420 N0 ₂ SOCHs CI H OCHs

A-4421 N0 ₂ SOCHs CI H OCFs

A-4422 N0 ₂ SOCHs CI H SCHs

A-4423 N0 ₂ SOCHs CI H SOCHs A-4535 N0 ₂ SO2CH3 F H SOCH3

A-4536 N0 ₂ SO2CH3 F H SO2CH3

A-4537 N0 ₂ SO2CH3 F H CH2OCH3

A-4538 N0 ₂ SO2CH3 F cyclopropyl H

A-4539 N0 ₂ SO2CH3 F OCH3 H

A-4540 N0 ₂ SO2CH3 F OCF3 H

A-4541 N0 ₂ SO2CH3 F SCH ₃ H

A-4542 N0 ₂ SO2CH3 F SOCH3 H

A-4543 N0 ₂ SO2CH3 F SO2CH3 H

A-4544 N0 ₂ SO2CH3 F CH2OCH3 H

A-4545 N0 ₂ SO2CH3 CF ₃ H CN

A-4546 N0 ₂ SO2CH3 CF ₃ H N0 ₂

A-4547 N0 ₂ SO2CH3 CF ₃ H cyclopropyl

A-4548 N0 ₂ SO2CH3 CF ₃ H OCH3

A-4549 N0 ₂ SO2CH3 CF ₃ H OCF3

A-4550 N0 ₂ SO2CH3 CF ₃ H SCH ₃

A-4551 N0 ₂ SO2CH3 CF ₃ H SOCH3

A-4552 N0 ₂ SO2CH3 CF ₃ H SO2CH3

A-4553 N0 ₂ SO2CH3 CF ₃ H CH2OCH3

A-4554 N0 ₂ SO2CH3 CF ₃ cyclopropyl H

A-4555 N0 ₂ SO2CH3 CF ₃ OCH3 H

A-4556 N0 ₂ SO2CH3 CF ₃ OCF3 H

A-4557 N0 ₂ SO2CH3 CF ₃ SCH ₃ H

A-4558 N0 ₂ SO2CH3 CF ₃ SOCH3 H

A-4559 N0 ₂ SO2CH3 CF ₃ SO2CH3 H

A-4560 N0 ₂ SO2CH3 CF ₃ CH2OCH3 H

A-4561 N0 ₂ SO2CH3 SO2CH3 H CN

A-4562 N0 ₂ SO2CH3 SO2CH3 H N0 ₂

A-4563 N0 ₂ SO2CH3 SO2CH3 H cyclopropyl

A-4564 N0 ₂ SO2CH3 SO2CH3 H OCH3

A-4565 N0 ₂ SO2CH3 SO2CH3 H OCF3

A-4566 N0 ₂ SO2CH3 SO2CH3 H SCH ₃

A-4567 N0 ₂ SO2CH3 SO2CH3 H SOCH3

A-4568 N0 ₂ SO2CH3 SO2CH3 H SO2CH3

A-4569 N0 ₂ SO2CH3 SO2CH3 H CH2OCH3

A-4570 N0 ₂ SO2CH3 SO2CH3 cyclopropyl H

A-4571 N0 ₂ SO2CH3 SO2CH3 OCH3 H A-4609 N0 ₂ CH2OCH2CF3 CI H CN

A-4610 N0 ₂ CH2OCH2CF3 CI H N0 ₂

A-461 1 N0 ₂ CH2OCH2CF3 CI H cyclopropyl

A-4612 N0 ₂ CH2OCH2CF3 CI H OCH3

A-4613 N0 ₂ CH2OCH2CF3 CI H OCF3

A-4614 N0 ₂ CH2OCH2CF3 CI H SCH ₃

A-4615 N0 ₂ CH2OCH2CF3 CI H SOCH3

A-4616 N0 ₂ CH2OCH2CF3 CI H SO2CH3

A-4617 N0 ₂ CH2OCH2CF3 CI H CH2OCH3

A-4618 N0 ₂ CH2OCH2CF3 CI cyclopropyl H

A-4619 N0 ₂ CH2OCH2CF3 CI OCH3 H

A-4620 N0 ₂ CH2OCH2CF3 CI OCF3 H

A-4621 N0 ₂ CH2OCH2CF3 CI SCH ₃ H

A-4622 N0 ₂ CH2OCH2CF3 CI SOCH3 H

A-4623 N0 ₂ CH2OCH2CF3 CI SO2CH3 H

A-4624 N0 ₂ CH2OCH2CF3 CI CH2OCH3 H

A-4625 N0 ₂ CH2OCH2CF3 F H CN

A-4626 N0 ₂ CH2OCH2CF3 F H N0 ₂

A-4627 N0 ₂ CH2OCH2CF3 F H cyclopropyl

A-4628 N0 ₂ CH2OCH2CF3 F H OCH3

A-4629 N0 ₂ CH2OCH2CF3 F H OCF3

A-4630 N0 ₂ CH2OCH2CF3 F H SCH ₃

A-4631 N0 ₂ CH2OCH2CF3 F H SOCH3

A-4632 N0 ₂ CH2OCH2CF3 F H SO2CH3

A-4633 N0 ₂ CH2OCH2CF3 F H CH2OCH3

A-4634 N0 ₂ CH2OCH2CF3 F cyclopropyl H

A-4635 N0 ₂ CH2OCH2CF3 F OCH3 H

A-4636 N0 ₂ CH2OCH2CF3 F OCF3 H

A-4637 N0 ₂ CH2OCH2CF3 F SCH ₃ H

A-4638 N0 ₂ CH2OCH2CF3 F SOCH3 H

A-4639 N0 ₂ CH2OCH2CF3 F SO2CH3 H

A-4640 N0 ₂ CH2OCH2CF3 F CH2OCH3 H

A-4641 N0 ₂ CH2OCH2CF3 CF ₃ H CN

A-4642 N0 ₂ CH2OCH2CF3 CF ₃ H N0 ₂

A-4643 N0 ₂ CH2OCH2CF3 CF ₃ H cyclopropyl

A-4644 N0 ₂ CH2OCH2CF3 CF ₃ H OCH3

A-4645 N0 ₂ CH2OCH2CF3 CF ₃ H OCF3 A-4646 N0 ₂ CH2OCH2CF3 CF ₃ H SCH ₃

A-4647 N0 ₂ CH2OCH2CF3 CF ₃ H SOCH3

A-4648 N0 ₂ CH2OCH2CF3 CF ₃ H SO2CH3

A-4649 N0 ₂ CH2OCH2CF3 CF ₃ H CH2OCH3

A-4650 N0 ₂ CH2OCH2CF3 CF ₃ cyclopropyl H

A-4651 N0 ₂ CH2OCH2CF3 CF ₃ OCH3 H

A-4652 N0 ₂ CH2OCH2CF3 CF ₃ OCF3 H

A-4653 N0 ₂ CH2OCH2CF3 CF ₃ SCH ₃ H

A-4654 N0 ₂ CH2OCH2CF3 CF ₃ SOCH3 H

A-4655 N0 ₂ CH2OCH2CF3 CF ₃ SO2CH3 H

A-4656 N0 ₂ CH2OCH2CF3 CF ₃ CH2OCH3 H

A-4657 N0 ₂ CH2OCH2CF3 SO2CH3 H CN

A-4658 N0 ₂ CH2OCH2CF3 SO2CH3 H N0 ₂

A-4659 N0 ₂ CH2OCH2CF3 SO2CH3 H cyclopropyl

A-4660 N0 ₂ CH2OCH2CF3 SO2CH3 H OCH3

A-4661 N0 ₂ CH2OCH2CF3 SO2CH3 H OCF3

A-4662 N0 ₂ CH2OCH2CF3 SO2CH3 H SCH ₃

A-4663 N0 ₂ CH2OCH2CF3 SO2CH3 H SOCH3

A-4664 N0 ₂ CH2OCH2CF3 SO2CH3 H SO2CH3

A-4665 N0 ₂ CH2OCH2CF3 SO2CH3 H CH2OCH3

A-4666 N0 ₂ CH2OCH2CF3 SO2CH3 cyclopropyl H

A-4667 N0 ₂ CH2OCH2CF3 SO2CH3 OCH3 H

A-4668 N0 ₂ CH2OCH2CF3 SO2CH3 OCF3 H

A-4669 N0 ₂ CH2OCH2CF3 SO2CH3 SCH ₃ H

A-4670 N0 ₂ CH2OCH2CF3 SO2CH3 SOCH3 H

A-4671 N0 ₂ CH2OCH2CF3 SO2CH3 SO2CH3 H

A-4672 N0 ₂ CH2OCH2CF3 SO2CH3 CH2OCH3 H

A-4673 N0 ₂ CH2OCH2CF3 CN H CN

A-4674 N0 ₂ CH2OCH2CF3 CN H N0 ₂

A-4675 N0 ₂ CH2OCH2CF3 CN H cyclopropyl

A-4676 N0 ₂ CH2OCH2CF3 CN H OCH3

A-4677 N0 ₂ CH2OCH2CF3 CN H OCF3

A-4678 N0 ₂ CH2OCH2CF3 CN H SCH ₃

A-4679 N0 ₂ CH2OCH2CF3 CN H SOCH3

A-4680 N0 ₂ CH2OCH2CF3 CN H SO2CH3

A-4681 N0 ₂ CH2OCH2CF3 CN H CH2OCH3

A-4682 N0 ₂ CH2OCH2CF3 CN cyclopropyl H A-4683 N0 ₂ CH2OCH2CF3 CN 0CH3 H

A-4684 N0 ₂ CH2OCH2CF3 CN 0CF3 H

A-4685 N0 ₂ CH2OCH2CF3 CN SCH3 H

A-4686 N0 ₂ CH2OCH2CF3 CN SOCH3 H

A-4687 N0 ₂ CH2OCH2CF3 CN S02CH3 H

A-4688 N0 ₂ CH2OCH2CF3 CN CH20CH3 H

A-4689 N0 ₂ CH2OCH2CF3 H H CN

A-4690 N0 ₂ CH2OCH2CF3 H H N0 ₂

A-4691 N0 ₂ CH2OCH2CF3 H H cyclopropyl

A-4692 N0 ₂ CH2OCH2CF3 H H OCH3

A-4693 N0 ₂ CH2OCH2CF3 H H OCF3

A-4694 N0 ₂ CH2OCH2CF3 H H SCH ₃

A-4695 N0 ₂ CH2OCH2CF3 H H SOCH3

A-4696 N0 ₂ CH2OCH2CF3 H H SO2CH3

A-4697 N0 ₂ CH2OCH2CF3 H H CH2OCH3

A-4698 N0 ₂ CH2OCH2CF3 H cyclopropyl H

A-4699 N0 ₂ CH2OCH2CF3 H OCH3 H

A-4700 N0 ₂ CH2OCH2CF3 H OCF3 H

A-4701 N0 ₂ CH2OCH2CF3 H SCH ₃ H

A-4702 N0 ₂ CH2OCH2CF3 H SOCH3 H

A-4703 N0 ₂ CH2OCH2CF3 H SO2CH3 H

A-4704 N0 ₂ CH2OCH2CF3 H CH2OCH3 H

A-4705 N0 ₂ lsoxazolin-3-yl CI H CN

A-4706 N0 ₂ lsoxazolin-3-yl CI H N0 ₂

A-4707 N0 ₂ lsoxazolin-3-yl CI H cyclopropyl

A-4708 N0 ₂ lsoxazolin-3-yl CI H OCH3

A-4709 N0 ₂ lsoxazolin-3-yl CI H OCF3

A-4710 N0 ₂ lsoxazolin-3-yl CI H SCH ₃

A-471 1 N0 ₂ lsoxazolin-3-yl CI H SOCH3

A-4712 N0 ₂ lsoxazolin-3-yl CI H SO2CH3

A-4713 N0 ₂ lsoxazolin-3-yl CI H CH2OCH3

A-4714 N0 ₂ lsoxazolin-3-yl CI cyclopropyl H

A-4715 N0 ₂ lsoxazolin-3-yl CI OCH3 H

A-4716 N0 ₂ lsoxazolin-3-yl CI OCF3 H

A-4717 N0 ₂ lsoxazolin-3-yl CI SCH ₃ H

A-4718 N0 ₂ lsoxazolin-3-yl CI SOCH3 H

A-4719 N0 ₂ lsoxazolin-3-yl CI SO2CH3 H A-4720 N0 ₂ lsoxazolin-3-yl CI CH2OCH3 H

A-4721 N0 ₂ lsoxazolin-3-yl F H CN

A-4722 N0 ₂ lsoxazolin-3-yl F H N0 ₂

A-4723 N0 ₂ lsoxazolin-3-yl F H cyclopropyl

A-4724 N0 ₂ lsoxazolin-3-yl F H OCH3

A-4725 N0 ₂ lsoxazolin-3-yl F H OCFs

A-4726 N0 ₂ lsoxazolin-3-yl F H SCHs

A-4727 N0 ₂ lsoxazolin-3-yl F H SOCHs

A-4728 N0 ₂ lsoxazolin-3-yl F H SO2CH3

A-4729 N0 ₂ lsoxazolin-3-yl F H CH2OCH3

A-4730 N0 ₂ lsoxazolin-3-yl F cyclopropyl H

A-4731 N0 ₂ lsoxazolin-3-yl F OCH3 H

A-4732 N0 ₂ lsoxazolin-3-yl F OCFs H

A-4733 N0 ₂ lsoxazolin-3-yl F SCHs H

A-4734 N0 ₂ lsoxazolin-3-yl F SOCHs H

A-4735 N0 ₂ lsoxazolin-3-yl F SO2CH3 H

A-4736 N0 ₂ lsoxazolin-3-yl F CH2OCH3 H

A-4737 N0 ₂ lsoxazolin-3-yl CFs H CN

A-4738 N0 ₂ lsoxazolin-3-yl CFs H N0 ₂

A-4739 N0 ₂ lsoxazolin-3-yl CFs H cyclopropyl

A-4740 N0 ₂ lsoxazolin-3-yl CFs H OCH3

A-4741 N0 ₂ lsoxazolin-3-yl CFs H OCFs

A-4742 N0 ₂ lsoxazolin-3-yl CFs H SCHs

A-4743 N0 ₂ lsoxazolin-3-yl CFs H SOCHs

A-4744 N0 ₂ lsoxazolin-3-yl CFs H SO2CH3

A-4745 N0 ₂ lsoxazolin-3-yl CFs H CH2OCH3

A-4746 N0 ₂ lsoxazolin-3-yl CFs cyclopropyl H

A-4747 N0 ₂ lsoxazolin-3-yl CFs OCH3 H

A-4748 N0 ₂ lsoxazolin-3-yl CFs OCFs H

A-4749 N0 ₂ lsoxazolin-3-yl CFs SCHs H

A-4750 N0 ₂ lsoxazolin-3-yl CFs SOCHs H

A-4751 N0 ₂ lsoxazolin-3-yl CFs SO2CH3 H

A-4752 N0 ₂ lsoxazolin-3-yl CFs CH2OCH3 H

A-4753 N0 ₂ lsoxazolin-3-yl SO2CH3 H CN

A-4754 N0 ₂ lsoxazolin-3-yl SO2CH3 H N0 ₂

A-4755 N0 ₂ lsoxazolin-3-yl SO2CH3 H cyclopropyl

A-4756 N0 ₂ lsoxazolin-3-yl SO2CH3 H OCH3 A-4757 N0 ₂ lsoxazolin-3-yl SO2CH3 H OCF3

A-4758 N0 ₂ lsoxazolin-3-yl SO2CH3 H SCH ₃

A-4759 N0 ₂ lsoxazolin-3-yl SO2CH3 H SOCH3

A-4760 N0 ₂ lsoxazolin-3-yl SO2CH3 H SO2CH3

A-4761 N0 ₂ lsoxazolin-3-yl SO2CH3 H CH2OCH3

A-4762 N0 ₂ lsoxazolin-3-yl SO2CH3 cyclopropyl H

A-4763 N0 ₂ lsoxazolin-3-yl SO2CH3 OCH3 H

A-4764 N0 ₂ lsoxazolin-3-yl SO2CH3 OCF3 H

A-4765 N0 ₂ lsoxazolin-3-yl SO2CH3 SCH ₃ H

A-4766 N0 ₂ lsoxazolin-3-yl SO2CH3 SOCH3 H

A-4767 N0 ₂ lsoxazolin-3-yl SO2CH3 SO2CH3 H

A-4768 N0 ₂ lsoxazolin-3-yl SO2CH3 CH2OCH3 H

A-4769 N0 ₂ lsoxazolin-3-yl CN H CN

A-4770 N0 ₂ lsoxazolin-3-yl CN H N0 ₂

A-4771 N0 ₂ lsoxazolin-3-yl CN H cyclopropyl

A-4772 N0 ₂ lsoxazolin-3-yl CN H OCH3

A-4773 N0 ₂ lsoxazolin-3-yl CN H OCF3

A-4774 N0 ₂ lsoxazolin-3-yl CN H SCH ₃

A-4775 N0 ₂ lsoxazolin-3-yl CN H SOCH3

A-4776 N0 ₂ lsoxazolin-3-yl CN H SO2CH3

A-4777 N0 ₂ lsoxazolin-3-yl CN H CH2OCH3

A-4778 N0 ₂ lsoxazolin-3-yl CN cyclopropyl H

A-4779 N0 ₂ lsoxazolin-3-yl CN OCH3 H

A-4780 N0 ₂ lsoxazolin-3-yl CN OCF3 H

A-4781 N0 ₂ lsoxazolin-3-yl CN SCH ₃ H

A-4782 N0 ₂ lsoxazolin-3-yl CN SOCH3 H

A-4783 N0 ₂ lsoxazolin-3-yl CN SO2CH3 H

A-4784 N0 ₂ lsoxazolin-3-yl CN CH2OCH3 H

A-4785 N0 ₂ lsoxazolin-3-yl H H CN

A-4786 N0 ₂ lsoxazolin-3-yl H H N0 ₂

A-4787 N0 ₂ lsoxazolin-3-yl H H cyclopropyl

A-4788 N0 ₂ lsoxazolin-3-yl H H OCH3

A-4789 N0 ₂ lsoxazolin-3-yl H H OCF3

A-4790 N0 ₂ lsoxazolin-3-yl H H SCH ₃

A-4791 N0 ₂ lsoxazolin-3-yl H H SOCH3

A-4792 N0 ₂ lsoxazolin-3-yl H H SO2CH3

A-4793 N0 ₂ lsoxazolin-3-yl H H CH2OCH3 A-4794 N0 ₂ lsoxazolin-3-yl H cyclopropyl H

A-4795 N0 ₂ lsoxazolin-3-yl H OCH3 H

A-4796 N0 ₂ lsoxazolin-3-yl H OCF3 H

A-4797 N0 ₂ lsoxazolin-3-yl H SCHs H

A-4798 N0 ₂ lsoxazolin-3-yl H SOCH3 H

A-4799 N0 ₂ lsoxazolin-3-yl H SO2CH3 H

A-4800 N0 ₂ lsoxazolin-3-yl H CH2OCH3 H

A-4801 N0 ₂ 5-Me-lsoxazolin-3-yl CI H CN

A-4802 N0 ₂ 5-Me-lsoxazolin-3-yl CI H N0 ₂

A-4803 N0 ₂ 5-Me-lsoxazolin-3-yl CI H cyclopropyl

A-4804 N0 ₂ 5-Me-lsoxazolin-3-yl CI H OCH3

A-4805 N0 ₂ 5-Me-lsoxazolin-3-yl CI H OCF3

A-4806 N0 ₂ 5-Me-lsoxazolin-3-yl CI H SCH ₃

A-4807 N0 ₂ 5-Me-lsoxazolin-3-yl CI H SOCH3

A-4808 N0 ₂ 5-Me-lsoxazolin-3-yl CI H SO2CH3

A-4809 N0 ₂ 5-Me-lsoxazolin-3-yl CI H CH2OCH3

A-4810 N0 ₂ 5-Me-lsoxazolin-3-yl CI cyclopropyl H

A-481 1 N0 ₂ 5-Me-lsoxazolin-3-yl CI OCH3 H

A-4812 N0 ₂ 5-Me-lsoxazolin-3-yl CI OCF3 H

A-4813 N0 ₂ 5-Me-lsoxazolin-3-yl CI SCH ₃ H

A-4814 N0 ₂ 5-Me-lsoxazolin-3-yl CI SOCH3 H

A-4815 N0 ₂ 5-Me-lsoxazolin-3-yl CI SO2CH3 H

A-4816 N0 ₂ 5-Me-lsoxazolin-3-yl CI CH2OCH3 H

A-4817 N0 ₂ 5-Me-lsoxazolin-3-yl F H CN

A-4818 N0 ₂ 5-Me-lsoxazolin-3-yl F H N0 ₂

A-4819 N0 ₂ 5-Me-lsoxazolin-3-yl F H cyclopropyl

A-4820 N0 ₂ 5-Me-lsoxazolin-3-yl F H OCH3

A-4821 N0 ₂ 5-Me-lsoxazolin-3-yl F H OCF3

A-4822 N0 ₂ 5-Me-lsoxazolin-3-yl F H SCH ₃

A-4823 N0 ₂ 5-Me-lsoxazolin-3-yl F H SOCH3

A-4824 N0 ₂ 5-Me-lsoxazolin-3-yl F H SO2CH3

A-4825 N0 ₂ 5-Me-lsoxazolin-3-yl F H CH2OCH3

A-4826 N0 ₂ 5-Me-lsoxazolin-3-yl F cyclopropyl H

A-4827 N0 ₂ 5-Me-lsoxazolin-3-yl F OCH3 H

A-4828 N0 ₂ 5-Me-lsoxazolin-3-yl F OCF3 H

A-4829 N0 ₂ 5-Me-lsoxazolin-3-yl F SCH ₃ H

A-4830 N0 ₂ 5-Me-lsoxazolin-3-yl F SOCH3 H A-4831 N0 ₂ 5-Me-lsoxazolin-3-yl F SO2CH3 H

