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Title:
【発明の名称】エンケファリナーゼ及びACEの阻害剤として有用な新規なメルカプトアセチルアミドピリダゾ[1,2]ピリダジン、ピラゾロ[1,2]ピリダジン、ピリダゾ[1,2‐a][1,2]ジアゼピン、及びピラゾロ[1,2‐a][1,2]ジアゼピン誘導体類
Document Type and Number:
Japanese Patent JPH07506832
Kind Code:
A
Abstract:
The present invention relates to certain novel mercaptoacetylamido pyridazo[1,2]pyridazine, pyrazolo[1,2]pyridazine, pyridazo[1,2- a] [1,2]diazepine and pyrazolo[1,2- a ][1,2]diazepine derivatives useful as inhibitors of enkephalinase and of ACE.

Inventors:
Flyin, Gary A.
Siam, Patrick W.
Application Number:
JP52023593A
Publication Date:
July 27, 1995
Filing Date:
April 21, 1993
Export Citation:
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Assignee:
Merrell Dow Pharmaceuticals Inc.
International Classes:
A61K31/415; A61K31/50; A61K31/5025; A61K31/55; A61P7/10; A61P9/00; A61P9/12; A61P25/04; A61P25/24; A61P25/28; A61P43/00; C07D487/04; C07K5/078; A61K38/00; (IPC1-7): C07D487/04; A61K31/415; A61K31/50; A61K31/55; C07D487/04
Attorney, Agent or Firm:
Katsuro Sasai



 
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