Title:
VORTIOXETINE ANALOGUE AND USE AND PREPARATION THEREOF
Document Type and Number:
WIPO Patent Application WO/2018/014880
Kind Code:
A1
Abstract:
Provided are a vortioxetine analogue as shown in formula I or a polymorph or a solvate thereof, a composition and a kit comprising the analogue, polymorph or solvate, the use of the analogue, polymorph or solvate in the preparation of a drug for treating depression, a method for preparing the analogue, and intermediates in the method.
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Inventors:
LI QINGENG (CN)
WANG TAO (CN)
LIAO JIAN (CN)
XU XIANGQING (CN)
REN LIANG (CN)
WANG TAO (CN)
LIAO JIAN (CN)
XU XIANGQING (CN)
REN LIANG (CN)
Application Number:
PCT/CN2017/094037
Publication Date:
January 25, 2018
Filing Date:
July 24, 2017
Export Citation:
Assignee:
LI QINGENG (CN)
International Classes:
C07D295/096; A61K31/495; A61P25/24; C07C319/02; C07C321/26; C07D295/185; C07D295/192; C07D295/205
Domestic Patent References:
| WO2015107057A1 | 2015-07-23 | |||
| WO1993016067A1 | 1993-08-19 |
Foreign References:
| CN1561336A | 2005-01-05 | |||
| CN101709045A | 2010-05-19 | |||
| GB281290A | 1928-11-01 |
Other References:
DATABASE CAS 4 December 2015 (2015-12-04), retrieved from STN Database accession no. 75.2659
BANDGAR, B.P. ET AL.: "Rapid Synthesis of Thiophenols Under Mild and Non-Aqueous Conditions", SULFUR LETTERS, vol. 24, no. 3, 31 December 2000 (2000-12-31), pages 123 - 126, XP009514644
See also references of EP 3489225A4
BANDGAR, B.P. ET AL.: "Rapid Synthesis of Thiophenols Under Mild and Non-Aqueous Conditions", SULFUR LETTERS, vol. 24, no. 3, 31 December 2000 (2000-12-31), pages 123 - 126, XP009514644
See also references of EP 3489225A4
Attorney, Agent or Firm:
NTD UNIVATION INTELLECTUAL PROPERTY AGENCY LTD. (CN)
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