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Title:
固体薬物剤形
Document Type and Number:
Japanese Patent JP5498411
Kind Code:
B2
Abstract:
A solid pharmaceutical dosage form providing improved oral bioavailability is disclosed for inhibitors of HIV protease. In particular, the dosage form comprises a solid dispersion of at least one HIV protease inhibitor in at least one pharmaceutically acceptable water-soluble polymer and at least one pharmaceutically acceptable surfactant.

Inventors:
Jörg Rosenberg
Ulrich Reinhold
Bernd Riport
Gunter Derndl
Jerck Breitenbach
Raman Alanie
Sumo Gite Gauille
Application Number:
JP2011032972A
Publication Date:
May 21, 2014
Filing Date:
February 18, 2011
Export Citation:
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Assignee:
AbbVie Incorporated
International Classes:
A61K31/427; A61K9/14; A61K9/20; A61K9/28; A61K31/425; A61K31/513; A61K47/14; A61K47/32; A61K47/34; A61P31/18; A61P43/00
Domestic Patent References:
JP2003513904A
JP2002524150A
Foreign References:
WO2001034119A1
WO2003063833A1
Other References:
Pharmaceutical Research,1996年,Vol.13, No.9,S-351,PDD7475
Attorney, Agent or Firm:
Kawaguchi International Patent Office