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JP4568400B2 |
A process for preparing 5,5'-bi-lH-tetrazolediammonium salts (BHT . 2NH3) maintaining a high yield through oxaldiimidic acid dihydrazide (OAH) from the starting materials which are cheaply available and are easy to handle. The 5,5'-bi-1H...
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JP2009542654T5 |
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JP4503232B2 |
The present invention relates to methods for the prophylaxis, management and treatment of certain diseases modulated by the inhibition of the enzyme malonyl-coenzyme A decarboxylase (malonyl-CoA decarboxylase, MCD) by the administration ...
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JP2010521505A |
Compounds of the formula (I), in which E, R3, R4, R5, X, Y, W, Q1, Q2, Z, s and m have the meanings indicated in claim 1, can be employed, inter alia, for the treatment of tumours.
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JP4485638B2 |
There is provided a process for the preparation of 2-aryl-5-(perfluoroalkyl)pyrrole compounds of formula I from N-Ä1-chloro-1-(perfluoroalkyl)methylÜarylimidoyl chloride compounds. The 2-aryl-5-(perfluoroalkyl)pyrrole compounds are use...
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JP2010520901A |
The present invention is for the 3,4-disubstituted phenoxyphenyl amidine of general formula (I), a method for producing the phenoxyphenyl amidine, the use of the amidine to suppress unwanted microorganisms, and the object comprising said...
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JP2010520900A |
The present invention relates to 3-substituted phenylamidines of the general formula (I), to a process for their preparation, to the use of the amidines according to the invention for controlling unwanted microorganisms and also to a com...
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JP2010520903A |
The substituted phenylamidine has general formula (I). The compound having general formula (I), is new. (I) Y : O, NH or a single bond; R 1> : H, linear or branched 1-12C alkyl, 2-12C alkenyl, 2-12C alkinyl, cyclic 3-8C alkyl, 4-8C alken...
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JP2010520898A |
The use of N2-phenylamidines of formula (I) as herbicides is described. In this formula (I), R2, R3, R4, R5 and R6 are different radicals and A is a bond or various 1- or polyatomic bridging elements.
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JP2010520904A |
The phenoxyphenyl amidine has general formula (I). The phenoxyphenyl amidine having general formula (I), is new. R 1>H, mercapto or methyl, linear or branched 1-8C alkyl, 1-12C alkyl, 2-12C alkenyl, 2-12C alkinyl, cyclic 3-8C alkyl, 4-8C...
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JP2010520899A |
The present invention relates to dihalophenoxyphenylamidine of general formula (I), methods for its preparation, use of the amidine to control unwanted microorganisms and agents for the purpose comprising the phenoxyamidine. The present ...
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JP4478157B2 |
A compound represented by the following general formula (1) or a salt thereof or a hydrate of the foregoing is safe while exhibiting suitable physicochemical stability, and is useful as therapeutic or prophylactic agents for diseases ass...
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JP4469280B2 |
The present invention provides crystalline biphenyl-4-carboxylic acid (R)-(6-(1-((4-fluorobenzyl)methylamino)ethylideneamino)-2(R)
-hydroxyindan-1-yl)amide hemihydrate, compositions thereof, methods of using the same, processes for makin...
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JP4464505B2 |
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JP2010513530A |
Provided are compounds that are modulators of C3a receptor activity, compositions containing the compounds and methods of use of the compounds and compositions. In certain embodiments, the compounds are pyridones. In certain embodiments,...
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JP2010090138A |
To provide a novel substituted tetracycline compound useful to treat numerous tetracycline compound-responsive states such as bacterial infections and neoplasms.The compound is represented by formula (I), wherein X is CH2, CH-alkyl or th...
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JP2010077150A |
To provide methods for prophylaxis, management and treatment of specific diseases modulated by inhibition of enzyme malonyl-coenzyme A decarboxylase (malonyl-CoA decarboxylase, MCD) by administration of a composition containing as an act...
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JP4434595B2 |
New metal complexes of iminohydroxamic acids are claimed. New metal complexes (I) of iminohydroxamic acids are of formula (1). Nu = O, S, NR4asterisk, PR4asterisk; M = Ni, Pd; h = 0-4; X = halo, 1-8C alkyl, 3-12C cycloalkyl, 7-13C aralky...
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JP4428900B2 |
The invention relates to a novel LTB4 antagonist, to a method for the production thereof and to its use as a medicament.
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JP4421818B2 |
An improved process for preparing arylethanoldiamines is described. Compounds of this type are known to be useful as agonists at atypical beta-adrenoceptors (also known as beta-3-adrenoceptors).
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JP4420416B2 |
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JP4414331B2 |
Non-natural amino acids such as 2-alkylated amino acids allow for the synthesis of a wider variety of peptidal and non-peptidal pharmaceutically active agents. A method of preparing a 2-alkyl amino acid involves a Michael-type addition o...
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JP4409290B2 |
The present invention relates to compounds of Formula I: Formula I which are agonists of the M-1 muscarinic receptor.
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JP4405389B2 |
A 1,2,4-Triazole derivative of formula 1 or a non-toxic salt thereof, a preparation method thereof, and a pharmaceutical composition containing the derivative or the salt as an active ingredient are provided.
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JP4393869B2 |
The present invention relates to a group of novel 1H-imidazole derivatives, to methods for the preparation of these compounds, and to pharmaceutical compositions containing one or more of these compounds as an active component. These 1H-...
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JP2009545552A |
The present invention relates to a novel process for preparing amidrazones of the formula (I) wherein R, R1, R2, A, B, W, Y and n have the meanings as indicated in the description. Further, the invention relates to novel compounds used a...