A-4832 N0 ₂ 5-Me-lsoxazolin-3-yl F CH2OCH3 H

A-4833 N0 ₂ 5-Me-lsoxazolin-3-yl CFs H CN

A-4834 N0 ₂ 5-Me-lsoxazolin-3-yl CFs H N0 ₂

A-4835 N0 ₂ 5-Me-lsoxazolin-3-yl CFs H cyclopropyl

A-4836 N0 ₂ 5-Me-lsoxazolin-3-yl CFs H OCH3

A-4837 N0 ₂ 5-Me-lsoxazolin-3-yl CFs H OCFs

A-4838 N0 ₂ 5-Me-lsoxazolin-3-yl CFs H SCHs

A-4839 N0 ₂ 5-Me-lsoxazolin-3-yl CFs H SOCHs

A-4840 N0 ₂ 5-Me-lsoxazolin-3-yl CFs H SO2CH3

A-4841 N0 ₂ 5-Me-lsoxazolin-3-yl CFs H CH2OCH3

A-4842 N0 ₂ 5-Me-lsoxazolin-3-yl CFs cyclopropyl H

A-4843 N0 ₂ 5-Me-lsoxazolin-3-yl CFs OCH3 H

A-4844 N0 ₂ 5-Me-lsoxazolin-3-yl CFs OCFs H

A-4845 N0 ₂ 5-Me-lsoxazolin-3-yl CFs SCHs H

A-4846 N0 ₂ 5-Me-lsoxazolin-3-yl CFs SOCHs H

A-4847 N0 ₂ 5-Me-lsoxazolin-3-yl CFs SO2CH3 H

A-4848 N0 ₂ 5-Me-lsoxazolin-3-yl CFs CH2OCH3 H

A-4849 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 H CN

A-4850 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 H N0 ₂

A-4851 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 H cyclopropyl

A-4852 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 H OCH3

A-4853 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 H OCFs

A-4854 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 H SCHs

A-4855 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 H SOCHs

A-4856 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 H SO2CH3

A-4857 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 H CH2OCH3

A-4858 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 cyclopropyl H

A-4859 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 OCH3 H

A-4860 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 OCFs H

A-4861 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 SCHs H

A-4862 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 SOCHs H

A-4863 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 SO2CH3 H

A-4864 N0 ₂ 5-Me-lsoxazolin-3-yl SO2CH3 CH2OCH3 H

A-4865 N0 ₂ 5-Me-lsoxazolin-3-yl CN H CN

A-4866 N0 ₂ 5-Me-lsoxazolin-3-yl CN H N0 ₂

A-4867 N0 ₂ 5-Me-lsoxazolin-3-yl CN H cyclopropyl A-4868 N0 ₂ 5-Me-lsoxazolin-3-yl CN H OCH3

A-4869 N0 ₂ 5-Me-lsoxazolin-3-yl CN H OCF3

A-4870 N0 ₂ 5-Me-lsoxazolin-3-yl CN H SCH ₃

A-4871 N0 ₂ 5-Me-lsoxazolin-3-yl CN H SOCH3

A-4872 N0 ₂ 5-Me-lsoxazolin-3-yl CN H SO2CH3

A-4873 N0 ₂ 5-Me-lsoxazolin-3-yl CN H CH2OCH3

A-4874 N0 ₂ 5-Me-lsoxazolin-3-yl CN cyclopropyl H

A-4875 N0 ₂ 5-Me-lsoxazolin-3-yl CN OCH3 H

A-4876 N0 ₂ 5-Me-lsoxazolin-3-yl CN OCF3 H

A-4877 N0 ₂ 5-Me-lsoxazolin-3-yl CN SCHs H

A-4878 N0 ₂ 5-Me-lsoxazolin-3-yl CN SOCH3 H

A-4879 N0 ₂ 5-Me-lsoxazolin-3-yl CN SO2CH3 H

A-4880 N0 ₂ 5-Me-lsoxazolin-3-yl CN CH2OCH3 H

A-4881 N0 ₂ 5-Me-lsoxazolin-3-yl H H CN

A-4882 N0 ₂ 5-Me-lsoxazolin-3-yl H H N0 ₂

A-4883 N0 ₂ 5-Me-lsoxazolin-3-yl H H cyclopropyl

A-4884 N0 ₂ 5-Me-lsoxazolin-3-yl H H OCH3

A-4885 N0 ₂ 5-Me-lsoxazolin-3-yl H H OCF3

A-4886 N0 ₂ 5-Me-lsoxazolin-3-yl H H SCH ₃

A-4887 N0 ₂ 5-Me-lsoxazolin-3-yl H H SOCH3

A-4888 N0 ₂ 5-Me-lsoxazolin-3-yl H H SO2CH3

A-4889 N0 ₂ 5-Me-lsoxazolin-3-yl H H CH2OCH3

A-4890 N0 ₂ 5-Me-lsoxazolin-3-yl H cyclopropyl H

A-4891 N0 ₂ 5-Me-lsoxazolin-3-yl H OCH3 H

A-4892 N0 ₂ 5-Me-lsoxazolin-3-yl H OCF3 H

A-4893 N0 ₂ 5-Me-lsoxazolin-3-yl H SCH ₃ H

A-4894 N0 ₂ 5-Me-lsoxazolin-3-yl H SOCH3 H

A-4895 N0 ₂ 5-Me-lsoxazolin-3-yl H SO2CH3 H

A-4896 N0 ₂ 5-Me-lsoxazolin-3-yl H CH2OCH3 H

A-4897 N0 ₂ lsoxazol-3-yl CI H CN

A-4898 N0 ₂ lsoxazol-3-yl CI H N0 ₂

A-4899 N0 ₂ lsoxazol-3-yl CI H cyclopropyl

A-4900 N0 ₂ lsoxazol-3-yl CI H OCH3

A-4901 N0 ₂ lsoxazol-3-yl CI H OCF3

A-4902 N0 ₂ lsoxazol-3-yl CI H SCH ₃

A-4903 N0 ₂ lsoxazol-3-yl CI H SOCH3

A-4904 N0 ₂ lsoxazol-3-yl CI H SO2CH3 A-4905 N0 ₂ lsoxazol-3-yl CI H CH2OCH3

A-4906 N0 ₂ lsoxazol-3-yl CI cyclopropyl H

A-4907 N0 ₂ lsoxazol-3-yl CI OCHs H

A-4908 N0 ₂ lsoxazol-3-yl CI OCFs H

A-4909 N0 ₂ lsoxazol-3-yl CI SCHs H

A-4910 N0 ₂ lsoxazol-3-yl CI SOCHs H

A-491 1 N0 ₂ lsoxazol-3-yl CI SO2CH3 H

A-4912 N0 ₂ lsoxazol-3-yl CI CH2OCH3 H

A-4913 N0 ₂ lsoxazol-3-yl F H CN

A-4914 N0 ₂ lsoxazol-3-yl F H N0 ₂

A-4915 N0 ₂ lsoxazol-3-yl F H cyclopropyl

A-4916 N0 ₂ lsoxazol-3-yl F H OCHs

A-4917 N0 ₂ lsoxazol-3-yl F H OCFs

A-4918 N0 ₂ lsoxazol-3-yl F H SCHs

A-4919 N0 ₂ lsoxazol-3-yl F H SOCHs

A-4920 N0 ₂ lsoxazol-3-yl F H SO2CH3

A-4921 N0 ₂ lsoxazol-3-yl F H CH2OCH3

A-4922 N0 ₂ lsoxazol-3-yl F cyclopropyl H

A-4923 N0 ₂ lsoxazol-3-yl F OCHs H

A-4924 N0 ₂ lsoxazol-3-yl F OCFs H

A-4925 N0 ₂ lsoxazol-3-yl F SCHs H

A-4926 N0 ₂ lsoxazol-3-yl F SOCHs H

A-4927 N0 ₂ lsoxazol-3-yl F SO2CH3 H

A-4928 N0 ₂ lsoxazol-3-yl F CH2OCH3 H

A-4929 N0 ₂ lsoxazol-3-yl CFs H CN

A-4930 N0 ₂ lsoxazol-3-yl CFs H N0 ₂

A-4931 N0 ₂ lsoxazol-3-yl CFs H cyclopropyl

A-4932 N0 ₂ lsoxazol-3-yl CFs H OCHs

A-4933 N0 ₂ lsoxazol-3-yl CFs H OCFs

A-4934 N0 ₂ lsoxazol-3-yl CFs H SCHs

A-4935 N0 ₂ lsoxazol-3-yl CFs H SOCHs

A-4936 N0 ₂ lsoxazol-3-yl CFs H SO2CH3

A-4937 N0 ₂ lsoxazol-3-yl CFs H CH2OCH3

A-4938 N0 ₂ lsoxazol-3-yl CFs cyclopropyl H

A-4939 N0 ₂ lsoxazol-3-yl CFs OCHs H

A-4940 N0 ₂ lsoxazol-3-yl CFs OCFs H

A-4941 N0 ₂ lsoxazol-3-yl CFs SCHs H A-4942 N0 ₂ lsoxazol-3-yl CFs SOCH3 H

A-4943 N0 ₂ lsoxazol-3-yl CFs SO2CH3 H

A-4944 N0 ₂ lsoxazol-3-yl CFs CH2OCH3 H

A-4945 N0 ₂ lsoxazol-3-yl SO2CH3 H CN

A-4946 N0 ₂ lsoxazol-3-yl SO2CH3 H N0 ₂

A-4947 N0 ₂ lsoxazol-3-yl SO2CH3 H cyclopropyl

A-4948 N0 ₂ lsoxazol-3-yl SO2CH3 H OCH3

A-4949 N0 ₂ lsoxazol-3-yl SO2CH3 H OCF3

A-4950 N0 ₂ lsoxazol-3-yl SO2CH3 H SCH ₃

A-4951 N0 ₂ lsoxazol-3-yl SO2CH3 H SOCH3

A-4952 N0 ₂ lsoxazol-3-yl SO2CH3 H SO2CH3

A-4953 N0 ₂ lsoxazol-3-yl SO2CH3 H CH2OCH3

A-4954 N0 ₂ lsoxazol-3-yl SO2CH3 cyclopropyl H

A-4955 N0 ₂ lsoxazol-3-yl SO2CH3 OCH3 H

A-4956 N0 ₂ lsoxazol-3-yl SO2CH3 OCF3 H

A-4957 N0 ₂ lsoxazol-3-yl SO2CH3 SCH ₃ H

A-4958 N0 ₂ lsoxazol-3-yl SO2CH3 SOCH3 H

A-4959 N0 ₂ lsoxazol-3-yl SO2CH3 SO2CH3 H

A-4960 N0 ₂ lsoxazol-3-yl SO2CH3 CH2OCH3 H

A-4961 N0 ₂ lsoxazol-3-yl CN H CN

A-4962 N0 ₂ lsoxazol-3-yl CN H N0 ₂

A-4963 N0 ₂ lsoxazol-3-yl CN H cyclopropyl

A-4964 N0 ₂ lsoxazol-3-yl CN H OCH3

A-4965 N0 ₂ lsoxazol-3-yl CN H OCF3

A-4966 N0 ₂ lsoxazol-3-yl CN H SCH ₃

A-4967 N0 ₂ lsoxazol-3-yl CN H SOCH3

A-4968 N0 ₂ lsoxazol-3-yl CN H SO2CH3

A-4969 N0 ₂ lsoxazol-3-yl CN H CH2OCH3

A-4970 N0 ₂ lsoxazol-3-yl CN cyclopropyl H

A-4971 N0 ₂ lsoxazol-3-yl CN OCH3 H

A-4972 N0 ₂ lsoxazol-3-yl CN OCF3 H

A-4973 N0 ₂ lsoxazol-3-yl CN SCH ₃ H

A-4974 N0 ₂ lsoxazol-3-yl CN SOCH3 H

A-4975 N0 ₂ lsoxazol-3-yl CN SO2CH3 H

A-4976 N0 ₂ lsoxazol-3-yl CN CH2OCH3 H

A-4977 N0 ₂ lsoxazol-3-yl H H CN

A-4978 N0 ₂ lsoxazol-3-yl H H N0 ₂ A-4979 N0 ₂ lsoxazol-3-yl H H cyclopropyl

A-4980 N0 ₂ lsoxazol-3-yl H H OCH3

A-4981 N0 ₂ lsoxazol-3-yl H H OCF3

A-4982 N0 ₂ lsoxazol-3-yl H H SCH ₃

A-4983 N0 ₂ lsoxazol-3-yl H H SOCH3

A-4984 N0 ₂ lsoxazol-3-yl H H SO2CH3

A-4985 N0 ₂ lsoxazol-3-yl H H CH2OCH3

A-4986 N0 ₂ lsoxazol-3-yl H cyclopropyl H

A-4987 N0 ₂ lsoxazol-3-yl H OCH3 H

A-4988 N0 ₂ lsoxazol-3-yl H OCF3 H

A-4989 N0 ₂ lsoxazol-3-yl H SCHs H

A-4990 N0 ₂ lsoxazol-3-yl H SOCH3 H

A-4991 N0 ₂ lsoxazol-3-yl H SO2CH3 H

A-4992 N0 ₂ lsoxazol-3-yl H CH2OCH3 H

A-4993 N0 ₂ 5-Me-lsoxazol-3-yl CI H CN

A-4994 N0 ₂ 5-Me-lsoxazol-3-yl CI H N0 ₂

A-4995 N0 ₂ 5-Me-lsoxazol-3-yl CI H cyclopropyl

A-4996 N0 ₂ 5-Me-lsoxazol-3-yl CI H OCH3

A-4997 N0 ₂ 5-Me-lsoxazol-3-yl CI H OCF3

A-4998 N0 ₂ 5-Me-lsoxazol-3-yl CI H SCH ₃

A-4999 N0 ₂ 5-Me-lsoxazol-3-yl CI H SOCH3

A-5000 N0 ₂ 5-Me-lsoxazol-3-yl CI H SO2CH3

A-5001 N0 ₂ 5-Me-lsoxazol-3-yl CI H CH2OCH3

A-5002 N0 ₂ 5-Me-lsoxazol-3-yl CI cyclopropyl H

A-5003 N0 ₂ 5-Me-lsoxazol-3-yl CI OCH3 H

A-5004 N0 ₂ 5-Me-lsoxazol-3-yl CI OCF3 H

A-5005 N0 ₂ 5-Me-lsoxazol-3-yl CI SCH ₃ H

A-5006 N0 ₂ 5-Me-lsoxazol-3-yl CI SOCH3 H

A-5007 N0 ₂ 5-Me-lsoxazol-3-yl CI SO2CH3 H

A-5008 N0 ₂ 5-Me-lsoxazol-3-yl CI CH2OCH3 H

A-5009 N0 ₂ 5-Me-lsoxazol-3-yl F H CN

A-5010 N0 ₂ 5-Me-lsoxazol-3-yl F H N0 ₂

A-501 1 N0 ₂ 5-Me-lsoxazol-3-yl F H cyclopropyl

A-5012 N0 ₂ 5-Me-lsoxazol-3-yl F H OCH3

A-5013 N0 ₂ 5-Me-lsoxazol-3-yl F H OCF3

A-5014 N0 ₂ 5-Me-lsoxazol-3-yl F H SCH ₃

A-5015 N0 ₂ 5-Me-lsoxazol-3-yl F H SOCH3 A-5016 N0 ₂ 5-Me-lsoxazol-3-yl F H SO2CH3

A-5017 N0 ₂ 5-Me-lsoxazol-3-yl F H CH2OCH3

A-5018 N0 ₂ 5-Me-lsoxazol-3-yl F cyclopropyl H

A-5019 N0 ₂ 5-Me-lsoxazol-3-yl F OCHs H

A-5020 N0 ₂ 5-Me-lsoxazol-3-yl F OCF3 H

A-5021 N0 ₂ 5-Me-lsoxazol-3-yl F SCHs H

A-5022 N0 ₂ 5-Me-lsoxazol-3-yl F SOCH3 H

A-5023 N0 ₂ 5-Me-lsoxazol-3-yl F SO2CH3 H

A-5024 N0 ₂ 5-Me-lsoxazol-3-yl F CH2OCH3 H

A-5025 N0 ₂ 5-Me-lsoxazol-3-yl CFs H CN

A-5026 N0 ₂ 5-Me-lsoxazol-3-yl CFs H N0 ₂

A-5027 N0 ₂ 5-Me-lsoxazol-3-yl CFs H cyclopropyl

A-5028 N0 ₂ 5-Me-lsoxazol-3-yl CFs H OCHs

A-5029 N0 ₂ 5-Me-lsoxazol-3-yl CFs H OCFs

A-5030 N0 ₂ 5-Me-lsoxazol-3-yl CFs H SCHs

A-5031 N0 ₂ 5-Me-lsoxazol-3-yl CFs H SOCHs

A-5032 N0 ₂ 5-Me-lsoxazol-3-yl CFs H SO2CH3

A-5033 N0 ₂ 5-Me-lsoxazol-3-yl CFs H CH2OCH3

A-5034 N0 ₂ 5-Me-lsoxazol-3-yl CFs cyclopropyl H

A-5035 N0 ₂ 5-Me-lsoxazol-3-yl CFs OCHs H

A-5036 N0 ₂ 5-Me-lsoxazol-3-yl CFs OCF3 H

A-5037 N0 ₂ 5-Me-lsoxazol-3-yl CFs SCHs H

A-5038 N0 ₂ 5-Me-lsoxazol-3-yl CFs SOCH3 H

A-5039 N0 ₂ 5-Me-lsoxazol-3-yl CFs SO2CH3 H

A-5040 N0 ₂ 5-Me-lsoxazol-3-yl CFs CH2OCH3 H

A-5041 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 H CN

A-5042 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 H N0 ₂

A-5043 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 H cyclopropyl

A-5044 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 H OCHs

A-5045 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 H OCFs

A-5046 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 H SCHs

A-5047 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 H SOCHs

A-5048 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 H SO2CH3

A-5049 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 H CH2OCH3

A-5050 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 cyclopropyl H

A-5051 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 OCHs H

A-5052 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 OCF3 H A-5053 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 SCH ₃ H

A-5054 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 SOCH3 H

A-5055 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 SO2CH3 H

A-5056 N0 ₂ 5-Me-lsoxazol-3-yl SO2CH3 CH2OCH3 H

A-5057 N0 ₂ 5-Me-lsoxazol-3-yl CN H CN

A-5058 N0 ₂ 5-Me-lsoxazol-3-yl CN H N0 ₂

A-5059 N0 ₂ 5-Me-lsoxazol-3-yl CN H cyclopropyl

A-5060 N0 ₂ 5-Me-lsoxazol-3-yl CN H OCH3

A-5061 N0 ₂ 5-Me-lsoxazol-3-yl CN H OCF3

A-5062 N0 ₂ 5-Me-lsoxazol-3-yl CN H SCH ₃

A-5063 N0 ₂ 5-Me-lsoxazol-3-yl CN H SOCH3

A-5064 N0 ₂ 5-Me-lsoxazol-3-yl CN H SO2CH3

A-5065 N0 ₂ 5-Me-lsoxazol-3-yl CN H CH2OCH3

A-5066 N0 ₂ 5-Me-lsoxazol-3-yl CN cyclopropyl H

A-5067 N0 ₂ 5-Me-lsoxazol-3-yl CN OCH3 H

A-5068 N0 ₂ 5-Me-lsoxazol-3-yl CN OCF3 H

A-5069 N0 ₂ 5-Me-lsoxazol-3-yl CN SCH ₃ H

A-5070 N0 ₂ 5-Me-lsoxazol-3-yl CN SOCH3 H

A-5071 N0 ₂ 5-Me-lsoxazol-3-yl CN SO2CH3 H

A-5072 N0 ₂ 5-Me-lsoxazol-3-yl CN CH2OCH3 H

A-5073 N0 ₂ 5-Me-lsoxazol-3-yl H H CN

A-5074 N0 ₂ 5-Me-lsoxazol-3-yl H H N0 ₂

A-5075 N0 ₂ 5-Me-lsoxazol-3-yl H H cyclopropyl

A-5076 N0 ₂ 5-Me-lsoxazol-3-yl H H OCH3

A-5077 N0 ₂ 5-Me-lsoxazol-3-yl H H OCF3

A-5078 N0 ₂ 5-Me-lsoxazol-3-yl H H SCH ₃

A-5079 N0 ₂ 5-Me-lsoxazol-3-yl H H SOCH3

A-5080 N0 ₂ 5-Me-lsoxazol-3-yl H H SO2CH3

A-5081 N0 ₂ 5-Me-lsoxazol-3-yl H H CH2OCH3

A-5082 N0 ₂ 5-Me-lsoxazol-3-yl H cyclopropyl H

A-5083 N0 ₂ 5-Me-lsoxazol-3-yl H OCH3 H

A-5084 N0 ₂ 5-Me-lsoxazol-3-yl H OCF3 H

A-5085 N0 ₂ 5-Me-lsoxazol-3-yl H SCH ₃ H

A-5086 N0 ₂ 5-Me-lsoxazol-3-yl H SOCH3 H

A-5087 N0 ₂ 5-Me-lsoxazol-3-yl H SO2CH3 H

A-5088 N0 ₂ 5-Me-lsoxazol-3-yl H CH2OCH3 H

A-5089 N0 ₂ 3-Me-lsoxazolin-5-yl CI H CN A-5090 N0 ₂ 3-Me-lsoxazolin-5-yl CI H N0 ₂

