Title:
SULFAMOYL BENZOIC ACID HETEROBICYCLIC DERIVATIVES AS TRPM8 ANTAGONISTS
Document Type and Number:
WIPO Patent Application WO/2012/042915
Kind Code:
A1
Abstract:
The present invention relates to sulfamoyl benzoic acid heterobicyclic derivatives of the formula (I) or a pharmaceutically acceptable salt thereof or a prodrug thereof, processes for their preparation, pharmaceutical compositions containing them and their use in the treatment of various disorders which are mediated via the TRPM8 receptor.
Inventors:
KAWAMURA KIYOSHI (JP)
SHISHIDO YUJI (JP)
OHMI MASASHI (JP)
SHISHIDO YUJI (JP)
OHMI MASASHI (JP)
Application Number:
PCT/JP2011/005588
Publication Date:
April 05, 2012
Filing Date:
October 03, 2011
Export Citation:
Assignee:
RAQUALIA PHARMA INC (JP)
KAWAMURA KIYOSHI (JP)
SHISHIDO YUJI (JP)
OHMI MASASHI (JP)
KAWAMURA KIYOSHI (JP)
SHISHIDO YUJI (JP)
OHMI MASASHI (JP)
International Classes:
C07D401/12; A61K31/443; A61K31/4439; A61K31/444; A61K31/4709; A61P13/00; A61P25/00; A61P29/00; A61P43/00; C07D209/08; C07D215/12; C07D231/56; C07D249/18; C07D307/79; C07D405/04; C07D405/12; C07D405/14; C07D471/04
Domestic Patent References:
| WO2009012430A1 | 2009-01-22 | |||
| WO2009025793A2 | 2009-02-26 | |||
| WO2011113861A2 | 2011-09-22 | |||
| WO2010151797A2 | 2010-12-29 | |||
| WO2009153285A2 | 2009-12-23 | |||
| WO2008157500A1 | 2008-12-24 |
Foreign References:
| JP2007505849A | 2007-03-15 | |||
| JP2006514614A | 2006-05-11 | |||
| JPH05323534A | 1993-12-07 | |||
| US5441563A | 1995-08-15 |
Other References:
DATABASE REGISTRY Database accession no. 310890-89-2
Attorney, Agent or Firm:
IWATANI, Ryo (1-31 Dojima 2-chome, Kita-ku, Osaka-sh, Osaka 03, JP)
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Claims: