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Matches 401 - 450 out of 457

Document Document Title
JP2847969B2
A cyclopentene derivative represented by general formula (I) and a pharmaceutically acceptable salt thereof: wherein Ar<1> and Ar<2> represent each independently phenyl, thienyl, pyridyl, indolyl, benzofuranyl or dihydrobenzofuranyl; A r...  
JPH11500717A
The application relates to novel heterocycloalkenes, to a number of processes for their preparation and to their use as fungicide.  
JPH10509140A
Pyrazole derivatives represented by formula (I) and physiologically acceptable salts thereof can suppress the production of both of prostaglandins and leukotrienes simultaneously, and, therefore, exhibit anti-inflammatory and analgesic e...  
JPH10508030A
Antihyperglycemic compounds selected from the group consisting of C-substituted pentacycloazoles and N-alkyl-substituted pentacycloazoles.  
JP2766421B2
The present invention relates to a novel antibacterial compound of formula (I) from the genus Alteromonas and which shares structural similarity with the pseudomonic acids. i  
JP2764784B2
PURPOSE: To provide the subject compound having wide range of vermin controlling effect without giving chemical damage to a cultivated plant and useful as insecticide. CONSTITUTION: The compound is expressed by formula I [A is a 5-member...  
JP2761441B2
The present invention provides certain 3-aryl-5,6-dihydro-1,4,2-ocathiazines and their oxides, useful for the long-term preservation of wood and composite wood materials against wood damaging and wood destroying materials. The present in...  
JPH10504275A
Compounds having the formulawhere R2 is a heteroaryl group linked to the remainder of the molecule via a carbon atom adjacent a nitrogen atom and R4 and R5 are both hydrogen atoms or together represent -SO- or -SO2- and A is C2-C4 alkyle...  
JPH1072444A
To obtain the subject new compound useful as a medicine having a pharmacological activity such as a growth hormone accelerating activity. A benzene condensed lactam derivative expressed by formula I [R1 is a lower alkyl; R3 is H or a low...  
JP2695132B2
PURPOSE: To obtain a new inhibitor which inhibits DNA gyrase activity in bacteria, has antibiotic properties, especially antibacterial activity against microorganisms and is useful for treatment or prophylaxis of infectious diseases. CON...  
JPH09511215A
Heteroarylpiperidines, pyrrolidines, and piperazines of the formula wherein X is -O-, -S-, -NH-, or -N(R 2 )- R 2 is selected from the group consisting of lower alkyl, aryl lower alkyl, aryl, cycloalkyl, aroyl, alkanoyl, alkoxycarbonyl a...  
JPH09221481A
To obtain a medicine comprising a new specific aromatic compound, containing thiazolidine-2,4-dion-5-ylmethyl group, etc., and useful as a therapeutic agent, a preventing agent, etc., for insulin-resistance diseases, hyperglycemia, hyper...  
JP2645962B2
Compounds shown by the above formula or salt thereof show a strong angiotensin II antagonistic activity and hypotensive action and CNS activity, and are useful as therapeutic agents of circulatory diseases such as hypertensive diseases a...  
JP2614981B2
PURPOSE: To provide new compds. having low toxicity, useful for agonist of 5-HT1 like acceptor, such as antimigraine medicine, etc. CONSTITUTION: The compds. have formula I (where R1 is H, halogen, 1-6C alkyl, 1-6C alkoxy, cyano or the l...  
JP2609122B2
A silver halide photographic material containing a compound having a structure represented by formula (I) (I) wherein EAG represents a group capable of accepting an electron from a reducing material; E represents an electron-attracting g...  
JP2610988B2
Novel heterocyclic compounds of the formula (I) wherein A, R<1>, E, Z, X and Y have the meanings as defined in the patent application and the use of the new compounds as insecticides.  
JPH0881463A
To obtain a novel compound that has activity against microorganisms, particularly Gram-positive bacteria, mycobacteria, anaerobic microorganisms and the like with low toxicity and is useful for prevention and treatment of systemic infect...  
JPH07121941B2
This invention relates to certain quinolinyl-benzoheterobicyclic compounds and their use as valuable pharmaceutical agents, particularly as lipoxygenase inhibitors and/or leukotriene antagonists and/or as mediator release inhibitors usef...  
