Title:
SYNTHESIS OF SUBSTITUTED PYRAZOLINE CARBOXAMIDINE DERIVATIVES
Document Type and Number:
WIPO Patent Application WO/2011/092226
Kind Code:
A8
Abstract:
This invention relates to organic chemistry, in particular to processes for the preparation of pyrazoline carboxamidine derivatives of formula (I), known as potent 5-HT6 antagonists. The invention also relates to novel intermediates of these compounds. wherein the symbols have the meanings given in the description.
Inventors:
VAN LOEVEZIJN ARNOLD (NL)
LANGE JOSEPHUS H M (NL)
BARF GERRIT A (NL)
DEN HARTOG ARNOLD P (NL)
LANGE JOSEPHUS H M (NL)
BARF GERRIT A (NL)
DEN HARTOG ARNOLD P (NL)
Application Number:
PCT/EP2011/051100
Publication Date:
September 07, 2012
Filing Date:
January 27, 2011
Export Citation:
Assignee:
ABBOTT HEALTHCARE PRODUCTS BV (NL)
VAN LOEVEZIJN ARNOLD (NL)
LANGE JOSEPHUS H M (NL)
BARF GERRIT A (NL)
DEN HARTOG ARNOLD P (NL)
VAN LOEVEZIJN ARNOLD (NL)
LANGE JOSEPHUS H M (NL)
BARF GERRIT A (NL)
DEN HARTOG ARNOLD P (NL)
International Classes:
C07D231/06; C07D231/54; C07D409/04; C07D409/12; C07D491/107; C07D513/10
Attorney, Agent or Firm:
JANSEN, C.M. et al. (Johan de Wittlaan 7, JR The Hague, NL)
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