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Title:
ETHENE DERIVATIVE
Document Type and Number:
Japanese Patent JPS6187653
Kind Code:
A
Abstract:
Ethene derivatives of the formula: [R5(R1CR4=CR2R3)m]n I wherein R5 represents optionally substituted heterocyclyl or a group -CR4=CR2R3, or optionally substituted aryl, heterocyclylalkyl or arylalkyl and R1 represents -NR6- wherein R6 represents hydrogen or optionally substituted alkyl or aryl, or R5 represents a quinonoidal group, and R1 represents =N-, R4 represents hydrogen, alkoxy, alkylthio, trifluoromethyl or optionally substituted alkyl or aryl, R2 represents cyano, formyl, alkoxycarbonyl, alkylsulphonyl, dialkylcarbamoyl, dialkylthiocarbamoyl, aryloxycarbonyl, arylsulphinyl or arylsulphonyl, R3 represents a group R2 or hydrogen, nitro or optionally substituted aryl or aroyl or alkanoyl, and m and n are 1 or 2, and pharmaceutically acceptable salts thereof, with the exclusion of certain compounds in which R5 represents pyridyl, 5-halogenopyrid-2-yl or 1,2,4-triazolo[4,3-a]-quinoline possess useful pharmacological properties.

Inventors:
ADONAN HATSUSAN ARUUSHIYAAA
BAABARA JIYOISU BUROOTON
ROBAATO KIISU CHIENBAAZU
DEIBITSUDO UIRUKINSON GIRUMOA
DAIAN MONITSUKU KERUSHII
PIITAA ROUDEN
EDOWAADO RUNTO
DEIBITSUDO JIYON RISUGOU
IAN MAKURENAGAN
RIBAATO KURINTON SOONDAAZU
KIISU ARUFURETSUDO JIEIMUZU SU
PIITAA JIEIMUZU UOON
Application Number:
JP19962985A
Publication Date:
May 06, 1986
Filing Date:
September 11, 1985
Export Citation:
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Assignee:
MAY & BAKER LTD
International Classes:
A61K31/135; A61K31/165; A61K31/195; A61K31/21; A61K31/22; A61K31/275; A61K31/34; A61K31/341; A61K31/357; A61K31/40; A61K31/403; A61K31/4035; A61K31/415; A61K31/44; A61K31/4402; A61K31/4406; A61K31/4409; A61K31/4418; A61K31/4425; A61K31/455; A61K31/47; A61K31/472; A61K31/495; A61P9/00; A61P11/00; A61P17/00; A61P25/28; A61P29/00; A61P37/00; A61P37/08; C07C67/00; C07C229/30; C07C231/00; C07C231/12; C07C233/43; C07C233/54; C07C237/30; C07C253/00; C07C255/30; C07C301/00; C07C303/40; C07C311/16; C07C313/00; C07C317/14; C07C317/32; C07C323/22; C07C323/54; C07C323/58; C07C323/60; C07C323/65; C07C323/67; C07D209/48; C07D213/74; C07D213/82; C07D215/06; C07D215/38; C07D215/42; C07D217/22; C07D231/38; C07D239/14; C07D239/42; C07D241/20; C07D241/26; C07D249/04; C07D249/14; C07D253/07; C07D257/06; C07D275/03; C07D277/20; C07D277/42; C07D277/82; C07D285/12; C07D285/135; C07D295/12; C07D295/30; C07D307/66; C07D317/46; C07D317/66; C07D471/04; C07D473/34; C07D521/00; C07D275/02; (IPC1-7): C07C101/28; A61K31/135; A61K31/165; A61K31/21; A61K31/275; A61K31/34; A61K31/40; A61K31/415; A61K31/44; A61K31/455; A61K31/47; A61K31/495; C07C103/44; C07C121/45; C07C121/78; C07C143/78; C07C147/04; C07C147/06; C07C149/40; C07D209/48; C07D213/74; C07D213/82; C07D215/38; C07D215/42; C07D217/22; C07D231/38; C07D239/42; C07D241/20; C07D277/42; C07D295/12; C07D307/66; C07D317/46; C07D473/34; C07D521/00