A-5091 N0 ₂ 3-Me-lsoxazolin-5-yl CI H cyclopropyl

A-5092 N0 ₂ 3-Me-lsoxazolin-5-yl CI H OCHs

A-5093 N0 ₂ 3-Me-lsoxazolin-5-yl CI H OCFs

A-5094 N0 ₂ 3-Me-lsoxazolin-5-yl CI H SCHs

A-5095 N0 ₂ 3-Me-lsoxazolin-5-yl CI H SOCHs

A-5096 N0 ₂ 3-Me-lsoxazolin-5-yl CI H SO2CH3

A-5097 N0 ₂ 3-Me-lsoxazolin-5-yl CI H CH2OCH3

A-5098 N0 ₂ 3-Me-lsoxazolin-5-yl CI cyclopropyl H

A-5099 N0 ₂ 3-Me-lsoxazolin-5-yl CI OCHs H

A-5100 N0 ₂ 3-Me-lsoxazolin-5-yl CI OCFs H

A-5101 N0 ₂ 3-Me-lsoxazolin-5-yl CI SCHs H

A-5102 N0 ₂ 3-Me-lsoxazolin-5-yl CI SOCHs H

A-5103 N0 ₂ 3-Me-lsoxazolin-5-yl CI SO2CH3 H

A-5104 N0 ₂ 3-Me-lsoxazolin-5-yl CI CH2OCH3 H

A-5105 N0 ₂ 3-Me-lsoxazolin-5-yl F H CN

A-5106 N0 ₂ 3-Me-lsoxazolin-5-yl F H N0 ₂

A-5107 N0 ₂ 3-Me-lsoxazolin-5-yl F H cyclopropyl

A-5108 N0 ₂ 3-Me-lsoxazolin-5-yl F H OCHs

A-5109 N0 ₂ 3-Me-lsoxazolin-5-yl F H OCFs

A-5110 N0 ₂ 3-Me-lsoxazolin-5-yl F H SCHs

A-511 1 N0 ₂ 3-Me-lsoxazolin-5-yl F H SOCHs

A-5112 N0 ₂ 3-Me-lsoxazolin-5-yl F H SO2CH3

A-5113 N0 ₂ 3-Me-lsoxazolin-5-yl F H CH2OCH3

A-5114 N0 ₂ 3-Me-lsoxazolin-5-yl F cyclopropyl H

A-5115 N0 ₂ 3-Me-lsoxazolin-5-yl F OCHs H

A-5116 N0 ₂ 3-Me-lsoxazolin-5-yl F OCFs H

A-5117 N0 ₂ 3-Me-lsoxazolin-5-yl F SCHs H

A-5118 N0 ₂ 3-Me-lsoxazolin-5-yl F SOCHs H

A-5119 N0 ₂ 3-Me-lsoxazolin-5-yl F SO2CH3 H

A-5120 N0 ₂ 3-Me-lsoxazolin-5-yl F CH2OCH3 H

A-5121 N0 ₂ 3-Me-lsoxazolin-5-yl CFs H CN

A-5122 N0 ₂ 3-Me-lsoxazolin-5-yl CFs H N0 ₂

A-5123 N0 ₂ 3-Me-lsoxazolin-5-yl CFs H cyclopropyl

A-5124 N0 ₂ 3-Me-lsoxazolin-5-yl CFs H OCHs

A-5125 N0 ₂ 3-Me-lsoxazolin-5-yl CFs H OCFs

A-5126 N0 ₂ 3-Me-lsoxazolin-5-yl CFs H SCHs A-5127 N0 ₂ 3-Me-lsoxazolin-5-yl CFs H SOCH3

A-5128 N0 ₂ 3-Me-lsoxazolin-5-yl CFs H SO2CH3

A-5129 N0 ₂ 3-Me-lsoxazolin-5-yl CFs H CH2OCH3

A-5130 N0 ₂ 3-Me-lsoxazolin-5-yl CFs cyclopropyl H

A-5131 N0 ₂ 3-Me-lsoxazolin-5-yl CFs OCHs H

A-5132 N0 ₂ 3-Me-lsoxazolin-5-yl CFs OCF3 H

A-5133 N0 ₂ 3-Me-lsoxazolin-5-yl CFs SCHs H

A-5134 N0 ₂ 3-Me-lsoxazolin-5-yl CFs SOCH3 H

A-5135 N0 ₂ 3-Me-lsoxazolin-5-yl CFs SO2CH3 H

A-5136 N0 ₂ 3-Me-lsoxazolin-5-yl CFs CH2OCH3 H

A-5137 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 H CN

A-5138 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 H N0 ₂

A-5139 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 H cyclopropyl

A-5140 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 H OCHs

A-5141 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 H OCF3

A-5142 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 H SCHs

A-5143 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 H SOCH3

A-5144 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 H SO2CH3

A-5145 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 H CH2OCH3

A-5146 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 cyclopropyl H

A-5147 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 OCHs H

A-5148 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 OCF3 H

A-5149 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 SCHs H

A-5150 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 SOCH3 H

A-5151 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 SO2CH3 H

A-5152 N0 ₂ 3-Me-lsoxazolin-5-yl SO2CH3 CH2OCH3 H

A-5153 N0 ₂ 3-Me-lsoxazolin-5-yl CN H CN

A-5154 N0 ₂ 3-Me-lsoxazolin-5-yl CN H N0 ₂

A-5155 N0 ₂ 3-Me-lsoxazolin-5-yl CN H cyclopropyl

A-5156 N0 ₂ 3-Me-lsoxazolin-5-yl CN H OCHs

A-5157 N0 ₂ 3-Me-lsoxazolin-5-yl CN H OCF3

A-5158 N0 ₂ 3-Me-lsoxazolin-5-yl CN H SCHs

A-5159 N0 ₂ 3-Me-lsoxazolin-5-yl CN H SOCH3

A-5160 N0 ₂ 3-Me-lsoxazolin-5-yl CN H SO2CH3

A-5161 N0 ₂ 3-Me-lsoxazolin-5-yl CN H CH2OCH3

A-5162 N0 ₂ 3-Me-lsoxazolin-5-yl CN cyclopropyl H

A-5163 N0 ₂ 3-Me-lsoxazolin-5-yl CN OCHs H A-5164 N0 ₂ 3-Me-lsoxazolin-5-yl CN 0CF3 H

A-5165 N0 ₂ 3-Me-lsoxazolin-5-yl CN SCHs H

A-5166 N0 ₂ 3-Me-lsoxazolin-5-yl CN SOCH3 H

A-5167 N0 ₂ 3-Me-lsoxazolin-5-yl CN SO2CH3 H

A-5168 N0 ₂ 3-Me-lsoxazolin-5-yl CN CH2OCH3 H

A-5169 N0 ₂ 3-Me-lsoxazolin-5-yl H H CN

A-5170 N0 ₂ 3-Me-lsoxazolin-5-yl H H N0 ₂

A-5171 N0 ₂ 3-Me-lsoxazolin-5-yl H H cyclopropyl

A-5172 N0 ₂ 3-Me-lsoxazolin-5-yl H H OCH3

A-5173 N0 ₂ 3-Me-lsoxazolin-5-yl H H OCF3

A-5174 N0 ₂ 3-Me-lsoxazolin-5-yl H H SCH ₃

A-5175 N0 ₂ 3-Me-lsoxazolin-5-yl H H SOCH3

A-5176 N0 ₂ 3-Me-lsoxazolin-5-yl H H SO2CH3

A-5177 N0 ₂ 3-Me-lsoxazolin-5-yl H H CH2OCH3

A-5178 N0 ₂ 3-Me-lsoxazolin-5-yl H cyclopropyl H

A-5179 N0 ₂ 3-Me-lsoxazolin-5-yl H OCH3 H

A-5180 N0 ₂ 3-Me-lsoxazolin-5-yl H OCF3 H

A-5181 N0 ₂ 3-Me-lsoxazolin-5-yl H SCH ₃ H

A-5182 N0 ₂ 3-Me-lsoxazolin-5-yl H SOCH3 H

A-5183 N0 ₂ 3-Me-lsoxazolin-5-yl H SO2CH3 H

A-5184 N0 ₂ 3-Me-lsoxazolin-5-yl H CH2OCH3 H

A-5185 N0 ₂ 3-Me-lsoxazol-5-yl CI H CN

A-5186 N0 ₂ 3-Me-lsoxazol-5-yl CI H N0 ₂

A-5187 N0 ₂ 3-Me-lsoxazol-5-yl CI H cyclopropyl

A-5188 N0 ₂ 3-Me-lsoxazol-5-yl CI H OCH3

A-5189 N0 ₂ 3-Me-lsoxazol-5-yl CI H OCF3

A-5190 N0 ₂ 3-Me-lsoxazol-5-yl CI H SCH ₃

A-5191 N0 ₂ 3-Me-lsoxazol-5-yl CI H SOCH3

A-5192 N0 ₂ 3-Me-lsoxazol-5-yl CI H SO2CH3

A-5193 N0 ₂ 3-Me-lsoxazol-5-yl CI H CH2OCH3

A-5194 N0 ₂ 3-Me-lsoxazol-5-yl CI cyclopropyl H

A-5195 N0 ₂ 3-Me-lsoxazol-5-yl CI OCH3 H

A-5196 N0 ₂ 3-Me-lsoxazol-5-yl CI OCF3 H

A-5197 N0 ₂ 3-Me-lsoxazol-5-yl CI SCH ₃ H

A-5198 N0 ₂ 3-Me-lsoxazol-5-yl CI SOCH3 H

A-5199 N0 ₂ 3-Me-lsoxazol-5-yl CI SO2CH3 H

A-5200 N0 ₂ 3-Me-lsoxazol-5-yl CI CH2OCH3 H A-5201 N0 ₂ 3-Me-lsoxazol-5-yl F H CN

A-5202 N0 ₂ 3-Me-lsoxazol-5-yl F H N0 ₂

A-5203 N0 ₂ 3-Me-lsoxazol-5-yl F H cyclopropyl

A-5204 N0 ₂ 3-Me-lsoxazol-5-yl F H OCH3

A-5205 N0 ₂ 3-Me-lsoxazol-5-yl F H OCFs

A-5206 N0 ₂ 3-Me-lsoxazol-5-yl F H SCHs

A-5207 N0 ₂ 3-Me-lsoxazol-5-yl F H SOCHs

A-5208 N0 ₂ 3-Me-lsoxazol-5-yl F H SO2CH3

A-5209 N0 ₂ 3-Me-lsoxazol-5-yl F H CH2OCH3

A-5210 N0 ₂ 3-Me-lsoxazol-5-yl F cyclopropyl H

A-521 1 N0 ₂ 3-Me-lsoxazol-5-yl F OCH3 H

A-5212 N0 ₂ 3-Me-lsoxazol-5-yl F OCFs H

A-5213 N0 ₂ 3-Me-lsoxazol-5-yl F SCHs H

A-5214 N0 ₂ 3-Me-lsoxazol-5-yl F SOCHs H

A-5215 N0 ₂ 3-Me-lsoxazol-5-yl F SO2CH3 H

A-5216 N0 ₂ 3-Me-lsoxazol-5-yl F CH2OCH3 H

A-5217 N0 ₂ 3-Me-lsoxazol-5-yl CFs H CN

A-5218 N0 ₂ 3-Me-lsoxazol-5-yl CFs H N0 ₂

A-5219 N0 ₂ 3-Me-lsoxazol-5-yl CFs H cyclopropyl

A-5220 N0 ₂ 3-Me-lsoxazol-5-yl CFs H OCH3

A-5221 N0 ₂ 3-Me-lsoxazol-5-yl CFs H OCFs

A-5222 N0 ₂ 3-Me-lsoxazol-5-yl CFs H SCHs

A-5223 N0 ₂ 3-Me-lsoxazol-5-yl CFs H SOCHs

A-5224 N0 ₂ 3-Me-lsoxazol-5-yl CFs H SO2CH3

A-5225 N0 ₂ 3-Me-lsoxazol-5-yl CFs H CH2OCH3

A-5226 N0 ₂ 3-Me-lsoxazol-5-yl CFs cyclopropyl H

A-5227 N0 ₂ 3-Me-lsoxazol-5-yl CFs OCH3 H

A-5228 N0 ₂ 3-Me-lsoxazol-5-yl CFs OCFs H

A-5229 N0 ₂ 3-Me-lsoxazol-5-yl CFs SCHs H

A-5230 N0 ₂ 3-Me-lsoxazol-5-yl CFs SOCHs H

A-5231 N0 ₂ 3-Me-lsoxazol-5-yl CFs SO2CH3 H

A-5232 N0 ₂ 3-Me-lsoxazol-5-yl CFs CH2OCH3 H

A-5233 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 H CN

A-5234 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 H N0 ₂

A-5235 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 H cyclopropyl

A-5236 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 H OCH3

A-5237 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 H OCFs A-5238 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 H SCH ₃

A-5239 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 H SOCH3

A-5240 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 H SO2CH3

A-5241 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 H CH2OCH3

A-5242 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 cyclopropyl H

A-5243 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 OCH3 H

A-5244 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 OCF3 H

A-5245 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 SCH ₃ H

A-5246 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 SOCH3 H

A-5247 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 SO2CH3 H

A-5248 N0 ₂ 3-Me-lsoxazol-5-yl SO2CH3 CH2OCH3 H

A-5249 N0 ₂ 3-Me-lsoxazol-5-yl CN H CN

A-5250 N0 ₂ 3-Me-lsoxazol-5-yl CN H N0 ₂

A-5251 N0 ₂ 3-Me-lsoxazol-5-yl CN H cyclopropyl

A-5252 N0 ₂ 3-Me-lsoxazol-5-yl CN H OCH3

A-5253 N0 ₂ 3-Me-lsoxazol-5-yl CN H OCF3

A-5254 N0 ₂ 3-Me-lsoxazol-5-yl CN H SCH ₃

A-5255 N0 ₂ 3-Me-lsoxazol-5-yl CN H SOCH3

A-5256 N0 ₂ 3-Me-lsoxazol-5-yl CN H SO2CH3

A-5257 N0 ₂ 3-Me-lsoxazol-5-yl CN H CH2OCH3

A-5258 N0 ₂ 3-Me-lsoxazol-5-yl CN cyclopropyl H

A-5259 N0 ₂ 3-Me-lsoxazol-5-yl CN OCH3 H

A-5260 N0 ₂ 3-Me-lsoxazol-5-yl CN OCF3 H

A-5261 N0 ₂ 3-Me-lsoxazol-5-yl CN SCH ₃ H

A-5262 N0 ₂ 3-Me-lsoxazol-5-yl CN SOCH3 H

A-5263 N0 ₂ 3-Me-lsoxazol-5-yl CN SO2CH3 H

A-5264 N0 ₂ 3-Me-lsoxazol-5-yl CN CH2OCH3 H

A-5265 N0 ₂ 3-Me-lsoxazol-5-yl H H CN

A-5266 N0 ₂ 3-Me-lsoxazol-5-yl H H N0 ₂

A-5267 N0 ₂ 3-Me-lsoxazol-5-yl H H cyclopropyl

A-5268 N0 ₂ 3-Me-lsoxazol-5-yl H H OCH3

A-5269 N0 ₂ 3-Me-lsoxazol-5-yl H H OCF3

A-5270 N0 ₂ 3-Me-lsoxazol-5-yl H H SCH ₃

A-5271 N0 ₂ 3-Me-lsoxazol-5-yl H H SOCH3

A-5272 N0 ₂ 3-Me-lsoxazol-5-yl H H SO2CH3

A-5273 N0 ₂ 3-Me-lsoxazol-5-yl H H CH2OCH3

A-5274 N0 ₂ 3-Me-lsoxazol-5-yl H cyclopropyl H A-5275 N0 ₂ 3-Me-lsoxazol-5-yl H OCH3 H

A-5276 N0 ₂ 3-Me-lsoxazol-5-yl H OCF3 H

A-5277 N0 ₂ 3-Me-lsoxazol-5-yl H SCHs H

A-5278 N0 ₂ 3-Me-lsoxazol-5-yl H SOCH3 H

A-5279 N0 ₂ 3-Me-lsoxazol-5-yl H SO2CH3 H

A-5280 N0 ₂ 3-Me-lsoxazol-5-yl H CH2OCH3 H

The compounds of formula I can be prepared by standard methods of organic chemistry, e.g. by the methods described hereinafter in schemes 1 to 8. The substituents, variables and indices in schemes 1 to 8 are as defined above for formula I, if not otherwise specified.

The compounds of formula I can be prepared analogous to Scheme 1 below.

Scheme 1 :

(III) (ll) (I)

5-Amino-1 -R-1 ,2,4-triazole or 5-amino-1 -R-tetrazole compounds of formula III can be reacted with benzoyl derivatives of formula II to afford compounds of formula I. X is a leaving group, such as halogen, in particular CI, an anhydride residue or an active ester residue. Especially in case of X being halogen the reaction is suitably carried out in the presence of a base. Suitable bases are for example carbonates, such as lithium, sodium or potassium carbonates, amines, such as trimethylamine or triethylamine, and basic N-heterocycles, such as pyridine, 2,6- dimethylpyridine or 2,4,6-trimethylpyridine. Suitable solvents are in particular aprotic solvents such as pentane, hexane, heptane, octane, cyclohexane, dichloromethane, chloroform, 1 ,2- dichlorethane, benzene, chlorobenzene, toluene, the xylenes, dichlorobenzene, trimethylben- zene, pyridine, 2,6-dimethylpyridine, 2,4,6-trimethylpyridine, acetonitrile, diethyl ether, tetrahy- drofuran, 2-methyl tetrahydrofuran, methyl tert-butylether, 1 ,4-dioxane, Ν,Ν-dimethyl formamide, N-methyl pyrrolidinone or mixtures thereof. The starting materials are generally reacted with one another in equimolar or nearly equimolar amounts at a reaction temperature usually in the range of -20°C to 100°C and preferably in the range of -5°C to 50°C.

Alternatively, compounds of formula I can also be prepared as shown in Scheme 2. Reaction of 5-amino-1 -R-1 ,2,4-triazole or 5-amino-1 -R-tetrazole of formula III with a benzoic acid derivative of formula IV yields compound I. The reaction is preferably carried out in the presence of a suitable activating agent, which converts the acid group of compound IV into an activated ester or amide. For this purpose activating agents known in the art, such as

1 ,1 ',carbonyldiimidazole (CDI), dicyclohexyl carbodiimide (DCC), 1 -ethyl-3-(3- dimethylaminopropyl)carbodiimide (EDC) or 2,4,6-tripropyl-1 ,3,5,2,4,6-trioxatriphosphorinane- 2,4,6-trioxide (T3P) can be employed. The activated ester or amide can be formed, depending in particular on the specific activating agent used, either in situ by contacting compound IV with the activating agent in the presence of compound III, or in a separate step prior to the reaction with compound III. It may be advantageous, especially in cases where DCC or EDC are used as activating agent, to include further additives in the activating reaction, such as hydroxybenzotri- azole (HOBt), nitrophenol, pentafluorophenol, 2,4,5-trichlorophenol or N-hydroxysuccinimide. It may further be advantageous to prepare the activated ester or amide in the presence of a base, for example a tertiary amine. The activated ester or amide is either in situ or subsequently reacted with the amine of formula III to afford the amide of formula I. The reaction normally takes place in anhydrous inert solvents, such as chlorinated hydrocarbons, e.g. dichloromethane or dichloroethane, ethers, e.g. tetrahydrofuran or 1 ,4-dioxane or carboxamides, e.g. N,N- dimethylformamide, Ν,Ν-dimethylacetamide or N-methylpyrrolidone. The reaction is ordinarily carried out at temperatures in the range from -20°C to +25°C.

Scheme 2:

(III) (IV) (I)

The compounds of formula II and their respective benzoic acid precursors of formula IV can be purchased or can be prepared by processes known in the art or disclosed in the literature, e.g. in WO 9746530, WO 9831676, WO 9831681 , WO 2002/018352, WO 2000/003988, US

2007/0191335, US 6277847.

Furthermore, compounds of formula I, can be obtained by treating N-(1 H-1 ,2,4-triazol-5- yl)benzamides or N-(1 H-tetrazol-5-yl)benzamides of formula V with, for example, alkylating agents such as alkyl halides according to Scheme 3.

Scheme 3.

The 5-amino-1 -R-tetrazoles of formula III, where R is for example alkyl, are either commercially available or are obtainable according to methods known from the literature. For example, 5- amino-1 -R-tetrazole can be prepared from 5-aminotetrazole according to the method described in the Journal of the American Chemical Society, 1954, 76, 923-924 (Scheme 4).

