Title:
THERAPEUTIC COMPOUNDS AND METHODS OF USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2018/072602
Kind Code:
A1
Abstract:
The invention provides a compound of formula I: or a pharmaceutically acceptable salt thereof, wherein the variables X, Y1-Y5, R1, R2, R3, R4, and Het have the meaning as described herein, and compositions containing such compounds and methods for using such compounds and compositions.
Inventors:
SUTHERLIN DANIEL (US)
MCKERRALL STEVEN (US)
WILSON MICHAEL SCOTT (CA)
LAI KWONG WAH (CN)
BERGERON PHILIPPE (US)
ZHANG BIRONG (US)
MCKERRALL STEVEN (US)
WILSON MICHAEL SCOTT (CA)
LAI KWONG WAH (CN)
BERGERON PHILIPPE (US)
ZHANG BIRONG (US)
Application Number:
PCT/CN2017/103499
Publication Date:
April 26, 2018
Filing Date:
September 26, 2017
Export Citation:
Assignee:
GENENTECH INC (US)
XENON PHARMACEUTICALS INC (CA)
SUTHERLIN DANIEL (US)
MCKERRALL STEVEN (US)
WILSON MICHAEL SCOTT (CA)
LAI KWONG WAH (CN)
BERGERON PHILIPPE (US)
ZHANG BIRONG (US)
XENON PHARMACEUTICALS INC (CA)
SUTHERLIN DANIEL (US)
MCKERRALL STEVEN (US)
WILSON MICHAEL SCOTT (CA)
LAI KWONG WAH (CN)
BERGERON PHILIPPE (US)
ZHANG BIRONG (US)
International Classes:
A61K31/427; C07D285/08; A61P19/02
Domestic Patent References:
WO2013064983A1 | 2013-05-10 |
Foreign References:
EP2813491A1 | 2014-12-17 | |||
EP2974730A1 | 2016-01-20 |
Other References:
See also references of EP 3526205A4
Attorney, Agent or Firm:
WU, FENG & ZHANG (CN)
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