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Matches 951 - 1,000 out of 1,390

Document Document Title
JPH0154344B2  
JPH01272581A
PURPOSE: To obtain the subject compound useful for remedy of chronic hepatitis, nephrotic syndrome, etc., in good recovery by extracting a phellodendron with alcohols, dissolving the extract in water, shaking with a water-insoluble solve...  
JPH01250380A
NEW MATERIAL:The (+)-isomer of the optically active compound of formula I (X1 is halogen; R1 and R2 are lower alkyl), its salt or their hydrate. EXAMPLE: (+)-9-Fluoro-5-methyl-8-(4-methyl-1-piperazinyl)-6,7-dihydro -1,7-dioxo-1 H,5H-benz...  
JPH01226883A
NEW MATERIAL: Compd. of formula I {where R1 is methyl, ethyl, propyl, vinyl, 2-hydroxyethyl or the like; R2 is H, 1-4C alkyl or (5-methyl-2-oxo-1,3-dioxol-4-yl)- methyl; R3 is H or amino; R4 is formula II or III [where (l) is 0-2; (m) is...  
JPH01226818A
PURPOSE: To provide a learning-promoting agent or a mnemonic agent comprising an arylamidoazabicycloalkane and capable of promoting memory of living animals and useful for curing hypomnesia and dysmnesia. CONSTITUTION: This mnemonic agen...  
JPH01224317A
PURPOSE: To provide a cellular antibody production inhibitor having a cellular antibody production-inhibiting action and effective against chronic hepatitis, nephrotic syndrome, etc., by comprising phellodendrine or a salt thereof as an ...  
JPH0141127B2  
JPH01203323A
PURPOSE: To inhibit or suppress the release of histamine from the mast cells of a mammalian by bringing the mast cells into contact with a benzo-C- phenanthridine alkaloid. CONSTITUTION: The mast cells of a mammalian are brought into con...  
JPH01203324A
PURPOSE: To control the alveolar osteoclasis by administering a benzo-C- phenanthridine alkaloid compound to a mammalian having a periodontal disease at a dose for inhibiting osteoclasis and collagenase release. CONSTITUTION: This method...  
JPH01502186A
The invention relates to the use of compounds which act as antagonists of 5-hydroxytryptamine (5-HT) at 5-HT3 receptors for the relief or prevention of a withdrawal syndrome resulting from addiction to a drug or substance of abuse and/or...  
JPH01193268A
NEW MATERIAL:A compound of formula I [R1 is carboxy, amidated carboxy, CN, thiocarbamoyl, tetrazolyi; R7 is H, aryl; R2 is H, OH, alkyl, alkoxy; R3 is R2, alkenyloxy, aryl which may be substituted, arylthio, aroyl, arenesulfonyl; R2 and ...  
JPH1175934A
To soften an impact to a bar-form cosmetic when an external impact is applied to a feeding out container for the bar-form cosmetic, and prevent the bar-form cosmetic from being damaged. This cartridge 7 for bar-form cosmetic is equipped ...  
JPH1165391A
To enhance the cleaning performance of a cleaning member and to prolong the service life thereof by setting the coating width of lubricant with respect to the surface of a photoreceptor to be longer than the length of a cleaning blade br...  
JP01165391A
PURPOSE: To efficiently mass-produce a berberine type alkaloid, by cultivating a plant cell and/or tissue thereof using a culture medium having an ammonium ion concentration of ≥50% based on the total inorganic nitrogen concentration. ...  
JPH01149782A
NEW MATERIAL:A compound expressed by formula I [R is (phenyl substituted) 1W6C alkyl; Y is 2W6C alkylene; Ar is (substituted) phenyl]. EXAMPLE: 3-Cyano-1-ethoxycarbonyl-2-[2-(4-sulfamoylphenyl)ethylamino] -4H- quinolidin-4-one. USE: A re...  
JPH01149784A
NEW MATERIAL:A compound expressed by formula I [R is (phenyl substituted) 1W6C alkyl; Y is single bond or 1W6C alkylene; A is (substituted) 3W7C cycloalkyl or 5-W7-membered saturated heterocyclic ring]. EXAMPLE: 3-Cyano-2-cyclohexylamino...  
JPH01149783A
NEW MATERIAL:A compound expressed by formula I [R is phenyl or (OH substituted) 1W6C alkyl; formula II is a 5-W6-membered heterocyclic ring optionally having 1W2 hetero atoms other than the linked N atom; the heterocyclic ring may have 1...  