Scheme 4.

(III)

Alternatively, 5-amino-1 -R-tetrazole compounds of formula III can be prepared according to the method described in the Journal of the American Chemical Society, 1954, 76, 88-89 (Scheme 5).

Scheme 5:

As shown in Scheme 6, 5-amino-1 -R-triazoles of formula III, where R is for example alkyl, are either commercially available or are obtainable according to methods described in the literature. For example, 5-amino-1 -R-triazole can be prepared from 5-aminotriazole according to the method described in Zeitschrift fur Chemie, 1990, 30, 12, 436-437.

Scheme 6:

(III)

5-Amino-1 -R-triazole compounds of formula III, can also be prepared analogous to the synthesis described in Chemische Berichte, 1964, 97, 2, 396-404, as shown in Scheme 7.

Scheme 7:

H ₂ N

Alternatively, 5-amino-1 -R-triazoles of formula III, can be prepared according to the synthesis described in Angewandte Chemie, 1963, 75, 918 (Scheme 8).

Scheme 8

'

As a rule, the compounds of formula I including their stereoisomers, salts, tautomers and N-oxides, and their precursors in the synthesis process, can be prepared by the methods described above. If individual compounds can not be prepared via the above-described routes, they can be prepared by derivatization of other compounds of formula I or the respective pre- cursor or by customary modifications of the synthesis routes described. For example, in individual cases, certain compounds of formula I can advantageously be prepared from other compounds of formula I by derivatization, e.g. by ester hydrolysis, amidation, esterification, ether cleavage, olefination, reduction, oxidation and the like, or by customary modifications of the syn- thesis routes described.

The reaction mixtures are worked up in the customary manner, for example by mixing with water, separating the phases, and, if appropriate, purifying the crude products by chromatography, for example on alumina or on silica gel. Some of the intermediates and end products may be obtained in the form of colorless or pale brown viscous oils which are freed or purified from volatile components under reduced pressure and at moderately elevated temperature. If the intermediates and end products are obtained as solids, they may be purified by recrystalliza- tion or trituration.

The compounds of formula I and their agriculturally suitable salts are useful as herbicides. They are useful as such or as an appropriately formulated composition. The herbicidal compositions comprising the compound I, in particular the preferred aspects thereof, control vegetation on non-crop areas very efficiently, especially at high rates of application. They act against broad-leaved weeds and weed grasses in crops such as wheat, rice, corn, soybeans and cotton without causing any significant damage to the crop plants. This effect is mainly observed at low rates of application.

Depending on the application method in question, the compounds of formula I, in particular the preferred aspects thereof, or compositions comprising them can additionally be employed in a further number of crop plants for eliminating unwanted plants. Examples of suitable crops are the following:

Allium cepa, Ananas comosus, Arachis hypogaea, Asparagus officinalis, Avena sativa,

Beta vulgaris spec, altissima, Beta vulgaris spec, rapa, Brassica napus var. napus, Brassica napus var. napobrassica, Brassica rapa var. silvestris, Brassica oleracea, Brassica nigra, Camellia sinensis, Carthamus tinctorius, Carya illinoinensis, Citrus limon, Citrus sinensis, Coffea arabica (Coffea canephora, Coffea liberica), Cucumis sativus, Cynodon dactylon, Daucus caro- ta, Elaeis guineensis, Fragaria vesca, Glycine max, Gossypium hirsutum, (Gossypium arbo- reum, Gossypium herbaceum, Gossypium vitifolium), Helianthus annuus, Hevea brasiliensis, Hordeum vulgare, Humulus lupulus, Ipomoea batatas, Juglans regia, Lens culinaris, Linum usi- tatissimum, Lycopersicon lycopersicum, Malus spec, Manihot esculenta, Medicago sativa, Mu- sa spec, Nicotiana tabacum (N.rustica), Olea europaea, Oryza sativa, Phaseolus lunatus, Phaseolus vulgaris, Picea abies, Pinus spec, Pistacia vera, Pisum sativum, Prunus avium, Prunus persica, Pyrus communis, Prunus armeniaca, Prunus cerasus, Prunus dulcis and Prunus domestica, Ribes sylvestre, Ricinus communis, Saccharum officinarum, Secale cereale, Sinapis alba, Solanum tuberosum, Sorghum bicolor (s. vulgare), Theobroma cacao, Trifolium pratense, Triticum aestivum, Triticale, Triticum durum, Vicia faba, Vitis vinifera, Zea mays.

The term "crop plants" also includes plants which have been modified by breeding, mutagenesis or genetic engineering. Genetically modified plants are plants whose genetic material has been modified in a manner which does not occur under natural conditions by crossing, mutations or natural recombination (i.e. reassembly of the genetic information). Here, in general, one or more genes are integrated into the genetic material of the plant to improve the properties of the plant.

Accordingly, the term "crop plants" also includes plants which, by breeding and genetic engineering, have acquired tolerance to certain classes of herbicides, such as hydroxy- phenylpyruvate dioxygenase (HPPD) inhibitors, acetolactate synthase (ALS) inhibitors, such as, for example, sulfonylureas (EP-A-0257993, US 5,013,659) or imidazolinones (see, for example, US 6,222,100, WO 01/82685, WO 00/26390, WO 97/41218, WO 98/02526, WO 98/02527, WO 04/106529, WO 05/20673, WO 03/14357, WO 03/13225, WO 03/14356, WO 04/16073), enolpyruvylshikimate 3-phosphate synthase (EPSPS) inhibitors, such as, for example, glypho- sate (see, for example, WO 92/00377), glutamine synthetase (GS) inhibitors, such as, for example, glufosinate (see, for example, EP-A-0242236, EP-A-242246), or oxynil herbicides (see, for example, US 5,559,024).

Numerous crop plants, for example Clearfield® oilseed rape, tolerant to imidazolinones, for example imazamox, have been generated with the aid of classic breeding methods (mutagenesis). Crop plants such as soybeans, cotton, corn, beet and oilseed rape, resistant to glyphosate or glufosinate, which are available under the tradenames RoundupReady ^® (glypho- sate) and Liberty Link ^® (glufosinate) have been generated with the aid of genetic engineering methods.

Accordingly, the term "crop plants" also includes plants which, with the aid of genetic engineering, produce one or more toxins, for example those of the bacterial strain Bacillus ssp. Toxins which are produced by such genetically modified plants include, for example, insecticidal proteins of Bacillus spp., in particular B. thuringiensis, such as the endotoxins CrylAb, Cry1 Ac, Cry1 F, Cry1 Fa2, Cry2Ab, Cry3A, Cry3Bb1 , Cry9c, Cry34Ab1 or Cry35Ab1 ; or vegetative insec- ticidal proteins (VIPs), for example VIP1 , VIP2, VIP3, or VIP3A; insecticidal proteins of nema- tode-colonizing bacteria, for example Photorhabdus spp. or Xenorhabdus spp.; toxins of animal organisms, for example wasp, spider or scorpion toxins; fungal toxins, for example from Strep- tomycetes; plant lectins, for example from peas or barley; agglutinins; proteinase inhibitors, for example trypsin inhibitors, serine protease inhibitors, patatin, cystatin or papain inhibitors, ribo- some-inactivating proteins (RIPs), for example ricin, corn-RIP, abrin, luffin, saporin or bryodin; steroid-metabolizing enzymes, for example 3-hydroxysteroid oxidase, ecdysteroid-IDP glycosyl transferase, cholesterol oxidase, ecdysone inhibitors, or HMG-CoA reductase; ion channel blockers, for example inhibitors of sodium channels or calcium channels; juvenile hormone esterase; receptors of the diuretic hormone (helicokinin receptors); stilbene synthase, bibenzyl synthase, chitinases and glucanases. In the plants, these toxins may also be produced as pre- toxins, hybrid proteins or truncated or otherwise modified proteins. Hybrid proteins are characterized by a novel combination of different protein domains (see, for example, WO

2002/015701 ). Further examples of such toxins or genetically modified plants which produce these toxins are disclosed in EP-A 374 753, WO 93/007278, WO 95/34656, EP-A 427 529, EP- A 451 878, WO 03/018810 and WO 03/052073. The methods for producing these genetically modified plants are known to the person skilled in the art and disclosed, for example, in the publications mentioned above. Numerous of the toxins mentioned above bestow, upon the plants by which they are produced, tolerance to pests from all taxonomic classes of arthropods, in particular to beetles (Coeleropta), dipterans (Diptera) and butterflies (Lepidoptera) and to nema- todes (Nematoda).

Genetically modified plants which produce one or more genes coding for insecticidal toxins are described, for example, in the publications mentioned above, and some of them are commercially available, such as, for example, YieldGard ^® (corn varieties producing the toxin CrylAb), YieldGard ^® Plus (corn varieties which produce the toxins CrylAb and Cry3Bb1 ), Star- link ^® (corn varieties which produce the toxin Cry9c), Herculex ^® RW (corn varieties which produce the toxins Cry34Ab1 , Cry35Ab1 and the enzyme phosphinothricin-N-acetyltransferase [PAT]); NuCOTN ^® 33B (cotton varieties which produce the toxin CrylAc), Bollgard ^® I (cotton varieties which produce the toxin CrylAc), Bollgard ^® II (cotton varieties which produce the toxins CrylAc and Cry2Ab2); VIPCOT ^® (cotton varieties which produce a VIP toxin); NewLeaf ^® (potato varieties which produce the toxin Cry3A); Bt-Xtra ^® , NatureGard ^® , KnockOut ^® , BiteGard ^® , Protecta ^® , Bt1 1 (for example Agrisure ^® CB) and Bt176 from Syngenta Seeds SAS, France (corn varieties which produce the toxin CrylAb and the PAT enyzme), MIR604 from Syngenta Seeds SAS, France (corn varieties which produce a modified version of the toxin Cry3A, see

WO 03/018810), MON 863 from Monsanto Europe S.A., Belgium (corn varieties which produce the toxin Cry3Bb1 ), IPC 531 from Monsanto Europe S.A., Belgium (cotton varieties which produce a modified version of the toxin CrylAc) and 1507 from Pioneer Overseas Corporation, Belgium (corn varieties which produce the toxin Cry1 F and the PAT enzyme).

Accordingly, the term "crop plants" also includes plants which, with the aid of genetic engineering, produce one or more proteins which are more robust or have increased resistance to bacterial, viral or fungal pathogens, such as, for example, pathogenesis-related proteins (PR proteins, see EP-A 0 392 225), resistance proteins (for example potato varieties producing two resistance genes against Phytophthora infestans from the wild Mexican potato Solanum bulbocastanum) or T4 lysozyme (for example potato cultivars which, by producing this protein, are resistant to bacteria such as Erwinia amylvora).

Accordingly, the term "crop plants" also includes plants whose productivity has been improved with the aid of genetic engineering methods, for example by enhancing the potential yield (for example biomass, grain yield, starch, oil or protein content), tolerance to drought, salt or other limiting environmental factors or resistance to pests and fungal, bacterial and viral pathogens.

The term "crop plants" also includes plants whose ingredients have been modified with the aid of genetic engineering methods in particular for improving human or animal diet, for ex- ample by oil plants producing health-promoting long-chain omega 3 fatty acids or monounsatu- rated omega 9 fatty acids (for example Nexera ^® oilseed rape).

The term "crop plants" also includes plants which have been modified with the aid of genetic engineering methods for improving the production of raw materials, for example by increasing the amylopectin content of potatoes (Amflora ^® potato).

Furthermore, it has been found that the compounds of formula I are also suitable for the defoliation and/or desiccation of plant parts, for which crop plants such as cotton, potato, oilseed rape, sunflower, soybean or field beans, in particular cotton, are suitable. In this regard, there have been found compositions for the desiccation and/or defoliation of plants, processes for preparing these compositions and methods for desiccating and/or defoliating plants using the compounds of formula I.

As desiccants, the compounds of formula I are particularly suitable for desiccating the above-ground parts of crop plants such as potato, oilseed rape, sunflower and soybean, but also cereals. This makes possible the fully mechanical harvesting of these important crop plants.

Also of economic interest is to facilitate harvesting, which is made possible by

concentrating within a certain period of time the dehiscence, or reduction of adhesion to the tree, in citrus fruit, olives and other species and varieties of pomaceous fruit, stone fruit and nuts. The same mechanism, i.e. the promotion of the development of abscission tissue between fruit part or leaf part and shoot part of the plants is also essential for the readily controllable defoliation of useful plants, in particular cotton.

Moreover, a shortening of the time interval in which the individual cotton plants mature leads to an increased fiber quality after harvesting.

The compounds of formula I, or the herbicidal compositions comprising the compounds of formula I, can be used, for example, in the form of ready-to-spray aqueous solutions, powders, suspensions, also highly concentrated aqueous, oily or other suspensions or dispersions, emulsions, oil dispersions, pastes, dusts, materials for broadcasting, or granules, by means of spraying, atomizing, dusting, spreading, watering or treatment of the seed or mixing with the seed. The use forms depend on the intended purpose; in each case, they should ensure the finest possible distribution of the active ingredients according to the invention.

The herbicidal compositions comprise a herbicidally effective amount of at least one compound of the formula I or an agriculturally useful salt of I, and auxiliaries which are customary for the formulation of crop protection agents.

Examples of auxiliaries customary for the formulation of crop protection agents are inert auxiliaries, solid carriers, surfactants (such as dispersants, protective colloids, emulsifiers, wetting agents and tackifiers), organic and inorganic thickeners, bactericides, antifreeze agents, antifoams, if appropriate colorants and, for seed formulations, adhesives.

Examples of thickeners (i.e. compounds which impart to the formulation modified flow properties, i.e. high viscosity in the state of rest and low viscosity in motion) are

polysaccharides, such as xanthan gum (Kelzan® from Kelco), Rhodopol® 23 (Rhone Poulenc) or Veegum® (from R.T. Vanderbilt), and also organic and inorganic sheet minerals, such as Attaclay® (from Engelhardt).

Examples of antifoams are silicone emulsions (such as, for example, Silikon ^® SRE,

Wacker or Rhodorsil® from Rhodia), long-chain alcohols, fatty acids, salts of fatty acids, organofluorine compounds and mixtures thereof.

Bactericides can be added for stabilizing the aqueous herbicidal formulation. Examples of bactericides are bactericides based on diclorophen and benzyl alcohol hemiformal (Proxel® from ICI or Acticide® RS from Thor Chemie and Kathon® MK from Rohm & Haas), and also isothiazolinone derivates, such as alkylisothiazolinones and benzisothiazolinones (Acticide MBS from Thor Chemie).

Examples of antifreeze agents are ethylene glycol, propylene glycol, urea or glycerol.

Examples of colorants are both sparingly water-soluble pigments and water-soluble dyes. Examples which may be mentioned are the dyes known under the names Rhodamin B, C.I. Pigment Red 1 12 and C.I. Solvent Red 1 , and also pigment blue 15:4, pigment blue 15:3, pigment blue 15:2, pigment blue 15:1 , pigment blue 80, pigment yellow 1 , pigment yellow 13, pigment red 1 12, pigment red 48:2, pigment red 48:1 , pigment red 57:1 , pigment red 53:1 , pigment orange 43, pigment orange 34, pigment orange 5, pigment green 36, pigment green 7, pigment white 6, pigment brown 25, basic violet 10, basic violet 49, acid red 51 , acid red 52, acid red 14, acid blue 9, acid yellow 23, basic red 10, basic red 108.

Examples of adhesives are polyvinylpyrrolidone, polyvinyl acetate, polyvinyl alcohol and tylose.

Suitable inert auxiliaries are, for example, the following:

mineral oil fractions of medium to high boiling point, such as kerosene and diesel oil, furthermore coal tar oils and oils of vegetable or animal origin, aliphatic, cyclic and aromatic hydrocarbons, for example paraffin, tetrahydronaphthalene, alkylated naphthalenes and their derivatives, alkylated benzenes and their derivatives, alcohols such as methanol, ethanol, propanol, butanol and cyclohexanol, ketones such as cyclohexanone or strongly polar solvents, for example amines such as N-methylpyrrolidone, and water.

Solid carriers are mineral earths such as silicas, silica gels, silicates, talc, kaolin, limestone, lime, chalk, bole, loess, clay, dolomite, diatomaceous earth, calcium sulfate, magnesium sulfate and magnesium oxide, ground synthetic materials, fertilizers such as ammonium sulfate, ammonium phosphate, ammonium nitrate and ureas, and products of vegetable origin, such as cereal meal, tree bark meal, wood meal and nutshell meal, cellulose powders, or other solid carriers.

Suitable surfactants (adjuvants, wetting agents, tackifiers, dispersants and also

emulsifiers) are the alkali metal salts, alkaline earth metal salts and ammonium salts of aromatic sulfonic acids, for example lignosulfonic acids (e.g. Borrespers-types, Borregaard),

phenolsulfonic acids, naphthalenesulfonic acids (Morwet types, Akzo Nobel) and

dibutylnaphthalenesulfonic acid (Nekal types, BASF SE), and of fatty acids, alkyl- and alkylarylsulfonates, alkyl sulfates, lauryl ether sulfates and fatty alcohol sulfates, and salts of sulfated hexa-, hepta- and octadecanols, and also of fatty alcohol glycol ethers, condensates of sulfonated naphthalene and its derivatives with formaldehyde, condensates of naphthalene or of the naphthalenesulfonic acids with phenol and formaldehyde, polyoxyethylene octylphenol ether, ethoxylated isooctyl-, octyl- or nonylphenol, alkylphenyl or tributylphenyl polyglycol ether, alkylaryl polyether alcohols, isotridecyl alcohol, fatty alcohol/ethylene oxide condensates, ethoxylated castor oil, polyoxyethylene alkyl ethers or polyoxypropylene alkyl ethers, lauryl alcohol polyglycol ether acetate, sorbitol esters, lignosulfite waste liquors and proteins, denatured proteins, polysaccharides (e.g. methylcellulose), hydrophobically modified starches, polyvinyl alcohol (Mowiol types Clariant), polycarboxylates (BASF SE, Sokalan types), polyalkoxylates, polyvinylamine (BASF SE, Lupamine types), polyethyleneimine (BASF SE, Lupasol types), polyvinylpyrrolidone and copolymers thereof.

Powders, materials for broadcasting and dusts can be prepared by mixing or grinding the active ingredients together with a solid carrier.

Granules, for example coated granules, impregnated granules and homogeneous granules, can be prepared by binding the active ingredients to solid carriers.

Aqueous use forms can be prepared from emulsion concentrates, suspensions, pastes, wettable powders or water-dispersible granules by adding water. To prepare emulsions, pastes or oil dispersions, the compounds of formula I or la, either as such or dissolved in an oil or solvent, can be homogenized in water by means of a wetting agent, tackifier, dispersant or emulsifier. Alternatively, it is also possible to prepare concentrates comprising active substance, wetting agent, tackifier, dispersant or emulsifier and, if desired, solvent or oil, which are suitable for dilution with water.

The concentrations of the compounds of formula I in the ready-to-use preparations can be varied within wide ranges. In general, the formulations comprise from 0.001 to 98% by weight, preferably 0.01 to 95% by weight of at least one active compound. The active compounds are employed in a purity of from 90% to 100%, preferably 95% to 100% (according to NMR spectrum).

The formulations or ready-to-use preparations may also comprise acids, bases or buffer systems, suitable examples being phosphoric acid or sulfuric acid, or urea or ammonia.

The compounds of formula I of the invention can for example be formulated as follows:

1 . Products for dilution with water

A. Water-soluble concentrates

10 parts by weight of active compound are dissolved in 90 parts by weight of water or a water-soluble solvent. As an alternative, wetters or other adjuvants are added. The active compound dissolves upon dilution with water. This gives a formulation with an active compound content of 10% by weight.

B. Dispersible concentrates

20 parts by weight of active compound are dissolved in 70 parts by weight of cyclohexa- none with addition of 10 parts by weight of a dispersant, for example polyvinylpyrrolidone. Dilution with water gives a dispersion. The active compound content is 20% by weight.

C. Emulsifiable concentrates

15 parts by weight of active compound are dissolved in 75 parts by weight of an organic solvent (e.g. alkylaromatics) with addition of calcium dodecylbenzenesulfonate and castor oil ethoxylate (in each case 5 parts by weight). Dilution with water gives an emulsion. The formulation has an active compound content of 15% by weight.

D. Emulsions

25 parts by weight of active compound are dissolved in 35 parts by weight of an organic solvent (e.g. alkylaromatics) with addition of calcium dodecylbenzenesulfonate and castor oil ethoxylate (in each case 5 parts by weight). This mixture is introduced into 30 parts by weight of water by means of an emulsifier (e.g. Ultraturrax) and made into a homogeneous emulsion. Dilution with water gives an emulsion. The formulation has an active compound content of 25% by weight.

E. Suspensions

In an agitated ball mill, 20 parts by weight of active compound are comminuted with addition of 10 parts by weight of dispersants and wetters and 70 parts by weight of water or an organic solvent to give a fine active compound suspension. Dilution with water gives a stable sus- pension of the active compound. The active compound content in the formulation is 20% by weight.

F. Water-dispersible granules and water-soluble granules 50 parts by weight of active compound are ground finely with addition of 50 parts by weight of dispersants and wetters and made into water-dispersible or water-soluble granules by means of technical appliances (for example extrusion, spray tower, fluidized bed). Dilution with water gives a stable dispersion or solution of the active compound. The formulation has an ac- tive compound content of 50% by weight.

