Title:
AMIDINOPHENYLPYRUVIC ACID DERIVATIVE
Document Type and Number:
WIPO Patent Application WO/2001/042199
Kind Code:
A1
Abstract:
An amidinophenylpyruvic acid derivative represented by the following formula, its analogs and pharmaceutically acceptable salts thereof which have an excellent effect of inhibiting activated blood coagulation factor VII.
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Inventors:
SUGIKI MASAYUKI (JP)
SAGI KAZUYUKI (JP)
FUJITA KOHICHI (JP)
KAYAHARA TAKASHI (JP)
TAKEHANA SHUNJI (JP)
SAKURAI KUNIYA (JP)
TASHIRO KAZUMI (JP)
SAGI KAZUYUKI (JP)
FUJITA KOHICHI (JP)
KAYAHARA TAKASHI (JP)
TAKEHANA SHUNJI (JP)
SAKURAI KUNIYA (JP)
TASHIRO KAZUMI (JP)
Application Number:
PCT/JP2000/008569
Publication Date:
June 14, 2001
Filing Date:
December 04, 2000
Export Citation:
Assignee:
AJINOMOTO KK (JP)
SUGIKI MASAYUKI (JP)
SAGI KAZUYUKI (JP)
FUJITA KOHICHI (JP)
KAYAHARA TAKASHI (JP)
TAKEHANA SHUNJI (JP)
SAKURAI KUNIYA (JP)
TASHIRO KAZUMI (JP)
SUGIKI MASAYUKI (JP)
SAGI KAZUYUKI (JP)
FUJITA KOHICHI (JP)
KAYAHARA TAKASHI (JP)
TAKEHANA SHUNJI (JP)
SAKURAI KUNIYA (JP)
TASHIRO KAZUMI (JP)
International Classes:
A61P7/02; A61P9/10; A61P43/00; C07C257/18; C07C279/14; C07C279/18; C07C279/22; C07D213/56; C07D213/73; C07D215/48; C07D233/60; C07D235/08; C07D235/30; C07D239/84; C07D277/64; C07D277/82; C07D307/79; C07D333/24; C07D333/38; C07D401/04; C07D521/00; (IPC1-7): C07C257/18; C07C279/14; C07C279/22; C07D215/48; C07D235/30; C07D235/08; C07D333/40; C07D333/24; C07D215/58; C07D213/74; C07D401/04; C07D277/82; C07D277/64; C07D233/60; C07D239/84; A61K31/166; A61K31/197; A61K31/47; A61K31/4184; A61K31/381; A61K31/44; A61K31/4453; A61K31/4545; A61K31/428; A61K31/4164; A61K31/517; A61P43/00; A61P7/02; A61P9/10
Domestic Patent References:
WO1998031661A1 | 1998-07-23 | |||
WO1999064392A1 | 1999-12-16 |
Foreign References:
Other References:
See also references of EP 1236712A4
Attorney, Agent or Firm:
Nakamura, Minoru (Shin-Tokyo Bldg 3-1 Marunouchi 3-Chome Chiyoda-Ku, Tokyo, JP)
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