JPH07113021B2
Compounds of formula I: in which R1, R2, R3, R4, R5, R6, R7, X, and n are defined in the description, their optical isomers and their addition salts with a pharmaceutically acceptable base or acid. Medicinal products.  
JPH0791280B2
Aminobenzosultam derivatives as inhibitors of lipoxygenase and useful in the treatment or alleviation of allergic and inflammatory diseases.  
JPH07242664A
PURPOSE: To obtain the subject novel compound having an antagonism against angiotensin II, useful for treatment of hypertension, aldosterone excessiveness, cardiac insufficiency, central nervous system diseases, or the like. CONSTITUTION...  
JPH0780998B2
Electrically conducting homo- and/or copolymers and/or tripolymers can be produced from novel monomers, such as a 3-substituted 2,5-di(2-thienyl)pyrrole. The polymers exhibit unexpectedly high stability and conductivities, and can be fun...  
JPH07173142A
PURPOSE: To obtain the subject novel inhibitor which inhibits the angiotensinogen-cleaving action of a natural proteolytic enzyme, renin, and is useful in treating or preventing renin-associated hypertension, hyperaldosteronism, glaucoma...  
JPH0751564B2
Spirocyclic compounds of the formula: are oxytocin and vasopressin antagonists useful in the treatment of pre-term labor, dysmenorrhea and for the stoppage of labor preparatory to cesarean delivery, timing of parturition, uterine hyperac...  
JPH0699423B2
PCT No. PCT/US91/01470 Sec. 371 Date Nov. 6, 1992 Sec. 102(e) Date Nov. 6, 1992 PCT Filed Mar. 4, 1991 PCT Pub. No. WO91/17156 PCT Pub. Date Nov. 14, 1991.5-(1-Hydroxy-2-piperidinopropyl)-2(1H,3H)-indolone derivatives and analogs; pharma...  
JPH06329637A
PURPOSE: To provide novel compounds useful as active compounds in medicaments, particularly as hypotensor and anti-artherosclerosis agents. CONSTITUTION: A compound of formula I [wherein A represents alkyl, alkenyl, or cycloalkyl; B repr...  
JPH0678339B2  
JPH06237790A
PURPOSE: To obtain an enantiomer of a heterodicyclic alcohol by stereoselectively resolving from its corresponding racemic body through a specific process having no need of an optically active reagent, while converting another enantiomer...  
JPH06507418A
Substituted 1-(2H)-isoquinolinones of the structural formula: (I) are angiotensin II antagonists which are useful in the treatment of hypertension and congestive heart failure.  
JPH06211654A
PURPOSE: To obtain a new compd. having selective affinity for the 5-HT receptor of a brain and much smaller affinity for other receptor and useful to treat motion sickness and emesis. CONSTITUTION: This compd. is represented by formula 1...  
JPH06211655A
PURPOSE: To obtain a new compd. having selective affinity for the 5-HT receptor of a brain and much smaller affinity for other receptor and useful to treat motion sickness and emesis. CONSTITUTION: This compd. is represented by formula 1...  
JPH0629248B2
(A) Bicyclic cpds. of formula (I) and their salts are new; where n = 0 or 1; m = 0-3; X = CH2, O, S, SO, SO2, NH or 1-4C alkylimino; X1 = CH2, O, S, SO or SO2; Y+Y1 = O, or Y = H and Y1 = OH or in-vivo hydrolysable acyloxy; Z = CH2, CHMe...  
JPH0656807A
PURPOSE: To provide a new compd. which is effective to treat, prevent or control renin-associated hypertension, hyperaldosteronism, congestive heart failure and galucoma. CONSTITUTION: This compd., for example a compd. expressed by formu...  
JPH064624B2
Compound of the formula:- wherein R is phenyl or phenyl substituted by one or more substituents selected from nitro, halo, C1-C4 alkyl, C1-C4 alkoxy, aryl(C1-C4 alkoxy), C1-C4 alkylthio, C1-C4 alkylsulphonyl, hydroxy, trifluormethyl and ...  
JPH05320153A
PURPOSE: To provide a new compd. useful as a prophylactic and therapeutic drug for diabetes and hyperglycemic obesity. CONSTITUTION: The compd. is expressed by formula I. In the formula I, R1, R4 are H, 1 to 4C alkyl, 1 to 4C alkoxy, etc...  