JPH01135785A
NEW MATERIAL:A compound expressed by formula I [R represents (phenyl- substituted) 1W6C alkyl; Y represents 1W6C alkylene; B represents single bond or -NH-; Het represents (substituted) 5W6 membered aromatic heterocyclic ring]. EXAMPLE: ...  
JPH01128982A
PURPOSE: To industrially advantageously obtain the subject compd. for antibacterial agents or the like by reacting specified 6-fluorotetrahydroquinoline with an orthoformic ester and 1,3-dioxan-4,6-diones together with a catalyst and the...  
JPH01104014A
PURPOSE: To obtain an antimicrobial agent represented by a specific formula. CONSTITUTION: A compound of formula I (R<1> is an alkyl, an alkenyl, a cycloalkyl, phenyl, etc.; R<2> is a halogen, an alkoxy, a heteroaryl, etc.; R<3> is H, a ...  
JPH01104073A
NEW MATERIAL:Crystallizable monohydrate of N-(1H-tetrazol-5-yl)-phenoxy-4H- quinolizin-4-one-carboxamide sodium salt. USE: An antiallergic drug and antitumor agent having excellent handleability because of extremely excellent water-vapor...  
JPH01103603A
PURPOSE: To provide a photopolymerizable composition which is colorless and is suitable for a photoresist, etc., by incorporating a photopolymerizable nongaseous ethylene series unsaturated compd., 2,4,5-triarylimidazolyl dimer initiator...  
JPS6490184A
NEW MATERIAL:A compound (salt or ester) expressed by formula I [R1 represents cycloalkyl, (substituted)phenyl, etc.; W represents formula II (R2 represents H, lower alkyl, etc.), N, etc.; Z represents formula III (R4WR6 repre sent H, low...  
JPS6483080A
NEW MATERIAL:The compound of formula I (R1 is lower alkyl, R2 is halogen, lower alkyl, lower alkoxy, OH, NO2, NH2, acylamino, lower alkylthio, phenyl, benzoyl, benzyloxy or methylenedioxy; n is 0W3). EXAMPLE: 3-Cyano-1-ethoxycarbonyl-2-p...  
JPH0116836B2  
JPS6475470A
NEW MATERIAL:A diphenylamine derivative shown by formula I [X is -(CH2)2- or -(CH2)3; R1, R2 and R3 are H or alkyl; R6, R7 and R8 are individually H or R1 and R6, R2 and R7 or R3 and R8 may be bonded to give -(CH2)2 or -(CH2)2; R4 and R5...  
JPH0113696B2
1,2,3,4,4a,4b,5,6,7,8,8a,12b-Dodecahydro-7-(oxo, hydroxy or amino)-9-hydroxy-11-(alkyl, alkoxy or alkoxyalkyl)triphenylenes, 2,3,3a,3b,4,5,6,7,7a,11b-decahydro-6-(oxo, hydroxy or amino)-8-hydroxy-10-(alkyl, alkoxy or alkoxyalkyl)-1H-cycl...  
JPS6412264B2  
JPS6450884A
NEW MATERIAL: The compd. of formulas I, II {Z is formulas III to V [(n) is 0 or 1; R5 and R6 are H, methyl, benzyl, etc., when R6 is H, n=1; R7 to R9 are H or methyl, when R6 is H, at least one of R8, R9 is methyl, R10 is methyl, ethyl, ...  
JPS6410514B2  
JPS647996B2
NEW MATERIAL:A compound of formulaI(R<1> is H, lower alkyl; R<2> is H, halogen; R<3> is H, lower alkyl, lower alkoxy, hydroxyl; n is 1,2; Z is O, S, methylene). EXAMPLE:9-Fluoro-8-(4-hydroxy-1-piperidyl)-5-methyl-6,7-dihy dro-oxo-1H ,5H-...  
JPS645024B2  
JPS643181A
NEW MATERIAL:A compound (salt or ester) expressed by formula I [R1 is lower alkyl, phenyl, etc.; R2 is lower alkyl; R3 and R4 are H or lower alkyl; A is N or expressed by the formula C-R6 (R6 is H, methyl, etc.)] or formula II (R5 is H o...  
JPS63313744A
1,2,3,4,4a,4b,5,6,7,8,8a,12b-Dodecahydro-7-(oxo, hydroxy or amino)-9-hydroxy-11-(alkyl, alkoxy or alkoxyalkyl)triphenylenes, 2,3,3a,3b,4,5,6,7,7a,11b-decahydro-6-(oxo, hydroxy or amino)-8-hydroxy-10-(alkyl, alkoxy or alkoxyalkyl)-1H-cycl...  
