Title:
THIOPHENE DERIVATIVE
Document Type and Number:
WIPO Patent Application WO/2010/126167
Kind Code:
A1
Abstract:
Disclosed are: a compound represented by formula (I), or a salt, solvate or physiologically functional derivative thereof; and a pharmaceutical composition comprising the compound or the salt, solvate or physiologically functional derivative thereof, which is useful for the treatment or prevention of conditions or disorders that are sensitive to selective androgen receptor modulation.
Inventors:
HARADA KOICHIRO (JP)
MOTONAGA KOZO (JP)
SAITO KOICHI (JP)
TANAKA AKIO (JP)
MOTONAGA KOZO (JP)
SAITO KOICHI (JP)
TANAKA AKIO (JP)
Application Number:
PCT/JP2010/057917
Publication Date:
November 04, 2010
Filing Date:
April 28, 2010
Export Citation:
Assignee:
SUMITOMO CHEMICAL CO (JP)
HARADA KOICHIRO (JP)
MOTONAGA KOZO (JP)
SAITO KOICHI (JP)
TANAKA AKIO (JP)
HARADA KOICHIRO (JP)
MOTONAGA KOZO (JP)
SAITO KOICHI (JP)
TANAKA AKIO (JP)
International Classes:
C07D333/36; A61K31/381; A61K31/4025; A61K31/4535; A61P3/04; A61P3/06; A61P3/10; A61P5/26; A61P9/10; A61P13/02; A61P13/06; A61P15/08; A61P15/10; A61P17/00; A61P17/08; A61P17/10; A61P17/14; A61P19/10; A61P21/00; A61P25/24; A61P25/28; A61P35/00; A61P43/00; C07D333/38; C07D409/04; C07D409/12
Domestic Patent References:
| WO2007076423A2 | 2007-07-05 | |||
| WO2000021928A1 | 2000-04-20 | |||
| WO2003062241A1 | 2003-07-31 | |||
| WO2002028353A2 | 2002-04-11 | |||
| WO2005073395A1 | 2005-08-11 |
Foreign References:
| GB1334015A | 1973-10-17 | |||
| JPS6447781A | 1989-02-22 | |||
| JPS4986361A | 1974-08-19 | |||
| US20030078248A1 | 2003-04-24 |
Other References:
HURD, CHARLES D. ET AL.: "Diazo reactions in the thiophene and furan series", JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, vol. 69, 1947, pages 859 - 864, XP008154665
MIGIANU, EVELYNE. ET AL.: "Regioselective Nucleophilic Aromatic Substitution: Unexpected Results in the Thiophene Series", SYNLETT, vol. 8, 2000, pages 459 - 462, XP008154672
STANETTY, PETER ET AL.: "Herbicidal thienylureas. I", MONATSHEFTE FUER CHEMIE, vol. 120, no. 1, 1989, pages 53 - 63, XP008154675
STANETTY, PETER ET AL.: "Herbicidal thienylureas. II", MONATSHEFTE FUER CHEMIE, vol. 120, no. 1, 1989, pages 65 - 72, XP008154674
CONSIGLIO, GIOVANNI ET AL.: "Secondary steric effects in SNAr of thiophenes: a coordinate kinetic, thermodynamic, UV-VIS, crystallographic and ab initio study", JOURNAL OF THE CHEMICAL SOCIETY, PERKIN TRANSACTIONS 2: PHYSICAL ORGANIC CHEMISTRY, vol. 2, 1997, pages 309 - 316, XP008154667
T. HIGUCHI; V. STELLA: "Prodrugs as Novel Delivery Systems", A.C.S. SYMPOSIUM SERIES, vol. 14
"Bioreversible Carriers in Drug Design", 1987, AMERICAN PHARMACEUTICAL ASSOCIATION AND PERGAMON
T. W. GREEN; P. G. M. NUTS: "Protecting Groups in Organic Synthesis", 1991, JOHN WILEY & SONS
PHARMACEUTICAL RESEARCH, vol. 3, no. 6, 1986, pages 318
See also references of EP 2426117A4
MIGIANU, EVELYNE. ET AL.: "Regioselective Nucleophilic Aromatic Substitution: Unexpected Results in the Thiophene Series", SYNLETT, vol. 8, 2000, pages 459 - 462, XP008154672
STANETTY, PETER ET AL.: "Herbicidal thienylureas. I", MONATSHEFTE FUER CHEMIE, vol. 120, no. 1, 1989, pages 53 - 63, XP008154675
STANETTY, PETER ET AL.: "Herbicidal thienylureas. II", MONATSHEFTE FUER CHEMIE, vol. 120, no. 1, 1989, pages 65 - 72, XP008154674
CONSIGLIO, GIOVANNI ET AL.: "Secondary steric effects in SNAr of thiophenes: a coordinate kinetic, thermodynamic, UV-VIS, crystallographic and ab initio study", JOURNAL OF THE CHEMICAL SOCIETY, PERKIN TRANSACTIONS 2: PHYSICAL ORGANIC CHEMISTRY, vol. 2, 1997, pages 309 - 316, XP008154667
T. HIGUCHI; V. STELLA: "Prodrugs as Novel Delivery Systems", A.C.S. SYMPOSIUM SERIES, vol. 14
"Bioreversible Carriers in Drug Design", 1987, AMERICAN PHARMACEUTICAL ASSOCIATION AND PERGAMON
T. W. GREEN; P. G. M. NUTS: "Protecting Groups in Organic Synthesis", 1991, JOHN WILEY & SONS
PHARMACEUTICAL RESEARCH, vol. 3, no. 6, 1986, pages 318
See also references of EP 2426117A4
Attorney, Agent or Firm:
NAKAYAMA, Tohru et al. (JP)
Toru Nakayama (JP)
Toru Nakayama (JP)
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