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Patent Searching and Data


Title:
TRPA1 ANTAGONIST COMPOUNDS
Document Type and Number:
WIPO Patent Application WO/2014/184248
Kind Code:
A3
Abstract:
Compounds of Formula (I), pharmaceutically acceptable salts thereof, diastereomers, enantiomers, or mixtures thereof: wherein R1, R2, R3, X, Yn and A are as defined in the specification, as well as pharmaceutical compositions including the compounds are prepared. They are useful in therapy, in particular in the management of pain.

Inventors:
SVENSSON MATS A (US)
WEIGELT DIRK (SE)
Application Number:
PCT/EP2014/059853
Publication Date:
December 31, 2014
Filing Date:
May 14, 2014
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Assignee:
ACTURUM LIFE SCIENCE AB (SE)
International Classes:
C07C275/18; C07D211/34; C07D217/06; C07D295/16; C07D401/04; C07D403/04; C07D413/04; C07D417/04
Domestic Patent References:
WO2012050512A12012-04-19
Other References:
VALLIN K S ET AL: "N-1-Alkyl-2-oxo-2-aryl amides as novel antagonists of the TRPA1 receptor", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, PERGAMON, AMSTERDAM, NL, vol. 22, no. 17, 1 September 2012 (2012-09-01), pages 5485 - 5492, XP002716178, ISSN: 0960-894X, [retrieved on 20120714], DOI: 10.1016/J.BMCL.2012.07.032
Attorney, Agent or Firm:
NEELISSEN-SUBNEL, Marianne (c/o NellpatBox 138, Hagford, SE)
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