JPS63313786A
1,2,3,4,4a,4b,5,6,7,8,8a,12b-Dodecahydro-7-(oxo, hydroxy or amino)-9-hydroxy-11-(alkyl, alkoxy or alkoxyalkyl)triphenylenes, 2,3,3a,3b,4,5,6,7,7a,11b-decahydro-6-(oxo, hydroxy or amino)-8-hydroxy-10-(alkyl, alkoxy or alkoxyalkyl)-1H-cycl...  
JPS6361941B2
NEW MATERIAL:A quinoline derivative of formula I (R<1> is lower alkyl; R<2> is halogen, nitro, amino, or lower alkanoylamino; R<3> is halogen or hydroxy) and its salt. EXAMPLE:5-Nitro-6-chloroquinaldine. USE:An antimicrobial agent and an...  
JPS63503223A  
JPS6360006B2
A perfluorobicyclo compound emulsion preparation having oxygen carrying ability containing a perfluorobicyclo compound of the general formula: wherein R represents a perfluoromethyl group or perfluoroethyl group, as an oxygen carrying co...  
JPS63284174A
NEW MATERIAL:A compound expressed by formula I [R1 is carboxy, amidated carboxy, CN, thiocarbamoyl or tetrazolyl; R7 is H or aryl; R2 is H, OH, alkyl or alkoxy; R3 is R2, alkenyloxy, (substituted) aryl, arylthio, aroyl, aralkyl, etc.; R2...  
JPS6358834B2
A perfluorobicyclo compound of the general formula: wherein either or both of Ring A and Ring B may optionally be substituted with lower perfluoroalkyl group(s) and m and n each represent 3 or 4.  
JPS63280068A
Solutions of quinolonecarboxylic acids for parenteral administration, of the formula I …… in which R<1>, R<2>, R<3>, X and A have the meaning given in the description, and a process for their preparation.  
JPS6357432B2  
JPS6351675B2
The invention relates to the enzyme S-tetrahydroprotoberberineoxidase, which oxidizes selectively S-tetrahydroprotoberberines and S-1-benzyl-1,2,3,4-tetrahydroisoquinoline in the presence of oxygen, resulting in the corresponding protobe...  
JPS63239269A
NEW MATERIAL:1,4-Dihydro-4-oxoquinoline of formula I (X, Y are identical or different and F or Cl). EXAMPLE: 8-Bromo-5-chloro-6-fluoro-4-oxo-1,4-dihydroquinoline. USE: It is used as a synthetic intermediate of a novel antibacterial, 9-ha...  
JPS63239268A
NEW MATERIAL:1,2,3,4-Tetrahydro-4-oxoquinoline compound of formula I (R1 is methyl, ethyl; X, Y is F, Cl). EXAMPLE: 5,6-Difluoro-2-methyl-4-oxo-1,2,3,4-tetrahydroquinoline. USE: It is used as a synthetic intermediate of 9-halogeno-5-alky...  
JPS63238072A
4-Chlorooxazole derivatives of the formula I …… which in the 2- or 5-position carry unsaturated groups, such as the -CH=CH- or -CH=CH-CH=CH- group. …R1 denotes phenyl which is optionally mono- or polysubstituted by (C1-C4)-alko...  
JPS63225375A
NEW MATERIAL:The quinolizinone derivative of formula I {R1 is carboxy; R2 is H or halogen; R3 is A-R4 {A is lower alkylene; R4 is NH2, OH, arylthio, arylsulfinyl or NHSO2R5 [R5 is group of formula II (X is H, halogen, alkoxy, etc.; Y is ...  
JPS6344156B2  
JPS6344157B2
NEW MATERIAL:Benzo[ij]quinolidine-2-carboxylic acid derivatives of formula I (R<1> is Br; R<2> is Cl, F) and their salts. EXAMPLE:9-Fluoro-8-bromo-5-methyl-6, 7-dihydro-1-oxo-1H, 5H-benzo[ ij ]quinolidine-2-carboxylic acid. USE:Antibacte...  
JPS63201126A
PURPOSE: To obtain the titled remedy having low toxicity, high safety and long-acting activity to suppress the production of immunoglobulin E antibody and useful as a remedy for bronchial asthma, by using a 4H-quinolizin-4-one derivative...  

Matches 951 - 1,000 out of 1,390