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Matches 701 - 750 out of 1,415

Document Document Title
JP3498372B2
PURPOSE: To obtain a new semicarbazone compound useful as a noxious organism-controlling agent, having excellent insecticidal or germicidal activity at low doses, land having little adverse effects on mammals, fish and beneficial insects...  
JP2004504270A
This invention relates to novel compounds of Formula (I), and compositions thereof, useful in the treatment of disease states mediated by the chemokine, Interleukin-8 (IL-8).  
JP2004043480A
To provide a medicine becoming a treating agent of diabetes mellitus and an intermediate for producing the same.This intermediate of a new 3-aryl-2-hydroxypropionic acid derivative is expressed by formula IV [wherein, Q is H; A is OH, a ...  
JP3491311B2
PURPOSE: To readily obtain an N-substituted-N-arylcyanamide derivative useful as intermediates for agricultural chemicals and medicines, especially herbicides, in high purity and high yield by reacting an N-arylcyanamide derivative with ...  
JP3487415B2
To obtain the subject new compound capable of binding to arachidonic acid cascade receptors, having a blood platelet coagulation-inhibiting action and useful for treating thrombosis, arteriosclerosis, or the like. A compound of formula I...  
JP2004501132A
This invention relates to compounds of the formula (I) which are thyroid receptor ligands, and are preferably selective for the thyroid hormone receptor beta, to methods of preparing such compounds and to methods for using such compounds...  
JP2004500330A
The present invention provides oligomers which are specifically hybridizable with a selected sequence of RNA or DNA wherein at least one of the nucleoside moieties of the oligomer is modified to include a guanidinium group. These oligome...  
JP2003342253A
To provide a method for producing a 2-alkyl-3-nitroisothiourea useful as a raw material for agrochemicals from an S-alkylisothiourea in a high yield. This method for producing the 2-alkyl-3-nitroisothiourea comprises reacting the S-alkyl...  
JP2003535915A
3,4-Dihydroxybenzyl-substituted carbonic acid derivatives (I) are new. Carbonic acid derivatives of formula (I) (including their tautomers) are new. [Image] X1-X3O, S or NR3; R1H, R4, OH or OR4; R4alkyl, alkenyl, 1-oxoalkyl or 1-oxoalken...  
JP2003535868A
New spisulosine derivatives of use in treating tumors are of the formula (I) wherein: each X is the same or different, and represents H, OH, OR', SH, SR', SOR', SO2R', NO2, NH2, NHR', N(R')2, CN, halogen, C(-O)H, C(-O)CH3, CO2H, CO2CH3, ...  
JP2003532705A
A method is provided for inhibiting free radical degradation in the skin of a human or nonhuman animal comprising contacting the skin with a skin treatment composition having a concentration of a 1-(3-methoxybenzyl)-3-substituted thioure...  
JP2003530429A
Methods and compositions for the treatment of pain using thiourea derivatives. Particularly disclosed are new compositions for the treatment of chronic pain, and methods for their use.  
JP2003530430A
Methods and compositions for the treatment of pain using this area derivatives. Particularly disclosed are new compositions for the treatment of chronic pain, and methods for their use.  
JP3457240B2
To provide a method for producing an episulfide compound by epithioation of the corresponding epoxy compound in high yield in such a way that the product episulfide compound does not run to tar. This method for producing an episulfide co...  
JP3446052B2  
JP3444306B2
PURPOSE: To economically and advantageously produce a solution of thiourea dioxide with small loss of chemicals and reduced energy consumption or to effectively bleach papermaking pulp with the produced solution of thiourea dioxide. CONS...  
JP2003525225A
The present invention relates to novel substituted imide derivatives of the general formula (I)in whichR<1 >represents optionally substituted cycloalkyl,R<2 >represents optionally substituted alkyl or optionally substituted cycloalkyl,R<...  
JP2003524574A
[Chemical 1]  
JP2003520843A
The present invention refers to new classes of polymerisable monomers, to molecularly imprinted polymers obtainable by polymerisation of at least one of the monomers and a crosslinking monomer in the presence of a template molecule. The ...  
JP2003146963A
To provide an antioxidation agent for cosmetic and pharmaceutical preparation having strong specific free radical scavenging action and antioxidation action to protect the cells and tissues of mammals and provide a method for the product...  
JP2003103655A
To provide an apparatus and a method for simply detecting and deciding a specific position of a cylindrical film close contact material in which cylindrical films are brought into close contact with each other without mistake.The apparat...  
JP2003513002A5  
JP2003509422A
This invention relates to a compound capable of binding to a picornavirus capsid comprising two or more capsid binding moieties.  
JP3383328B2
PURPOSE: To provide a compsn. useful to inhibit and/or treat infections by HIV and to treat or inhibit AIDS. CONSTITUTION: The compsn. contains as an effective component, a compd. expressed by formula I or its salt, or a compd. expressed...  
JP2003506355A5  
JP2003506355A
Compounds of formula (I), are useful in treating diseases prevented by or ameliorated with potassium channel openers. Also disclosed are potassium channel opening compositions and a method of opening potassium channels in a mammal.  
JP2003506348A
Urea and thiourea derivatives inhibit cell function of the chemokine receptor CCR-3. These compounds offer an effective means for treating a range of diseases thought to be mediated by the CCR-3 receptor. A variety of useful urea and thi...  
