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Title:
TRICYCLIC DIHYDROIMIDAZOPYRIMIDONE DERIVATIVE, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND USE THEREOF
Document Type and Number:
WIPO Patent Application WO/2021/089032
Kind Code:
A1
Abstract:
Disclosed are a compound as represented by general formula (I), a cis-trans isomer thereof, an enantiomer thereof, a diastereoisomer thereof, a racemate thereof, a solvate thereof, a hydrate thereof, or a pharmaceutically acceptable salt thereof or a prodrug thereof, a preparation method therefor, a pharmaceutical composition comprising the compound and the use of the compound as an Lp-PLA2 inhibitor.

Inventors:
JIN YUN (CN)
WU JINHUA (CN)
PENG JUN (CN)
SUN YONG (CN)
Application Number:
PCT/CN2020/127426
Publication Date:
May 14, 2021
Filing Date:
November 09, 2020
Export Citation:
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Assignee:
SHANGHAI SIMR BIOTECHNOLOGY CO LTD (CN)
SHANGHAI SIMRD BIOTECHNOLOGY CO LTD (CN)
International Classes:
C07D487/14; A61K31/519; A61K31/527; A61P9/10; A61P25/28; C07D487/20; C07D491/20; C07D513/12
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See also references of EP 4056571A4
Attorney, Agent or Firm:
CCPIT PATENT AND TRADEMARK LAW OFFICE (CN)
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