G. Water-dispersible powders and water-soluble powders

75 parts by weight of active compound are ground in a rotor-stator mill with addition of 25 parts by weight of dispersants, wetters and silica gel. Dilution with water gives a stable dispersion or solution of the active compound. The active compound content of the formulation is 75% by weight.

H. Gel formulations

In a ball mill, 20 parts by weight of active compound, 10 parts by weight of dispersant, 1 part by weight of gelling agent and 70 parts by weight of water or of an organic solvent are ground to give a fine suspension. Dilution with water gives a stable suspension with active com- pound content of 20% by weight.

2. Products to be applied undiluted

I. Dusts

5 parts by weight of active compound are ground finely and mixed intimately with 95 parts by weight of finely divided kaolin. This gives a dusting powder with an active compound content of 5% by weight.

J. Granules (GR, FG, GG, MG)

0.5 parts by weight of active compound are ground finely and associated with 99.5 parts by weight of carriers. Current methods here are extrusion, spray-drying or the fluidized bed. This gives granules to be applied undiluted with an active compound content of 0.5% by weight.

K. ULV solutions (UL)

10 parts by weight of active compound are dissolved in 90 parts by weight of an organic solvent, for example xylene. This gives a product to be applied undiluted with an active compound content of 10% by weight.

The compounds of formula I or the herbicidal compositions comprising them can be applied pre- or post-emergence, or together with the seed of a crop plant. It is also possible to apply the herbicidal compositions or active compounds by applying seed, pretreated with the herbicidal compositions or active compounds, of a crop plant. If the active compounds are less well tolerated by certain crop plants, application techniques may be used in which the herbicidal compositions are sprayed, with the aid of the spraying equipment, in such a way that as far as possible they do not come into contact with the leaves of the sensitive crop plants, while the active compounds reach the leaves of undesirable plants growing underneath, or the bare soil surface (post-directed, lay-by).

In a further embodiment, the compounds of formula I or the herbicidal compositions can be applied by treating seed.

The treatment of seed comprises essentially all procedures familiar to the person skilled in the art (seed dressing, seed coating, seed dusting, seed soaking, seed film coating, seed multilayer coating, seed encrusting, seed dripping and seed pelleting) based on the compounds of formula I according to the invention or the compositions prepared therefrom. Here, the herbicid- al compositions can be applied diluted or undiluted.

The term seed comprises seed of all types, such as, for example, corns, seeds, fruits, tubers, cuttings and similar forms. Here, preferably, the term seed describes corns and seeds.

The seed used can be seed of the useful plants mentioned above, but also the seed of transgenic plants or plants obtained by customary breeding methods.

The rates of application of active compound are from 0.001 to 3.0, preferably 0.01 to 1.0, kg/ha of active substance (a.s.), depending on the control target, the season, the target plants and the growth stage. To treat the seed, the compounds of formula I are generally employed in amounts of from 0.001 to 10 kg per 100 kg of seed.

It may also be advantageous to use the compounds of formula I in combination with saf- eners. Safeners are chemical compounds which prevent or reduce damage to useful plants without substantially affecting the herbicidal action of the compounds of formula I on unwanted plants. They can be used both before sowing (for example in the treatment of seed, or on cut- tings or seedlings) and before or after the emergence of the useful plant. The safeners and the compounds of formula I can be used simultaneously or in succession.

Suitable safeners are, for example, (quinolin-8-oxy)acetic acids, 1 -phenyl-5-haloalkyl-1 H- 1 ,2,4-triazole-3-carboxylic acids, 1 -phenyl-4,5-dihydro-5-alkyl-1 H-pyrazole-3,5-dicarboxylic acids, 4,5-dihydro-5,5-diaryl-3-isoxazolecarboxylic acids, dichloroacetamides, alpha- oximinophenylacetonitriles, acetophenone oximes, 4,6-dihalo-2-phenylpyrimidines, N-[[4-

(aminocarbonyl)phenyl]sulfonyl]-2-benzamides, 1 ,8-naphthalic anhydride, 2-halo-4-(haloalkyl)-5- thiazolecarboxylic acids, phosphorothiolates and O-phenyl N-alkylcarbamates and their agriculturally useful salts and, provided that they have an acid function, their agriculturally useful derivatives, such as amides, esters and thioesters.

To broaden the activity spectrum and to obtain synergistic effects, the compounds of the formula I can be mixed and jointly applied with numerous representatives of other herbicidal or growth-regulating groups of active compounds or with safeners. Suitable mixing partners are, for example, 1 ,2,4-thiadiazoles, 1 ,3,4-thiadiazoles, amides, aminophosphoric acid and its derivatives, aminotriazoles, anilides, aryloxy/heteroaryloxyalkanoic acids and their derivatives, ben- zoic acid and its derivatives, benzothiadiazinones, 2-(hetaroyl/aroyl)-1 ,3-cyclohexanediones, heteroaryl aryl ketones, benzylisoxazolidinones, meta-CF3-phenyl derivatives, carbamates, quinoline carboxylic acid and its derivatives, chloroacetanilides, cyclohexenone oxime ether derivates, diazines, dichloropropionic acid and its derivatives, dihydrobenzofurans, dihydrofu- ran-3-ones, dinitroanilines, dinitrophenols, diphenyl ethers, dipyridyls, halocarboxylic acids and their derivatives, ureas, 3-phenyluracils, imidazoles, imidazolinones, N-phenyl-3,4,5,6- tetrahydrophthalimides, oxadiazoles, oxiranes, phenols, aryloxy- and heteroaryloxyphenoxypro- pionic esters, phenylacetic acid and its derivatives, 2-phenylpropionic acid and its derivatives, pyrazoles, phenylpyrazoles, pyridazines, pyridinecarboxylic acid and its derivatives, pyrimidyl ethers, sulfonamides, sulfonylureas, triazines, triazinones, triazolinones, triazolecarboxamides, uracils and also phenylpyrazolines and isoxazolines and their derivatives.

Moreover, it may be useful to apply the compounds of formula I alone or in combination with other herbicides or else also mixed with further crop protection agents, jointly, for example with compositions for controlling pests or phytopathogenic fungi or bacteria. Also of interest is the miscibility with mineral salt solutions which are employed for alleviating nutritional and trace element deficiencies. Other additives such as nonphytotoxic oils and oil concentrates may also be added.

Examples of herbicides which can be used in combination with the N-(tetrazol-5-yl)- and

N-(triazol-5-yl)arylcarboxamide compounds of formula I according to the present invention are: b1 ) from the group of the lipid biosynthesis inhibitors:

alloxydim, alloxydim-sodium, butroxydim, clethodim, clodinafop, clodinafop-propargyl, cy- cloxydim, cyhalofop, cyhalofop-butyl, diclofop, diclofop-methyl, fenoxaprop, fenoxaprop-ethyl, fenoxaprop-P, fenoxaprop-P-ethyl, fluazifop, fluazifop-butyl, fluazifop-P, fluazifop-P-butyl, halox- yfop, haloxyfop-methyl, haloxyfop-P, haloxyfop-P-methyl, metamifop, pinoxaden, profoxydim, propaquizafop, quizalofop, quizalofop-ethyl, quizalofop-tefuryl, quizalofop-P, quizalofop-P-ethyl, quizalofop-P-tefuryl, sethoxydim, tepraloxydim, tralkoxydim, benfuresate, butylate, cycloate, dalapon, dimepiperate, EPTC, esprocarb, ethofumesate, flupropanate, molinate, orbencarb, pebulate, prosulfocarb, TCA, thiobencarb, tiocarbazil, triallate and vernolate;

b2) from the group of the ALS inhibitors:

amidosulfuron, azimsulfuron, bensulfuron, bensulfuron-methyl, bispyribac, bispyribac- sodium, chlorimuron, chlorimuron-ethyl, chlorsulfuron, cinosulfuron, cloransulam, cloransulam- methyl, cyclosulfamuron, diclosulam, ethametsulfuron, ethametsulfuron-methyl, ethoxysulfuron, flazasulfuron, florasulam, flucarbazone, flucarbazone-sodium, flucetosulfuron, flumetsulam, flupyrsulfuron, flupyrsulfuron-methyl-sodium, foramsulfuron, halosulfuron, halosulfuron-methyl, imazamethabenz, imazamethabenz-methyl, imazamox, imazapic, imazapyr, imazaquin, ima- zethapyr, imazosulfuron, iodosulfuron, iodosulfuron-methyl-sodium, mesosulfuron, metosulam, metsulfuron, metsulfuron-methyl, nicosulfuron, orthosulfamuron, oxasulfuron, penoxsulam, primisulfuron, primisulfuron-methyl, propoxycarbazone, propoxycarbazone-sodium, prosulfuron, pyrazosulfuron, pyrazosulfuron-ethyl, pyribenzoxim, pyrimisulfan, pyriftalid, pyriminobac, pyrimi- nobac-methyl, pyrithiobac, pyrithiobac-sodium, pyroxsulam, rimsulfuron, sulfometuron, sulfome- turon-methyl, sulfosulfuron, thiencarbazone, thiencarbazone-methyl, thifensulfuron, thifensulfu- ron-methyl, triasulfuron, tribenuron, tribenuron-methyl, trifloxysulfuron, triflusulfuron, triflusulfu- ron-methyl and tritosulfuron;

b3) from the group of the photosynthesis inhibitors:

ametryn, amicarbazone, atrazine, bentazone, bentazone-sodium, bromacil, bromofenox- im, bromoxynil and its salts and esters, chlorobromuron, chloridazone, chlorotoluron, chloroxuron, cyanazine, desmedipham, desmetryn, dimefuron, dimethametryn, diquat, diquat- dibromide, diuron, fluometuron, hexazinone, ioxynil and its salts and esters, isoproturon, isouron, karbutilate, lenacil, linuron, metamitron, methabenzthiazuron, metobenzuron, me- toxuron, metribuzin, monolinuron, neburon, paraquat, paraquat-dichloride, paraquat- dimetilsulfate, pentanochlor, phenmedipham, phenmedipham-ethyl, prometon, prometryn, pro- panil, propazine, pyridafol, pyridate, siduron, simazine, simetryn, tebuthiuron, terbacil, ter- bumeton, terbuthylazine, terbutryn, thidiazuron and trietazine;

b4) from the group of the protoporphyrinogen-IX oxidase inhibitors: acifluorfen, acifluorfen-sodium, azafenidin, bencarbazone, benzfendizone, bifenox, bu- tafenacil, carfentrazone, carfentrazone-ethyl, chlomethoxyfen, cinidon-ethyl, fluazolate, flufenpyr, flufenpyr-ethyl, flumiclorac, flumiclorac-pentyl, flumioxazin, fluoroglycofen, fluorogly- cofen-ethyl, fluthiacet, fluthiacet-methyl, fomesafen, halosafen, lactofen, oxadiargyl, oxadiazon, oxyfluorfen, pentoxazone, profluazol, pyraclonil, pyraflufen, pyraflufen-ethyl, saflufenacil, sulfen- trazone, thidiazimin, 2-chloro-5-[3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluoromethy l)-1 (2H)- pyrimidinyl]-4-fluoro-N-[(isopropyl)methylsulfamoyl]benzamid e (H-1 ; CAS 372137-35-4), ethyl [3-[2-chloro-4-fluoro-5-(1 -methyl-6-trifluoromethyl-2,4-dioxo-1 ,2,3,4-tetrahydropyrimidin-3- yl)phenoxy]-2-pyridyloxy]acetate (H-2; CAS 353292-31 -6), N-ethyl-3-(2,6-dichloro-4-trifluoro- methylphenoxy)-5-methyl-1 H-pyrazole-1 -carboxamide (H-3; CAS 452098-92-9),

N-tetrahydrofurfuryl-3-(2,6-dichloro-4-trifluoromethylphenox y)-5-methyl-1 H-pyrazole-1 - carboxamide (H-4; CAS 915396-43-9), N-ethyl-3-(2-chloro-6-fluoro-4-trifluoromethylphenoxy)-5- methyl-1 H-pyrazole-1 -carboxamide (H-5; CAS 452099-05-7), N-tetrahydrofurfuryl-3-(2-chloro-6- fluoro-4-trifluoromethylphenoxy)-5-methyl-1 H-pyrazole-1 -carboxamide (H-6; CAS 45100-03-7), 3-[7-fluoro-3-oxo-4-(prop-2-ynyl)-3,4-dihydro-2H-benzo[1 ,4]oxazin-6-yl]-1 ,5-dimethyl-6-thioxo- [1 ,3,5]triazinan-2,4-dione, 1 ,5-dimethyl-6-thioxo-3-(2,2,7-trifluoro-3-oxo-4-(prop-2-ynyl )-3,4- dihydro-2H-benzo[b][1 ,4]oxazin-6-yl)-1 ,3,5-triazinane-2,4-dione, 2-(2,2,7-Trifluoro-3-oxo-4-prop- 2-ynyl-3,4-dihydro-2H-benzo[1 ,4]oxazin-6-yl)-4,5,6,7-tetrahydro-isoindole-1 ,3-dione and 1 - Methyl-6-trifluoromethyl-3-(2,2,7-trifluoro-3-oxo-4-prop-2-y nyl-3,4-dihydro-2H-benzo[1 ,4]oxazin 6-yl)-1 H-pyrimidine-2,4-dione;

b5) from the group of the bleacher herbicides:

aclonifen, amitrol, beflubutamid, benzobicyclon, benzofenap, clomazone, diflufenican, flu- ridone, flurochloridone, flurtamone, isoxaflutole, mesotrione, norflurazon, picolinafen, pyrasulfu- tole, pyrazolynate, pyrazoxyfen, sulcotrione, tefuryltrione, tembotrione, topramezone, 4-hydroxy- 3-[[2-[(2-methoxyethoxy)methyl]-6-(trifluoromethyl)-3-pyridy l]carbonyl]bicyclo[3.2.1]oct-3-en-2- one (H-7; CAS 352010-68-5) and 4-(3-trifluoromethylphenoxy)-2-(4- trifluoromethylphenyl)pyrimidine (H-8; CAS 180608-33-7);

b6) from the group of the EPSP synthase inhibitors:

glyphosate, glyphosate-isopropylammonium and glyphosate-trimesium (sulfosate);

b7) from the group of the glutamine synthase inhibitors:

bilanaphos (bialaphos), bilanaphos-sodium, glufosinate and glufosinate-ammonium;

b8) from the group of the DHP synthase inhibitors:

asulam;

b9) from the group of the mitose inhibitors:

amiprophos, amiprophos-methyl, benfluralin, butamiphos, butralin, carbetamide, chlor- propham, chlorthal, chlorthal-dimethyl, dinitramine, dithiopyr, ethalfluralin, fluchloralin, oryzalin, pendimethalin, prodiamine, propham, propyzamide, tebutam, thiazopyr and trifluralin;

b10) from the group of the VLCFA inhibitors:

acetochlor, alachlor, anilofos, butachlor, cafenstrole, dimethachlor, dimethanamid, dime- thenamid-P, diphenamid, fentrazamide, flufenacet, mefenacet, metazachlor, metolachlor, metolachlor-S, naproanilide, napropamide, pethoxamid, piperophos, pretilachlor, propachlor, propisochlor, pyroxasulfone (KIH-485) and thenylchlor; Compounds of the formula 2:

in which the variables have the following meanings:

Y is phenyl or 5- or 6-membered heteroaryl as defined at the outset, which radicals may be substituted by one to three groups R ^aa ; R ²¹ ,R ²² ,R ²³ ,R ²⁴ are H, halogen or Ci-C ₄ -alkyl; X is O or NH; N is 0 or 1 .

Compounds of the formula 2 have in particular the following meanings:

where # denotes the bond to the skeleton of the molecule; and

R ² ,R ²² ,R ²³ ,R ²⁴ are H, CI, F or CH ₃ ; R ²⁵ is halogen, Ci-C ₄ -alkyl or Ci-C ₄ -haloalkyl; R ²⁶ is Ci-C ₄ - alkyl; R ²⁷ is halogen, Ci-C ₄ -alkoxy or Ci-C ₄ -haloalkoxy; R ²⁸ is H, halogen, Ci-C ₄ -alkyl, Ci-C ₄ - haloalkyl or Ci-C ₄ -haloalkoxy; M is 0, 1 , 2 or 3; X is oxygen; N is 0 or 1.

Preferred compounds of the formula 2 have the following meanings:

R ²¹ is H; R ²² ,R ²³ are F; R ²⁴ is H or F; X is oxygen; N is 0 or 1 .

Particularly preferred compounds of the formula 2 are:

3-[5-(2,2-difluoroethoxy)-1 -methyl-3-trifluoromethyl-1 H-pyrazol-4-ylmethane- sulfonyl]-4-fluoro-5,5-dimethyl-4,5-dihydroisoxazole (2-1 ); 3-{[5-(2,2-difluoroethoxy)-1 -methyl-3- trifluoromethyl-1 H-pyrazol-4-yl]fluoromethanesulfonyl}-5,5-dimethyl-4,5-dihyd roisoxazole (2-2); 4-(4-fluoro-5,5-dimethyl-4,5-dihydroisoxazole-3-sulfonylmeth yl)-2-methyl-5-trifluoromethyl-2H- [1 ,2,3]triazole (2-3); 4-[(5,5-dimethyl-4,5-dihydroisoxazole-3-sulfonyl)fluoromethy l]-2-methyl-5- trifluoromethyl-2H-[1 ,2,3]triazole (2-4); 4-(5,5-dimethyl-4,5-dihydroisoxazole-3-sulfonylmethyl)-2- methyl-5-trifluoromethyl-2H-[1 ,2,3]triazole (2-5); 3-{[5-(2,2-difluoroethoxy)-1 -methyl-3- trifluoromethyl-1 H-pyrazol-4-yl]difluoromethanesulfonyl}-5,5-dimethyl-4,5-dih ydroisoxazole (2-6); 4-[(5,5-dimethyl-4,5-dihydroisoxazole-3-sulfonyl)difluoromet hyl]-2-methyl-5-trifluoromethyl-2H- [1 ,2,3]triazole (2-7); 3-{[5-(2,2-difluoroethoxy)-1 -methyl-3-trifluoromethyl-1 H-pyrazol-4- yl]difluoromethanesulfonyl}-4-fluoro-5,5-dimethyl-4,5-dihydr oisoxazole (2-8); 4-[difluoro-(4- fluoro-5,5-dimethyl-4,5-dihydroisoxazole-3-sulfonyl)methyl]- 2-methyl-5-trifluoromethyl-2H- [1 ,2,3]triazole (2-9);

b1 1 ) from the group of the cellulose biosynthesis inhibitors:

chlorthiamid, dichlobenil, flupoxam and isoxaben; b12) from the group of the decoupler herbicides:

dinoseb, dinoterb and DNOC and its salts;

b13) from the group of the auxin herbicides:

2,4-D and its salts and esters, 2,4-DB and its salts and esters, aminopyralid and its salts such as aminopyralid-tris(2-hydroxypropyl)ammonium and its esters, benazolin, benazolin-ethyl, chloramben and its salts and esters, clomeprop, clopyralid and its salts and esters, dicamba and its salts and esters, dichlorprop and its salts and esters, dichlorprop-P and its salts and esters, fluroxypyr, fluroxypyr-butometyl, fluroxypyr-meptyl, MCPA and its salts and esters, MCPA- thioethyl, MCPB and its salts and esters, mecoprop and its salts and esters, mecoprop-P and its salts and esters, picloram and its salts and esters, quinclorac, quinmerac, TBA (2,3,6) and its salts and esters, triclopyr and its salts and esters, and 5,6-dichloro-2-cyclopropyl-4- pyrimidinecarboxylic acid (H-9; CAS 858956-08-8) and its salts and esters;

b14) from the group of the auxin transport inhibitors: diflufenzopyr, diflufenzopyr-sodium, naptalam and naptalam-sodium;

b15) from the group of the other herbicides: bromobutide, chlorflurenol, chlorflurenol- methyl, cinmethylin, cumyluron, dalapon, dazomet, difenzoquat, difenzoquat-metilsulfate, dime- thipin, DSMA, dymron, endothal and its salts, etobenzanid, flamprop, flamprop-isopropyl, flam- prop-methyl, flamprop-M-isopropyl, flamprop-M-methyl, flurenol, flurenol-butyl, flurprimidol, fos- amine, fosamine-ammonium, indanofan, maleic hydrazide, mefluidide, metam, methyl azide, methyl bromide, methyl-dymron, methyl iodide, MSMA, oleic acid, oxaziclomefone, pelargonic acid, pyributicarb, quinoclamine, triaziflam, tridiphane and 6-chloro-3-(2-cyclopropyl-6- methylphenoxy)-4-pyridazinol (H-10; CAS 499223-49-3) and its salts and esters.

Examples of preferred safeners C are benoxacor, cloquintocet, cyometrinil, cyprosulfa- mide, dichlormid, dicyclonone, dietholate, fenchlorazole, fenclorim, flurazole, fluxofenim, furi- lazole, isoxadifen, mefenpyr, mephenate, naphthalic anhydride, oxabetrinil, 4-(dichloroacetyl)-1 - oxa-4-azaspiro[4.5]decane (H-1 1 ; MON4660, CAS 71526-07-3) and 2,2,5-trimethyl-3- (dichloroacetyl)-1 ,3-oxazolidine (H-12; R-29148, CAS 52836-31 -4).