JP2003503350A
Compounds that selectively inhibit the binding of ligands to alpha 4 beta 1 integrin (VLA-4) and methods for their preparation are disclosed. In one embodiment, compounds of the invention are represented by formula (I). As selective inhi...  
JP3365633B2
The compounds of the formula (I) (I) in which R1-R4, W, X, Y and Z are as defined in claim 1 are suitable for controlling harmful plants in crops. Their preparation may employ the intermediates of the formulae II and III: (II) (III)  
JP2003500381A
Compounds of formula I are useful for treating conditions associated with hyperglycemia, especially Type II diabetes. These compounds are useful in stimulating the kinase activity of the insulin receptor, activating the insulin receptor,...  
JP3354090B2
To obtain a new benzamide derivative having differentiation inducing acton, useful as a medicine for treating and improving malignant tumor, autoimmune disease, dermatitis and parasitic infectious disease. This compound is shown by formu...  
JP2002540086A
This invention provides combinatorial chemistry libraries containing thiourea and urea compounds. In addition, the invention relates to methods for constructing combinatorial chemistry libraries containing thiourea and urea compounds. Fu...  
JP3350035B2
A process for preparing a compound represented by formula (I), wherein R1 represents straight-chain or branched C1-5 alkyl, C1-5 haloalkyl, or C3-6 cycloalkyl, and R2 represents C1-3 alkyl or C1-3 haloalkyl.  
JP2002332266A
To provide an excellent prophylactic and therapeutic agent for osteoporosis and the like.A compound represented by the following general formula (I) (A=phenyl or the like, B=aryl or the like, X=O or the like, n=0, 1) and a prophylactic a...  
JP2002533301A
Compounds of formula (I) wherein R1-R5 are independently selected from hydrogen, or substituents R9-R12 are independently hydrogen, or substituents provided that at least one of R9-12 is not hydrogen; G is a monocyclic heteroaryl: X is a...  
JP2002532465A
The present invention relates to biphenyl and biphenyl-analogous compounds, their preparation and use as pharmaceutical compositions, as integrin antagonists and in particular for the production of pharmaceutical compositions for the tre...  
JP3330374B2
The present invention relates to compounds exhibiting central nervous system (CNS) activity which are useful in the treatment of epilepsy and other CNS disorders. The compounds of this invention have the following general formula: and ph...  
JP2002531545A
Compounds of formula (I), wherein R1-R5 are independently selected from hydrogen, alkyl of 1 to 6 carbon atoms, alkenyl of 2 to 6 carbon atoms, alkynyl of 2 to 6 carbon atoms, perhaloalkyl of 1 to 6 carbon atoms, cycloalkyl of 3 to 10 ca...  
JP2002531544A
Compounds of formula (I) wherein R1-R5 are independently selected from hydrogen, alkyl of 1 to 6 carbon atoms, alkenyl of 2 to 6 carbon atoms, alkynyl of 2 to 6 carbon atoms, perhaloalkyl of 1 to 6 carbon atoms, cycloalkyl of 3 to 10 car...  
JP2002531557A
Compounds of formula (I) wherein A is heteroaryl; R9-R12 are independently hydrogen, alkyl of 1 to 4 carbon atoms, perhaloalkyl of 1 to 4 carbon atoms, halogen, alkoxy of 1 to 4 carbon atoms, or cyano, or R9 and R10 or R11 and R12 may be...  
JP2002531555A
Compounds having formula (I) wherein R1-R5 are independently selected from hydrogen, alkyl of 1 to 6 carbon atoms, alkenyl of 2 to 6 carbon atoms, alkynyl of 2 to 6 carbon atoms, perhaloalkyl of 1 to 6 carbon atoms, cycloalkyl of 3 to 10...  
JP2002241355A
To obtain a new compound capable of acting on a central nerve, especially having an antispasmodic action.The compounds are represented by formula (I) [R is an aryl, an aryl lower alkyl group or the like; R1 is hydrogen, a lower alkyl, a ...  
JP3309104B2
Sulfonic acid stilbenes are disclosed which block the infection of cells by HSV, HIV and CMV.  
JP2002193924A
To provide a new agent for agricultural and horticultural use.The phenylacetic acid compound represented by formula (1) [A is hydrogen atom, a 1-6C alkyl or the like, B is -NU3U4, Y is hydrogen atom or the like, Z is -OR1 or the like, X ...  
JP2002520387A5  
JP2002517458A
(57) [Summary] Methods for synthesizing large collections of diverse multimeric compounds and iterative processes for assessing key molecular constraints that confer multibinding properties on multimeric compounds are disclosed. A librar...  
JP2002517422A
This invention relates to novel multibinding compounds (agents) that are antibacterial agents. The multibinding compounds of the invention comprise from 2-10 ligands covalently connected by a linker or linkers, wherein each of said ligan...  
JP2002517423A
Disclosed are multibinding compounds which inhibit cyclooxygenase-2 (COX-2), an enzyme which catalyzes the first committed step in the biosynthesis of prostaglandins. The multibinding compounds of this invention containing from 2 to 10 l...  
JP2002517465A
This invention relates to novel multibinding compounds (agents) that are antibacterial agents. The multibinding compounds of the invention comprise from 2-10 ligands covalently connected by a linker or linkers, wherein each of said ligan...  
JP2002513385A
Compounds useful as potassium channel inhibitors and especially useful for the treatment of cardiac arrhythmias and cell proliferative disorders are described.  

Matches 701 - 750 out of 1,415