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Title:
ESTROGENIC COMPOUND AS ANTI-MITOTIC AGENT
Document Type and Number:
Japanese Patent JP2008120839
Kind Code:
A
Abstract:

To provide a compound useful for treating mammalian diseases characterized by undesired cell mitosis.

A new estradiol derivative binds to tubulin, inhibits microtubule formation or exhibits anti-mitotic properties.


Inventors:
D AMATO ROBERT JOHN
FOLKMAN MOSES JUDAH
Application Number:
JP2008041709A
Publication Date:
May 29, 2008
Filing Date:
February 22, 2008
Export Citation:
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Assignee:
CHILDRENS MEDICAL CT CORP
International Classes:
A61K31/565; A61K31/05; A61K31/27; A61K31/56; A61K31/567; A61K31/59; A61P5/30; A61P9/00; A61P9/10; A61P17/02; A61P19/02; A61P19/06; A61P25/00; A61P25/02; A61P27/02; A61P27/16; A61P29/00; A61P35/00; A61P37/00; A61P43/00; C07J1/00; C07J3/00; C07J5/00; C07J7/00; C07J9/00; C07J13/00; C07J31/00; C07J41/00; C07J63/00
Foreign References:
WO1993010141A21993-05-27
Attorney, Agent or Firm:
Yoshiyuki Kawaguchi
Hidemi Matsukura
Mayuko Wakuda
Tsutomu Toyama