The active compounds of groups b1 ) to b15) and the safeners C are known herbicides and safeners, see, for example, The Compendium of Pesticide Common Names

(http://www.alanwood.net/pesticides/); B. Hock, C. Fedtke, R. R. Schmidt, Herbizide

[Herbicides], Georg Thieme Verlag, Stuttgart, 1995. Further herbicidally active compounds are known from WO 96/26202, WO 97/41 1 16, WO 97/41 1 17, WO 97/41 1 18, WO 01/83459 and WO 2008/074991 and from W. Kramer et al. (ed.) "Modern Crop Protection Compounds", Vol. 1 , Wiley VCH, 2007 and the literature quoted therein.

The invention also relates to compositions in the form of a crop protection composition formulated as a 1 -component composition comprising an active compound combination comprising at least one N-(tetrazol-5-yl)- and N-(triazol-5-yl)arylcarboxamide compound of the formula I and at least one further active compound, preferably selected from the active compounds of groups b1 to b15, and at least one solid or liquid carrier and/or one or more surfactants and, if desired, one or more further auxiliaries customary for crop protection compositions.

The invention also relates to compositions in the form of a crop protection composition formulated as a 2-component composition comprising a first component comprising at least one com- pound of the formula I, a solid or liquid carrier and/or one or more surfactants and a second component comprising at least one further active compound selected from the active compounds of groups b1 to b15, a solid or liquid carrier and/or one or more surfactants, where additionally both components may also comprise further auxiliaries customary for crop protection compositions.

In binary compositions comprising at least one compound of the formula I as component A and at least one herbicide B, the weight ratio of the active compounds A:B is generally in the range of from 1 :1000 to 1000:1 , preferably in the range of from 1 :500 to 500:1 , in particular in the range of from 1 :250 to 250:1 and particularly preferably in the range of from 1 :75 to 75:1.

In binary compositions comprising at least one compound of the formula I as component A and at least one safener C, the weight ratio of the active compounds A:C is generally in the range of from 1 :1000 to 1000:1 , preferably in the range of from 1 :500 to 500:1 , in particular in the range of from 1 :250 to 250:1 and particularly preferably in the range of from 1 :75 to 75:1 .

In ternary compositions comprising both at least one compound of the formula I as com- ponent A, at least one herbicide B and at least one safener C, the relative parts by weight of the components A:B are generally in the range of from 1 :1000 to 1000:1 , preferably in the range of from 1 :500 to 500:1 , in particular in the range of from 1 :250 to 250:1 and particularly preferably in the range of from 1 :75 to 75:1 ; the weight ratio of the components A:C is generally in the range of from 1 :1000 to 1000:1 , preferably in the range of from 1 :500 to 500:1 , in particular in the range of from 1 :250 to 250:1 and particularly preferably in the range of from 1 :75 to 75:1 ; and the weight ratio of the components B:C is generally in the range of from 1 :1000 to 1000:1 , preferably in the range of from 1 :500 to 500:1 , in particular in the range of from 1 :250 to 250:1 and particularly preferably in the range of from 1 :75 to 75:1. Preferably, the weight ratio of the components A + B to the component C is in the range of from 1 :500 to 500:1 , in particular in the range of from 1 :250 to 250:1 and particularly preferably in the range of from 1 :75 to 75:1.

Examples of particularly preferred compositions according to the invention comprising in each case one individualized compound of the formula I and one mixing partner or a mixing partner combination are given in Table B below.

A further aspect of the invention relates to the compositions B-1 to B-1236 listed in Table B below, where in each case one row of Table B corresponds to a herbicidal composition comprising one of the compounds of formula I individualized in the above description (component 1 ) and the further active compound from groups b1 ) to b15) and/or safener C stated in each case in the row in question (component 2). The active compounds in the compositions described are in each case preferably present in synergistically effective amounts.

Table B:

Herbicide(s) B Safener C

B-1 clodinafop-propargyl —

B-2 cycloxydim —

B-3 cyhalofop-butyl —

B-4 fenoxaprop-P-ethyl —

B-5 pinoxaden — Herbicide(s) B Safener C

B-6 profoxydim —

B-7 tepraloxydim —

B-8 tralkoxydim —

B-9 esprocarb —

B-10 prosulfocarb —

B-1 1 thiobencarb —

B-12 triallate —

B-13 bensulfuron-methyl —

B-14 bispyribac-sodium —

B-15 cyclosulfamuron —

B-16 flumetsulam —

B-17 flupyrsulfuron-methyl-sodium —

B-18 foramsulfuron —

B-19 imazamox —

B-20 imazapic —

B-21 imazapyr —

B-22 imazaquin —

B-23 imazethapyr —

B-24 imazosulfuron —

B-25 iodosulfuron-methyl-sodium —

B-26 mesosulfuron —

B-27 nicosulfuron —

B-28 penoxsulam —

B-29 propoxycarbazone-sodium —

B-30 pyrazosulfuron-ethyl —

B-31 pyroxsulam —

B-32 rimsulfuron —

B-33 sulfosulfuron —

B-34 thiencarbazone-methyl —

B-35 tritosulfuron —

B-36 2,4-D and its salts and esters —

B-37 aminopyralid and its salts and esters —

B-38 clopyralid and its salts and esters —

B-39 dicamba and its salts and esters —

B-40 fluroxypyr-meptyl —

B-41 quinclorac —

B-42 quinmerac —

B-43 H-9 —

B-44 diflufenzopyr —

B-45 diflufenzopyr-sodium — Herbicide(s) B Safener C

B-46 clomazone —

B-47 diflufenican —

B-48 fluorochloridone —

B-49 isoxaflutol —

B-50 mesotrione —

B-51 picolinafen —

B-52 sulcotrione —

B-53 tefuryltrione —

B-54 tembotrione —

B-55 topramezone —

B-56 H-7 —

B-57 atrazine —

B-58 diuron —

B-59 fluometuron —

B-60 hexazinone —

B-61 isoproturon —

B-62 metribuzin —

B-63 propanil —

B-64 terbuthylazine —

B-65 paraquat dichloride —

B-66 flumioxazin —

B-67 oxyfluorfen —

B-68 saflufenacil —

B-69 sulfentrazone —

B-70 H-1 —

B-71 H-2 —

B-72 glyphosate —

B-73 glyphosate-isopropylammonium —

B-74 glyphosate-trimesium (sulfosate) —

B-75 glufosinate —

B-76 glufosinate-ammonium —

B-77 pendimethalin —

B-78 trifluralin —

B-79 acetochlor —

B-80 cafenstrole —

B-81 dimethenamid-P —

B-82 fentrazamide —

B-83 flufenacet —

B-84 mefenacet —

B-85 metazachlor — Herbicide(s) B Safener C

B-86 metolachlor-S —

B-87 pyroxasulfone —

B-88 isoxaben —

B-89 dymron —

B-90 indanofan —

B-91 oxaziclomefone —

B-92 triaziflam —

B-93 chlorotoluron —

B-94 atrazine + H-1 —

B-95 atrazine + glyphosate —

B-96 atrazine + mesotrione —

B-97 atrazine + nicosulfuron —

B-98 atrazine + tembotrione —

B-99 atrazine + topramezone —

B-100 clomazone + glyphosate —

B-101 diflufenican + clodinafop-propargyl —

B-102 diflufenican + fenoxaprop-P-ethyl —

B-103 diflufenican + flupyrsulfuron-methyl-sodium —

B-104 diflufenican + glyphosate —

B-105 diflufenican + mesosulfuron-methyl —

B-106 diflufenican + pinoxaden —

B-107 diflufenican + pyroxsulam —

B-108 flumetsulam + glyphosate —

B-109 flumioxazin + glyphosate —

B-1 10 imazapic + glyphosate —

B-1 1 1 imazethapyr + glyphosate —

B-1 12 isoxaflutol + H-1 —

B-1 13 isoxaflutol + glyphosate —

B-1 14 metazachlor + H-1 —

B-1 15 metazachlor + glyphosate —

B-1 16 metazachlor + mesotrione —

B-1 17 metazachlor + nicosulfuron —

B-1 18 metazachlor + terbuthylazine —

B-1 19 metazachlor + topramezone —

B-120 metribuzin + glyphosate —

B-121 pendimethalin + H-1 —

B-122 pendimethalin + clodinafop-propargyl —

B-123 pendimethalin + fenoxaprop-P-ethyl —

B-124 pendimethalin + flupyrsulfuron-methyl-sodium —

B-125 pendimethalin + glyphosate — Herbicide(s) B Safener C

B-126 pendimethalin + mesosulfuron-methyl —

B-127 pendimethalin + mesotrione —

B-128 pendimethalin + nicosulfuron —

B-129 pendimethalin + pinoxaden —

B-130 pendimethalin + pyroxsulam —

B-131 pendimethalin + tembotrione —

B-132 pendimethalin + topramezone —

B-133 pyroxasulfone + tembotrione —

B-134 pyroxasulfone + topramezone —

B-135 sulfentrazone + glyphosate —

B-136 terbuthylazine + H-1 —

B-137 terbuthylazine + foramsulfuron —

B-138 terbuthylazine + glyphosate —

B-139 terbuthylazine + mesotrione —

B-140 terbuthylazine + nicosulfuron —

B-141 terbuthylazine + tembotrione —

B-142 terbuthylazine + topramezone —

B-143 trifluralin + glyphosate —

B-144 — benoxacor

B-145 — cloquintocet

B-146 — cyprosulfamide

B-147 — dichlormid

B-148 — fenchlorazole

B-149 — isoxadifen

B-150 — mefenpyr

B-151 — H-1 1

B-152 — H-12

B-153 clodinafop-propargyl benoxacor

B-154 cycloxydim benoxacor

B-155 cyhalofop-butyl benoxacor

B-156 fenoxaprop-P-ethyl benoxacor

B-157 pinoxaden benoxacor

B-158 profoxydim benoxacor

B-159 tepraloxydim benoxacor

B-160 tralkoxydim benoxacor

B-161 esprocarb benoxacor

B-162 prosulfocarb benoxacor

B-163 thiobencarb benoxacor

B-164 triallate benoxacor

B-165 bensulfuron-methyl benoxacor Herbicide(s) B Safener C

B-166 bispyribac-sodium benoxacor

B-167 cyclosulfamuron benoxacor

B-168 flumetsulam benoxacor

B-169 flupyrsulfuron-methyl-sodium benoxacor

B-170 foramsulfuron benoxacor

B-171 imazamox benoxacor

B-172 imazapic benoxacor

B-173 imazapyr benoxacor

B-174 imazaquin benoxacor

B-175 imazethapyr benoxacor

B-176 imazosulfuron benoxacor

B-177 iodosulfuron-methyl-sodium benoxacor

B-178 mesosulfuron benoxacor

B-179 nicosulfuron benoxacor

B-180 penoxsulam benoxacor

B-181 propoxycarbazone-sodium benoxacor

B-182 pyrazosulfuron-ethyl benoxacor

B-183 pyroxsulam benoxacor

B-184 rimsulfuron benoxacor

B-185 sulfosulfuron benoxacor

B-186 thiencarbazone-methyl benoxacor

B-187 tritosulfuron benoxacor

B-188 2,4-D and its salts and esters benoxacor

B-189 aminopyralid and its salts and esters benoxacor

B-190 clopyralid and its salts and esters benoxacor

B-191 dicamba and its salts and esters benoxacor

B-192 fluroxypyr-meptyl benoxacor

B-193 quinclorac benoxacor

B-194 quinmerac benoxacor

B-195 H-9 benoxacor

B-196 diflufenzopyr benoxacor

B-197 diflufenzopyr-sodium benoxacor

B-198 clomazone benoxacor

B-199 diflufenican benoxacor

B-200 fluorochloridone benoxacor

B-201 isoxaflutol benoxacor

B-202 mesotrione benoxacor

B-203 picolinafen benoxacor

B-204 sulcotrione benoxacor

B-205 tefuryltrione benoxacor Herbicide(s) B Safener C

B-206 tembotrione benoxacor

B-207 topramezone benoxacor

B-208 H-7 benoxacor

B-209 atrazine benoxacor

B-210 diuron benoxacor

B-21 1 fluometuron benoxacor

B-212 hexazinone benoxacor

B-213 isoproturon benoxacor

B-214 metribuzin benoxacor

B-215 propanil benoxacor

B-216 terbuthylazine benoxacor

B-217 paraquat dichloride benoxacor

B-218 flumioxazin benoxacor

B-219 oxyfluorfen benoxacor

B-220 saflufenacil benoxacor

B-221 sulfentrazone benoxacor

B-222 H-1 benoxacor

B-223 H-2 benoxacor

B-224 glyphosate benoxacor

B-225 glyphosate-isopropylammonium benoxacor

B-226 glyphosate-trimesium (sulfosate) benoxacor

B-227 glufosinate benoxacor

B-228 glufosinate-ammonium benoxacor

B-229 pendimethalin benoxacor

B-230 trifluralin benoxacor

B-231 acetochlor benoxacor

B-232 cafenstrole benoxacor

B-233 dimethenamid-P benoxacor

B-234 fentrazamide benoxacor

B-235 flufenacet benoxacor

B-236 mefenacet benoxacor

B-237 metazachlor benoxacor

B-238 metolachlor-S benoxacor

B-239 pyroxasulfone benoxacor

B-240 isoxaben benoxacor

B-241 dymron benoxacor

B-242 indanofan benoxacor

B-243 oxaziclomefone benoxacor

B-244 triaziflam benoxacor

B-245 atrazine + H-1 benoxacor Herbicide(s) B Safener C

B-246 atrazine + glyphosate benoxacor

B-247 atrazine + mesotrione benoxacor

B-248 atrazine + nicosulfuron benoxacor

B-249 atrazine + tembotrione benoxacor

B-250 atrazine + topramezone benoxacor

B-251 clomazone + glyphosate benoxacor

B-252 diflufenican + clodinafop-propargyl benoxacor

B-253 diflufenican + fenoxaprop-P-ethyl benoxacor

B-254 diflufenican + flupyrsulfuron-methyl-sodium benoxacor

B-255 diflufenican + glyphosate benoxacor

B-256 diflufenican + mesosulfuron-methyl benoxacor

B-257 diflufenican + pinoxaden benoxacor

B-258 diflufenican + pyroxsulam benoxacor

B-259 flumetsulam + glyphosate benoxacor

B-260 flumioxazin + glyphosate benoxacor

B-261 imazapic + glyphosate benoxacor

B-262 imazethapyr + glyphosate benoxacor

B-263 isoxaflutol + H-1 benoxacor

B-264 isoxaflutol + glyphosate benoxacor

B-265 metazachlor + H-1 benoxacor

B-266 metazachlor + glyphosate benoxacor

B-267 metazachlor + mesotrione benoxacor

B-268 metazachlor + nicosulfuron benoxacor

B-269 metazachlor + terbuthylazine benoxacor

B-270 metazachlor + topramezone benoxacor

B-271 metribuzin + glyphosate benoxacor

B-272 pendimethalin + H-1 benoxacor

B-273 pendimethalin + clodinafop-propargyl benoxacor

B-274 pendimethalin + fenoxaprop-P-ethyl benoxacor

B-275 pendimethalin + flupyrsulfuron-methyl-sodium benoxacor

B-276 pendimethalin + glyphosate benoxacor

B-277 pendimethalin + mesosulfuron-methyl benoxacor

B-278 pendimethalin + mesotrione benoxacor

B-279 pendimethalin + nicosulfuron benoxacor

B-280 pendimethalin + pinoxaden benoxacor

B-281 pendimethalin + pyroxsulam benoxacor

B-282 pendimethalin + tembotrione benoxacor

B-283 pendimethalin + topramezone benoxacor

B-284 pyroxasulfone + tembotrione benoxacor

B-285 pyroxasulfone + topramezone benoxacor Herbicide(s) B Safener C

B-286 sulfentrazone + glyphosate benoxacor

B-287 terbuthylazine + H-1 benoxacor

B-288 terbuthylazine + foramsulfuron benoxacor

B-289 terbuthylazine + glyphosate benoxacor

B-290 terbuthylazine + mesotrione benoxacor

B-291 terbuthylazine + nicosulfuron benoxacor

B-292 terbuthylazine + tembotrione benoxacor

B-293 terbuthylazine + topramezone benoxacor

B-294 trifluralin + glyphosate benoxacor

B-295 clodinafop-propargyl cloquintocet

B-296 cycloxydim cloquintocet

B-297 cyhalofop-butyl cloquintocet

B-298 fenoxaprop-P-ethyl cloquintocet

B-299 pinoxaden cloquintocet

B-300 profoxydim cloquintocet

B-301 tepraloxydim cloquintocet

B-302 tralkoxydim cloquintocet

B-303 esprocarb cloquintocet

B-304 prosulfocarb cloquintocet

B-305 thiobencarb cloquintocet

B-306 triallate cloquintocet

B-307 bensulfuron-methyl cloquintocet

B-308 bispyribac-sodium cloquintocet

B-309 cyclosulfamuron cloquintocet

B-310 flumetsulam cloquintocet

B-31 1 flupyrsulfuron-methyl-sodium cloquintocet

B-312 foramsulfuron cloquintocet

B-313 imazamox cloquintocet

B-314 imazapic cloquintocet

B-315 imazapyr cloquintocet

B-316 imazaquin cloquintocet

B-317 imazethapyr cloquintocet

B-318 imazosulfuron cloquintocet

B-319 iodosulfuron-methyl-sodium cloquintocet

B-320 mesosulfuron cloquintocet

B-321 nicosulfuron cloquintocet

B-322 penoxsulam cloquintocet

B-323 propoxycarbazone-sodium cloquintocet

B-324 pyrazosulfuron-ethyl cloquintocet

B-325 pyroxsulam cloquintocet Herbicide(s) B Safener C

B-326 rimsulfuron cloquintocet

B-327 sulfosulfuron cloquintocet

B-328 thiencarbazone-methyl cloquintocet

B-329 tritosulfuron cloquintocet

B-330 2,4-D and its salts and esters cloquintocet

B-331 aminopyralid and its salts and esters cloquintocet

B-332 clopyralid and its salts and esters cloquintocet

B-333 dicamba and its salts and esters cloquintocet

B-334 fluroxypyr-meptyl cloquintocet

B-335 quinclorac cloquintocet

B-336 quinmerac cloquintocet

B-337 H-9 cloquintocet

B-338 diflufenzopyr cloquintocet

B-339 diflufenzopyr-sodium cloquintocet

B-340 clomazone cloquintocet

B-341 diflufenican cloquintocet

B-342 fluorochloridone cloquintocet

B-343 isoxaflutol cloquintocet

B-344 mesotrione cloquintocet

B-345 picolinafen cloquintocet

B-346 sulcotrione cloquintocet

B-347 tefuryltrione cloquintocet

B-348 tembotrione cloquintocet

B-349 topramezone cloquintocet

B-350 H-7 cloquintocet

B-351 atrazine cloquintocet

B-352 diuron cloquintocet

B-353 fluometuron cloquintocet

B-354 hexazinone cloquintocet

B-355 isoproturon cloquintocet

B-356 metribuzin cloquintocet

B-357 propanil cloquintocet

B-358 terbuthylazine cloquintocet

B-359 paraquat dichloride cloquintocet

B-360 flumioxazin cloquintocet

B-361 oxyfluorfen cloquintocet

B-362 saflufenacil cloquintocet

B-363 sulfentrazone cloquintocet

B-364 H-1 cloquintocet

B-365 H-2 cloquintocet Herbicide(s) B Safener C

B-366 glyphosate cloquintocet

B-367 glyphosate-isopropylammonium cloquintocet

B-368 glyphosate-trimesium (sulfosate) cloquintocet

B-369 glufosinate cloquintocet

B-370 glufosinate-ammonium cloquintocet

B-371 pendimethalin cloquintocet

B-372 trifluralin cloquintocet

B-373 acetochlor cloquintocet

B-374 cafenstrole cloquintocet

B-375 dimethenamid-P cloquintocet

B-376 fentrazamide cloquintocet

B-377 flufenacet cloquintocet

B-378 mefenacet cloquintocet

B-379 metazachlor cloquintocet

B-380 metolachlor-S cloquintocet

B-381 pyroxasulfone cloquintocet

B-382 isoxaben cloquintocet

B-383 dymron cloquintocet

B-384 indanofan cloquintocet

B-385 oxaziclomefone cloquintocet

B-386 triaziflam cloquintocet

B-387 atrazine + H-1 cloquintocet

B-388 atrazine + glyphosate cloquintocet

B-389 atrazine + mesotrione cloquintocet

B-390 atrazine + nicosulfuron cloquintocet

B-391 atrazine + tembotrione cloquintocet

B-392 atrazine + topramezone cloquintocet

B-393 clomazone + glyphosate cloquintocet

B-394 diflufenican + clodinafop-propargyl cloquintocet

B-395 diflufenican + fenoxaprop-p-ethyl cloquintocet

B-396 diflufenican + flupyrsulfuron-methyl-sodium cloquintocet

B-397 diflufenican + glyphosate cloquintocet

B-398 diflufenican + mesosulfuron-methyl cloquintocet

B-399 diflufenican + pinoxaden cloquintocet

B-400 diflufenican + pyroxsulam cloquintocet

B-401 flumetsulam + glyphosate cloquintocet

B-402 flumioxazin + glyphosate cloquintocet

B-403 imazapic + glyphosate cloquintocet

B-404 imazethapyr + glyphosate cloquintocet

B-405 isoxaflutol + H-1 cloquintocet Herbicide(s) B Safener C

B-406 isoxaflutol + glyphosate cloquintocet

B-407 metazachlor + H-1 cloquintocet

B-408 metazachlor + glyphosate cloquintocet

B-409 metazachlor + mesotrione cloquintocet

B-410 metazachlor + nicosulfuron cloquintocet

B-41 1 metazachlor + terbuthylazine cloquintocet

B-412 metazachlor + topramezone cloquintocet

B-413 metribuzin + glyphosate cloquintocet

B-414 pendimethalin + H-1 cloquintocet

B-415 pendimethalin + clodinafop-propargyl cloquintocet

B-416 pendimethalin + fenoxaprop-P-ethyl cloquintocet

B-417 pendimethalin + flupyrsulfuron-methyl-sodium cloquintocet

B-418 pendimethalin + glyphosate cloquintocet

B-419 pendimethalin + mesosulfuron-methyl cloquintocet

B-420 pendimethalin + mesotrione cloquintocet

B-421 pendimethalin + nicosulfuron cloquintocet

B-422 pendimethalin + pinoxaden cloquintocet

B-423 pendimethalin + pyroxsulam cloquintocet

B-424 pendimethalin + tembotrione cloquintocet

B-425 pendimethalin + topramezone cloquintocet

B-426 pyroxasulfone + tembotrione cloquintocet

B-427 pyroxasulfone + topramezone cloquintocet

B-428 sulfentrazone + glyphosate cloquintocet

B-429 terbuthylazine + H-1 cloquintocet

B-430 terbuthylazine + foramsulfuron cloquintocet

B-431 terbuthylazine + glyphosate cloquintocet

B-432 terbuthylazine + mesotrione cloquintocet

B-433 terbuthylazine + nicosulfuron cloquintocet

B-434 terbuthylazine + tembotrione cloquintocet

B-435 terbuthylazine + topramezone cloquintocet

B-436 trifluralin + glyphosate cloquintocet

B-437 clodinafop-propargyl dichlormid

B-438 cycloxydim dichlormid

B-439 cyhalofop-butyl dichlormid

B-440 fenoxaprop-P-ethyl dichlormid

B-441 pinoxaden dichlormid

B-442 profoxydim dichlormid

B-443 tepraloxydim dichlormid

B-444 tralkoxydim dichlormid

B-445 esprocarb dichlormid Herbicide(s) B Safener C

B-446 prosulfocarb dichlormid

B-447 thiobencarb dichlormid

B-448 triallate dichlormid

B-449 bensulfuron-methyl dichlormid

B-450 bispyribac-sodium dichlormid

B-451 cyclosulfamuron dichlormid

B-452 flumetsulam dichlormid

B-453 flupyrsulfuron-methyl-sodium dichlormid

B-454 foramsulfuron dichlormid

B-455 imazamox dichlormid

B-456 imazapic dichlormid

B-457 imazapyr dichlormid

B-458 imazaquin dichlormid

B-459 imazethapyr dichlormid

B-460 imazosulfuron dichlormid

B-461 iodosulfuron-methyl-sodium dichlormid

B-462 mesosulfuron dichlormid

B-463 nicosulfuron dichlormid

B-464 penoxsulam dichlormid

B-465 propoxycarbazone-sodium dichlormid

B-466 pyrazosulfuron-ethyl dichlormid

B-467 pyroxsulam dichlormid

B-468 rimsulfuron dichlormid

B-469 sulfosulfuron dichlormid

B-470 thiencarbazone-methyl dichlormid

B-471 tritosulfuron dichlormid

B-472 2,4-D and its salts and esters dichlormid

B-473 aminopyralid and its salts and esters dichlormid

B-474 clopyralid and its salts and esters dichlormid

B-475 dicamba and its salts and esters dichlormid

B-476 fluroxypyr-meptyl dichlormid

B-477 quinclorac dichlormid

B-478 quinmerac dichlormid

B-479 H-9 dichlormid

B-480 diflufenzopyr dichlormid

B-481 diflufenzopyr-sodium dichlormid

B-482 clomazone dichlormid

B-483 diflufenican dichlormid

B-484 fluorochloridone dichlormid

B-485 isoxaflutol dichlormid Herbicide(s) B Safener C

B-486 mesotrione dichlormid

B-487 picolinafen dichlormid

B-488 sulcotrione dichlormid

B-489 tefuryltrione dichlormid

B-490 tembotrione dichlormid

B-491 topramezone dichlormid

B-492 H-7 dichlormid

B-493 atrazine dichlormid

B-494 diuron dichlormid

B-495 fluometuron dichlormid

B-496 hexazinone dichlormid

B-497 isoproturon dichlormid

B-498 metribuzin dichlormid

B-499 propanil dichlormid

B-500 terbuthylazine dichlormid

B-501 paraquat dichloride dichlormid

B-502 flumioxazin dichlormid

B-503 oxyfluorfen dichlormid

B-504 saflufenacil dichlormid

B-505 sulfentrazone dichlormid

B-506 H-1 dichlormid

B-507 H-2 dichlormid

B-508 glyphosate dichlormid

B-509 glyphosate-isopropylammonium dichlormid

B-510 glyphosate-trimesium (sulfosate) dichlormid

B-51 1 glufosinate dichlormid

B-512 glufosinate-ammonium dichlormid

B-513 pendimethalin dichlormid

B-514 trifluralin dichlormid

B-515 acetochlor dichlormid

B-516 cafenstrole dichlormid

B-517 dimethenamid-P dichlormid

B-518 fentrazamide dichlormid

B-519 flufenacet dichlormid

B-520 mefenacet dichlormid

B-521 metazachlor dichlormid

B-522 metolachlor-S dichlormid

B-523 pyroxasulfone dichlormid

B-524 isoxaben dichlormid

B-525 dymron dichlormid Herbicide(s) B Safener C

B-526 indanofan dichlormid

B-527 oxaziclomefone dichlormid

B-528 triaziflam dichlormid

B-529 atrazine + H-1 dichlormid

B-530 atrazine + glyphosate dichlormid

B-531 atrazine + mesotrione dichlormid

B-532 atrazine + nicosulfuron dichlormid

B-533 atrazine + tembotrione dichlormid

B-534 atrazine + topramezone dichlormid

B-535 clomazone + glyphosate dichlormid

B-536 diflufenican + clodinafop-propargyl dichlormid

B-537 diflufenican + fenoxaprop-p-ethyl dichlormid

B-538 diflufenican + flupyrsulfuron-methyl-sodium dichlormid

B-539 diflufenican + glyphosate dichlormid

B-540 diflufenican + mesosulfuron-methyl dichlormid

B-541 diflufenican + pinoxaden dichlormid

B-542 diflufenican + pyroxsulam dichlormid

B-543 flumetsulam + glyphosate dichlormid

B-544 flumioxazin + glyphosate dichlormid

B-545 imazapic + glyphosate dichlormid

B-546 imazethapyr + glyphosate dichlormid

B-547 isoxaflutol + H-1 dichlormid

B-548 isoxaflutol + glyphosate dichlormid

B-549 metazachlor + H-1 dichlormid

B-550 metazachlor + glyphosate dichlormid

B-551 metazachlor + mesotrione dichlormid

B-552 metazachlor + nicosulfuron dichlormid

B-553 metazachlor + terbuthylazine dichlormid

B-554 metazachlor + topramezone dichlormid

B-555 metribuzin + glyphosate dichlormid

B-556 pendimethalin + H-1 dichlormid

B-557 pendimethalin + clodinafop-propargyl dichlormid

B-558 pendimethalin + fenoxaprop-P-ethyl dichlormid

B-559 pendimethalin + flupyrsulfuron-methyl-sodium dichlormid

B-560 pendimethalin + glyphosate dichlormid

B-561 pendimethalin + mesosulfuron-methyl dichlormid

B-562 pendimethalin + mesotrione dichlormid

B-563 pendimethalin + nicosulfuron dichlormid

B-564 pendimethalin + pinoxaden dichlormid

B-565 pendimethalin + pyroxsulam dichlormid Herbicide(s) B Safener C

B-566 pendimethalin + tembotrione dichlormid

B-567 pendimethalin + topramezone dichlormid

B-568 pyroxasulfone + tembotrione dichlormid

B-569 pyroxasulfone + topramezone dichlormid

B-570 sulfentrazone + glyphosate dichlormid

B-571 terbuthylazine + H-1 dichlormid

B-572 terbuthylazine + foramsulfuron dichlormid

B-573 terbuthylazine + glyphosate dichlormid

B-574 terbuthylazine + mesotrione dichlormid

B-575 terbuthylazine + nicosulfuron dichlormid

B-576 terbuthylazine + tembotrione dichlormid

B-577 terbuthylazine + topramezone dichlormid

B-578 trifluralin + glyphosate dichlormid

B-579 clodinafop-propargyl fenchlorazole

B-580 cycloxydim fenchlorazole

B-581 cyhalofop-butyl fenchlorazole

B-582 fenoxaprop-P-ethyl fenchlorazole

B-583 pinoxaden fenchlorazole

B-584 profoxydim fenchlorazole

B-585 tepraloxydim fenchlorazole

B-586 tralkoxydim fenchlorazole

B-587 esprocarb fenchlorazole

B-588 prosulfocarb fenchlorazole

B-589 thiobencarb fenchlorazole

B-590 triallate fenchlorazole

B-591 bensulfuron-methyl fenchlorazole

B-592 bispyribac-sodium fenchlorazole

B-593 cyclosulfamuron fenchlorazole

B-594 flumetsulam fenchlorazole

B-595 flupyrsulfuron-methyl-sodium fenchlorazole

B-596 foramsulfuron fenchlorazole

B-597 imazamox fenchlorazole

B-598 imazapic fenchlorazole

B-599 imazapyr fenchlorazole

B-600 imazaquin fenchlorazole

B-601 imazethapyr fenchlorazole

B-602 imazosulfuron fenchlorazole

B-603 iodosulfuron-methyl-sodium fenchlorazole

B-604 mesosulfuron fenchlorazole

B-605 nicosulfuron fenchlorazole Herbicide(s) B Safener C

B-606 penoxsulam fenchlorazole

B-607 propoxycarbazone-sodium fenchlorazole

B-608 pyrazosulfuron-ethyl fenchlorazole

B-609 pyroxsulam fenchlorazole

B-610 rimsulfuron fenchlorazole

B-61 1 sulfosulfuron fenchlorazole

B-612 thiencarbazone-methyl fenchlorazole

B-613 tritosulfuron fenchlorazole

B-614 2,4-D and its salts and esters fenchlorazole

B-615 aminopyralid and its salts and esters fenchlorazole

B-616 clopyralid and its salts and esters fenchlorazole

B-617 dicamba and its salts and esters fenchlorazole

B-618 fluroxypyr-meptyl fenchlorazole

B-619 quinclorac fenchlorazole

B-620 quinmerac fenchlorazole

B-621 H-9 fenchlorazole

B-622 diflufenzopyr fenchlorazole

B-623 diflufenzopyr-sodium fenchlorazole

B-624 clomazone fenchlorazole

B-625 diflufenican fenchlorazole

B-626 fluorochloridone fenchlorazole

B-627 isoxaflutol fenchlorazole

B-628 mesotrione fenchlorazole

B-629 picolinafen fenchlorazole

B-630 sulcotrione fenchlorazole

B-631 tefuryltrione fenchlorazole

B-632 tembotrione fenchlorazole

B-633 topramezone fenchlorazole

B-634 H-7 fenchlorazole

B-635 atrazine fenchlorazole

B-636 diuron fenchlorazole

B-637 fluometuron fenchlorazole

B-638 hexazinone fenchlorazole

B-639 isoproturon fenchlorazole

B-640 metribuzin fenchlorazole

B-641 propanil fenchlorazole

B-642 terbuthylazine fenchlorazole

B-643 paraquat dichloride fenchlorazole

B-644 flumioxazin fenchlorazole

B-645 oxyfluorfen fenchlorazole Herbicide(s) B Safener C

B-646 saflufenacil fenchlorazole

B-647 sulfentrazone fenchlorazole

B-648 H-1 fenchlorazole

B-649 H-2 fenchlorazole

B-650 glyphosate fenchlorazole

B-651 glyphosate-isopropylammonium fenchlorazole

B-652 glyphosate-trimesium (sulfosate) fenchlorazole

B-653 glufosinate fenchlorazole

