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Patent Searching and Data

Document Type and Number:
Japanese Patent JP2006508985
Kind Code:
A method for modifying at least one non-ester-containing parent compound, and the compounds produced using such method, which compounds are deployed to temporarily incapacitate at least one subject are disclosed. The modified compounds are rapidly metabolized to inactive and non-toxic metabolites when exposure to the modified compounds is halted. One or more of a predetermined chemical arrangement is incorporated into the parent compound having the formula: phi-R-X-R'; where phi is a phenyl, substituted aryl or heteroaryl system present in the parent compound or is added to the parent compound; R is an alkyl or alkene containing chain either branched or unbranched from 0 to 10 carbons present in the parent compound or is added to phi; X is a carboxyl, sulfoxyl or phosphatyl function added to R; and, R' is an alkyl, alkenyl or aralkyl group either branched or unbranched containing from 1 to 10 carbons is added to X in a metabolically labile manner, or is a structural element already present as an inherent portion of the parent compound that is connected to X in a metabolically labile manner.

Airhart, Paul W
Application Number:
Publication Date:
March 16, 2006
Filing Date:
November 17, 2003
Export Citation:
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The University of Toledo
International Classes:
A61K31/4535; C07D499/68; A61K31/185; A61K31/195; A61K31/216; A61K31/235; A61K31/245; A61K31/255; A61K31/277; A61K31/325; A61K31/401; A61K31/4025; A61K31/405; A61K31/4166; A61K31/4168; A61K31/421; A61K31/426; A61K31/43; A61K31/4422; A61K31/454; A61K31/46; A61K31/517; A61K31/519; A61K31/522; A61K31/55; A61K31/58; A61K31/65; A61K31/66; A61K45/00; A61K47/48; A61P9/06; A61P17/02; A61P17/06; A61P25/02; A61P25/20; A61P29/00; A61P31/10; A61P35/00; A61P43/00; C07C217/40; C07C219/10; C07C219/14; C07C229/60; C07C237/04; C07D207/16; C07D209/26; C07D209/28; C07D211/90; C07D223/22; C07D233/26; C07D233/50; C07D233/76; C07D261/16; C07D277/20; C07D277/56; C07D295/14; C07D401/06; C07D405/12; C07D407/06; C07D451/06; C07D451/10; C07D473/06; C07D475/08; C07D501/22; C07J43/00; A61K47/46
Attorney, Agent or Firm:
Kazuo Shamoto
Tadashi Masui
Yasushi Kobayashi
Akio Chiba
Hiroyuki Tomita
Nakamura Yoshiya