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Title:
二重作用性降圧剤
Document Type and Number:
Japanese Patent JP2010538071
Kind Code:
A
Abstract:
The invention relates to compounds having the formula: wherein: Ar, r, R3, Z, X, and R5-7 are as defined in the specification, or a pharmaceutically acceptable salt thereof. These compounds have AT1 receptor antagonist activity and neprilysin inhibition activity. The invention also relates to pharmaceutical compositions comprising such compounds; methods of using such compounds; and process and intermediates for preparing such compounds.

Inventors:
Choi, Suk-ki
Fathery, Paul Earl.
Gendron, Roland
Hudson, ryan
McKinell, Robert Murray
Sasikmar, Bibeck
Application Number:
JP2010524042A
Publication Date:
December 09, 2010
Filing Date:
September 05, 2008
Export Citation:
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Assignee:
Theravans, Incorporated
International Classes:
C07C239/14; A61K31/192; A61K31/401; A61K31/41; A61K38/00; A61K45/00; A61P9/04; A61P9/12; A61P43/00; C07C237/08; C07C237/10; C07C237/12; C07C319/12; C07C323/41; C07D207/16; C07D257/04; C07D403/12
Domestic Patent References:
JPH0748360A1995-02-21
JPH06184086A1994-07-05
JP2003048874A2003-02-21
JP2010518003A2010-05-27
Attorney, Agent or Firm:
Hidesaku Yamamoto
Takaaki Yasumura
Natsuki Morishita