B-654 glufosinate-ammonium fenchlorazole

B-655 pendimethalin fenchlorazole

B-656 trifluralin fenchlorazole

B-657 acetochlor fenchlorazole

B-658 cafenstrole fenchlorazole

B-659 dimethenamid-P fenchlorazole

B-660 fentrazamide fenchlorazole

B-661 flufenacet fenchlorazole

B-662 mefenacet fenchlorazole

B-663 metazachlor fenchlorazole

B-664 metolachlor-S fenchlorazole

B-665 pyroxasulfone fenchlorazole

B-666 isoxaben fenchlorazole

B-667 dymron fenchlorazole

B-668 indanofan fenchlorazole

B-669 oxaziclomefone fenchlorazole

B-670 triaziflam fenchlorazole

B-671 atrazine + H-1 fenchlorazole

B-672 atrazine + glyphosate fenchlorazole

B-673 atrazine + mesotrione fenchlorazole

B-674 atrazine + nicosulfuron fenchlorazole

B-675 atrazine + tembotrione fenchlorazole

B-676 atrazine + topramezone fenchlorazole

B-677 clomazone + glyphosate fenchlorazole

B-678 diflufenican + clodinafop-propargyl fenchlorazole

B-679 diflufenican + fenoxaprop-P-ethyl fenchlorazole

B-680 diflufenican + flupyrsulfuron-methyl-sodium fenchlorazole

B-681 diflufenican + glyphosate fenchlorazole

B-682 diflufenican + mesosulfuron-methyl fenchlorazole

B-683 diflufenican + pinoxaden fenchlorazole

B-684 diflufenican + pyroxsulam fenchlorazole

B-685 flumetsulam + glyphosate fenchlorazole Herbicide(s) B Safener C

B-686 flumioxazin + glyphosate fenchlorazole

B-687 imazapic + glyphosate fenchlorazole

B-688 imazethapyr + glyphosate fenchlorazole

B-689 isoxaflutol + H-1 fenchlorazole

B-690 isoxaflutol + glyphosate fenchlorazole

B-691 metazachlor + H-1 fenchlorazole

B-692 metazachlor + glyphosate fenchlorazole

B-693 metazachlor + mesotrione fenchlorazole

B-694 metazachlor + nicosulfuron fenchlorazole

B-695 metazachlor + terbuthylazine fenchlorazole

B-696 metazachlor + topramezone fenchlorazole

B-697 metribuzin + glyphosate fenchlorazole

B-698 pendimethalin + H-1 fenchlorazole

B-699 pendimethalin + clodinafop-propargyl fenchlorazole

B-700 pendimethalin + fenoxaprop-P-ethyl fenchlorazole

B-701 pendimethalin + flupyrsulfuron-methyl-sodium fenchlorazole

B-702 pendimethalin + glyphosate fenchlorazole

B-703 pendimethalin + mesosulfuron-methyl fenchlorazole

B-704 pendimethalin + mesotrione fenchlorazole

B-705 pendimethalin + nicosulfuron fenchlorazole

B-706 pendimethalin + pinoxaden fenchlorazole

B-707 pendimethalin + pyroxsulam fenchlorazole

B-708 pendimethalin + tembotrione fenchlorazole

B-709 pendimethalin + topramezone fenchlorazole

B-710 pyroxasulfone + tembotrione fenchlorazole

B-71 1 pyroxasulfone + topramezone fenchlorazole

B-712 sulfentrazone + glyphosate fenchlorazole

B-713 terbuthylazine + H-1 fenchlorazole

B-714 terbuthylazine + foramsulfuron fenchlorazole

B-715 terbuthylazine + glyphosate fenchlorazole

B-716 terbuthylazine + mesotrione fenchlorazole

B-717 terbuthylazine + nicosulfuron fenchlorazole

B-718 terbuthylazine + tembotrione fenchlorazole

B-719 terbuthylazine + topramezone fenchlorazole

B-720 trifluralin + glyphosate fenchlorazole

B-721 clodinafop-propargyl isoxadifen

B-722 cycloxydim isoxadifen

B-723 cyhalofop-butyl isoxadifen

B-724 fenoxaprop-P-ethyl isoxadifen

B-725 pinoxaden isoxadifen Herbicide(s) B Safener C

B-726 profoxydim isoxadifen

B-727 tepraloxydim isoxadifen

B-728 tralkoxydim isoxadifen

B-729 esprocarb isoxadifen

B-730 prosulfocarb isoxadifen

B-731 thiobencarb isoxadifen

B-732 triallate isoxadifen

B-733 bensulfuron-methyl isoxadifen

B-734 bispyribac-sodium isoxadifen

B-735 cyclosulfamuron isoxadifen

B-736 flumetsulam isoxadifen

B-737 flupyrsulfuron-methyl-sodium isoxadifen

B-738 foramsulfuron isoxadifen

B-739 imazamox isoxadifen

B-740 imazapic isoxadifen

B-741 imazapyr isoxadifen

B-742 imazaquin isoxadifen

B-743 imazethapyr isoxadifen

B-744 imazosulfuron isoxadifen

B-745 iodosulfuron-methyl-sodium isoxadifen

B-746 mesosulfuron isoxadifen

B-747 nicosulfuron isoxadifen

B-748 penoxsulam isoxadifen

B-749 propoxycarbazone-sodium isoxadifen

B-750 pyrazosulfuron-ethyl isoxadifen

B-751 pyroxsulam isoxadifen

B-752 rimsulfuron isoxadifen

B-753 sulfosulfuron isoxadifen

B-754 thiencarbazone-methyl isoxadifen

B-755 tritosulfuron isoxadifen

B-756 2,4-D and its salts and esters isoxadifen

B-757 aminopyralid and its salts and esters isoxadifen

B-758 clopyralid and its salts and esters isoxadifen

B-759 dicamba and its salts and esters isoxadifen

B-760 fluroxypyr-meptyl isoxadifen

B-761 quinclorac isoxadifen

B-762 quinmerac isoxadifen

B-763 H-9 isoxadifen

B-764 diflufenzopyr isoxadifen

B-765 diflufenzopyr-sodium isoxadifen Herbicide(s) B Safener C

B-766 clomazone isoxadifen

B-767 diflufenican isoxadifen

B-768 fluorochloridone isoxadifen

B-769 isoxaflutol isoxadifen

B-770 mesotrione isoxadifen

B-771 picolinafen isoxadifen

B-772 sulcotrione isoxadifen

B-773 tefuryltrione isoxadifen

B-774 tembotrione isoxadifen

B-775 topramezone isoxadifen

B-776 H-7 isoxadifen

B-777 atrazine isoxadifen

B-778 diuron isoxadifen

B-779 fluometuron isoxadifen

B-780 hexazinone isoxadifen

B-781 isoproturon isoxadifen

B-782 metribuzin isoxadifen

B-783 propanil isoxadifen

B-784 terbuthylazine isoxadifen

B-785 paraquat dichloride isoxadifen

B-786 flumioxazin isoxadifen

B-787 oxyfluorfen isoxadifen

B-788 saflufenacil isoxadifen

B-789 sulfentrazone isoxadifen

B-790 H-1 isoxadifen

B-791 H-2 isoxadifen

B-792 glyphosate isoxadifen

B-793 glyphosate-isopropylammonium isoxadifen

B-794 glyphosate-trimesium (sulfosate) isoxadifen

B-795 glufosinate isoxadifen

B-796 glufosinate-ammonium isoxadifen

B-797 pendimethalin isoxadifen

B-798 trifluralin isoxadifen

B-799 acetochlor isoxadifen

B-800 cafenstrole isoxadifen

B-801 dimethenamid-P isoxadifen

B-802 fentrazamide isoxadifen

B-803 flufenacet isoxadifen

B-804 mefenacet isoxadifen

B-805 metazachlor isoxadifen Herbicide(s) B Safener C

B-806 metolachlor-S isoxadifen

B-807 pyroxasulfone isoxadifen

B-808 isoxaben isoxadifen

B-809 dymron isoxadifen

B-810 indanofan isoxadifen

B-81 1 oxaziclomefone isoxadifen

B-812 triaziflam isoxadifen

B-813 atrazine + H-1 isoxadifen

B-814 atrazine + glyphosate isoxadifen

B-815 atrazine + mesotrione isoxadifen

B-816 atrazine + nicosulfuron isoxadifen

B-817 atrazine + tembotrione isoxadifen

B-818 atrazine + topramezone isoxadifen

B-819 clomazone + glyphosate isoxadifen

B-820 diflufenican + clodinafop-propargyl isoxadifen

B-821 diflufenican + fenoxaprop-P-ethyl isoxadifen

B-822 diflufenican + flupyrsulfuron-methyl-sodium isoxadifen

B-823 diflufenican + glyphosate isoxadifen

B-824 diflufenican + mesosulfuron-methyl isoxadifen

B-825 diflufenican + pinoxaden isoxadifen

B-826 diflufenican + pyroxsulam isoxadifen

B-827 flumetsulam + glyphosate isoxadifen

B-828 flumioxazin + glyphosate isoxadifen

B-829 imazapic + glyphosate isoxadifen

B-830 imazethapyr + glyphosate isoxadifen

B-831 isoxaflutol + H-1 isoxadifen

B-832 isoxaflutol + glyphosate isoxadifen

B-833 metazachlor + H-1 isoxadifen

B-834 metazachlor + glyphosate isoxadifen

B-835 metazachlor + mesotrione isoxadifen

B-836 metazachlor + nicosulfuron isoxadifen

B-837 metazachlor + terbuthylazine isoxadifen

B-838 metazachlor + topramezone isoxadifen

B-839 metribuzin + glyphosate isoxadifen

B-840 pendimethalin + H-1 isoxadifen

B-841 pendimethalin + clodinafop-propargyl isoxadifen

B-842 pendimethalin + fenoxaprop-P-ethyl isoxadifen

B-843 pendimethalin + flupyrsulfuron-methyl-sodium isoxadifen

B-844 pendimethalin + glyphosate isoxadifen

B-845 pendimethalin + mesosulfuron-methyl isoxadifen Herbicide(s) B Safener C

B-846 pendimethalin + mesotrione isoxadifen

B-847 pendimethalin + nicosulfuron isoxadifen

B-848 pendimethalin + pinoxaden isoxadifen

B-849 pendimethalin + pyroxsulam isoxadifen

B-850 pendimethalin + tembotrione isoxadifen

B-851 pendimethalin + topramezone isoxadifen

B-852 pyroxasulfone + tembotrione isoxadifen

B-853 pyroxasulfone + topramezone isoxadifen

B-854 sulfentrazone + glyphosate isoxadifen

B-855 terbuthylazine + H-1 isoxadifen

B-856 terbuthylazine + foramsulfuron isoxadifen

B-857 terbuthylazine + glyphosate isoxadifen

B-858 terbuthylazine + mesotrione isoxadifen

B-859 terbuthylazine + nicosulfuron isoxadifen

B-860 terbuthylazine + tembotrione isoxadifen

B-861 terbuthylazine + topramezone isoxadifen

B-862 trifluralin + glyphosate isoxadifen

B-863 clodinafop-propargyl mefenpyr

B-864 cycloxydim mefenpyr

B-865 cyhalofop-butyl mefenpyr

B-866 fenoxaprop-P-ethyl mefenpyr

B-867 pinoxaden mefenpyr

B-868 profoxydim mefenpyr

B-869 tepraloxydim mefenpyr

B-870 tralkoxydim mefenpyr

B-871 esprocarb mefenpyr

B-872 prosulfocarb mefenpyr

B-873 thiobencarb mefenpyr

B-874 triallate mefenpyr

B-875 bensulfuron-methyl mefenpyr

B-876 bispyribac-sodium mefenpyr

B-877 cyclosulfamuron mefenpyr

B-878 flumetsulam mefenpyr

B-879 flupyrsulfuron-methyl-sodium mefenpyr

B-880 foramsulfuron mefenpyr

B-881 imazamox mefenpyr

B-882 imazapic mefenpyr

B-883 imazapyr mefenpyr

B-884 imazaquin mefenpyr

B-885 imazethapyr mefenpyr Herbicide(s) B Safener C

B-886 imazosulfuron mefenpyr

B-887 iodosulfuron-methyl-sodium mefenpyr

B-888 mesosulfuron mefenpyr

B-889 nicosulfuron mefenpyr

B-890 penoxsulam mefenpyr

B-891 propoxycarbazone-sodium mefenpyr

B-892 pyrazosulfuron-ethyl mefenpyr

B-893 pyroxsulam mefenpyr

B-894 rimsulfuron mefenpyr

B-895 sulfosulfuron mefenpyr

B-896 thiencarbazone-methyl mefenpyr

B-897 tritosulfuron mefenpyr

B-898 2,4-D and its salts and esters mefenpyr

B-899 aminopyralid and its salts and esters mefenpyr

B-900 clopyralid and its salts and esters mefenpyr

B-901 dicamba and its salts and esters mefenpyr

B-902 fluroxypyr-meptyl mefenpyr

B-903 quinclorac mefenpyr

B-904 quinmerac mefenpyr

B-905 H-9 mefenpyr

B-906 diflufenzopyr mefenpyr

B-907 diflufenzopyr-sodium mefenpyr

B-908 clomazone mefenpyr

B-909 diflufenican mefenpyr

B-910 fluorochloridone mefenpyr

B-91 1 isoxaflutol mefenpyr

B-912 mesotrione mefenpyr

B-913 picolinafen mefenpyr

B-914 sulcotrione mefenpyr

B-915 tefuryltrione mefenpyr

B-916 tembotrione mefenpyr

B-917 topramezone mefenpyr

B-918 H-7 mefenpyr

B-919 atrazine mefenpyr

B-920 diuron mefenpyr

B-921 fluometuron mefenpyr

B-922 hexazinone mefenpyr

B-923 isoproturon mefenpyr

B-924 metribuzin mefenpyr

B-925 propanil mefenpyr Herbicide(s) B Safener C

B-926 terbuthylazine mefenpyr

B-927 paraquat dichloride mefenpyr

B-928 flumioxazin mefenpyr

B-929 oxyfluorfen mefenpyr

B-930 saflufenacil mefenpyr

B-931 sulfentrazone mefenpyr

B-932 H-1 mefenpyr

B-933 H-2 mefenpyr

B-934 glyphosate mefenpyr

B-935 glyphosate-isopropylammonium mefenpyr

B-936 glyphosate-trimesium (sulfosate) mefenpyr

B-937 glufosinate mefenpyr

B-938 glufosinate-ammonium mefenpyr

B-939 pendimethalin mefenpyr

B-940 trifluralin mefenpyr

B-941 acetochlor mefenpyr

B-942 cafenstrole mefenpyr

B-943 dimethenamid-P mefenpyr

B-944 fentrazamide mefenpyr

B-945 flufenacet mefenpyr

B-946 mefenacet mefenpyr

B-947 metazachlor mefenpyr

B-948 metolachlor-S mefenpyr

B-949 pyroxasulfone mefenpyr

B-950 isoxaben mefenpyr

B-951 dymron mefenpyr

B-952 indanofan mefenpyr

B-953 oxaziclomefone mefenpyr

B-954 triaziflam mefenpyr

B-955 atrazine + H-1 mefenpyr

B-956 atrazine + glyphosate mefenpyr

B-957 atrazine + mesotrione mefenpyr

B-958 atrazine + nicosulfuron mefenpyr

B-959 atrazine + tembotrione mefenpyr

B-960 atrazine + topramezone mefenpyr

B-961 clomazone + glyphosate mefenpyr

B-962 diflufenican + clodinafop-propargyl mefenpyr

B-963 diflufenican + fenoxaprop-P-ethyl mefenpyr

B-964 diflufenican + flupyrsulfuron-methyl-sodium mefenpyr

B-965 diflufenican + glyphosate mefenpyr Herbicide(s) B Safener C

B-966 diflufenican + mesosulfuron-methyl mefenpyr

B-967 diflufenican + pinoxaden mefenpyr

B-968 diflufenican + pyroxsulam mefenpyr

B-969 flumetsulam + glyphosate mefenpyr

B-970 flumioxazin + glyphosate mefenpyr

B-971 imazapic + glyphosate mefenpyr

B-972 imazethapyr + glyphosate mefenpyr

B-973 isoxaflutol + H-1 mefenpyr

B-974 isoxaflutol + glyphosate mefenpyr

B-975 metazachlor + H-1 mefenpyr

B-976 metazachlor + glyphosate mefenpyr

B-977 metazachlor + mesotrione mefenpyr

B-978 metazachlor + nicosulfuron mefenpyr

B-979 metazachlor + terbuthylazine mefenpyr

B-980 metazachlor + topramezone mefenpyr

B-981 metribuzin + glyphosate mefenpyr

B-982 pendimethalin + H-1 mefenpyr

B-983 pendimethalin + clodinafop-propargyl mefenpyr

B-984 pendimethalin + fenoxaprop-P-ethyl mefenpyr

B-985 pendimethalin + flupyrsulfuron-methyl-sodium mefenpyr

B-986 pendimethalin + glyphosate mefenpyr

B-987 pendimethalin + mesosulfuron-methyl mefenpyr

B-988 pendimethalin + mesotrione mefenpyr

B-989 pendimethalin + nicosulfuron mefenpyr

B-990 pendimethalin + pinoxaden mefenpyr

B-991 pendimethalin + pyroxsulam mefenpyr

B-992 pendimethalin + tembotrione mefenpyr

B-993 pendimethalin + topramezone mefenpyr

B-994 pyroxasulfone + tembotrione mefenpyr

B-995 pyroxasulfone + topramezone mefenpyr

B-996 sulfentrazone + glyphosate mefenpyr

B-997 terbuthylazine + H-1 mefenpyr

B-998 terbuthylazine + foramsulfuron mefenpyr

B-999 terbuthylazine + glyphosate mefenpyr

B-1000 terbuthylazine + mesotrione mefenpyr

B-1001 terbuthylazine + nicosulfuron mefenpyr

B-1002 terbuthylazine + tembotrione mefenpyr

B-1003 terbuthylazine + topramezone mefenpyr

B-1004 trifluralin + glyphosate mefenpyr

B-1005 clodinafop-propargyl H-12 Herbicide(s) B Safener C

B-1006 cycloxydim H-12

B-1007 cyhalofop-butyl H-12

B-1008 fenoxaprop-P-ethyl H-12

B-1009 pinoxaden H-12

B-1010 profoxydim H-12

B-101 1 tepraloxydim H-12

B-1012 tralkoxydim H-12

B-1013 esprocarb H-12

B-1014 prosulfocarb H-12

B-1015 thiobencarb H-12

B-1016 triallate H-12

B-1017 bensulfuron-methyl H-12

B-1018 bispyribac-sodium H-12

B-1019 cyclosulfamuron H-12

B-1020 flumetsulam H-12

B-1021 flupyrsulfuron-methyl-sodium H-12

B-1022 foramsulfuron H-12

B-1023 imazamox H-12

B-1024 imazapic H-12

B-1025 imazapyr H-12

B-1026 imazaquin H-12

B-1027 imazethapyr H-12

B-1028 imazosulfuron H-12

B-1029 iodosulfuron-methyl-sodium H-12

B-1030 mesosulfuron H-12

B-1031 nicosulfuron H-12

B-1032 penoxsulam H-12

B-1033 propoxycarbazone-sodium H-12

B-1034 pyrazosulfuron-ethyl H-12

B-1035 pyroxsulam H-12

B-1036 rimsulfuron H-12

B-1037 sulfosulfuron H-12

B-1038 thiencarbazone-methyl H-12

B-1039 tritosulfuron H-12

B-1040 2,4-D and its salts and esters H-12

B-1041 aminopyralid and its salts and esters H-12

B-1042 clopyralid and its salts and esters H-12

B-1043 dicamba and its salts and esters H-12

B-1044 fluroxypyr-meptyl H-12

B-1045 quinclorac H-12 Herbicide(s) B Safener C

B-1046 quinmerac H-12

B-1047 B-9 H-12

B-1048 diflufenzopyr H-12

B-1049 diflufenzopyr-sodium H-12

B-1050 clomazone H-12

B-1051 diflufenican H-12

B-1052 fluorochloridone H-12

B-1053 isoxaflutol H-12

B-1054 mesotrione H-12

B-1055 picolinafen H-12

B-1056 sulcotrione H-12

B-1057 tefuryltrione H-12

B-1058 tembotrione H-12

B-1059 topramezone H-12

B-1060 H-7 H-12

B-1061 atrazine H-12

B-1062 diuron H-12

B-1063 fluometuron H-12

B-1064 hexazinone H-12

B-1065 isoproturon H-12

B-1066 metribuzin H-12

B-1067 propanil H-12

B-1068 terbuthylazine H-12

B-1069 paraquat dichloride H-12

B-1070 flumioxazin H-12

B-1071 oxyfluorfen H-12

B-1072 saflufenacil H-12

B-1073 sulfentrazone H-12

B-1074 H-1 H-12

B-1075 H-2 H-12

B-1076 glyphosate H-12

B-1077 glyphosate-isopropylammonium H-12

B-1078 glyphosate-trimesium (sulfosate) H-12

B-1079 glufosinate H-12

B-1080 glufosinate-ammonium H-12

B-1081 pendimethalin H-12

B-1082 trifluralin H-12

B-1083 acetochlor H-12

B-1084 cafenstrole H-12

B-1085 dimethenamid-P H-12 Herbicide(s) B Safener C

B-1086 fentrazamide H-12

B-1087 flufenacet H-12

B-1088 mefenacet H-12

B-1089 metazachlor H-12

B-1090 metolachlor-S H-12

B-1091 pyroxasulfone H-12

B-1092 isoxaben H-12

B-1093 dymron H-12

B-1094 indanofan H-12

B-1095 oxaziclomefone H-12

B-1096 triaziflam H-12

B-1097 atrazine + H-1 H-12

B-1098 atrazine + glyphosate H-12

B-1099 atrazine + mesotrione H-12

B-1100 atrazine + nicosulfuron H-12

B-1101 atrazine + tembotrione H-12

B-1102 atrazine + topramezone H-12

B-1103 clomazone + glyphosate H-12

B-1104 diflufenican + clodinafop-propargyl H-12

B-1105 diflufenican + fenoxaprop-P-ethyl H-12

B-1106 diflufenican + flupyrsulfuron-methyl-sodium H-12

B-1107 diflufenican + glyphosate H-12

B-1108 diflufenican + mesosulfuron-methyl H-12

B-1109 diflufenican + pinoxaden H-12

B-1110 diflufenican + pyroxsulam H-12

B-1111 flumetsulam + glyphosate H-12

B-1112 flumioxazin + glyphosate H-12

B-1113 imazapic + glyphosate H-12

B-1114 imazethapyr + glyphosate H-12

B-1115 isoxaflutol + H-1 H-12

B-1116 isoxaflutol + glyphosate H-12

B-1117 metazachlor + H-1 H-12

B-1118 metazachlor + glyphosate H-12

B-1119 metazachlor + mesotrione H-12

B-1120 metazachlor + nicosulfuron H-12

B-1121 metazachlor + terbuthylazine H-12

B-1122 metazachlor + topramezone H-12

B-1123 metribuzin + glyphosate H-12

B-1124 pendimethalin + H-1 H-12

B-1125 pendimethalin + clodinafop-propargyl H-12 Herbicide(s) B Safener C

B-1126 pendimethalin + fenoxaprop-P-ethyl H-12

B-1127 pendimethalin + flupyrsulfuron-methyl-sodium H-12

B-1128 pendimethalin + glyphosate H-12

B-1129 pendimethalin + mesosulfuron-methyl H-12

B-1130 pendimethalin + mesotrione H-12

B-1131 pendimethalin + nicosulfuron H-12

B-1132 pendimethalin + pinoxaden H-12

B-1133 pendimethalin + pyroxsulam H-12

B-1134 pendimethalin + tembotrione H-12

B-1135 pendimethalin + topramezone H-12

B-1136 pyroxasulfone + tembotrione H-12

B-1137 pyroxasulfone + topramezone H-12

B-1138 sulfentrazone + glyphosate H-12

B-1139 terbuthylazine + H-1 H-12

B-1140 terbuthylazine + foramsulfuron H-12

B-1141 terbuthylazine + glyphosate H-12

B-1142 terbuthylazine + mesotrione H-12

B-1143 terbuthylazine + nicosulfuron H-12

B-1144 terbuthylazine + tembotrione H-12

B-1145 terbuthylazine + topramezone H-12

B-1146 trifluralin + glyphosate H-12

B-1147 2-1 —

B-1148 2-2 —

B-1149 2-3 —

B-1150 2-4 —

B-1151 2-5 —

B-1152 2-6 —

B-1153 2-7 —

B-1154 2-8 —

B-1155 2-9 —

B-1156 2-1 benoxacor

B-1157 2-2 benoxacor

B-1158 2-3 benoxacor

B-1159 2-4 benoxacor

B-1160 2-5 benoxacor

B-1161 2-6 benoxacor

B-1162 2-7 benoxacor

B-1163 2-8 benoxacor

B-1164 2-9 benoxacor

B-1165 2-1 cloquintocet Herbicide(s) B Safener C

B-1166 2-2 cloquintocet

B-1167 2-3 cloquintocet

B-1168 2-4 cloquintocet

B-1169 2-5 cloquintocet

B-1170 2-6 cloquintocet

B-1171 2-7 cloquintocet

B-1172 2-8 cloquintocet

B-1173 2-9 cloquintocet

B-1174 2-1 cyprosulfamide

B-1175 2-2 cyprosulfamide

B-1176 2-3 cyprosulfamide

B-1177 2-4 cyprosulfamide

B-1178 2-5 cyprosulfamide

B-1179 2-6 cyprosulfamide

B-1180 2-7 cyprosulfamide

B-1181 2-8 cyprosulfamide

B-1182 2-9 cyprosulfamide

B-1183 2-1 dichlormid

B-1184 2-2 dichlormid

B-1185 2-3 dichlormid

B-1186 2-4 dichlormid

B-1187 2-5 dichlormid

B-1188 2-6 dichlormid

B-1189 2-7 dichlormid

B-1190 2-8 dichlormid

B-1191 2-9 dichlormid

B-1192 2-1 fenchlorazole

B-1193 2-2 fenchlorazole

B-1194 2-3 fenchlorazole

B-1195 2-4 fenchlorazole

B-1196 2-5 fenchlorazole

B-1197 2-6 fenchlorazole

B-1198 2-7 fenchlorazole

B-1199 2-8 fenchlorazole

B-1200 2-9 fenchlorazole

B-1201 2-1 isoxadifen

B-1202 2-2 isoxadifen

B-1203 2-3 isoxadifen

B-1204 2-4 isoxadifen

B-1205 2-5 isoxadifen Herbicide(s) B Safener C

B-1206 2-6 isoxadifen

B-1207 2-7 isoxadifen

B-1208 2-8 isoxadifen

B-1209 2-9 isoxadifen

B-1210 2-1 mefenpyr

B-121 1 2-2 mefenpyr

B-1212 2-3 mefenpyr

B-1213 2-4 mefenpyr

B-1214 2-5 mefenpyr

B-1215 2-6 mefenpyr

B-1216 2-7 mefenpyr

B-1217 2-8 mefenpyr

B-1218 2-9 mefenpyr

B-1219 2-1 H-1 1

B-1220 2-2 H-1 1

B-1221 2-3 H-1 1

B-1222 2-4 H-1 1

B-1223 2-5 H-1 1

B-1224 2-6 H-1 1

B-1225 2-7 H-1 1

B-1226 2-8 H-1 1

B-1227 2-9 H-1 1

B-1228 2-1 H-12

B-1229 2-2 H-12

B-1230 2-3 H-12

B-1231 2-4 H-12

B-1232 2-5 H-12

B-1233 2-6 H-12

B-1234 2-7 H-12

B-1235 2-8 H-12

B-1236 2-9 H-12

The compounds of formula I and the compositions according to the invention may also have a plant-strengthening action. Accordingly, they are suitable for mobilizing the defense system of the plants against attack by unwanted microorganisms, such as harmful fungi, but also viruses and bacteria. Plant-strengthening (resistance-inducing) substances are to be understood as meaning, in the present context, those substances which are capable of stimulating the defense system of treated plants in such a way that, when subsequently inoculated by unwanted microorganisms, the treated plants display a substantial degree of resistance to these microorganisms. The compounds of formula I can be employed for protecting plants against attack by unwanted microorganisms within a certain period of time after the treatment. The period of time within which their protection is effected generally extends from 1 to 28 days, preferably from 1 to

14 days, after the treatment of the plants with the compounds of formula I, or, after treatment of the seed, for up to 9 months after sowing.

The compounds of formula I and the compositions according to the invention are also suitable for increasing the harvest yield.

Moreover, they have reduced toxicity and are tolerated well by the plants. Use examples

The herbicidal activity of the compunds of the formula I was demonstrated by the following greenhouse experiments:

The culture containers used were plastic flowerpots containing loamy sand with approximately 3.0% of humus as the substrate. The seeds of the test plants were sown separately for each species.

For the pre-emergence treatment, the active ingredients, which had been suspended or emulsified in water, were applied directly after sowing by means of finely distributing nozzles. The containers were irrigated gently to promote germination and growth and subsequently cov- ered with transparent plastic hoods until the plants had rooted. This cover caused uniform germination of the test plants, unless this has been impaired by the active ingredients.

For the post-emergence treatment, the test plants were first grown to a height of 3 to

15 cm, depending on the plant habit, and only then treated with the active ingredients which had been suspended or emulsified in water. For this purpose, the test plants were either sown directly and grown in the same containers, or they were first grown separately as seedlings and transplanted into the test containers a few days prior to treatment.

Depending on the species, the plants were kept at 10-25°C or 20-35°C. The test period extended over 2 to 4 weeks. During this time, the plants were tended, and their response to the individual treatments was evaluated.

Evaluation was carried out using a scale from 0 to 100. 100 means no emergence of the plants, or complete destruction of at least the aerial moieties, and 0 means no damage, or normal course of growth. A good herbicidal activity is given at values of at least 70 and a very good herbicidal activity is given at values of at least 85.