JPH05508167A
Compounds of the formula II in which P is hydroxy and T is the group -X2-CR7aR7b-CHR8-OH or T is hydrogen and P is the group O-CHR8-CR7aR7b-X2-OH and, wherein X1, X2, R1, R2, R3, R4, R5, R6, R7a, R7b, and R8 are as defined in the specifi...  
JPH05222005A
PURPOSE: To provide the subject compound which has the ability to inhibit angiotensinogen-cleaving action of the natural proteolytic enzyme, renin and is useful for preventing and treating renin-associated hypertension, hyperaldosteronis...  
JPH0552309B2
Compounds of the formulawherein C' and N4 are in trans configuration to each other, Y is OH, R'COO, R2R3NCOO- or R4O whereby R' is an aliphatic hydrocarbon residue having 1-17 carbon atoms, a phenyl, 2,6-dimethylphenyl or 3- or 4-hydroxy...  
JPH05155867A
PURPOSE: To obtain a new substd. quinazolinone having angiotensin II antagonistic action which is useful for treatment of hypertension and congestive failure. CONSTITUTION: This compd. is a compd. of formula I [wherein L is bonded to J a...  
JPH04234881A
PURPOSE: To provide a novel compd. which is excellent as a selective herbicide by treatments before germination and after germination. CONSTITUTION: This compd. is a triazolopyridine type one expressed by formula I (X, Y and Z are each H...  
JPH04128276A
NEW MATERIAL:The compound of formula I [Z is A, group of formula II, CR2=N, etc., (A is O, S, SO, etc.; R2 and R3 are H, OH, halogen, etc.; R2 and R3 may be independently 3-6C cycloalkyl); R1 is H, 1-5C alkyl, alkanoyl or benzyl; (m) is ...  
JPH04500969A
(57) [Abstract] Since this gazette is application data in front of an electronic application, the data of an abstract is not recorded.  
JPH0316951B2
Title compds. I [Het=aromatic heterocycle R1=H, alkyl, alkanoyl, R2=H, alkenyl, are prepd. Thus, 2-[5-(1-tertiany -butoxyformamide)- 3-(1,2,4-thiacliazolyl) -2-[[(Z)-(tertiarybutoxycarbonyl) methoxyl imino!acetate 2-benzthiazollyl thio e...  
JPH02229157A
NEW MATERIAL:A compound of formula I [X is H, F; Z is formula II (R1 is 1-6C alkyl), formula III (R2, R3, R4 are 1-4C alkyl, N(CH3)2]. EXAMPLE: 2-[2-Chloro-4-fluoro-5-(4,5,6,7,2H-tetrahydroisoindole-1,3-d ione-2-yl) phenyl-4-t-butyl-1,3,...  
JPH01305082A
NEW MATERIAL: Compds. of formula I [wherein R1 is a (substd.) aliphatic, aromatic or alicyclic group; R2 is a (substd.) aliphatic group; and R3 is a (substd.) phenyl group united with a heterocyclic ring]. EXAMPLE: 1-(2,2-Dimethylpropyl)...  
JPS63284173A
NEW MATERIAL:A benzothiazole derivative expressed by formula I [R is 2-(1- methyl)imidazolyl or formula IIWIV; R' is H, NH2, 1W4C alkyl or 1W4C alkylthio; n is 0, 1 or 2]. EXAMPLE: 2-[2'-(5'-Methyl-1',3',4'-thiadiazolyl)thio]benzothiazol...  
JPS6335632B2
A compound of the formula where R<6> is either wherein R' is (C1-C4)alkyl or phenyl; wherein W is hydrogen or halo, and n is 1 or 2; wherein Q is sulfur or oxygen; and V is hydrogen or (C1-C3)alkyl; or wherein Y is sulfur or oxygen; X is...  
JPS62226978A
(57) [Abstract] Since this gazette is application data in front of an electronic application, the data of an abstract is not recorded.  
JPS61280491A
(57) [Abstract] Since this gazette is application data in front of an electronic application, the data of an abstract is not recorded.  
JPS61212568A
Fungicidally active novel piperazinylmethyl-1,2,4-triazolylmethyl-carbinols of the formula in which R represents optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkinyl, optionally substituted cycloal...  

Matches 401 - 450 out of 457