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Matches 551 - 600 out of 4,769

Document Document Title
JP3647041B2
Modified amino acid compounds useful for the delivery of active agents are provided. The amino acids, non-alpha-amino acids, have been modified by acylation on the amino group particularly with phenyl or cyclohexyl groups. These groups h...  
JP3639313B2
PURPOSE: To obtain the subject new compounds useful for antibiotic agents or the like indicating excellent antimicrobial activity against tetralin resistant microbe or the like. CONSTITUTION: The compound of formula I or II (X is a halog...  
JP2005509590A
Disclosed is a compound represented by Structural Formula (I): Ar is a substituted or unsubstituted aromatic group. Q is a covalent bond, -CH2- or -CH2CH2-; W is a substituted or unsubstituted alkylene or a substituted or unsubstituted h...  
JP3637924B2
PURPOSE: To provide an industrially advantageous method capable of producing crystal of a high-purity N-chloro aromatic carboxylic acid amide having excellent stirring properties and filtering characteristics by a reaction of short time ...  
JP2005089458A
To provide another method to perform oxidative reaction of an organic substrate in the presence of an organorhenium oxide and its derivative when an easily available rhenium catalyst is used to lower the whole cost for preparation of the...  
JP3633640B2
PURPOSE: To obtain a new compound having strong antibacterial action particularly on tetracycline resistant bacteria and which is useful as an antibiotic. CONSTITUTION: This compound of formula I (R is H, a 1-8C alkyl, an α-hydroxy (1-4...  
JP3634749B2
The present invention relates to a pharmaceutical composition comprising as an active ingredient a compound of formula (I), wherein Ring A is an aromatic or a heterocyclic ring; Q is a bond, carbonyl, lower alkylene, lower alkenylene, -O...  
JP2005002116A
To provide an α4 (including α4β7) mediated cell adhesion inhibitor effective for treating asthma, diabetes, and pathologic conditions associated with leukocyte invasion in the gastrointestinal tract and other epithelial tissue.A compo...  
JP3596041B2  
JP2004534018A
This invention relates to novel triazolopyrimidines of the formula in which R1, R2, R3, R4and X have the meanings given in the disclosure, to a plurality of processes for preparing these novel substances, and to their use for controlling...  
JP2004534019A
Novel triazolopyrimidines of the formula in which R<1>, R<2>, R<3>, R<4>, X and n have the meanings given in the description, a plurality of processes for preparing these novel substances and their use for controlling unwanted microorgan...  
JP2004533436A
The invention relates to novel triazolopyrimidines of the formula in which R1, R2, R3 and X have the meanings given in the disclosure, and acid addition salts thereof, to a plurality of processes for preparing these novel substances, and...  
JP2004256511A
To provide a reduction reaction process for converting imines to corresponding amines by using α-picoline borane or γ-picoline borane that is stable and easily handleable as a reductant.In this process for reducing imines represented b...  
JP3565878B2
PURPOSE: To obtain new cyclopentane- and -pentene-β-amino acids having antimicrobial and antimitotic actions. CONSTITUTION: The cyclopentane- and -pentene-β-amino acids are compds. of formula I [A, B, D, E, G, L, M and T are each H, ha...  
JP2004524266A
Compounds of formula I: wherein A, B, D, and R are as defined herein and their agriculturally acceptable salts are disclosed as effective insecticides. In addition, compositions comprising an insecticidally effective amount of a compound...  
JP3545338B2
Substituted carbamoylmethyl-azulene derivatives (I) are new. 6-(Substituted carbamoylmethyl)-azulene derivatives of formula (I) and their tautomers, enantiomers, diastereomers, racemates, salts, esters and derivatives which are hydrolyse...  
JP2004518765A
The object of the invention are (p-aminohydroxyphenyl)acrylamide derivatives of general formula (I) or the physiologically tolerated, water-soluble salts thereof and oxidative coloring agents for keratin fibers, containing these compounds.  
JP3529106B2
PURPOSE: To obtain a new antibiotic agent useful for preventing, treating or inhibiting bacterial infectious diseases in warm-blooded animals. CONSTITUTION: This compound is represented by formulae I or II [X is a halogen or trifluoromet...  
JP2004512805A
A process for producing nitrosonium ions is described, in which a nitroxyl compound such as TEMPO is oxidized using an oxidizing agent in the presence of a complex of a transition metal such as Mn, Fe, Cu, and a complexing agent such as ...  
JP2004107320A
To provide a method for producing a functionalized alkoxyamine initiator and its use in radical polymerization process.The invention provides a one-pot process for the production of a functionalized alkoxyamine of general formula (I) (fo...  
JP2004509845A
Novel "bispolyamine" inhibitor compounds of polyamine transport are disclosed. These compounds are useful pharmaceutical agents for treating diseases where it is desired to inhibit polyamine transport or other polyamine binding proteins,...  
JP2004505934A
A process for preparing alkoxyamines in a biphasic medium comprises mixing an ionic liquid, an organic solvent, a metal salt, a ligand for the metal, a halocarbon compound ZX and a nitroxide, keeping the reaction medium stirring at a tem...  
JP2004505125A
An initiator system for radical polymerization, which comprises a combination of compounds of the formulae:  
JP2004051614A
To provide a new vermin-controlling agent, especially an insecticide or acaricide.This vermin-controlling agent contains a substituted amide compound expressed by general formula (1) [wherein, A is carbon atom or the like; G is G-1 or G-...  
JP3492763B2
PURPOSE: To obtain a new platinum complex, capable of manifesting excellent antitumor effects, having high safety, good in water solubility and useful as a therapeutic agent for malignant tumor. CONSTITUTION: This platinum complex is of ...  
JP2004502665A
The present invention is substituted amine s of formula (XV) useful in treating Alzheimer's ease and other similar disease.  
JP2004502664A
The present invention is substituted amine s of formula (XV) useful in treating Alzheimer's ease and other similar disease.  
JP2004502669A
The present invention is substituted amines of formula (X) and of the formula (X') useful in treating Alzheimer's disease and other similar diseases.  
JP3487415B2
To obtain the subject new compound capable of binding to arachidonic acid cascade receptors, having a blood platelet coagulation-inhibiting action and useful for treating thrombosis, arteriosclerosis, or the like. A compound of formula I...  
JP2004500413A
The instant invention provides a process for the selective N-formylation of N-hydroxylamines.  
JP3481623B2
PCT No. PCT/EP93/03597 Sec. 371 Date Jun. 6, 1995 Sec. 102(e) Date Jun. 6, 1995 PCT Filed Dec. 17, 1993 PCT Pub. No. WO94/14757 PCT Pub. Date Jul. 7, 1994Hydroxylamine ethers I I (where X is NO2, CN, halogen, alkyl or haloalkyl, Y is H, ...  
JP2003313157A
To provide a simple and readily prepared system technique being not expensive and capable of delivering an active agent in a wide range.A modified amino acid compound useful in the delivery of the active agent is provided. The active age...  
JP2003531897A
Sterically hindered N-substituted aryloxyamines are prepared by the transition-metal-catalyzed decomposition of diazonium salts in the presence of a sterically hindered nitroxyl radical. These compounds are useful as thermal and light st...  
JP2003531110A
Synthetic methods for lactone-containing compounds such as the discodermolides are provided, as are compounds which mimic the chemical and/or biological activity thereof, and methods and intermediates useful in their preparation.  
JP3382297B2
A process for the preparation of high-purity deferoxamine salts from filtered fermentation liquors containing deferoxamine B as active ingredient by the adsorption of the active ingredient onto an ion exchange resin and the subsequent di...  
JP2003500377A
(57) Summary book invention relates to those use for processing a plant that a plant should be protected against the attack from new halogenated compounds, those production methods, the microbe of vegetable pathogenicity, and an insect. ...  
JP2003500378A
The invention relates to polyalcoxyamines obtained from beta-substituted nitroxides of formula (1) wherein A represents a di- or polyvalent structure, R1 represents a molar mass of more than 15 and is a monovalent radical, and n>2. The i...  
JP2002541197A
Compounds of formula (I) are antibacterial agents:wherein Z represents a radical of formula -N(OH)CH(=O) or of formula -C(=O)NH(OH), and R1-R4 are as defined in the specification. A method for the treatment of bacterial or protozoal infe...  
JP2002537283A
New Phenylalaninol derivatives (I). Phenylalaninol derivatives of formula (I) are new: [Image] X : a benzamide group of formula (i), a heterocyclyl-amide group of formula (ii) or an imidazolin-3-yl-4-one group of formula (iii): [Image] R...  
JP2002537374A
A process for producing nitrosonium ions is described, in which a nitroxyl compound such as TEMPO is oxidized using an oxidizing agent in the presence of a complex of a transition metal such as Mn, Fe, Cu, and a complexing agent such as ...  
JP2002302439A
To obtain an excellent ileum-type bile acid transporter inhibitor containing a cyclobutene derivative, a pharmacologically acceptable salt thereof, or an ester or other derivative thereof.This ileum-type bile acid transporter inhibitor c...  
JP3330374B2
The present invention relates to compounds exhibiting central nervous system (CNS) activity which are useful in the treatment of epilepsy and other CNS disorders. The compounds of this invention have the following general formula: and ph...  
JP2002241355A
To obtain a new compound capable of acting on a central nerve, especially having an antispasmodic action.The compounds are represented by formula (I) [R is an aryl, an aryl lower alkyl group or the like; R1 is hydrogen, a lower alkyl, a ...  
JP3311840B2
PURPOSE: To obtain a 3-halogeno aromatic compound useful as an intermediate for medicines and agrochemicals in high yield while suppressing by-products by subjecting an aromatic compound such as 2-amino-5-trifluoromethylpyridine to speci...  
JP2002522415A
The invention relates to a compound of formula Ia, Ib or IcThe open chain alkoxyamine compounds are useful for the polymerization of ethylenically unsaturated monomers. The compounds of the present invention provide polymeric resin produ...  
JP2002205984A
To develop an insecticide having extremely excellent insecticidal activities against various injurious insects and a novel molecular structure.This N-substituted spirodihydropyrrole derivative is a compound represented by formula (I) (wh...  
JP2002521529A
A compound of formula (I) where R 1 is CH and R 6 is a bond, or R 1 and R 6 together form an electron withdrawing group; R 2 and R 3 are independently selected from (CR 7 R 8 ) n , or a group CR 9 R 10 , -(CR 7 R 8 CR 9 R 10 )- or -(CR 9...  
JP2002521317A
Synthetic methods for lactone-containing compounds such as the discodermolides are provided, as are compounds which mimic the chemical and/or biological activity thereof, and methods and intermediates useful in their preparation.  
JP2002195990A
To provide a carbonyl compound collecting material and a collector tube using it enabling easier and high-precision microanalysis of aldehyde compound without requiring any complicated operation.In this carbonyl compound collecting mater...  
JP2002520306A
Novel salts of N-tert-butylhydroxylamine with lower carboxylic acids are disclosed, together with processes for their preparation. The salts possess advantageous properties that render them useful in synthesis.  

Matches 551 - 600 out of 4,769