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JP4384617B2 |
The present invention is related to novel intermediates and processes which are useful in the preparation of certain antihistaminic piperidine derivatives of formula (I) wherein W represents -C(=O)- or -CH(OH)-; R 1 represents hydrogen o...
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JP4369978B2 |
Disclosed herein is a benzylformamidine compound having high ultraviolet light absorption and superior thermal stability that can be suitably used as an ultraviolet light absorber for plastic products which undergo high-temperature treat...
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JP4361137B2 |
Battery has an electrolyte comprising a solvent and a salt (I) comprising a hydroxonium, nitrosonium, ammonium, metal, organic or organometallic cation and a 5-membered (hetero)cyclic anion. Battery has an electrolyte comprising a solven...
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JP4356111B2 |
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JP4342178B2 |
Compounds of formula (I) are useful as inhibitors of trypsin like serine protease enzymes such as thrombin, factor VIIa, factor Xa, TF/FVIIa, and trypsin. These compounds could be useful to treat and/or prevent clotting disorders, and as...
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JP2009227655A |
To provide a compound having an excellent controlling effect on pests.Provided are a compound expressed by formula (I) and its agronomically allowable salt having excellent controlling effect on pests. In formula (I), A and E are each in...
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JP2009209090A |
To provide an insecticide which exhibits a high insecticidal effect even in a low dosage.There are provided a compound represented by general formula (1) and an insecticide containing the compound as an active ingredient. In the formula ...
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JP4334016B2 |
PCT No. PCT/EP96/05529 Sec. 371 Date Jul. 31, 1998 Sec. 102(e) Date Jul. 31, 1998 PCT Filed Dec. 11, 1996 PCT Pub. No. WO97/21670 PCT Pub. Date Jun. 19, 1997The invention relates to new phenylamidine derivatives, processes for preparing ...
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JP4320260B2 |
Arylamide derivatives (I) are new. Arylamide derivatives of formula (I) and their salts are new. [Image] X : optionally substituted lower alkylene or alkenylene; G 1O, S or NH; G 2C or N; R aH, halo or optionally substituted alkyl, cyclo...
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JP4320249B2 |
Sulfonamide and urea compounds having an inhibitory effect on Src kinase including enantiomers, stereoisomers and tautomers thereof, as well as pharmaceutically acceptable salts or solvates of said compound, said compound having the gene...
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JP4306806B2 |
3-(Substituted phenyl)-5-(thienyl or furyl)-1,2,4-triazole compounds are useful as insecticides and acaricides. New synthetic procedures and intermediates for preparing the compounds, pesticide compositions containing the compounds, and ...
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JP4288299B2 |
Benzamidine derivatives of formula (I), and their salts, are new: A =O(2-4C alkylene)O or (1-3C alkylene)O; R1 = 1-6C alkyl or halo; R2 = H, 1-6C alkyl or halo; R3, R4 = H, 1-6C alkyl, 1-6C alkoxy, OH, CF3; or R3+R4 = part of a condensed...
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JP4271657B2 |
The invention is concerned with novel mandelic acid derivatives of formula (I) wherein R1 to R10, X and Y are as defined in the description and in the claims, as well as pharmaceutically acceptable salts thereof. These compounds inhibit ...
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JP4267920B2 |
The present invention relates to novel compounds (I), their prodrugs, and the pharmaceutically acceptable salts as well as pharmaceutical compositions containing such compounds useful in treating certain metabolic diseases and diseases m...
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JP4253897B2 |
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JP2009514830A |
The present invention relates to a novel crystalline modification of N-ethyl-2,2-dichloro-1-methylcyclopropane-carboxamide-2-(2,6
-dichloro-alpha,alpha,alpha-trifluoro-p-tolyl)hydrazone, to a process for its preparation and to its use fo...
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JP4243101B2 |
A new and distinct hybrid of artichoke named ‘PS-H2015’, characterized by its numerous bud numbers, fleshiness of bracts, fleshiness of hearts, uniformity of head shapes; strong violet blush coloration; and ability to bolt in warm su...
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JP2009508827A |
The present invention relates to 2,5-di-substituted-4-naphthyloxy-substituted-phenyl-amidine derivatives of formula (I) wherein the substituents are as in the description, their process of preparation, their use as fungicide or insectici...
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JP2009507813A |
The present invention relates to bi-phenyl-amidine derivatives of formula (I) in which the substituents are as in the description, their process of preparation, their use as fungicide or insecticide active agents, particularly in the for...
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JP2009507895A |
The present invention relates to benzyloxy- and phenethyl-substituted phenyl-amidine derivatives of formula (I) wherein the substituents are as in the description, their process of preparation, their use as fungicide or insecticide activ...
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JP2009505973A |
A compound of formula (III): or a salt, solvate and chemically protected form thereof, wherein: R5 is an optionally substituted C5-20 aryl or C4-20alkyl group; L′ is a single bond, —O— or —C(═O)—; A is selected from the group...
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JP2009504913A |
This invention is directed to processes for the formation of ruthenium-containing films on surfaces in atomic layer deposition (ALD) processes. The ALD process includes depositing a surface-activating group on the surface; exposing the d...
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JP4209659B2 |
Amidino derivatives represented by the following general formula (I): {where X is a group represented by R1SO2NR2- (wherein R1 represents optionally substituted C6-14 aryl, etc. and R2 represents hydrogen atom, etc.), etc., Ar1 represent...
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JP2009004374A |
To provide a proton conductor which has a melting point lower than room temperature and a low vapor pressure and a similar conductivity with what can be obtained in an aqueous medium.The proton conductor of a liquid form contains a mixtu...
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